Page last updated: 2024-08-23

penfluridol and pimozide

penfluridol has been researched along with pimozide in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-199014 (58.33)18.7374
1990's5 (20.83)18.2507
2000's2 (8.33)29.6817
2010's2 (8.33)24.3611
2020's1 (4.17)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Bleich, S; Gulbins, E; Kornhuber, J; Reichel, M; Terfloth, L; Tripal, P; Wiltfang, J1
Cho, YS; Hwang, EM; Jung, SY; Lim, SM; Min, SJ; Pae, AN; Park, KD; Viswanath, AN1
Nose, T; Takemoto, H1
Ahlenius, S; Engel, J; Lundborg, P1
Pluym, A1
Carlsson, A1
König, L; Lange, E1
Janssen, PA; Lenaerts, FM; Niemegeers, CJ; Schellekens, KH; Wauquier, A1
Kourounakis, PN; Rekka, E; Tani, E1
Stárková, L; Wiedermann, J1
Biagi, BA; Day, RN; Enyeart, JJ; Maurer, RA; Sheu, SS1
Brannan, MD; Flaim, SF; Gleason, MM; Muschek, LD; Swigart, SC1
Hopkała, H; Przyborowski, L1
Lackington, I; Orrego, F1
Key, KA; Oakley, AC; Pizzo, SV1
Judd, AM; MacLeod, RM; Schettini, G1
Blum, JJ; Keegan, FP1
Shapiro, AK; Shapiro, E1
Enyeart, JA; Enyeart, JJ; Mlinar, B1
Canchola-Martínez, E; Mercado-Sánchez, G; Rodríguez-Medina, MA; Vergara-Onofre, M1
Cayabyab, FS; Hamming, KS; McRory, JE; Mezeyova, J; Parker, D; Santi, CM; Snutch, TP; Stea, A; Sutton, KG1
Enyeart, JA; Enyeart, JJ1
Abou Farraj, R; Al Batran, R; Chahade, JJ; Chan, JSF; Crawford, PA; Eaton, F; Glover, JNM; Gopal, K; Greenwell, AA; Lee, C; Saed, CT; Tabatabaei Dakhili, SA; Ussher, JR; Velázquez-Martínez, CA; Yang, K1

Other Studies

24 other study(ies) available for penfluridol and pimozide

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Identification of new functional inhibitors of acid sphingomyelinase using a structure-property-activity relation model.
    Journal of medicinal chemistry, 2008, Jan-24, Volume: 51, Issue:2

    Topics: Algorithms; Animals; Cell Line; Cell Line, Tumor; Chemical Phenomena; Chemistry, Physical; Enzyme Inhibitors; Humans; Hydrogen-Ion Concentration; Molecular Conformation; Quantitative Structure-Activity Relationship; Rats; Sphingomyelin Phosphodiesterase

2008
Identification of the first in silico-designed TREK1 antagonists that block channel currents dose dependently.
    Chemical biology & drug design, 2016, Volume: 88, Issue:6

    Topics: Animals; Computer Simulation; Crystallography, X-Ray; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Mice; Mice, Knockout; Molecular Docking Simulation; Potassium Channels, Tandem Pore Domain

2016
The effect of penfluridol and some psychotropic drugs on monoamine metabolism in central nervous system.
    European journal of pharmacology, 1975, Volume: 31, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Biogenic Amines; Brain; Brain Chemistry; Chlordiazepoxide; Chlorpromazine; Diazepam; Dopamine; Haloperidol; Homovanillic Acid; Hydroxyindoleacetic Acid; Male; Mice; Norepinephrine; Penfluridol; Pimozide; Piperazines; Piperidines; Psychotropic Drugs; Rats; Serotonin

1975
Antagonism by d-amphetamine of learning deficits in rats induced by exposure to antipsychotic drugs during early postnatal life.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 288, Issue:2-3

    Topics: Animals; Animals, Newborn; Antipsychotic Agents; Avoidance Learning; Dextroamphetamine; Discrimination Learning; Female; Learning; Light; Male; Penfluridol; Pimozide; Rats

1975
TLC differentiation of butyrophenone and diphenylbutylpiperidine compounds from phenothiazine derivatives.
    Journal of pharmaceutical sciences, 1979, Volume: 68, Issue:8

    Topics: Butyrophenones; Chromatography, Thin Layer; Fluspirilene; Indicators and Reagents; Penfluridol; Phenothiazines; Pimozide; Piperidines

1979
Age-dependent changes in central dopaminergic and other monoaminergic systems.
    Advances in experimental medicine and biology, 1978, Volume: 113

