pentagastrin has been researched along with l 365260 in 32 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 1 (3.13) | 18.7374 |
| 1990's | 29 (90.63) | 18.2507 |
| 2000's | 1 (3.13) | 29.6817 |
| 2010's | 1 (3.13) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Drysdale, MJ; Horwell, DC; Pritchard, MC | 1 |
| Horwell, DC; Hughes, J; Hunter, JC; Pritchard, MC; Richardson, RS; Roberts, E; Woodruff, GN | 1 |
| Boden, PR; Higginbottom, M; Hill, DR; Horwell, DC; Hughes, J; Rees, DC; Roberts, E; Singh, L; Suman-Chauhan, N; Woodruff, GN | 1 |
| Honda, K; Ito, H; Kamato, T; Miyata, K; Nishida, A; Tsutsumi, R; Yamano, M; Yuki, H | 1 |
| Arnold, R; Bothe-Sandfort, E; Eissele, R; Koop, H | 1 |
| Harro, J; Männistö, PT; Peuranen, E; Vasar, E | 1 |
| Field, MJ; Hughes, J; Menzies, R; Oles, RJ; Singh, L; Vass, CA; Woodruff, GN | 1 |
| Ameglio, PJ; McHugh, PR; Moran, TH; Schwartz, GJ | 1 |
| Elliott, KJ; Hirst, BH; Ryder, H; Szelke, M | 1 |
| Field, MJ; Hughes, J; Lewis, AS; Singh, L; Woodruff, GN | 1 |
| Barnes, S; Hughes, J; Marshall, FH; Pinnock, RD | 1 |
| Chang, RS; Lotti, VJ | 1 |
| Challenor, J; Lines, C; Traub, M | 1 |
| Fantaskey, AP; Liu, G; Smith, JP; Zagon, IS | 1 |
| Bishop, LA; Black, JW; Gerskowitch, VP; Hull, RA; Shankley, NP | 1 |
| Akuzawa, S; Ito, H; Kamato, T; Katuyama, Y; Kobayashi, A; Miyata, K; Nishida, A; Tsutsumi, R; Yamano, M; Yuki, H | 1 |
| Chapman, KL; Fletcher, AE; Hargreaves, RJ; Iversen, LL; Iversen, SD; Kemp, JA; Marshall, GR; Patel, S; Ryecroft, W; Smith, AJ | 1 |
| Freedman, SB; Patel, S; Smith, AJ | 1 |
| Bentley, G; Bourson, A; Hargreaves, R; Iversen, S; Jackson, A; Rycroft, W; Tattersall, D; Tricklebank, M | 1 |
| Ewanik, D; Gertz, BJ; Kovacs, TO; Lin, JH; Mertz, H; Murphy, MG; Shingo, S; Sytnik, B; Walsh, JH | 1 |
| Eklund, A; Lindholm, M | 1 |
| Bado, A; Blommaert, AG; Böhme, A; Ducos, B; Garbay, C; Moizo, L; Roques, BP; Weng, JH | 1 |
| Black, JW; Gerskowitch, VP; Harper, EA; Hull, RA; Roberts, SP; Shankley, NP; Watt, GF | 1 |
| Akuzawa, S; Batt, AR; Kendrick, DA; Miyata, K; Nishida, A; Ohta, M; Rooker, DP; Ryder, H; Satoh, M; Semple, G; Szelke, M | 1 |
| Bradwejn, J; Frankland, PW; Josselyn, SA; Vaccarino, FJ; Yeomans, JS | 1 |
| Akuzawa, S; Ito, H; Miyake, A; Miyata, K; Nishida, A; Takemoto, Y; Takinami, Y; Yuki, H | 1 |
| Hirata, T; Ishihara, Y; Ishikawa, M; Kunikata, T; Takeuchi, K; Yamamoto, H | 1 |
| Lainé, J; Mimeau-Worthington, T; Morisset, J | 1 |
| Impicciatore, M; Letari, O; Makovec, F; Mennuni, L; Revel, L | 1 |
| Black, JW; Harper, EA; Shankley, NP | 1 |
| Dunstone, DJ; Kalindjian, SB; Low, CM; Pether, MJ; Roberts, SP; Shankley, NP; Tozer, MJ; Watt, GF | 1 |
| El-Kouhen, K; Morisset, J | 1 |
2 trial(s) available for pentagastrin and l 365260
| Article | Year |
|---|---|
Cholecystokinin and anxiety in normal volunteers: an investigation of the anxiogenic properties of pentagastrin and reversal by the cholecystokinin receptor subtype B antagonist L-365,260.
