Page last updated: 2024-08-23

penfluridol and piperidines

penfluridol has been researched along with piperidines in 82 studies

Research

Studies (82)

TimeframeStudies, this research(%)All Research%
pre-199077 (93.90)18.7374
1990's3 (3.66)18.2507
2000's1 (1.22)29.6817
2010's1 (1.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Daigle, L; Furlong, W; Grof, P; Jacques, W; Kingstone, E; Virc, L1
Kane, J; Klein, DF; Quitkin, F; Ramos-Lorenzi, JR; Rifkin, A1
Fontaine, P; Jus, A; Jus, K1
Kuschinsky, K; Seeber, U1
Gallant, DM1
Nose, T; Takemoto, H1
Hanus, H; Kindernayová, H; Stránský, P; Valach, M; Zapletálek, M1
James, NM1
Abuzzahab, FS1
Klein, DF; Quitkin, F; Rifkin, A1
Woggon, B1
Donlon, PT; Meyer, JE1
Claghorn, JL; Mathew, RJ; Mirabi, M1
Grindel, JM; Heykants, JJ; Janssen, PA; Migdalof, BH1
Haring, C1
Gerbino, L; Klein, H; Selzer, G; Shopsin, B1
Pluym, A1
Dlabac, A; Metys, J1
Annunziato, LA; Moore, KE; Wuerthele, SM1
Engel, J; Lundborg, P2
Charles, J; Elgart, B; Iqbal, MJ; Simpson, GM; Von Greiff, H; Young, MA1
Doongaji, DR1
Annable, L; Chouinard, G; Cooper, S1
Fleischhauer, J1
Lapierre, YD1
Chung, PM; Lee, HK; Wang, SC1
Edenius, B; Jacobsson, L; Kettner, B; Magnusson, KE; Mattsson, B; Mjörndal, T; Oreland, L; Perris, C; Rapp, W; Villemoes, P; von Knorring, L1
Delvecchio, FR; Fracassi, MJ1
Hargrave, R; Rousos, AP1
Floru, L; Heinrich, K; Wittek, F1
Dlavac, A; Kazdová, E; Metys, J1
Ishida, R; Ito, K; Kowa, Y; Nurimoto, S; Shintomi, K; Yamamura, M1
d'Elia, G; Jacobsson, L; Mattsson, B; Mjörndal, T; Oreland, L; Perris, C; Rapp, W; von Knorring, L1
Ahlenius, S; Engel, J; Hård, E; Larsson, K; Lundborg, P; Sinnerstedt, P1
Klein, H; Selzer, G; Shopsin, B1
Annable, L; Chouinard, G1
Edenius, B; Jacobsson, L; Kettner, B; Magnusson, KE; Mattsson, B; Perris, C; Rapp, W; Villemoes, P; Von Knorring, L1
Canero, E; Mario Zelaschi, N; Suárez Richards, M1
Degenhardt, T; Glitschka, A; Graf, K; König, L; Kühne, GE; Lange, E; Niedermeyer, K; Schmidt, P; Waldmann, KD; Zielonka, VS1
Kuribara, H; Tadokoro, S1
Horiuchi, M; Ito, K; Nurimoto, S; Ochiai, T; Suzuki, S1
Ishida, R; Nakamura, S; Sugihara, J1
Aguirre Cárdenas, JJ; Hernández Cruz, S1
Kurland, AA; Ota, KY1
Gerlach, J; Kramp, P; Kristjansen, P; Lauritsen, B; Lühdorf, K; Munkvad, I1
Albert, JM; Bertrand, M; Cooper, SF; Dugal, R1
Deutsch, M; Nair, NP; Saarma, J1
Gerlach, J1
Albert, JM; Cooper, SF; Dugal, R1
Shintomi, K; Yamamura, M1
Kuribara, H; Okuizumi, K; Shirota, M; Tadokoro, S1
Andén, NE; Engel, J; Jackson, DM; Liljequist, S1
Janssen, PA; Lenaerts, FM; Niemegeers, CJ; Schellekens, KH; Wauquier, A1
Biagi, BA; Day, RN; Enyeart, JJ; Maurer, RA; Sheu, SS1
Lavoie, PA1
Hopkała, H; Przyborowski, L1
Chen, YG2
Bao, XQ1
Li, Y1
Munitz, H; Shalev, A1
Kruse, A; Lühdorf, K; Schulz, V1
Likhobabenko, IuM1
Mjörndal, T; Oreland, L; Perris, C; Rapp, W1
Asnis, GM; Dyrenfurth, I; Halbreich, U; Halpern, FS; Nathan, RS; Ostrow, LC; Sachar, EJ1
Rubin, RT1
Levy, V; Morales, E; Schilkrut, R1
Key, KA; Oakley, AC; Pizzo, SV1
Asnis, GM; Halbreich, U; Halpern, F; Nathan, RS; Ostrow, L; Renzi, NL; Sachar, EJ; Slotnick, V1
Judd, AM; MacLeod, RM; Schettini, G1
Blum, JJ; Keegan, FP1
Chodura, V1
Miranda, GF; Roncucci, R; Verry, M1
Shu, L1
Shapiro, AK; Shapiro, E1
Ciani, S; Fiume, S1
Jin, HM1
Cano-Abad, MF; Gandía, L; García, AG; Hernández-Guijo, JM; López, MG; Sánchez-García, P; Zapater, P1
Enyeart, JJ; Gomora, JC1
Cayabyab, FS; Hamming, KS; McRory, JE; Mezeyova, J; Parker, D; Santi, CM; Snutch, TP; Stea, A; Sutton, KG1
Enyeart, JA; Enyeart, JJ1

