Page last updated: 2024-09-03

pd 81723 and draflazine

pd 81723 has been researched along with draflazine in 3 studies

Compound Research Comparison

Studies
(pd 81723)
Trials
(pd 81723)
Recent Studies (post-2010)
(pd 81723)
Studies
(draflazine)
Trials
(draflazine)
Recent Studies (post-2010) (draflazine)
550125452

Protein Interaction Comparison

ProteinTaxonomypd 81723 (IC50)draflazine (IC50)
Equilibrative nucleoside transporter 1Homo sapiens (human)0.0053

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Belardinelli, L; Bruns, RF; Dennis, D; Kollias-Baker, C; Linden, J; Ruble, J1
Belardinelli, L; Kollias-Baker, C; Pelleg, A; Xu, J1
Belardinelli, L; Dennis, DM; Martens, JR; Raatikainen, MJ1

Other Studies

3 other study(ies) available for pd 81723 and draflazine

ArticleYear
Allosteric enhancer PD 81,723 acts by novel mechanism to potentiate cardiac actions of adenosine.
    Circulation research, 1994, Volume: 75, Issue:6

    Topics: Adenosine; Allosteric Regulation; Animals; Binding Sites; Brain; Bundle of His; Drug Synergism; Female; Guinea Pigs; Heart; Humans; In Vitro Techniques; Male; Membranes; Myocardium; Piperazines; Radioligand Assay; Receptors, Purinergic P1; Thiophenes

1994
Novel approach for enhancing atrioventricular nodal conduction delay mediated by endogenous adenosine.
    Circulation research, 1994, Volume: 75, Issue:6

    Topics: Adenosine; Animals; Atrioventricular Node; Bundle of His; Coronary Vessels; Female; Guinea Pigs; Hypoxia; In Vitro Techniques; Male; Piperazines; Receptors, Purinergic P1; Thiophenes; Tubercidin; Vasodilation

1994
Modulation of atrioventricular nodal function by metabolic and allosteric regulators of endogenous adenosine in guinea pig heart.
    Circulation, 1996, Nov-15, Volume: 94, Issue:10

    Topics: Adenosine; Allosteric Regulation; Animals; Atrioventricular Node; Biological Transport; Body Fluids; Enzyme Inhibitors; Guinea Pigs; Heart; Heart Conduction System; In Vitro Techniques; Myocardium; Nucleosides; Pericardium; Piperazines; Platelet Aggregation Inhibitors; Thiophenes; Tubercidin

1996