Topics: Adult; Analysis of Variance; Anti-Anxiety Agents; Anxiety; Benzodiazepinones; Blood Pressure; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Female; Heart Rate; Humans; Injections, Intravenous; Male; Middle Aged; Pentagastrin; Phenylurea Compounds; Receptors, Cholecystokinin | 1995 |
The gastrin-receptor antagonist L-365,260 inhibits stimulated acid secretion in humans.
Topics: Adolescent; Adult; Analysis of Variance; Benzodiazepinones; Dose-Response Relationship, Drug; Double-Blind Method; Gastric Acid; Gastrins; Humans; Male; Middle Aged; Pentagastrin; Phenylurea Compounds; Receptors, Cholecystokinin; Reference Values | 1993 |
30 other study(ies) available for pentagastrin and l 365260
| Article | Year |
|---|---|
Rationally designed "dipeptoid" analogues of CCK. Acid mimics of the potent and selective non-peptide CCK-B receptor antagonist CI-988.
Topics: Animals; Carboxylic Acids; Cholecystokinin; Dipeptides; Drug Design; Indoles; Male; Meglumine; Mice; Rats; Receptors, Cholecystokinin | 1992 |
Rationally designed "dipeptoid" analogues of CCK. alpha-Methyltryptophan derivatives as highly selective and orally active gastrin and CCK-B antagonists with potent anxiolytic properties.
Topics: Animals; Anti-Anxiety Agents; Cerebral Cortex; Cholecystokinin; Gastrins; Indicators and Reagents; Male; Mice; Receptors, Cholecystokinin; Structure-Activity Relationship | 1991 |
Cholecystokinin dipeptoid antagonists: design, synthesis, and anxiolytic profile of some novel CCK-A and CCK-B selective and "mixed" CCK-A/CCK-B antagonists.
Topics: Amino Acid Sequence; Amylases; Animals; Anti-Anxiety Agents; Anxiety; Electrophysiology; Hypothalamus; Male; Mice; Molecular Sequence Data; Molecular Structure; Pancreas; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Structure-Activity Relationship | 1993 |
L-365,260, a potent CCK-B/gastrin receptor antagonist, suppresses gastric acid secretion induced by histamine and bethanechol as well as pentagastrin in rats.
Topics: Animals; Benzodiazepinones; Bethanechol; Bethanechol Compounds; Cimetidine; Devazepide; Dose-Response Relationship, Drug; Gastric Acidity Determination; Gastric Mucosa; Histamine; Male; Pentagastrin; Perfusion; Phenylurea Compounds; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin | 1992 |
Effect of gastrin receptor antagonists on gastric acid secretion and gastrin and somatostatin release in the rat stomach.
Topics: Animals; Benzodiazepinones; Dose-Response Relationship, Drug; Female; Gastric Acid; Gastric Mucosa; Gastrins; Indoles; Pentagastrin; Phenethylamines; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Somatostatin; Stomach; Time Factors | 1992 |
Possible role of cholecystokinin-A receptors in regulation of thyrotropin (TSH) secretion in male rats.
Topics: Animals; Benzodiazepinones; Ceruletide; Cholecystokinin; Cold Temperature; Devazepide; Dose-Response Relationship, Drug; Male; Pentagastrin; Phenylurea Compounds; Prolactin; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide; Tetragastrin; Thyrotropin | 1992 |
The behavioural properties of CI-988, a selective cholecystokininB receptor antagonist.
Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Behavior, Animal; Benzodiazepinones; Carbolines; Central Nervous System Depressants; Cholecystokinin; Conflict, Psychological; Devazepide; Drug Interactions; Ethanol; Hypnotics and Sedatives; Indoles; Injections, Intraventricular; Male; Meglumine; Mice; Motor Activity; Pentagastrin; Pentobarbital; Pentylenetetrazole; Phenylurea Compounds; Postural Balance; Rats; Receptors, Cholecystokinin; Social Behavior | 1991 |
Blockade of type A, not type B, CCK receptors attenuates satiety actions of exogenous and endogenous CCK.
Topics: Animals; Benzodiazepinones; Cholecystokinin; Drinking; Gastric Acid; Glucose; Male; Pentagastrin; Phenylurea Compounds; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Satiety Response; Solutions | 1992 |
Inhibition of gastrin- and histamine-stimulated gastric acid secretion by gastrin and cholecystokinin antagonists in the rat.
Topics: Animals; Benzodiazepinones; Cholecystokinin; Devazepide; Gastric Acid; Gastric Mucosa; Gastrins; Histamine Antagonists; Injections, Intravenous; Male; Oligopeptides; Pentagastrin; Phenylurea Compounds; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin | 1991 |
Evidence for an involvement of the brain cholecystokinin B receptor in anxiety.
Topics: Animals; Anxiety; Benzodiazepinones; Cerebral Ventricles; Ceruletide; Chlordiazepoxide; Cholecystokinin; Devazepide; Indoles; Injections, Intraventricular; Male; Meglumine; Pentagastrin; Phenylurea Compounds; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin | 1991 |
Characterization of cholecystokinin octapeptide-stimulated endogenous dopamine release from rat nucleus accumbens in vitro.
Topics: Animals; Benzodiazepinones; Chromatography, High Pressure Liquid; Corpus Striatum; Devazepide; Dopamine; In Vitro Techniques; Male; Nucleus Accumbens; Pentagastrin; Phenylurea Compounds; Potassium; Rats; Rats, Inbred Strains; Receptors, Cholecystokinin; Septal Nuclei; Sincalide | 1990 |
A new potent and selective non-peptide gastrin antagonist and brain cholecystokinin receptor (CCK-B) ligand: L-365,260.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Brain Chemistry; Carbachol; Cholecystokinin; Dogs; Exocrine Glands; Female; Gastric Emptying; Gastrins; Guinea Pigs; Histamine; Humans; In Vitro Techniques; Iodine Radioisotopes; Mice; Pentagastrin; Phenylurea Compounds; Pylorus; Rats; Receptors, Cholecystokinin; Species Specificity; Structure-Activity Relationship | 1989 |
Identification of gastrin as a growth peptide in human pancreatic cancer.
Topics: Animals; Benzodiazepinones; Cell Division; Cell Line; Cholecystokinin; Devazepide; Gastrins; Growth Substances; Humans; Male; Mice; Mice, Nude; Pancreatic Neoplasms; Pentagastrin; Phenylurea Compounds; Receptors, Cholecystokinin; Transplantation, Heterologous; Tumor Cells, Cultured | 1995 |
The use of receptor desensitization to analyse CCKA and CCKB/gastrin receptors coupled to contraction in guinea-pig stomach muscle.
Topics: Animals; Benzodiazepinones; Binding, Competitive; Cholecystokinin; Devazepide; Gallbladder; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pentagastrin; Phenylurea Compounds; Receptors, Cholecystokinin; Stomach; Tetragastrin | 1995 |
Pharmacological profile of (R)-1-[2,3-dihydro-1-(2'-methylphenacyl)-2-oxo- 5-phenyl-1H-1,4-benzodiazepin-3-yl]-3-(3-methylphenyl)urea (YM022), a new potent and selective gastrin/cholecystokinin-B receptor antagonist, in vitro and in vivo.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Bethanechol; Bethanechol Compounds; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Indoles; Male; Meglumine; Pentagastrin; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Sincalide | 1994 |
Biological properties of the benzodiazepine amidine derivative L-740,093, a cholecystokinin-B/gastrin receptor antagonist with high affinity in vitro and high potency in vivo.
