Page last updated: 2024-08-24

pemirolast and pyrimidinones

pemirolast has been researched along with pyrimidinones in 44 studies

Research

Studies (44)

TimeframeStudies, this research(%)All Research%
pre-19906 (13.64)18.7374
1990's18 (40.91)18.2507
2000's14 (31.82)29.6817
2010's5 (11.36)24.3611
2020's1 (2.27)2.80

Authors

AuthorsStudies
Furui, T; Imai, A; Matsuda, T; Matsunami, K; Ohno, T; Tamaya, T1
Bernstein, IL; Bierman, CW; Kemp, JP; Li, JT; Siegel, SC; Spangenberg, RD; Tinkelman, DG1
Fujimiya, H; Miyata, H; Nakashima, S; Nozawa, Y1
Berkowitz, RB; Tinkelman, DG1
Kasai, H; Shida, T; Yanagihara, Y1
Kasai, H; Kawashima, T; Shida, T; Yanagihara, Y1
Kawashima, T; Tomioka, H; Yoshida, S1
Kasai, H; Matsui, S; Ninomiya, K; Yanagihara, Y1
Kasai, H; Kawashima, T; Ninomiya, K; Yanagihara, Y1
Cheng, H; Dandekar, KA; Pittman, KA1
Higasida, M; Jikuhara, Y; Nakagawa, Y; Yuasa, T1
Fujimiya, H; Kumada, T; Miyata, H; Nakamura, Y; Nakashima, S; Nozawa, Y; Ojio, K1
Fujimiya, H; Kato, Y; Kumada, T; Miyata, H; Nakamura, Y; Nakashima, S; Nozawa, Y1
Hasegawa, T; Nabeshima, T; Nadai, M; Ogura, Y; Takagi, K1
Iwamoto, I; Kawashima, T; Nakagawa, N; Tomioka, H; Yoshida, S1
Fujimiya, H; Kumada, T; Miyata, H; Nakamura, Y; Nakashima, S; Nozawa, Y1
Eura, M; Ishikawa, T; Masuyama, K; Minoda, R; Toriya, T; Uno, K1
Fujita, J; Hirashima, M; Ohnishi, T; Okada, H; Takahara, J; Todani, T; Yamaji, Y1
Kondo, K; Miyazawa, N; Nakashima, M; Umemura, K1
Gamache, DA; Miller, ST; Sharif, NA; Spellman, JM; Xu, S; Yanni, JM1
Iijima, H; Liu, Y; Shirato, K; Tamura, G; Taniguchi, H1
Aoyagi, K; Hitsumoto, T; Kanai, M; Kawamura, K; Mineoka, K; Noike, H; Ohsawa, H; Sakurai, T; Sato, S; Tokuhiro, K; Tomioka, H; Uchi, T; Uchida, Y; Yoshinuma, M1
Jin, D; Miyazaki, M; Shiota, N; Takai, S1
Yoshinuma, M1
Abelson, MB; Amdahl, LD; Berdy, GJ; Graves, AL; Mundorf, T1
Amdahl, L; Graves, A; Shulman, DG; Washington, C1
Aoyagi, K; Hitsumoto, T; Iizuka, T; Kaku, M; Kanai, M; Matsumoto, J; Noike, H; Ohsawa, H; Sakuragawa, H; Sakurai, T; Shimizu, K; Sugiyama, Y; Takahashi, M; Tokuhiro, K; Tomaru, T; Yoshinaga, K1
Goromaru, T; Hirakawa, T; Itoh, Y; Nakano, H; Oishi, R; Sendo, T; Takasaki, S1
Gous, P; Ropo, A1
Hossen, MA; Kamei, C; Minami, K1
Kunitomo, M; Otsuka, H1
Hirakawa, T; Itoh, Y; Nakano, H; Oishi, R; Saito, M; Sendo, T; Uchida, M; Yahata, H1
Audus, KL; Proudfoot, J; Yazdanian, M; Young, AM1
Hwang, DG; Magone, MT; Maric, I1
Inaba, T; Shishikura, T; Shito, K; Uchida, M1
Gohda, T; Hamada, C; Kawachi, H; Ra, C; Tomino, Y; Tsuge, T1
Fujishima, H; Fukagawa, K; Fukushima, A; Miyazaki, D; Nakagawa, Y; Okamoto, S; Takamura, E; Tanaka, M; Uchio, E; Yokoi, N1
Li, J; Yan, XM1
Egashira, N; Kawashiri, T; Kurobe, K; Matsushita, N; Oishi, R; Tatsushima, Y; Yano, T1
Egashira, N; Kawashiri, T; Oishi, R; Yano, T1
Bredahl, K; Eldrup, N; Hultgren, R; Lindeman, J; Sillesen, H; Swedenborg, J; Thompson, M; Wanhainen, A; Wingren, U1
Ben-Eli, H; Solomon, A1
Shen, T; Yang, Z1

