pentamidine and quinacrine

pentamidine has been researched along with quinacrine in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19902 (12.50)18.7374
1990's0 (0.00)18.2507
2000's6 (37.50)29.6817
2010's7 (43.75)24.3611
2020's1 (6.25)2.80

Authors

AuthorsStudies
Chibale, K; Croft, SL; Fairlamb, AH; Haupt, H; Kendrick, H; Saravanamuthu, A; Yardley, V1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Lombardo, F; Obach, RS; Waters, NJ1
Adrián, F; Anderson, P; Brinker, A; Caldwell, JS; Chatterjee, A; Gray, NS; Henson, K; Janes, J; Kato, N; Kuhen, K; Matzen, JT; McNamara, C; Nagle, A; Nam, TG; Plouffe, D; Schultz, PG; Trager, R; Winzeler, EA; Yan, SF; Zhou, Y1
González-Díaz, H; Orallo, F; Quezada, E; Santana, L; Uriarte, E; Viña, D; Yáñez, M1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Barnes, SW; Bonamy, GM; Bopp, SE; Borboa, R; Bright, AT; Chatterjee, A; Che, J; Cohen, S; Dharia, NV; Diagana, TT; Fidock, DA; Froissard, P; Gagaring, K; Gettayacamin, M; Glynne, RJ; Gordon, P; Groessl, T; Kato, N; Kuhen, KL; Lee, MC; Mazier, D; McNamara, CW; Meister, S; Nagle, A; Nam, TG; Plouffe, DM; Richmond, W; Roland, J; Rottmann, M; Sattabongkot, J; Schultz, PG; Tuntland, T; Walker, JR; Winzeler, EA; Wu, T; Zhou, B; Zhou, Y1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Brun, R; Buckner, FS; Chatterjee, AK; Creason, SA; Duster, NA; Gelb, MH; Gillespie, JR; Glynne, R; Hulverson, MA; McQueen, J; Molteni, V; Nagendar, P; Nagle, A; Norcross, NR; Ranade, RM; Supek, F; Tatipaka, HB; Wenzler, T1
Barros-Álvarez, X; Buckner, FS; Creason, SA; Fan, E; Gillespie, JR; Hol, WGJ; Huang, W; Koh, CY; Ranade, RM; Shibata, S; Verlinde, CLMJ; Zhang, Z1
Buckner, FS; Gelb, MH; Gillespie, JR; Herbst, ZM; Montanari, CA; Nguyen, UTT; Ranade, RM; Silva, DG1
Buckner, FS; Faghih, O; Gelb, MH; Gillespie, JR; Herbst, ZM; Molasky, NMR; Nagendar, P; Ranade, RM; Turner, RM1
Barros-Álvarez, X; Buckner, FS; Choy, RKM; de Hostos, E; Faghih, O; Fan, E; Gillespie, JR; Hol, WGJ; Huang, W; Molasky, NMR; Mushtaq, A; Ranade, RM; Shibata, S; Verlinde, CLMJ; Zhang, Z1
Mattock, NM; Peters, W1
Musil, R; Wachtler, F1
Chan, KF; Chan, TH; Chow, LM; Wong, IL; Zhao, Y1

Other Studies

16 other study(ies) available for pentamidine and quinacrine

ArticleYear
Antiprotozoal and cytotoxicity evaluation of sulfonamide and urea analogues of quinacrine.
    Bioorganic & medicinal chemistry letters, 2001, Oct-08, Volume: 11, Issue:19

    Topics: Animals; Antiprotozoal Agents; Leishmania; Parasitic Sensitivity Tests; Plasmodium; Quinacrine; Sulfonamides; Trypanosoma; Urea

2001
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
In silico activity profiling reveals the mechanism of action of antimalarials discovered in a high-throughput screen.
    Proceedings of the National Academy of Sciences of the United States of America, 2008, Jul-01, Volume: 105, Issue:26

    Topics: Animals; Antimalarials; Cluster Analysis; Computational Biology; Drug Evaluation, Preclinical; Drug Resistance; Folic Acid Antagonists; Malaria; Models, Molecular; Parasites; Plasmodium falciparum; Reproducibility of Results; Structure-Activity Relationship; Tetrahydrofolate Dehydrogenase

