Page last updated: 2024-09-03

pd 81723 and sch-202676

pd 81723 has been researched along with sch-202676 in 2 studies

Compound Research Comparison

Studies
(pd 81723)
Trials
(pd 81723)
Recent Studies (post-2010)
(pd 81723)
Studies
(sch-202676)
Trials
(sch-202676)
Recent Studies (post-2010) (sch-202676)
550122008

Protein Interaction Comparison

ProteinTaxonomypd 81723 (IC50)sch-202676 (IC50)
Replicase polyprotein 1abSevere acute respiratory syndrome coronavirus 20.98
FascinHomo sapiens (human)0.5
N-terminal Xaa-Pro-Lys N-methyltransferase 1Homo sapiens (human)0.46

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Göblyös, A; Heitman, L; IJzerman, AP; Pietra, D; van den Nieuwendijk, AM1
Beukers, MW; de Grip, WJ; Ijzerman, AP; Klaasse, EC; Roerink, SF; van den Hout, G1

Other Studies

2 other study(ies) available for pd 81723 and sch-202676

ArticleYear
Synthesis and biological evaluation of 2,3,5-substituted [1,2,4]thiadiazoles as allosteric modulators of adenosine receptors.
    Journal of medicinal chemistry, 2004, Jan-29, Volume: 47, Issue:3

    Topics: Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Agonists; Adenosine A3 Receptor Antagonists; Allosteric Regulation; Animals; Binding, Competitive; Cell Line; Cricetinae; Humans; Kinetics; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Radioligand Assay; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptor, Adenosine A3; Receptors, Purinergic P1; Thiadiazoles; Thiazoles

2004
Allosteric modulators affect the internalization of human adenosine A1 receptors.
    European journal of pharmacology, 2005, Oct-17, Volume: 522, Issue:1-3

    Topics: Adenosine; Allosteric Regulation; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Endocytosis; Humans; Luminescent Proteins; Microscopy, Confocal; Radioligand Assay; Receptor, Adenosine A1; Recombinant Fusion Proteins; Thiadiazoles; Thiazoles; Thiophenes; Transfection; Tritium; Xanthines

2005