Reviews

1 review(s) available for pemirolast and pyrimidinones

ArticleYear
Topical antihistamines, mast cell stabilizers, and dual-action agents in ocular allergy: current trends.
    Current opinion in allergy and clinical immunology, 2018, Volume: 18, Issue:5

    Topics: Administration, Ophthalmic; Anti-Allergic Agents; Benzazepines; Conjunctivitis, Allergic; Cromolyn Sodium; Dibenzazepines; Histamine Antagonists; Humans; Hyperemia; Imidazoles; Ketotifen; Nedocromil; Olopatadine Hydrochloride; Phthalazines; Piperidines; Pruritus; Pyridines; Pyrimidinones

2018

Trials

11 trial(s) available for pemirolast and pyrimidinones

ArticleYear
Pemirolast, a new oral nonbronchodilator drug for chronic asthma.
    Annals of allergy, 1992, Volume: 68, Issue:6

    Topics: Administration, Oral; Adolescent; Adult; Aged; Asthma; Bronchial Spasm; Chronic Disease; Double-Blind Method; Forced Expiratory Volume; Histamine Antagonists; Humans; Middle Aged; Placebos; Pyridines; Pyrimidinones

1992
A pilot study of pemirolast in patients with seasonal allergic rhinitis.
    Annals of allergy, 1991, Volume: 66, Issue:2

    Topics: Adolescent; Adult; Eosinophils; Female; Follow-Up Studies; Histamine Antagonists; Humans; Leukocyte Count; Male; Middle Aged; Nasal Mucosa; Pyridines; Pyrimidinones; Rhinitis, Allergic, Seasonal

1991
Kinetic interaction between theophylline and a newly developed anti-allergic drug, pemirolast potassium.
    European journal of clinical pharmacology, 1994, Volume: 46, Issue:1

    Topics: Adult; Delayed-Action Preparations; Drug Interactions; Half-Life; Histamine Antagonists; Humans; Liver; Male; Pyridines; Pyrimidinones; Theophylline

1994
Preventive effects of an antiallergic drug, pemirolast potassium, on restenosis after percutaneous transluminal coronary angioplasty.
    American heart journal, 1998, Volume: 136, Issue:6

    Topics: Aged; Angioplasty, Balloon, Coronary; Cell Division; Coronary Angiography; Coronary Disease; Female; Histamine Antagonists; Humans; Male; Middle Aged; Muscle, Smooth, Vascular; Prospective Studies; Pyridines; Pyrimidinones; Secondary Prevention

1998
[Preventive mechanisms and effects of pemirolast potassium on restenosis after percutaneous transluminal coronary angioplasty: serial coronary angiography and intravascular ultrasound studies].
    Journal of cardiology, 1999, Volume: 33, Issue:2

    Topics: Angioplasty, Balloon, Coronary; Coronary Angiography; Coronary Disease; Endosonography; Female; Follow-Up Studies; Histamine Antagonists; Humans; Male; Middle Aged; Pyridines; Pyrimidinones; Recurrence

1999
Pemirolast potassium 0.1% ophthalmic solution is an effective treatment for allergic conjunctivitis: a pooled analysis of two prospective, randomized, double-masked, placebo-controlled, phase III studies.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 2002, Volume: 18, Issue:5