Reviews

2 review(s) available for penfluridol and piperidines

ArticleYear
Penfluridol: a neuroleptic drug designed for long duration of action.
    Drug metabolism reviews, 1979, Volume: 9, Issue:2

    Topics: Animals; Chemistry, Pharmaceutical; Delayed-Action Preparations; Feces; Humans; Kinetics; Penfluridol; Piperidines; Time Factors

1979
[A new long-acting psychotropic substance in oral administration: penfluridol].
    La Clinica terapeutica, 1981, Feb-15, Volume: 96, Issue:3

    Topics: Adult; Delayed-Action Preparations; Female; Humans; Male; Mental Disorders; Middle Aged; Penfluridol; Piperidines

1981

Trials

21 trial(s) available for penfluridol and piperidines

ArticleYear
Long-acting oral vs injectable antipsychotic drugs in schizophrenics: a one-year double-blind comparison in multiple episode schizophrenics.
    Archives of general psychiatry, 1978, Volume: 35, Issue:7

    Topics: Administration, Oral; Adult; Clinical Trials as Topic; Double-Blind Method; Female; Fluphenazine; Humans; Injections, Intravenous; Long-Term Care; Male; Penfluridol; Piperidines; Recurrence; Schizophrenia

1978
Polygraphic sleep pattern during penfluridol treatment.
    Current therapeutic research, clinical and experimental, 1975, Volume: 18, Issue:1 pt 2

    Topics: Adult; Chronic Disease; Clinical Trials as Topic; Drug Evaluation; Electroencephalography; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia; Sleep; Sleep Stages; Sleep, REM; Time Factors

1975
Potential value of penfluridol and pipothiazine palmitate.
    Psychopharmacology bulletin, 1975, Volume: 11, Issue:1

    Topics: Antipsychotic Agents; Clinical Trials as Topic; Humans; Injections, Intramuscular; Penfluridol; Phenothiazines; Piperidines; Placebos; Psychiatric Status Rating Scales; Schizophrenia

1975
Penfluridol: a double blind trial in chronic schizophrenia.
    The New Zealand medical journal, 1977, Jan-26, Volume: 85, Issue:580

    Topics: Administration, Oral; Adult; Chronic Disease; Clinical Trials as Topic; Drug Administration Schedule; Female; Fluphenazine; Humans; Male; Middle Aged; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Schizophrenia

1977
The treatment of schizophrenia with long-acting oral neuroleptics: a six-month double-blind investigation of penfluridol versus trifluoperazine.
    Psychopharmacology bulletin, 1977, Volume: 13, Issue:3

    Topics: Adult; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Drug Evaluation; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia; Trifluoperazine

1977
A one-year double-blind comparison of long-acting oral (penfluridol) versus long-acting injectable (fluphenazine decanoate) antipsychotic drugs in multiple-episode schizophrenics.
    Psychopharmacology bulletin, 1977, Volume: 13, Issue:3

    Topics: Administration, Oral; Clinical Trials as Topic; Double-Blind Method; Drug Evaluation; Fluphenazine; Humans; Injections; Penfluridol; Piperidines; Recurrence; Schizophrenia

1977
[Penfluridol. Results of a year-long clinical trial].
    International pharmacopsychiatry, 1978, Volume: 13, Issue:1

    Topics: Adult; Clinical Trials as Topic; Female; Humans; Male; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Schizophrenia; Time Factors

1978
A twelve month comparison of penfluridol and trifluoperazine in chronic schizophrenic outpatients.
    The Journal of clinical psychiatry, 1978, Volume: 39, Issue:6

    Topics: Adult; Chronic Disease; Clinical Trials as Topic; Double-Blind Method; Drug Evaluation; Female; Humans; Interpersonal Relations; Male; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Schizophrenia; Trifluoperazine

1978
Penfluridol: a long acting oral antipsychotic drug.
    The Journal of clinical psychiatry, 1979, Volume: 40, Issue:2