Topics: Animals; Benzodiazepinones; Brain; Female; Gastric Acid; Guinea Pigs; In Vitro Techniques; Male; Mice; Pentagastrin; Phenylurea Compounds; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Receptors, Cholecystokinin | 1994 |
Characterisation of CCKB receptors on GH3 pituitary cells: receptor activation is linked to Ca2+ mobilisation.
Topics: Animals; Benzodiazepinones; Biotransformation; Calcium; Cell Line; Devazepide; Guanine Nucleotides; Iodine Radioisotopes; Kinetics; Pancreas; Pentagastrin; Phenylurea Compounds; Pituitary Gland, Anterior; Radioligand Assay; Rats; Receptors, Cholecystokinin; Second Messenger Systems; Sincalide; Succinimides | 1994 |
An investigation into the discriminative stimulus and reinforcing properties of the CCKB-receptor antagonist, L-365,260 in rats.
Topics: Animals; Behavior, Animal; Benzodiazepinones; Cocaine; Diazepam; Discrimination, Psychological; Drug Synergism; Gastric Acid; Male; Morphine; Naloxone; Pentagastrin; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Self Administration; Sodium Chloride | 1994 |
Inhibitory effect of gastrin and cholecystokinin fragments on the secretion of triacylglycerol in rat hepatocytes.
Topics: Animals; Benzodiazepinones; Cells, Cultured; Depression, Chemical; Devazepide; Gastrins; Liver; Male; Pentagastrin; Peptide Fragments; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide; Triglycerides | 1993 |
Role of N- and C-terminal substituents on the CCK-B agonist-antagonist pharmacological profile of Boc-Trp-Phg-Asp-Nal-NH2 derivatives.
Topics: Amino Acid Sequence; Animals; Anti-Anxiety Agents; Benzodiazepinones; CHO Cells; Cholecystokinin; Cricetinae; Dose-Response Relationship, Drug; Electrophysiology; Gastric Acid; Gastrointestinal Agents; Hippocampus; Indoles; Inositol Phosphates; Male; Meglumine; Molecular Sequence Data; Neurons; Neurotransmitter Agents; Oligopeptides; Pentagastrin; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Structure-Activity Relationship; Time Factors; Transfection | 1996 |
Analysis of the variation in the action of L-365,260 at CCKB/gastrin receptors in rat, guinea-pig and mouse isolated gastric tissue assays.
Topics: Animals; Benzodiazepinones; Binding, Competitive; Famotidine; Gastric Mucosa; Guinea Pigs; Histamine; Histamine H2 Antagonists; In Vitro Techniques; Mice; Muscle, Smooth; Pentagastrin; Phenylurea Compounds; Rats; Rats, Wistar; Receptors, Cholecystokinin; Species Specificity; Stomach | 1996 |
(3R)-N-(1-(tert-butylcarbonylmethyl)-2,3-dihydro-2-oxo-5-(2-pyridyl)-1H-1,4-benzodiazepin-3-yl)-N'-(3-(methylamino)phenyl)urea (YF476): a potent and orally active gastrin/CCK-B antagonist.
Topics: Administration, Oral; Animals; Benzodiazepines; Benzodiazepinones; Binding, Competitive; Brain; Devazepide; Dogs; Gastric Acid; Hormone Antagonists; Molecular Structure; Pancreas; Pentagastrin; Phenylurea Compounds; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Sincalide; Structure-Activity Relationship | 1997 |
Activation of amygdala cholecystokininB receptors potentiates the acoustic startle response in the rat.