    Topics: Adolescent; Adult; Aged; Child; Conjunctivitis, Allergic; Double-Blind Method; Female; Histamine Antagonists; Humans; Male; Middle Aged; Ophthalmic Solutions; Prospective Studies; Pyridines; Pyrimidinones; Treatment Outcome

2002
A combined analysis of two studies assessing the ocular comfort of antiallergy ophthalmic agents.
    Clinical therapeutics, 2003, Volume: 25, Issue:4

    Topics: Administration, Topical; Adult; Anti-Allergic Agents; Conjunctivitis, Allergic; Cromolyn Sodium; Double-Blind Method; Female; Histamine Antagonists; Humans; Ketorolac; Male; Middle Aged; Nedocromil; Ophthalmic Solutions; Patient Compliance; Pyridines; Pyrimidinones; Treatment Outcome

2003
A comparative trial of the safety and efficacy of 0.1 percent pemirolast potassium ophthalmic solution dosed twice or four times a day in patients with seasonal allergic conjunctivitis.
    Journal of ocular pharmacology and therapeutics : the official journal of the Association for Ocular Pharmacology and Therapeutics, 2004, Volume: 20, Issue:2

    Topics: Adolescent; Adult; Aged; Child; Conjunctivitis, Allergic; Drug Administration Schedule; Female; Histamine Antagonists; Humans; Instillation, Drug; Male; Middle Aged; Ophthalmic Solutions; Prospective Studies; Pyridines; Pyrimidinones; Seasons; Treatment Outcome

2004
Prophylactic effect of pemirolast, an antiallergic agent, against hypersensitivity reactions to paclitaxel in patients with ovarian cancer.
    International journal of cancer, 2006, May-15, Volume: 118, Issue:10

    Topics: Administration, Oral; Antineoplastic Agents, Phytogenic; Antineoplastic Combined Chemotherapy Protocols; Carboplatin; Drug Hypersensitivity; Female; Histamine Antagonists; Humans; Ovarian Neoplasms; Paclitaxel; Placebos; Pyridines; Pyrimidinones

2006
The effect of a combined therapy with a histamine H1 antagonist and a chemical mediator release inhibitor on allergic conjunctivitis.
    Ophthalmologica. Journal international d'ophtalmologie. International journal of ophthalmology. Zeitschrift fur Augenheilkunde, 2008, Volume: 222, Issue:4

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Child; Conjunctivitis, Allergic; Drug Therapy, Combination; Eosinophils; Female; Histamine H1 Antagonists, Non-Sedating; Humans; Leukocyte Count; Male; Middle Aged; Ophthalmic Solutions; Piperidines; Pyridines; Pyrimidinones; Treatment Outcome

2008
Randomized clinical trial of mast cell inhibition in patients with a medium-sized abdominal aortic aneurysm.
    The British journal of surgery, 2015, Volume: 102, Issue:8

    Topics: Aged; Aged, 80 and over; Anti-Inflammatory Agents; Aortic Aneurysm, Abdominal; Double-Blind Method; Female; Humans; Male; Mast Cells; Middle Aged; Pyridines; Pyrimidinones; Ultrasonography

2015

Other Studies

32 other study(ies) available for pemirolast and pyrimidinones

ArticleYear
Evidence of a role for phosphatidylinositol synthesis in human amnion cell proliferation.
    Biology of reproduction, 1992, Volume: 47, Issue:5

    Topics: Amnion; Calcimycin; Calcium; CDP-Diacylglycerol-Inositol 3-Phosphatidyltransferase; Cell Division; Cell Line; DNA; Dose-Response Relationship, Drug; Egtazic Acid; Gene Expression; Histamine Antagonists; Humans; Inositol; Magnesium; Membrane Proteins; Phosphatidylinositols; Phosphotransferases; Pyridines; Pyrimidinones; Time Factors; Transferases (Other Substituted Phosphate Groups)

1992
Effect of a novel antiallergic drug, pemirolast, on activation of rat peritoneal mast cells: inhibition of exocytotic response and membrane phospholipid turnover.
    International archives of allergy and applied immunology, 1991, Volume: 96, Issue:1