    Topics: Adult; Chlorpromazine; Clinical Trials as Topic; Dose-Response Relationship, Drug; Double-Blind Method; Drug Evaluation; Female; Humans; Male; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Psychotic Disorders; Schizophrenia

1979
[Long term treatment of schizophrenia with penfluridol].
    Die Medizinische Welt, 1977, Apr-01, Volume: 28, Issue:13

    Topics: Adult; Aged; Clinical Trials as Topic; Depressive Disorder, Major; Female; Humans; Long-Term Care; Male; Middle Aged; Obsessive-Compulsive Disorder; Penfluridol; Piperidines; Schizophrenia

1977
A long term comparative trial of penfluridol and fluphenazine decanoate in schizophrenic outpatients.
    The Journal of clinical psychiatry, 1978, Volume: 39, Issue:4

    Topics: Adult; Ambulatory Care; Chronic Disease; Double-Blind Method; Drug Evaluation; Female; Fluphenazine; Humans; Male; Middle Aged; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Schizophrenia

1978
Penfluridol and thiothixene. Dosage, plasma levels and changes in psychopathology.
    International pharmacopsychiatry, 1976, Volume: 11, Issue:4

    Topics: Adult; Chromatography, Gas; Chronic Disease; Clinical Trials as Topic; Dose-Response Relationship, Drug; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia; Thiothixene

1976
[Clinical evaluation of a weekly maintenance neuroleptic: penfluridol (R16341)].
    Acta psiquiatrica y psicologica de America latina, 1976, Volume: 22, Issue:4

    Topics: Adolescent; Adult; Clinical Trials as Topic; Drug Evaluation; Female; Humans; Intellectual Disability; Male; Middle Aged; Penfluridol; Piperidines; Psychotic Disorders; Schizophrenia; Tablets; Time Factors

1976
A preliminary study with penfluridol in hospitalized chronic schizophrenic patients.
    Current therapeutic research, clinical and experimental, 1975, Volume: 18, Issue:5

    Topics: Adult; Chronic Disease; Clinical Trials as Topic; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Schizophrenia; Time Factors

1975
The problem of post-psychotic schizophrenic depressions and their pharmacological induction. Long-term studies with fluspirilene and penfluridol and single-blind trial with fluphenazine-decanoate and flupenthixol-decanoate.
    International pharmacopsychiatry, 1975, Volume: 10, Issue:4

    Topics: Adult; Antidepressive Agents; Clinical Trials as Topic; Depression; Female; Flupenthixol; Fluphenazine; Fluspirilene; Humans; Long-Term Care; Male; Penfluridol; Personality Inventory; Piperidines; Schizophrenia; Spiro Compounds; Thioxanthenes

1975
Penfluridol: once-a-week oral maintenance neuroleptic in the management of chronic schizophrenics.
    Psychopharmacology bulletin, 1975, Volume: 11, Issue:1

    Topics: Administration, Oral; Chronic Disease; Clinical Trials as Topic; Humans; Penfluridol; Piperidines; Placebos; Psychiatric Status Rating Scales; Schizophrenia

1975
Peroral and parenteral administration of long-acting neuroleptics: a double-blind study of penfluridol compared to flupenthixol decanoate in the treatment of schizophrenia.
    Acta psychiatrica Scandinavica, 1975, Volume: 52, Issue:2

    Topics: Administration, Oral; Adolescent; Adult; Aged; Clinical Trials as Topic; Delayed-Action Preparations; Drug Evaluation; Flupenthixol; Humans; Injections; Male; Middle Aged; Penfluridol; Piperidines; Placebos; Schizophrenia; Thioxanthenes

1975
Penfluridol steady-state kinetics in psychiatric patients.
    Clinical pharmacology and therapeutics, 1975, Volume: 18, Issue:3

    Topics: Administration, Oral; Adult; Clinical Trials as Topic; Dose-Response Relationship, Drug; Female; Humans; Kinetics; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia

1975
Proceedings: Penfluridol in the treatment of schizophrenia: clinical and psychometric findings.
    Psychopharmacology bulletin, 1976, Volume: 12, Issue:1

    Topics: Adult; Clinical Trials as Topic; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Schizophrenia

1976
[A double-blind study on the effect of clozapine penfluridol and chlorpromazine in the treatment of schizophrenia].
    Zhonghua shen jing jing shen ke za zhi = Chinese journal of neurology and psychiatry, 1988, Volume: 21, Issue:5

    Topics: Adolescent; Adult; Chlorpromazine; Clinical Trials as Topic; Clozapine; Dibenzazepines; Double-Blind Method; Humans; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia

1988
[Application of NOSIE in the study of neuroleptic treatment].
    Zhonghua shen jing jing shen ke za zhi = Chinese journal of neurology and psychiatry, 1987, Volume: 20, Issue:6