    Topics: Aging; Animals; Avoidance Learning; Biogenic Amines; Castration; Child; Dihydroxyphenylalanine; Dopamine; Female; Humans; Male; Neurons; Penfluridol; Pimozide; Rats; Receptors, Dopamine; Tyrosine

1978
[Significance and advantages of Orap in the ambulatory care of schizophrenic psychoses].
    Psychiatrie, Neurologie, und medizinische Psychologie, 1976, Volume: 28, Issue:2

    Topics: Adolescent; Adult; Aged; Ambulatory Care; Cyclothymic Disorder; Depression; Depressive Disorder, Major; Female; Fluphenazine; Fluspirilene; Haloperidol; Humans; Male; Middle Aged; Penfluridol; Pimozide; Remission, Spontaneous; Schizophrenia; Therapeutic Equivalency

1976
Clopimozide (R 29 764), a new highly potent and orally long-acting neuroleptic of the diphenylbutylpiperidine series.
    Arzneimittel-Forschung, 1975, Volume: 25, Issue:8

    Topics: Animals; Apomorphine; Avoidance Learning; Behavior, Animal; Benzimidazoles; Blepharoptosis; Body Temperature Regulation; Body Weight; Catalepsy; Dextroamphetamine; Dogs; Escape Reaction; Female; Guinea Pigs; Haloperidol; Humans; Lethal Dose 50; Male; Mice; Norepinephrine; Penfluridol; Pimozide; Piperidines; Rats; Self Stimulation; Stereotyped Behavior; Tranquilizing Agents

1975
Modification of lipid peroxidation by some known substituted imidazole derivatives. An attempt to correlate their antioxidant activity with lipophilicity.
    Die Pharmazie, 1991, Volume: 46, Issue:2

    Topics: Animals; Antioxidants; Astemizole; Benzimidazoles; Chemical Phenomena; Chemistry, Physical; Chromatography, Thin Layer; Imidazoles; In Vitro Techniques; Lipid Peroxidation; Lipids; Microsomes, Liver; Penfluridol; Pimozide; Piperazines; Rats

1991
Our experience with incisive neuroleptic drugs in child psychiatry.
    Acta Universitatis Palackianae Olomucensis Facultatis Medicae, 1991, Volume: 131

    Topics: Antipsychotic Agents; Autistic Disorder; Child; Haloperidol; Humans; Mental Disorders; Obsessive-Compulsive Disorder; Penfluridol; Pimozide; Psychotic Disorders; Sulpiride; Tic Disorders

1991
Blockade of low and high threshold Ca2+ channels by diphenylbutylpiperidine antipsychotics linked to inhibition of prolactin gene expression.
    The Journal of biological chemistry, 1990, Sep-25, Volume: 265, Issue:27

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Cell Line; Fluspirilene; Gene Expression; Kinetics; Luciferases; Membrane Potentials; Penfluridol; Pimozide; Piperidines; Pituitary Neoplasms; Prolactin; Recombinant Fusion Proteins; Spiro Compounds; Thyrotropin-Releasing Hormone

1990
Neuroleptic drugs attenuate calcium influx and tension development in rabbit thoracic aorta: effects of pimozide, penfluridol, chlorpromazine, and haloperidol.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:4

    Topics: Animals; Antipsychotic Agents; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Chlorpromazine; Haloperidol; In Vitro Techniques; Ion Channels; Male; Muscle Contraction; Penfluridol; Pimozide; Rabbits

1985
Determination of drugs containing fluorine with ion-selective electrode. Part 2: Butyrophenones and bis(4-fluorophenyl)butylpiperidines.
    Die Pharmazie, 1989, Volume: 44, Issue:1

    Topics: Butyrophenones; Electrodes; Fluorine; Penfluridol; Pimozide; Piperidines; Potentiometry; Spectrophotometry, Ultraviolet

1989
Inhibition of calcium-activated potassium conductance of human erythrocytes by calmodulin inhibitory drugs.
    FEBS letters, 1981, Oct-12, Volume: 133, Issue:1

    Topics: Adenosine Triphosphatases; Ca(2+) Mg(2+)-ATPase; Calcimycin; Calcium; Calcium-Binding Proteins; Calcium-Transporting ATPases; Calmodulin; Erythrocyte Membrane; Erythrocytes; Fluspirilene; Humans; Kinetics; Penfluridol; Phenothiazines; Pimozide; Potassium