    Topics: Animals; Antigens, Helminth; Ascaris; Cell Degranulation; Cell Membrane; Exocytosis; Histamine Antagonists; Histamine Release; Mast Cells; p-Methoxy-N-methylphenethylamine; Peritoneal Cavity; Phospholipids; Pyridines; Pyrimidinones; Rats; Rats, Inbred Strains; Serotonin

1991
Immunopharmacological studies on TBX, a new antiallergic drug (2). Inhibitory effects on histamine release from peritoneal mast cells and lung fragments of rats.
    Japanese journal of pharmacology, 1988, Volume: 48, Issue:1

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Antigens; Calcimycin; Cromolyn Sodium; Cyclic AMP; Histamine Release; In Vitro Techniques; Lung; Male; Mast Cells; p-Methoxy-N-methylphenethylamine; Peritoneal Cavity; Pyridines; Pyrimidinones; Rats; Rats, Inbred Strains

1988
Immunopharmacological studies on TBX, a new antiallergic drug (1). Inhibitory effects on passive cutaneous anaphylaxis in rats and guinea pigs.
    Japanese journal of pharmacology, 1988, Volume: 48, Issue:1

    Topics: Animals; Cromolyn Sodium; Guinea Pigs; Immunoglobulin E; Immunoglobulin G; Male; ortho-Aminobenzoates; Passive Cutaneous Anaphylaxis; Pyridines; Pyrimidinones; Rats; Rats, Inbred Strains

1988
[Inhibition of chemical mediator release from human leukocytes and lung fragments by TBX].
    Arerugi = [Allergy], 1988, Volume: 37, Issue:7

    Topics: Animals; Depression, Chemical; Female; Guinea Pigs; Histamine Release; Humans; Leukocytes; Lung; Male; Pyridines; Pyrimidinones; SRS-A

1988
Immunopharmacological studies on TBX, a new antiallergic drug (3). Inhibitory effects on histamine release from lung fragments and bronchoconstriction in guinea pigs.
    Japanese journal of pharmacology, 1989, Volume: 51, Issue:1

    Topics: Animals; Asthma; Bronchi; Dinoprost; Guinea Pigs; Histamine Antagonists; Histamine Release; In Vitro Techniques; Lung; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Platelet Activating Factor; Platelet Aggregation; Pyridines; Pyrimidinones; SRS-A; Trachea

1989
Immunopharmacological studies on TBX, a new antiallergic drug (4). Effects on type II to IV allergic reactions and immunological functions in animal models.
    Japanese journal of pharmacology, 1989, Volume: 51, Issue:1

    Topics: Animals; Arthus Reaction; Cell Division; Complement System Proteins; Erythrocytes; Forssman Antigen; Guinea Pigs; Hemolysis; Histamine Antagonists; Hypersensitivity; Immunity, Cellular; Male; Mice; Mice, Inbred BALB C; Mice, Inbred ICR; Passive Cutaneous Anaphylaxis; Pyridines; Pyrimidinones; Rats; Rats, Inbred Strains; Sheep; Tuberculin Test

1989
Liquid chromatographic determination of 9-methyl-3-(1H-tetrazol-5-yl)-4H-pyrido[1,2-a]pyrimidin-4-one in human plasma with fluorescence detection.
    Journal of pharmaceutical sciences, 1987, Volume: 76, Issue:12

    Topics: Anti-Ulcer Agents; Chemical Phenomena; Chemistry; Chromatography, High Pressure Liquid; Drug Stability; Histamine H2 Antagonists; Humans; Pyridines; Pyridones; Pyrimidinones; Spectrometry, Fluorescence

1987
[Suppression of conjunctival provocation by 0.1% pemirolast potassium ophthalmic solution in VKC].
    Arerugi = [Allergy], 1994, Volume: 43, Issue:12

    Topics: Adolescent; Adult; Antigens; Conjunctiva; Conjunctivitis, Allergic; Female; Histamine Antagonists; Histamine Release; Humans; Male; Ophthalmic Solutions; Pyridines; Pyrimidinones

