pd 169316 and u 0126

pd 169316 has been researched along with u 0126 in 16 studies

Research

Studies (16)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's14 (87.50)29.6817
2010's2 (12.50)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bullock, AN; Fedorov, O; Knapp, S; Marsden, B; Müller, S; Pogacic, V; Rellos, P; Schwaller, J; Sundström, M1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Inaguma, Y; Ito, H; Iwamoto, I; Kato, K; Lida, K1
Hisaoka, K; Koda, T; Miyata, M; Morinobu, S; Nishida, A; Ohta, M; Yamawaki, S; Zensho, H1
Hatakeyama, D; Kozawa, O; Uematsu, T1
Akamatsu, S; Hatakeyama, D; Kozawa, O; Shibata, T; Tanabe, K; Tokuda, H; Yoshida, M1
Almazan, G; Athlan, E; Fragoso, G; Mushynski, WE; Robertson, J; Tam, E1
Chue, SC; Duan, W; Koh, AH; Seow, CJ; Wong, WS; Yeo, KS2
Shafer, LM; Slice, LW1
Collman, RG; Freedman, BD; Lee, C; Tomkowicz, B1
Montesano, R1
Hong, HY; Kim, BC1
Carrozzino, F; Féraille, E; Montesano, R; Pugnale, P1
Alamdary, SZ; Ansari, N; Ashabi, G; Azizi, P; Haghparast, A; Khodagholi, F; Motamedi, F; Ramin, M; Taslimi, Z1
Alamdary, SZ; Ashabi, G; Khodagholi, F; Ramin, M1

Other Studies

16 other study(ies) available for pd 169316 and u 0126

ArticleYear
A systematic interaction map of validated kinase inhibitors with Ser/Thr kinases.
    Proceedings of the National Academy of Sciences of the United States of America, 2007, Dec-18, Volume: 104, Issue:51

    Topics: Amino Acid Sequence; Binding Sites; Clinical Trials as Topic; Drug Evaluation, Preclinical; Enzyme Stability; Humans; Molecular Sequence Data; Phylogeny; Protein Array Analysis; Protein Conformation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Protein kinase inhibitors can suppress stress-induced dissociation of Hsp27.
    Cell stress & chaperones, 2001, Volume: 6, Issue:1

    Topics: Anisomycin; Arsenites; Butadienes; Cadmium Chloride; Carcinogens; Dithiothreitol; Enzyme Inhibitors; Flavonoids; Glioma; Heat-Shock Proteins; Humans; Hydrogen Peroxide; Imidazoles; MAP Kinase Kinase Kinases; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Nitriles; Osmotic Pressure; Oxidants; p38 Mitogen-Activated Protein Kinases; Protein Kinase C; Protein Synthesis Inhibitors; Pyridines; Sodium Compounds; Sorbitol; Staurosporine; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured

2001
Antidepressant drug treatments induce glial cell line-derived neurotrophic factor (GDNF) synthesis and release in rat C6 glioblastoma cells.
    Journal of neurochemistry, 2001, Volume: 79, Issue:1

    Topics: Amitriptyline; Animals; Antidepressive Agents; Astrocytes; Butadienes; Cell Line; Cells, Cultured; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glial Cell Line-Derived Neurotrophic Factor; Glioblastoma; Imidazoles; Isoquinolines; Kinetics; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Naphthalenes; Nerve Growth Factors; Nerve Tissue Proteins; Nitriles; p38 Mitogen-Activated Protein Kinases; Protein Kinase C; Psychotropic Drugs; Rats; Sulfonamides

2001
Divergent regulation by p44/p42 MAP kinase and p38 MAP kinase of bone morphogenetic protein-4-stimulated osteocalcin synthesis in osteoblasts.
    Journal of cellular biochemistry, 2002, Volume: 84, Issue:3

