pd 81723 has been researched along with sch-202676 in 2 studies
Studies (pd 81723) | Trials (pd 81723) | Recent Studies (post-2010) (pd 81723) | Studies (sch-202676) | Trials (sch-202676) | Recent Studies (post-2010) (sch-202676) |
---|---|---|---|---|---|
55 | 0 | 12 | 20 | 0 | 8 |
Protein | Taxonomy | pd 81723 (IC50) | sch-202676 (IC50) |
---|---|---|---|
Replicase polyprotein 1ab | Severe acute respiratory syndrome coronavirus 2 | 0.98 | |
Fascin | Homo sapiens (human) | 0.5 | |
N-terminal Xaa-Pro-Lys N-methyltransferase 1 | Homo sapiens (human) | 0.46 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (100.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Göblyös, A; Heitman, L; IJzerman, AP; Pietra, D; van den Nieuwendijk, AM | 1 |
Beukers, MW; de Grip, WJ; Ijzerman, AP; Klaasse, EC; Roerink, SF; van den Hout, G | 1 |
2 other study(ies) available for pd 81723 and sch-202676
Article | Year |
---|---|
Synthesis and biological evaluation of 2,3,5-substituted [1,2,4]thiadiazoles as allosteric modulators of adenosine receptors.
Topics: Adenosine A1 Receptor Agonists; Adenosine A1 Receptor Antagonists; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adenosine A3 Receptor Agonists; Adenosine A3 Receptor Antagonists; Allosteric Regulation; Animals; Binding, Competitive; Cell Line; Cricetinae; Humans; Kinetics; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Radioligand Assay; Receptor, Adenosine A1; Receptor, Adenosine A2A; Receptor, Adenosine A3; Receptors, Purinergic P1; Thiadiazoles; Thiazoles | 2004 |
Allosteric modulators affect the internalization of human adenosine A1 receptors.
Topics: Adenosine; Allosteric Regulation; Animals; Binding, Competitive; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Endocytosis; Humans; Luminescent Proteins; Microscopy, Confocal; Radioligand Assay; Receptor, Adenosine A1; Recombinant Fusion Proteins; Thiadiazoles; Thiazoles; Thiophenes; Transfection; Tritium; Xanthines | 2005 |