1994
[Effects of antiallergic drug, pemirolast potassium on phospholipase D activation in antigen-stimulated rat basophilic leukemia (RBL-2H3) cells].
    Arerugi = [Allergy], 1995, Volume: 44, Issue:6

    Topics: Animals; Antigens; Depression, Chemical; Enzyme Activation; Histamine Antagonists; Leukemia, Basophilic, Acute; Phospholipase D; Pyridines; Pyrimidinones; Rats; Tumor Cells, Cultured

1995
Effects of an antiallergic drug, pemirolast potassium on tyrosine phosphorylation and map kinase activation in antigen-stimulated rat basophilic leukemia (RBL-2H3) cells.
    Arerugi = [Allergy], 1995, Volume: 44, Issue:1

    Topics: Animals; Antigens; Calcium-Calmodulin-Dependent Protein Kinases; Enzyme Activation; Histamine Antagonists; Leukemia, Basophilic, Acute; Phosphorylation; Pyridines; Pyrimidinones; Rats; Tumor Cells, Cultured; Tyrosine

1995
Inhibitory effect of pemirolast, a novel antiallergic drug, on leukotriene C4 and granule protein release from human eosinophils.
    International archives of allergy and immunology, 1994, Volume: 103, Issue:4

    Topics: Asthma; Blood Proteins; Calcimycin; Eosinophil Granule Proteins; Eosinophils; Humans; In Vitro Techniques; Leukotriene C4; N-Formylmethionine Leucyl-Phenylalanine; Platelet Activating Factor; Pyridines; Pyrimidinones; Ribonucleases; Secretory Rate

1994
An antiallergic drug, pemirolast potassium, inhibits inositol 1,4,5-trisphosphate production and Ca2+ mobilization in antigen-stimulated rat basophilic leukemia (RBL-2H3) cells.
    Arerugi = [Allergy], 1994, Volume: 43, Issue:2 Pt 1

    Topics: Animals; Antigens; Calcium; Histamine Antagonists; Inositol 1,4,5-Trisphosphate; Leukemia, Basophilic, Acute; Phospholipases; Pyridines; Pyrimidinones; Rats; Tumor Cells, Cultured

1994
Recurrent hearing impairment and nystagmus induced by repeated antigen exposure in actively sensitized guinea pigs.
    International archives of allergy and immunology, 1996, Volume: 111, Issue:2

    Topics: Anaphylaxis; Animals; Cochlea; Dinitrophenols; Ear, Inner; Endolymphatic Hydrops; Guinea Pigs; Hearing Loss, Bilateral; Histamine Antagonists; Male; Nystagmus, Pathologic; Postural Balance; Pyridines; Pyrimidinones; Vaccination

1996
Anti-asthma effect of an antiviral drug, acyclovir: a clinical case and experimental study.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 1997, Volume: 27, Issue:4

    Topics: Acyclovir; Aminophylline; Animals; Anti-Asthmatic Agents; Antiviral Agents; Asthma; Bronchi; Bronchoalveolar Lavage Fluid; Bronchoconstriction; Calcimycin; Eosinophils; Guinea Pigs; Histamine Antagonists; Humans; Male; Middle Aged; Peak Expiratory Flow Rate; Pyridines; Pyrimidinones; Time Factors

1997
Effects of pemirolast and tranilast on intimal thickening after arterial injury in the rat.
    Journal of cardiovascular pharmacology, 1997, Volume: 30, Issue:2

    Topics: Animals; Antimetabolites; Arteries; Bromodeoxyuridine; Cell Division; Cell Movement; Cells, Cultured; Endothelium, Vascular; Histamine Antagonists; Histamine H1 Antagonists; ortho-Aminobenzoates; Pyridines; Pyrimidinones; Rats; Tunica Intima

1997
Comparative effects of topical ocular anti-allergy drugs on human conjunctival mast cells.
    Annals of allergy, asthma & immunology : official publication of the American College of Allergy, Asthma, & Immunology, 1997, Volume: 79, Issue:6