    Topics: Adolescent; Adult; Chlorpromazine; Clinical Trials as Topic; Clozapine; Dibenzazepines; Double-Blind Method; Humans; Male; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Schizophrenia

1987

Other Studies

59 other study(ies) available for penfluridol and piperidines

ArticleYear
Penfluridol, a peroral long-acting neuroleptic, for the maintenance treatment of schizophrenic patients who relapse.
    Journal of clinical pharmacology, 1977, Volume: 17, Issue:4

    Topics: Adult; Brief Psychiatric Rating Scale; Drug Evaluation; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Recurrence; Schizophrenia; Time Factors

1977
Effects of penfluridol of dopamine-sensitive adenylate cyclase in corpus striatum and substantia nigra of rats.
    Experientia, 1976, Dec-15, Volume: 32, Issue:12

    Topics: Adenylyl Cyclases; Animals; Corpus Striatum; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Male; Penfluridol; Piperidines; Rats; Substantia Nigra

1976
The effect of penfluridol and some psychotropic drugs on monoamine metabolism in central nervous system.
    European journal of pharmacology, 1975, Volume: 31, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Biogenic Amines; Brain; Brain Chemistry; Chlordiazepoxide; Chlorpromazine; Diazepam; Dopamine; Haloperidol; Homovanillic Acid; Hydroxyindoleacetic Acid; Male; Mice; Norepinephrine; Penfluridol; Pimozide; Piperazines; Piperidines; Psychotropic Drugs; Rats; Serotonin

1975
[Electroencephalographic picture in patients treated with penfluridol].
    Sbornik vedeckych praci Lekarske fakulty Karlovy university v Hradci Kralove, 1978, Volume: 21, Issue:5

    Topics: Adolescent; Adult; Brain; Electroencephalography; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines

1978
Penfluridol: an open phase III study in acute newly admitted hospitalized schizophrenic patients.
    Psychopharmacology, 1977, Dec-19, Volume: 55, Issue:2

    Topics: Acute Disease; Adult; Drug Evaluation; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Schizophrenia; Schizophrenia, Paranoid

1977
TLC differentiation of butyrophenone and diphenylbutylpiperidine compounds from phenothiazine derivatives.
    Journal of pharmaceutical sciences, 1979, Volume: 68, Issue:8

    Topics: Butyrophenones; Chromatography, Thin Layer; Fluspirilene; Indicators and Reagents; Penfluridol; Phenothiazines; Pimozide; Piperidines

1979
Interspecies differences in sensitivity to the neuroleptic drug penfluridol.
    Activitas nervosa superior, 1977, Volume: 19 Suppl 2

    Topics: Animals; Apomorphine; Behavior, Animal; Dogs; Macaca fascicularis; Macaca mulatta; Mice; Penfluridol; Piperidines; Rabbits; Rats; Receptors, Dopamine; Species Specificity

1977
Comparative effects of penfluridol on circling behavior and striatal DOPAC and serum prolactin concentrations in the rat.
    European journal of pharmacology, 1978, Aug-01, Volume: 50, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Apomorphine; Behavior; Corpus Striatum; Drug Interactions; Humans; Male; Penfluridol; Phenylacetates; Piperidines; Prolactin; Rats; Stereotyped Behavior; Time Factors

1978
Increased mesolimbic 3H-spiroperidol binding in 4 week old offspring of nursing rat mothers treated with penfluridol.
    European journal of pharmacology, 1979, Dec-20, Volume: 60, Issue:4

    Topics: Animal Population Groups; Animals; Animals, Suckling; Butyrophenones; Female; Lactation; Limbic System; Penfluridol; Piperidines; Pregnancy; Rats; Receptors, Dopamine; Spiperone

1979
The treatment of tardive dyskinesia with penfluridol. A case report.
    Neurology India, 1977, Volume: 25, Issue:4

    Topics: Adult; Chlorpromazine; Dyskinesia, Drug-Induced; Humans; Male; Penfluridol; Piperidines; Trifluoperazine

1977
Antiparkinsonian drug administration and plasma levels of penfluridol, a new long-acting neuroleptic.
    Communications in psychopharmacology, 1977, Volume: 1, Issue:4

    Topics: Adult; Antiparkinson Agents; Double-Blind Method; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Procyclidine; Schizophrenia; Time Factors

1977
Treatment of chronic schizophrenics with the oral long-term neuroleptic penfluridol in an open study.
    Progress in neuro-psychopharmacology, 1977, Volume: 1, Issue:1-2

    Topics: Administration, Oral; Adult; Aged; Evaluation Studies as Topic; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia

1977
A controlled study of penfluridol in the treatment of chronic schizophrenia.
    The American journal of psychiatry, 1978, Volume: 135, Issue:8