Topics: Acoustic Stimulation; Amygdala; Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepinones; Corpus Striatum; Fear; Indoles; Injections, Intraperitoneal; Injections, Intraventricular; Meglumine; Nucleus Accumbens; Pentagastrin; Phenylurea Compounds; Rats; Rats, Wistar; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Reflex, Startle | 1997 |
YM022, a potent and selective gastrin/CCK-B receptor antagonist, inhibits peptone meal-induced gastric acid secretion in Heidenhain pouch dogs.
Topics: Animals; Atropine; Benzodiazepines; Benzodiazepinones; Devazepide; Dogs; Dose-Response Relationship, Drug; Eating; Famotidine; Gastric Acid; Histamine; Histamine H2 Antagonists; Hormone Antagonists; Male; Methacholine Chloride; Muscarinic Antagonists; Pentagastrin; Peptones; Phenylurea Compounds; Receptors, Cholecystokinin; Sincalide; Stomach | 1997 |
Effects of S-0509, a novel CCKB/gastrin receptor antagonist, on acid secretion and experimental duodenal ulcers in rats.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzodiazepinones; Benzophenones; Dose-Response Relationship, Drug; Duodenal Ulcer; Epirizole; Gastric Acid; Gastric Mucosa; Hydrogen-Ion Concentration; Male; Pentagastrin; Peptones; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin | 1999 |
Hormonal control of rat fetal pancreas development.
Topics: Animals; Benzodiazepinones; Ceruletide; DNA; Female; Gastrin-Releasing Peptide; Hormones; Hydrocortisone; Maternal-Fetal Exchange; Organ Size; Pancreas; Pentagastrin; Phenylurea Compounds; Pregnancy; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Receptors, Cholecystokinin | 1999 |
Characterization of antisecretory and antiulcer activity of CR 2945, a new potent and selective gastrin/CCK(B) receptor antagonist.
Topics: Animals; Anti-Anxiety Agents; Anti-Ulcer Agents; Benzodiazepines; Benzodiazepinones; Calcium; Cats; Chronic Disease; Cysteamine; Dose-Response Relationship, Drug; Ethanol; Gastric Acid; Gastric Fistula; Gastric Mucosa; Gastrins; Histamine H2 Antagonists; Indomethacin; Male; Omeprazole; Parietal Cells, Gastric; Pentagastrin; Perfusion; Phenylurea Compounds; Rabbits; Ranitidine; Rats; Receptors, Cholecystokinin; Stomach; Stomach Ulcer | 1999 |
Characterization of the binding of a novel radioligand to CCKB/gastrin receptors in membranes from rat cerebral cortex.
Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Bridged-Ring Compounds; Cerebral Cortex; Dipeptides; Dose-Response Relationship, Drug; Hormone Antagonists; Indoles; Kinetics; Male; Meglumine; Membranes; Nootropic Agents; Pentagastrin; Phenylurea Compounds; Radioligand Assay; Rats; Rats, Wistar; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Sincalide; Tritium | 1999 |
Nonpeptide cholecystokinin-2 receptor agonists.
Topics: Adamantane; Animals; Benzodiazepinones; Binding, Competitive; Cerebral Cortex; In Vitro Techniques; Indoles; Ligands; Mice; Models, Molecular; Pentagastrin; Phenylurea Compounds; Radioligand Assay; Rats; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Stereoisomerism; Stomach | 2001 |
Control of somatostatin (SS) secretion by CCK-1 and CCK-2 receptors' occupation in RIN-14B cells, a rat pancreatic islet cell line.
Topics: Animals; Benzodiazepinones; Brefeldin A; Cell Line; Ceruletide; Cholecystokinin; Cycloheximide; Devazepide; Dose-Response Relationship, Drug; Enzyme-Linked Immunosorbent Assay; Fluorescent Antibody Technique; Gastrins; Islets of Langerhans; Pentagastrin; Phenylurea Compounds; Protein Precursors; Protein Synthesis Inhibitors; Protein Transport; Rats; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Sincalide; Somatostatin | 2010 |