Page last updated: 2024-09-04

pd 85639 and piperidines

pd 85639 has been researched along with piperidines in 5 studies

Compound Research Comparison

Studies
(pd 85639)
Trials
(pd 85639)
Recent Studies (post-2010)
(pd 85639)
Studies
(piperidines)
Trials
(piperidines)
Recent Studies (post-2010) (piperidines)
50040,2355,22114,545

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Campbell, GW; Dooley, DJ; Hays, SJ; Probert, AW; Roufos, I; Schwarz, RD1
Catterall, WA; Numann, R; Ragsdale, DS; Scheuer, T1
Catterall, WA; Hays, SJ; Hicks, JL; Schwarz, RD; Thomsen, W1
Hays, S; Roufos, I; Schwarz, RD1
Obrenovitch, TP1

Reviews

1 review(s) available for pd 85639 and piperidines

ArticleYear
Sodium and potassium channel modulators: their role in neuroprotection.
    International review of neurobiology, 1997, Volume: 40

    Topics: Animals; Benzeneacetamides; Cell Survival; Disease Models, Animal; Lamotrigine; Neurons; Neuroprotective Agents; Piperazines; Piperidines; Potassium Channels; Pyrimidines; Riluzole; Sodium Channels; Thiazoles; Triazines

1997

Other Studies

4 other study(ies) available for pd 85639 and piperidines

ArticleYear
Synthesis and pharmacological evaluation of phenylacetamides as sodium-channel blockers.
    Journal of medicinal chemistry, 1994, Jan-21, Volume: 37, Issue:2

    Topics: Acetamides; Animals; Batrachotoxins; Benzeneacetamides; Cell Hypoxia; Cells, Cultured; Cerebral Cortex; CHO Cells; Cricetinae; L-Lactate Dehydrogenase; Male; Piperidines; Rats; Rats, Sprague-Dawley; Sodium; Sodium Channel Blockers; Structure-Activity Relationship; Veratridine

1994
Inhibition of Na+ channels by the novel blocker PD85,639.
    Molecular pharmacology, 1993, Volume: 43, Issue:6

    Topics: Animals; Benzeneacetamides; Binding Sites; Brain Chemistry; CHO Cells; Cricetinae; DNA; Electrophysiology; Membrane Potentials; Piperidines; Rats; Sodium Channels; Transfection

1993
Specific binding of the novel Na+ channel blocker PD85,639 to the alpha subunit of rat brain Na+ channels.
    Molecular pharmacology, 1993, Volume: 43, Issue:6

    Topics: Anesthetics, Local; Animals; Anticonvulsants; Batrachotoxins; Benzeneacetamides; Binding Sites; Binding, Competitive; Brain; CHO Cells; Cricetinae; Hydrogen-Ion Concentration; Neurotoxins; Piperidines; Rats; Sodium Channels; Synaptosomes

1993
A structure-activity relationship study of novel phenylacetamides which are sodium channel blockers.
    Journal of medicinal chemistry, 1996, Mar-29, Volume: 39, Issue:7

    Topics: Acetamides; Animals; Benzeneacetamides; CHO Cells; Cricetinae; Magnetic Resonance Spectroscopy; Molecular Structure; Piperidines; Sodium; Sodium Channel Blockers; Sodium Channels; Structure-Activity Relationship; Veratridine

1996