    Topics: Adult; Ambulatory Care; Chronic Disease; Female; Fluphenazine; Humans; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia

1978
Mechanism of antiemetic action of penfluridol in the dog.
    European journal of pharmacology, 1978, Dec-15, Volume: 53, Issue:1

    Topics: Administration, Oral; Animals; Antiemetics; Apomorphine; Dogs; Drug Antagonism; Female; Injections, Intravenous; Injections, Intraventricular; Levodopa; Male; Medulla Oblongata; Penfluridol; Piperidines

1978
Proceedings: Pharmacological properties of a new oral long-acting neuroleptic drug penfluridol.
    Activitas nervosa superior, 1975, Volume: 17, Issue:4

    Topics: Animals; Apomorphine; Behavior, Animal; Haplorhini; Macaca mulatta; Mice; Penfluridol; Piperidines; Rats; Species Specificity

1975
[Pharmacological studies of an antipschotic agent, penfluridol. (1). The central pharmacological actions].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1976, Volume: 72, Issue:7

    Topics: Agonistic Behavior; Animals; Apomorphine; Avoidance Learning; Blepharoptosis; Body Temperature; Catalepsy; Cats; Central Nervous System; Chlorpromazine; Conditioning, Classical; Cooperative Behavior; Dogs; Dose-Response Relationship, Drug; Drug Synergism; Female; Haloperidol; Haplorhini; Hexobarbital; Humans; Locomotion; Male; Methamphetamine; Mice; Parasympatholytics; Penfluridol; Piperidines; Rats

1976
Changes in psychopathology in relation to EEG variables and visual averaged evoked responses (V.AER) in schizophrenic patients treated with penfluridol or thiothixene.
    Acta psychiatrica Scandinavica, 1977, Volume: 55, Issue:4

    Topics: Adult; Electroencephalography; Evoked Potentials; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia; Thiothixene

1977
Open field behavior and gross motor development in offspring of nursing rat mothers given penfluridol.
    Pharmacology, biochemistry, and behavior, 1977, Volume: 6, Issue:3

    Topics: Age Factors; Animals; Dopamine; Female; Male; Milk; Motor Activity; Penfluridol; Piperidines; Pregnancy; Rats; Reflex, Startle

1977
High-dose penfluridol (SEMAP) in acute hospitalized schizophrenic patients.
    Psychopharmacology bulletin, 1977, Volume: 13, Issue:3

    Topics: Acute Disease; Adult; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Schizophrenia

1977
Penfluridol in the treatment of newly admitted schizophrenic patients in a brief therapy unit.
    The American journal of psychiatry, 1976, Volume: 133, Issue:7

    Topics: Basal Ganglia Diseases; Chlorpromazine; Consciousness Disorders; Humans; Length of Stay; Penfluridol; Piperidines; Psychiatric Status Rating Scales; Schizophrenia

1976
Reduced turnover in mesolimbic dopamine neurons in 4-week-old offspring of nursing mothers treated with penfluridol.
    Brain research, 1976, Jul-09, Volume: 110, Issue:2

    Topics: Age Factors; Animals; Animals, Newborn; Avoidance Learning; Corpus Striatum; Dopamine; Female; Lactation; Limbic System; Male; Methyltyrosines; Neurons; Norepinephrine; Penfluridol; Piperidines; Pregnancy; Rats

1976
Controlled trial of penfluridol and thiothixene in the maintenance treatment of chronic schizophrenic syndromes.
    Acta psychiatrica Scandinavica, 1976, Volume: 54, Issue:2

    Topics: Adolescent; Adult; Aged; Biperiden; Chlorpromazine; Chronic Disease; Drug Evaluation; Female; Humans; Hypnotics and Sedatives; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia; Thiothixene

1976
[Activity of a new neuroleptic, penfluridol (R-16341) in long-term treatments].
    Acta psiquiatrica y psicologica de America latina, 1976, Volume: 22, Issue:3

    Topics: Administration, Oral; Adolescent; Adult; Drug Evaluation; Female; Humans; Mental Disorders; Middle Aged; Penfluridol; Piperidines

1976
[Position of the delayed-action neuroleptic penfluridol (Longperidol/Janssen) in psychiatric therapy].
    Psychiatrie, Neurologie, und medizinische Psychologie, 1976, Volume: 28, Issue:8

    Topics: Delayed-Action Preparations; Humans; Penfluridol; Piperidines; Schizophrenia

1976
Cumulative effects of penfluridol, a long-acting neuroleptic drug, as assayed by its behavioral actions.
    Japanese journal of pharmacology, 1976, Volume: 26, Issue:6

    Topics: Animals; Avoidance Learning; Behavior, Animal; Male; Penfluridol; Piperidines; Rats; Time Factors