    Topics: Bone Morphogenetic Protein 4; Bone Morphogenetic Proteins; Butadienes; Cells, Cultured; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Imidazoles; JNK Mitogen-Activated Protein Kinases; Kinetics; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nitriles; Osteoblasts; Osteocalcin; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines

2002
Involvement of MAP kinases in TGF-beta-stimulated vascular endothelial growth factor synthesis in osteoblasts.
    Archives of biochemistry and biophysics, 2003, Jul-01, Volume: 415, Issue:1

    Topics: 3T3 Cells; Angiogenesis Inducing Agents; Animals; Butadienes; Dose-Response Relationship, Drug; Drug Synergism; Endothelial Growth Factors; Flavonoids; Imidazoles; Intercellular Signaling Peptides and Proteins; Lymphokines; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nitriles; Osteoblasts; Pyridines; Transforming Growth Factor beta; Vascular Endothelial Growth Factor A; Vascular Endothelial Growth Factors

2003
Inhibition of p38 mitogen-activated protein kinase interferes with cell shape changes and gene expression associated with Schwann cell myelination.
    Experimental neurology, 2003, Volume: 183, Issue:1

    Topics: Animals; Ascorbic Acid; Butadienes; Cell Death; Cell Division; Cell Size; Cells, Cultured; Coculture Techniques; Enzyme Inhibitors; Extracellular Matrix; Ganglia, Spinal; Gene Expression; Heat-Shock Proteins; HSP27 Heat-Shock Proteins; Imidazoles; Laminin; Mitogen-Activated Protein Kinases; Myelin Sheath; Neoplasm Proteins; Nitriles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Rats; Rats, Sprague-Dawley; Schwann Cells

2003
Inhibitor of p42/44 mitogen-activated protein kinase, but not p38 MAPK, attenuated antigen challenge of guinea pig airways in vitro.
    International immunopharmacology, 2004, Volume: 4, Issue:8

    Topics: Anaphylaxis; Animals; Bronchi; Bronchoconstriction; Butadienes; Calcium-Calmodulin-Dependent Protein Kinases; Enzyme Inhibitors; Guinea Pigs; Histamine; Imidazoles; In Vitro Techniques; Leukotrienes; Male; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Muscle Contraction; Muscle, Smooth; Nitriles; Ovalbumin; p38 Mitogen-Activated Protein Kinases; Pyrimidines; Time Factors

2004
Effects of inhibitors of the tyrosine signalling cascade on antigen challenge of guinea pig airways in vitro.
    Annals of the Academy of Medicine, Singapore, 2004, Volume: 33, Issue:5 Suppl

    Topics: Animals; Asthma; Butadienes; Calcium-Calmodulin-Dependent Protein Kinases; Enzyme Inhibitors; Guinea Pigs; Imidazoles; Nitriles; Protein-Tyrosine Kinases; Pyrimidines; Signal Transduction; Stilbenes

2004
Anisomycin induces COX-2 mRNA expression through p38(MAPK) and CREB independent of small GTPases in intestinal epithelial cells.
    Biochimica et biophysica acta, 2005, Sep-30, Volume: 1745, Issue:3

    Topics: Animals; Anisomycin; Bacterial Proteins; Bacterial Toxins; Blotting, Western; Butadienes; Cyclic AMP Response Element-Binding Protein; Cyclooxygenase 2; DNA Primers; Flavonoids; Gene Expression Regulation; Imidazoles; Intestinal Mucosa; Monomeric GTP-Binding Proteins; Nitriles; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Rats; RNA Interference; RNA, Messenger; RNA, Small Interfering; Signal Transduction; Sorbitol

2005
HIV-1 gp120-induced TNF-{alpha} production by primary human macrophages is mediated by phosphatidylinositol-3 (PI-3) kinase and mitogen-activated protein (MAP) kinase pathways.
    Journal of leukocyte biology, 2005, Volume: 78, Issue:4

