pd168393 and erlotinib

pd168393 has been researched along with erlotinib in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (66.67)29.6817
2010's1 (33.33)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Grütter, C; Klüter, S; Michalczyk, A; Rabiller, M; Rauh, D; Rode, HB; Simard, JR1
Balk, SP; Didonato, M; Flatauer, L; Gray, NS; Hur, W; Jiang, X; Kim, S; Larson, B; Mason, DE; Nagle, A; Peters, EC; Suzuki, M; Valente, D; Velentza, A; Warmuth, M; Zagorska, A; Zhang, J1
Heynck, S; Pawar, VG; Rabiller, M; Rauh, D; Rode, HB; Sos, ML; Thomas, RK; van Otterlo, WA1

Other Studies

3 other study(ies) available for pd168393 and erlotinib

ArticleYear
Structural insights into how irreversible inhibitors can overcome drug resistance in EGFR.
    Bioorganic & medicinal chemistry, 2008, Apr-01, Volume: 16, Issue:7

    Topics: Crystallography, X-Ray; Drug Resistance; ErbB Receptors; Erlotinib Hydrochloride; Models, Molecular; Molecular Structure; Mutation; Protein Kinase Inhibitors; Quinazolines; Structure-Activity Relationship

2008
Clinical stage EGFR inhibitors irreversibly alkylate Bmx kinase.
    Bioorganic & medicinal chemistry letters, 2008, Nov-15, Volume: 18, Issue:22

    Topics: Animals; Cysteine; ErbB Receptors; Mice; Molecular Structure; Morpholines; Protein-Tyrosine Kinases; Quinazolines; Sequence Homology, Amino Acid

2008
Synthesis and biological evaluation of 4-anilinoquinolines as potent inhibitors of epidermal growth factor receptor.
    Journal of medicinal chemistry, 2010, Apr-08, Volume: 53, Issue:7

    Topics: Animals; Cell Line, Tumor; Drug Evaluation, Preclinical; ErbB Receptors; Inhibitory Concentration 50; Models, Molecular; Molecular Conformation; Mutation; Protein Kinase Inhibitors; Quinolines; Structure-Activity Relationship

2010