1976
[Pharmacological studies of antipsychotic drug, penfluridol. 2. General pharmacological properties].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1976, Volume: 72, Issue:5

    Topics: Animals; Autonomic Nervous System; Cats; Digestive System; Dogs; Electrolytes; Female; Gastrointestinal Motility; Guinea Pigs; Heart; Hemodynamics; In Vitro Techniques; Male; Mice; Muscle Contraction; Nerve Endings; Penfluridol; Piperidines; Rabbits; Rats; Respiration; Urination

1976
[Biological fate of 3H-labeled penfluridol. (3) Correlation between concentration of 3H-penfluridol in the brain and its anti-methamphetamine activity].
    Radioisotopes, 1976, Volume: 25, Issue:10

    Topics: Animals; Brain Chemistry; Mastication; Methamphetamine; Penfluridol; Piperidines; Rats; Tritium

1976
[Evaluation of penfluridol in hospitalized chronic psychotic patients].
    Neurologia, neurocirugia, psiquiatria, 1975, Volume: 16, Issue:4

    Topics: Adult; Drug Evaluation; Female; Humans; Penfluridol; Piperidines; Psychotic Disorders

1975
[Penfluridolum (Semap). An oral depotneuroleptic].
    Ugeskrift for laeger, 1975, May-26, Volume: 137, Issue:22

    Topics: Delayed-Action Preparations; Humans; Parkinson Disease, Secondary; Penfluridol; Piperidines; Schizophrenia

1975
Gas-liquid chromatographic determination of penfluridol in plasma. A new specific technique.
    International pharmacopsychiatry, 1975, Volume: 10, Issue:2

    Topics: Chromatography, Gas; Humans; Male; Penfluridol; Piperidines; Schizophrenia

1975
Effects of penfluridol and other drugs on apomorphine-induced stereotyped behavior in monkeys.
    European journal of pharmacology, 1975, Volume: 31, Issue:2

    Topics: Animals; Apomorphine; Behavior; Chlorpromazine; Dose-Response Relationship, Drug; Haloperidol; Humans; Injections, Subcutaneous; Macaca fascicularis; Male; Methyltyrosines; Nialamide; Penfluridol; Piperidines; Reserpine; Stereotyped Behavior; Time Factors

1975
[Effects of penfluridol, a psychotropic agent, on operant behavior of rats].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1975, Volume: 71, Issue:5

    Topics: Animals; Avoidance Learning; Chlorpromazine; Conditioning, Operant; Haloperidol; Male; Penfluridol; Piperidines; Rats; Reinforcement Schedule

1975
The effect of long-term penfluridol treatment on the sensitivity of the dopamine receptors in the nucleus accumbens and in the corpus striatum.
    Psychopharmacologia, 1975, Dec-31, Volume: 45, Issue:2

    Topics: Animals; Corpus Striatum; Dopamine; Dopamine Antagonists; Drug Synergism; Haloperidol; Humans; Male; Motor Activity; Nialamide; Penfluridol; Piperidines; Rats; Receptors, Drug; Septal Nuclei; Septum Pellucidum; Stereotyped Behavior

1975
Clopimozide (R 29 764), a new highly potent and orally long-acting neuroleptic of the diphenylbutylpiperidine series.
    Arzneimittel-Forschung, 1975, Volume: 25, Issue:8

    Topics: Animals; Apomorphine; Avoidance Learning; Behavior, Animal; Benzimidazoles; Blepharoptosis; Body Temperature Regulation; Body Weight; Catalepsy; Dextroamphetamine; Dogs; Escape Reaction; Female; Guinea Pigs; Haloperidol; Humans; Lethal Dose 50; Male; Mice; Norepinephrine; Penfluridol; Pimozide; Piperidines; Rats; Self Stimulation; Stereotyped Behavior; Tranquilizing Agents

1975
Blockade of low and high threshold Ca2+ channels by diphenylbutylpiperidine antipsychotics linked to inhibition of prolactin gene expression.
    The Journal of biological chemistry, 1990, Sep-25, Volume: 265, Issue:27

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Cell Line; Fluspirilene; Gene Expression; Kinetics; Luciferases; Membrane Potentials; Penfluridol; Pimozide; Piperidines; Pituitary Neoplasms; Prolactin; Recombinant Fusion Proteins; Spiro Compounds; Thyrotropin-Releasing Hormone

1990
Penfluridol, chlorprothixene and haloperidol block fast axonal transport in an order of potency consistent with a mechanism related to inhibition of calmodulin.
    Neuropharmacology, 1987, Volume: 26, Issue:9

    Topics: Adenosine Triphosphate; Animals; Axonal Transport; Axons; Biomechanical Phenomena; Calmodulin; Chlorprothixene; Haloperidol; In Vitro Techniques; Microtubules; Penfluridol; Phosphocreatine; Piperidines; Rana catesbeiana; Spinal Nerves; Time Factors