    Topics: Androstadienes; Butadienes; Cells, Cultured; Chromones; Flavonoids; HIV Envelope Protein gp120; Humans; Imidazoles; Macrophages; Mitogen-Activated Protein Kinases; Morpholines; Nitriles; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Receptors, CCR5; RNA, Messenger; Signal Transduction; Tumor Necrosis Factor-alpha; Wortmannin

2005
Bone morphogenetic protein-4 abrogates lumen formation by mammary epithelial cells and promotes invasive growth.
    Biochemical and biophysical research communications, 2007, Feb-16, Volume: 353, Issue:3

    Topics: Animals; Anthracenes; Bone Morphogenetic Protein 4; Bone Morphogenetic Proteins; Butadienes; Cell Transformation, Neoplastic; Cells, Cultured; Epithelial Cells; Female; Humans; Imidazoles; Mammary Glands, Animal; Mice; Mitogen-Activated Protein Kinases; Neoplasm Invasiveness; Nitriles

2007
Mixed lineage kinase 3 connects reactive oxygen species to c-Jun NH2-terminal kinase-induced mitochondrial apoptosis in genipin-treated PC3 human prostate cancer cells.
    Biochemical and biophysical research communications, 2007, Oct-19, Volume: 362, Issue:2

    Topics: Apoptosis; Blotting, Western; Butadienes; Cell Line, Tumor; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flow Cytometry; Green Fluorescent Proteins; Humans; Imidazoles; Iridoid Glycosides; Iridoids; JNK Mitogen-Activated Protein Kinases; Male; MAP Kinase Kinase Kinases; Membrane Potential, Mitochondrial; Mitochondria; Mitogen-Activated Protein Kinase Kinase Kinase 11; Nitriles; Prostatic Neoplasms; Reactive Oxygen Species; Recombinant Fusion Proteins; Signal Transduction; Transfection

2007
Inhibition of basal p38 or JNK activity enhances epithelial barrier function through differential modulation of claudin expression.
    American journal of physiology. Cell physiology, 2009, Volume: 297, Issue:3

    Topics: Animals; Anthracenes; Butadienes; Cell Line; Dogs; Epithelium; Female; Imidazoles; Mammary Glands, Animal; MAP Kinase Kinase 4; Membrane Proteins; Mice; Nitriles; p38 Mitogen-Activated Protein Kinases

2009
ERK and p38 inhibitors attenuate memory deficits and increase CREB phosphorylation and PGC-1α levels in Aβ-injected rats.
    Behavioural brain research, 2012, Jun-15, Volume: 232, Issue:1

    Topics: Amyloid beta-Peptides; Animals; Blotting, Western; Butadienes; CA1 Region, Hippocampal; Cyclic AMP Response Element-Binding Protein; Enzyme Inhibitors; Imidazoles; Male; MAP Kinase Signaling System; Maze Learning; Memory Disorders; Microinjections; Mitochondria; NF-E2-Related Factor 1; Nitriles; p38 Mitogen-Activated Protein Kinases; Peroxisome Proliferator-Activated Receptor Gamma Coactivator 1-alpha; Phosphorylation; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; RNA-Binding Proteins; Stereotaxic Techniques; Transcription Factors

2012
Reduction of hippocampal apoptosis by intracerebroventricular administration of extracellular signal-regulated protein kinase and/or p38 inhibitors in amyloid beta rat model of Alzheimer's disease: involvement of nuclear-related factor-2 and nuclear facto
    Basic & clinical pharmacology & toxicology, 2013, Volume: 112, Issue:3

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Apoptosis; Blotting, Western; Butadienes; Disease Models, Animal; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Hippocampus; Imidazoles; In Situ Nick-End Labeling; Injections, Intraventricular; Male; MAP Kinase Signaling System; NF-E2-Related Factor 2; NF-kappa B; Nitriles; p38 Mitogen-Activated Protein Kinases; Rats; Rats, Wistar

2013
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