    Topics: Administration, Topical; Anti-Allergic Agents; Antibodies, Anti-Idiotypic; Conjunctiva; Dibenzoxepins; Histamine Release; Humans; Mast Cells; Nedocromil; Olopatadine Hydrochloride; Pyridines; Pyrimidinones; Receptors, Histamine H1

1997
[Antigen-induced airway hyperresponsiveness in infantile guinea pigs].
    Arerugi = [Allergy], 1998, Volume: 47, Issue:8

    Topics: Animals; Anti-Allergic Agents; Antigens; Arylsulfonates; Asthma; Bronchoalveolar Lavage Fluid; Disease Models, Animal; Guinea Pigs; Histamine Antagonists; Leukocyte Count; Male; Ovalbumin; Pyridines; Pyrimidinones; Respiratory Hypersensitivity; Sulfonium Compounds

1998
Tranilast, an anti-allergic drug, possesses antagonistic potency to angiotensin II.
    European journal of pharmacology, 1998, Nov-20, Volume: 361, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Adult; Aged; Aged, 80 and over; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Anti-Allergic Agents; Anti-Asthmatic Agents; Aorta; Arteries; Cromolyn Sodium; Dose-Response Relationship, Drug; Histamine Antagonists; Humans; In Vitro Techniques; Male; Middle Aged; Muscle, Smooth, Vascular; Norepinephrine; ortho-Aminobenzoates; Potassium Chloride; Pyridines; Pyrimidinones; Rabbits; Vasoconstriction

1998
New drugs for allergic conjunctivitis.
    The Medical letter on drugs and therapeutics, 2000, May-01, Volume: 42, Issue:1077

    Topics: Adult; Anti-Allergic Agents; Child; Child, Preschool; Clinical Trials as Topic; Conjunctivitis, Allergic; Headache; Histamine H1 Antagonists; Humans; Ketotifen; Nedocromil; Pyridines; Pyrimidinones; Rhinitis

2000
Preventive effect of an antiallergic drug, pemirolast potassium, on restenosis after stent placement: quantitative coronary angiography and intravascular ultrasound studies.
    Journal of cardiology, 2003, Volume: 42, Issue:1

    Topics: Aged; Angioplasty, Balloon, Coronary; Anti-Allergic Agents; Coronary Angiography; Coronary Disease; Coronary Restenosis; Coronary Vessels; Female; Humans; Male; Middle Aged; Pyridines; Pyrimidinones; Stents; Ultrasonography, Interventional

2003
Pemirolast potently attenuates paclitaxel hypersensitivity reactions through inhibition of the release of sensory neuropeptides in rats.
    Neuropharmacology, 2004, Volume: 46, Issue:6

    Topics: Animals; Calcitonin Gene-Related Peptide; Dose-Response Relationship, Drug; Drug Hypersensitivity; Male; Neurokinin A; Neuropeptides; Paclitaxel; Pyridines; Pyrimidinones; Rats; Rats, Sprague-Dawley; Substance P

2004
Increasing effect by simultaneous use of levocabastine and pemirolast on experimental allergic conjunctivitis in rats.
    Biological & pharmaceutical bulletin, 2005, Volume: 28, Issue:3

    Topics: Animals; Conjunctivitis, Allergic; Drug Synergism; Drug Therapy, Combination; Histamine Release; Male; Piperidines; Pyridines; Pyrimidinones; Rats; Rats, Wistar

2005
Comparison of antigen-induced leukotriene and histamine release from nasal scrapings in allergic rhinitis.
    Rhinology, 2005, Volume: 43, Issue:3

    Topics: Adolescent; Adult; Antigens, Dermatophagoides; Child; Female; Histamine Antagonists; Histamine Release; Humans; Leukotrienes; Male; Mast Cells; Nasal Mucosa; Pyridines; Pyrimidinones; Rhinitis, Allergic, Perennial; Time Factors; Tissue Culture Techniques

2005
Tetrazole compounds: the effect of structure and pH on Caco-2 cell permeability.
    Journal of pharmaceutical sciences, 2006, Volume: 95, Issue:4