1987
Determination of drugs containing fluorine with ion-selective electrode. Part 2: Butyrophenones and bis(4-fluorophenyl)butylpiperidines.
    Die Pharmazie, 1989, Volume: 44, Issue:1

    Topics: Butyrophenones; Electrodes; Fluorine; Penfluridol; Pimozide; Piperidines; Potentiometry; Spectrophotometry, Ultraviolet

1989
[Malignant syndromes due to psychotherapeutic agents].
    Zhonghua shen jing jing shen ke za zhi = Chinese journal of neurology and psychiatry, 1987, Volume: 20, Issue:6

    Topics: Adult; Antidepressive Agents; Antipsychotic Agents; Bipolar Disorder; Female; Humans; Imipramine; Male; Neuroleptic Malignant Syndrome; Penfluridol; Piperidines; Schizophrenia

1987
Loading--a beneficial therapeutic effect using an oral long-acting drug, Penfluridol (SEMAP). A pilot study.
    The Israel journal of psychiatry and related sciences, 1986, Volume: 23, Issue:3

    Topics: Administration, Oral; Adult; Delayed-Action Preparations; Drug Administration Schedule; Humans; Penfluridol; Piperidines; Schizophrenia

1986
Neuroleptic malignant syndrome due to combination of penfluridol and sulpiride?
    Acta psychiatrica Scandinavica, 1987, Volume: 75, Issue:3

    Topics: Aged; Drug Interactions; Female; Humans; Middle Aged; Neuroleptic Malignant Syndrome; Penfluridol; Piperidines; Sulpiride

1987
[Semap treatment of paranoid schizophrenics].
    Vrachebnoe delo, 1986, Issue:8

    Topics: Adult; Chronic Disease; Drug Evaluation; Humans; Male; Penfluridol; Piperidines; Schizophrenia, Paranoid; Time Factors

1986
Concentration in plasma of an orally long-acting new neuroleptic, penfluridol.
    Acta psychiatrica Scandinavica. Supplementum, 1974, Volume: 255

    Topics: Half-Life; Humans; Penfluridol; Piperidines; Schizophrenia

1974
Plasma prolactin and testosterone during penfluridol treatment.
    Lancet (London, England), 1980, Jul-12, Volume: 2, Issue:8185

    Topics: Adult; Humans; Male; Penfluridol; Piperidines; Prolactin; Schizophrenia; Testosterone

1980
Plasma prolactin and testosterone during penfluridol treatment.
    Lancet (London, England), 1980, Aug-16, Volume: 2, Issue:8190

    Topics: Humans; Male; Penfluridol; Piperidines; Prolactin; Schizophrenia; Testosterone

1980
[Evaluation of a long-acting neuroleptic: penfluridol. Clinical and psychosocial evolution at a year follow-up].
    Acta psiquiatrica y psicologica de America latina, 1981, Volume: 27, Issue:3

    Topics: Adolescent; Adult; Brief Psychiatric Rating Scale; Family; Female; Follow-Up Studies; Humans; Male; Penfluridol; Piperidines; Rehabilitation, Vocational; Schizophrenia; Social Adjustment; Socioeconomic Factors; Surveys and Questionnaires

1981
Effects of pimozide and penfluridol on the binding and endocytosis of alpha 2-macroglobulin-CH3NH2 by mouse peritoneal macrophages.
    Biochemical pharmacology, 1984, Nov-15, Volume: 33, Issue:22

    Topics: alpha-Macroglobulins; Animals; Calcium; Endocytosis; Kinetics; Low Density Lipoprotein Receptor-Related Protein-1; Macrophages; Methylamines; Mice; Penfluridol; Pimozide; Piperidines; Receptors, Immunologic

1984
A preliminary study of sex-related differences in prolactin responses to dopamine blockade and insulin hypoglycemia and in penfluridol plasma levels in schizophrenic patients.
    Psychopharmacology, 1983, Volume: 80, Issue:1

    Topics: Adult; Female; Humans; Hypoglycemia; Insulin; Kinetics; Male; Middle Aged; Penfluridol; Piperidines; Prolactin; Receptors, Dopamine; Schizophrenia; Sex Factors

1983
Penfluridol decreases secretagogue-induced TSH, GH, and LH secretion in vitro: a possible role for calcium-calmodulin.
    Neuroendocrinology, 1983, Volume: 37, Issue:3

    Topics: Animals; Calmodulin; Dose-Response Relationship, Drug; Female; Growth Hormone; Luteinizing Hormone; Penfluridol; Piperidines; Pituitary Gland, Anterior; Pituitary Hormones, Anterior; Rats; Rats, Inbred Strains; Thyrotropin; Thyrotropin-Releasing Hormone