1981
Effects of pimozide and penfluridol on the binding and endocytosis of alpha 2-macroglobulin-CH3NH2 by mouse peritoneal macrophages.
    Biochemical pharmacology, 1984, Nov-15, Volume: 33, Issue:22

    Topics: alpha-Macroglobulins; Animals; Calcium; Endocytosis; Kinetics; Low Density Lipoprotein Receptor-Related Protein-1; Macrophages; Methylamines; Mice; Penfluridol; Pimozide; Piperidines; Receptors, Immunologic

1984
In vitro studies on basal and stimulated prolactin release by rat anterior pituitary: a possible role for calmodulin.
    Endocrinology, 1983, Volume: 112, Issue:1

    Topics: Animals; Bucladesine; Calcimycin; Calcium-Binding Proteins; Calmodulin; Haloperidol; Penfluridol; Pimozide; Pituitary Gland, Anterior; Potassium; Prolactin; Rats; Rats, Inbred Strains; Theophylline; Thyrotropin-Releasing Hormone

1983
Inhibition of growth and of thymidine incorporation into DNA in Tetrahymena by chlorpromazine, pimozide and penfluridol.
    The Journal of protozoology, 1983, Volume: 30, Issue:2

    Topics: Animals; Chlorpromazine; DNA; Dose-Response Relationship, Drug; Penfluridol; Pimozide; Piperidines; Tetrahymena pyriformis; Thymidine; Thymine Nucleotides

1983
Clinical efficacy of haloperidol, pimozide, penfluridol, and clonidine in the treatment of tourette syndrome.
    Advances in neurology, 1982, Volume: 35

    Topics: Child; Child, Preschool; Clonidine; Haloperidol; Humans; Penfluridol; Pimozide; Piperidines; Tourette Syndrome

1982
T-type Ca2+ channels are required for adrenocorticotropin-stimulated cortisol production by bovine adrenal zona fasciculata cells.
    Molecular endocrinology (Baltimore, Md.), 1993, Volume: 7, Issue:8

    Topics: Adrenocorticotropic Hormone; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cattle; Cells, Cultured; Cyclic AMP; Dihydropyridines; Hydrocortisone; Insulin-Like Growth Factor I; Male; Penfluridol; Pimozide; Signal Transduction; Zona Fasciculata

1993
[Inhibitors of calcium-calmodulin system and hypothalamic sex differentiation in rats. Biochemical parameters].
    Ginecologia y obstetricia de Mexico, 1997, Volume: 65

    Topics: Animals; Animals, Newborn; Antipsychotic Agents; Calcium Channel Blockers; Calmodulin; DNA; Dopamine Antagonists; Female; Haloperidol; Hypothalamus; Male; Organ Size; Ovary; Penfluridol; Pimozide; Proteins; Rats; RNA; Sex Differentiation; Testis; Trifluoperazine; Verapamil

1997
Differential inhibition of T-type calcium channels by neuroleptics.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Jan-15, Volume: 22, Issue:2

    Topics: Antipsychotic Agents; Calcium Channel Blockers; Calcium Channels, T-Type; Cell Line; Dose-Response Relationship, Drug; Flunarizine; Haloperidol; Humans; Ion Channel Gating; Kidney; Patch-Clamp Techniques; Penfluridol; Pimozide; Piperidines; Transfection

2002
Adrenal fasciculata cells express T-type and rapidly and slowly activating L-type Ca2+ channels that regulate cortisol secretion.
    American journal of physiology. Cell physiology, 2015, Jun-01, Volume: 308, Issue:11

    Topics: Action Potentials; Adrenocorticotropic Hormone; Angiotensin II; Animals; Benzamides; Calcium; Calcium Channel Blockers; Calcium Channels, L-Type; Calcium Channels, T-Type; Cattle; Cyclic AMP; Dihydropyridines; Fluspirilene; Gene Expression; Hydrocortisone; Microelectrodes; Nifedipine; Patch-Clamp Techniques; Penfluridol; Pimozide; Piperidines; Protein Isoforms; Single-Cell Analysis; Zona Fasciculata

2015
The Antipsychotic Dopamine 2 Receptor Antagonist Diphenylbutylpiperidines Improve Glycemia in Experimental Obesity by Inhibiting Succinyl-CoA:3-Ketoacid CoA Transferase.
    Diabetes, 2023, 01-01, Volume: 72, Issue:1

    Topics: Animals; Antipsychotic Agents; Coenzyme A-Transferases; Diabetes Mellitus, Type 2; Dopamine; Fluspirilene; Hyperglycemia; Mice; Mice, Obese; Penfluridol; Pimozide; Receptors, Dopamine

2023