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Benzimidazoles; Caco-2 Cells; Cell Line; Cell Membrane Permeability; Cell Polarity; Dogs; Drug Design; Humans; Hydrogen-Ion Concentration; Losartan; Membrane Transport Proteins; Multidrug Resistance-Associated Protein 2; Multidrug Resistance-Associated Proteins; Pyridines; Pyrimidinones; Structure-Activity Relationship; Tetrazoles; Transfection

2006
Peripheral interstitial keratitis: a novel manifestation of ocular mastocytosis.
    Cornea, 2006, Volume: 25, Issue:3

    Topics: Adult; Corneal Neovascularization; Corneal Stroma; Female; Glucocorticoids; Histamine Antagonists; Humans; Keratitis; Mast Cells; Prednisolone; Pyridines; Pyrimidinones; Urticaria Pigmentosa

2006
A late cutaneous response in actively sensitized rats: a new method for evaluating the efficacy of antiallergic drugs.
    Journal of pharmacological sciences, 2006, Volume: 101, Issue:4

    Topics: Aminopyridines; Animals; Anti-Allergic Agents; Antigens; Cromolyn Sodium; Cyclosporine; Dinitrobenzenes; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Evaluation, Preclinical; Edema; Haptens; Hindlimb; Hypersensitivity, Delayed; Male; ortho-Aminobenzoates; Ovalbumin; Passive Cutaneous Anaphylaxis; Promethazine; Pyridines; Pyrimidinones; Quinolones; Rats; Rats, Wistar

2006
Suppressive activity of pemirolast potassium, an antiallergic drug, on glomerulonephritis. Studies in glomerulonephritis model rats and in patients with chronic glomerulonephritis concurrently affected by allergic rhinitis.
    Arzneimittel-Forschung, 2008, Volume: 58, Issue:1

    Topics: Adolescent; Adult; Animals; Anti-Allergic Agents; Autoantibodies; Disease Models, Animal; Female; Glomerulonephritis; Histamine Antagonists; Humans; Kidney; Male; Middle Aged; Nephrectomy; Pilot Projects; Proteinuria; Pyridines; Pyrimidinones; Rats; Rats, Sprague-Dawley; Rats, Wistar; Rhinitis, Allergic, Seasonal; Thyroid Gland

2008
[Toxicity of topical ocular anti-allergic agents on human corneal epithelial cells in vitro].
    [Zhonghua yan ke za zhi] Chinese journal of ophthalmology, 2010, Volume: 46, Issue:1

    Topics: Anti-Allergic Agents; Cell Membrane Permeability; Cell Survival; Cells, Cultured; Dibenzoxepins; Epithelial Cells; Epithelium, Corneal; Humans; Ketotifen; Olopatadine Hydrochloride; Ophthalmic Solutions; Pyridines; Pyrimidinones

2010
Pemirolast reduces cisplatin-induced kaolin intake in rats.
    European journal of pharmacology, 2011, Jul-01, Volume: 661, Issue:1-3

    Topics: Animals; Antineoplastic Agents; Aprepitant; Biological Transport; Body Weight; Cisplatin; Dexamethasone; Eating; Kaolin; Male; Morpholines; Ondansetron; Pyridines; Pyrimidinones; Rats; Substance P

2011
[Substance P in antitumor drug-induced adverse reactions].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2013, Volume: 142, Issue:5

    Topics: Animals; Antineoplastic Agents; Carboplatin; Histamine Antagonists; Humans; Nausea; Neuropeptides; Paclitaxel; Pyridines; Pyrimidinones; Substance P; Vomiting

2013
In vivo and in vitro Evaluation of in situ Gel Formulation of Pemirolast Potassium in Allergic Conjunctivitis.
    Drug design, development and therapy, 2021, Volume: 15

    Topics: Animals; Conjunctivitis, Allergic; Drug Compounding; Gels; Mice; Mice, Inbred BALB C; Ophthalmic Solutions; Pyridines; Pyrimidinones; Rabbits; Viscosity

2021