1983
Inhibition of growth and of thymidine incorporation into DNA in Tetrahymena by chlorpromazine, pimozide and penfluridol.
    The Journal of protozoology, 1983, Volume: 30, Issue:2

    Topics: Animals; Chlorpromazine; DNA; Dose-Response Relationship, Drug; Penfluridol; Pimozide; Piperidines; Tetrahymena pyriformis; Thymidine; Thymine Nucleotides

1983
[Penfluridol in outpatient psychiatric practice].
    Ceskoslovenska psychiatrie, 1984, Volume: 80, Issue:3

    Topics: Adult; Ambulatory Care; Female; Humans; Male; Penfluridol; Piperidines; Schizophrenia

1984
Two novel agents affecting eating through an action on monoaminergic systems.
    International journal of obesity, 1984, Volume: 8 Suppl 1

    Topics: Animals; Appetite Depressants; Dextroamphetamine; Drug Tolerance; Eating; Female; Fenfluramine; Lethal Dose 50; Metergoline; Methysergide; Penfluridol; Phentolamine; Piperazines; Piperidines; Propranolol; Pyridines; Rats; Rats, Inbred Strains; Serotonin

1984
[Treatment of 326 cases of schizophrenia with domestic penfluridol].
    Zhonghua shen jing jing shen ke za zhi = Chinese journal of neurology and psychiatry, 1983, Volume: 16, Issue:2

    Topics: Adolescent; Adult; Aged; Child; Dose-Response Relationship, Drug; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia

1983
[Double-blind study of domestic penfluridol and fluphenazine decanoate].
    Zhonghua shen jing jing shen ke za zhi = Chinese journal of neurology and psychiatry, 1983, Volume: 16, Issue:3

    Topics: Adolescent; Adult; Basal Ganglia Diseases; Double-Blind Method; Fluphenazine; Humans; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia

1983
Clinical efficacy of haloperidol, pimozide, penfluridol, and clonidine in the treatment of tourette syndrome.
    Advances in neurology, 1982, Volume: 35

    Topics: Child; Child, Preschool; Clonidine; Haloperidol; Humans; Penfluridol; Pimozide; Piperidines; Tourette Syndrome

1982
[Clinical observation on 81 cases of schizophrenia treated with domestic penfluridol (author's transl)].
    Zhonghua shen jing jing shen ke za zhi = Chinese journal of neurology and psychiatry, 1981, Volume: 14, Issue:3

    Topics: Adult; Dose-Response Relationship, Drug; Female; Humans; Male; Middle Aged; Penfluridol; Piperidines; Schizophrenia; Time Factors

1981
Effects of the neuroprotectant lubeluzole on the cytotoxic actions of veratridine, barium, ouabain and 6-hydroxydopamine in chromaffin cells.
    British journal of pharmacology, 1998, Volume: 124, Issue:6

    Topics: Adrenal Glands; Animals; Barium; Calcium; Cattle; Chromaffin Cells; Cytosol; Neuroprotective Agents; Ouabain; Oxidopamine; Penfluridol; Piperidines; Sodium; Thiazoles; Veratridine

1998
Dual pharmacological properties of a cyclic AMP-sensitive potassium channel.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:1

    Topics: Animals; Antipsychotic Agents; Calcium Channel Blockers; Cattle; Cyclic AMP; Cyclic Nucleotide-Gated Cation Channels; Diltiazem; In Vitro Techniques; Ion Channel Gating; Ion Channels; Male; Membrane Potentials; Patch-Clamp Techniques; Penfluridol; Piperidines; Potassium Channel Blockers; Potassium Channels; Zona Fasciculata

1999
Differential inhibition of T-type calcium channels by neuroleptics.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Jan-15, Volume: 22, Issue:2

    Topics: Antipsychotic Agents; Calcium Channel Blockers; Calcium Channels, T-Type; Cell Line; Dose-Response Relationship, Drug; Flunarizine; Haloperidol; Humans; Ion Channel Gating; Kidney; Patch-Clamp Techniques; Penfluridol; Pimozide; Piperidines; Transfection

2002
Adrenal fasciculata cells express T-type and rapidly and slowly activating L-type Ca2+ channels that regulate cortisol secretion.
    American journal of physiology. Cell physiology, 2015, Jun-01, Volume: 308, Issue:11

    Topics: Action Potentials; Adrenocorticotropic Hormone; Angiotensin II; Animals; Benzamides; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, T-Type; Cattle; Cyclic AMP; Dihydropyridines; Fluspirilene; Gene Expression; Hydrocortisone; Microelectrodes; Nifedipine; Patch-Clamp Techniques; Penfluridol; Pimozide; Piperidines; Protein Isoforms; Single-Cell Analysis; Zona Fasciculata

2015