2008
Quantitative structure-activity relationship and complex network approach to monoamine oxidase A and B inhibitors.
    Journal of medicinal chemistry, 2008, Nov-13, Volume: 51, Issue:21

    Topics: Computational Biology; Drug Design; Humans; Isoenzymes; Molecular Structure; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Quantitative Structure-Activity Relationship

2008
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Imaging of Plasmodium liver stages to drive next-generation antimalarial drug discovery.
    Science (New York, N.Y.), 2011, Dec-09, Volume: 334, Issue:6061

    Topics: Animals; Antimalarials; Cell Line, Tumor; Drug Discovery; Drug Evaluation, Preclinical; Drug Resistance; Erythrocytes; Humans; Imidazoles; Liver; Malaria; Mice; Mice, Inbred BALB C; Molecular Structure; Piperazines; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Plasmodium yoelii; Polymorphism, Single Nucleotide; Protozoan Proteins; Random Allocation; Small Molecule Libraries; Sporozoites

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Substituted 2-phenylimidazopyridines: a new class of drug leads for human African trypanosomiasis.
    Journal of medicinal chemistry, 2014, Feb-13, Volume: 57, Issue:3

    Topics: Administration, Oral; Animals; Biological Availability; Cell Line, Tumor; Cell Membrane Permeability; Databases, Chemical; Dogs; Female; Humans; Imidazoles; Madin Darby Canine Kidney Cells; Mice; Microsomes, Liver; Pyridines; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2014
Structure-guided design of novel Trypanosoma brucei Methionyl-tRNA synthetase inhibitors.
    European journal of medicinal chemistry, 2016, Nov-29, Volume: 124

    Topics: Animals; Brain; Chemistry Techniques, Synthetic; Drug Design; Enzyme Inhibitors; Hep G2 Cells; Humans; Methionine-tRNA Ligase; Mice; Permeability; Protein Conformation; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei

2016
New Class of Antitrypanosomal Agents Based on Imidazopyridines.
    ACS medicinal chemistry letters, 2017, Jul-13, Volume: 8, Issue:7

    Topics:

2017
Triazolopyrimidines and Imidazopyridines: Structure-Activity Relationships and in Vivo Efficacy for Trypanosomiasis.
    ACS medicinal chemistry letters, 2019, Jan-10, Volume: 10, Issue:1

    Topics:

2019
Structure-guided discovery of selective methionyl-tRNA synthetase inhibitors with potent activity against
    RSC medicinal chemistry, 2020, Aug-01, Volume: 11, Issue:8

    Topics:

2020
The experimental chemotherapy of leishmaniasis. II. The activity in tissue culture of some antiparasitic and antimicrobial compounds in clinical use.
    Annals of tropical medicine and parasitology, 1975, Volume: 69, Issue:3

    Topics: Aminoquinolines; Animals; Anti-Bacterial Agents; Antimalarials; Antimony; Antiprotozoal Agents; Ascitic Fluid; Cell Line; Chloroquine; Cricetinae; Culture Techniques; Dogs; Drug Evaluation, Preclinical; Folic Acid Antagonists; Leishmania; Niridazole; Pentamidine; Primaquine; Quinacrine; Quinine; Sarcoma; Sulfonamides; Sulfones; Suramin

1975
On the structure and polymorphism of the human chromosome no. 15.
    Human genetics, 1980, Volume: 56, Issue:1

    Topics: Chromosome Banding; Chromosomes, Human, 13-15; Humans; Pentamidine; Plicamycin; Polymorphism, Genetic; Quinacrine; Silver; Staining and Labeling

1980
Quinacrine and a novel apigenin dimer can synergistically increase the pentamidine susceptibility of the protozoan parasite Leishmania.
    The Journal of antimicrobial chemotherapy, 2009, Volume: 63, Issue:6

    Topics: Animals; Antiprotozoal Agents; Apigenin; Drug Resistance; Drug Synergism; Inhibitory Concentration 50; Leishmania donovani; Leishmania enriettii; Pentamidine; Quinacrine

2009