Page last updated: 2024-09-04

pd 151242 and bq 3020

pd 151242 has been researched along with bq 3020 in 10 studies

Compound Research Comparison

Studies
(pd 151242)
Trials
(pd 151242)
Recent Studies (post-2010)
(pd 151242)
Studies
(bq 3020)
Trials
(bq 3020)
Recent Studies (post-2010) (bq 3020)
21008702

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (80.00)18.2507
2000's2 (20.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Davenport, AP; Peter, MG1
Bacon, CR; Cameron, IT; Davenport, AP; Morrison, JJ; O'Reilly, G1
Berryman, K; Davenport, AP; Doherty, AM; Fitzgerald, F; Kuc, RE; Maguire, JJ1
Davenport, AP; Pickard, JD; Yu, JC1
Davenport, AP; Harland, SP; Kuc, RE; Pickard, JD1
Davenport, AP; Pierre, LN1
Dashwood, MR; Khan, MA; Mikhailidis, DP; Morgan, RJ; Mumtaz, FH; Thompson, CS1
Drimal, J; Kovacik, V; Patoprsty, V1
Champion, HC; Malendowicz, LK; Mazzocchi, G; Nussdorfer, GG; Rossi, GP1
Davenport, AP; Kuc, R1

Other Studies

10 other study(ies) available for pd 151242 and bq 3020

ArticleYear
Selectivity of [125I]-PD151242 for human, rat and porcine endothelin ETA receptors in the heart.
    British journal of pharmacology, 1995, Volume: 114, Issue:2

    Topics: Adult; Animals; Azepines; Binding, Competitive; Endothelin Receptor Antagonists; Endothelins; Heart; Heart Ventricles; Humans; In Vitro Techniques; Indoles; Iodine Radioisotopes; Ligands; Male; Middle Aged; Myocardium; Oligopeptides; Peptide Fragments; Rats; Rats, Sprague-Dawley; Species Specificity; Swine

1995
ETA and ETB endothelin receptors in human myometrium characterized by the subtype selective ligands BQ123, BQ3020, FR139317 and PD151242.
    The Journal of endocrinology, 1995, Volume: 144, Issue:1

    Topics: Azepines; Base Sequence; DNA Primers; Endothelin Receptor Antagonists; Endothelins; Female; Humans; Indoles; Ligands; Molecular Sequence Data; Myometrium; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Polymerase Chain Reaction; Receptors, Endothelin

1995
[125I]-PD151242: a selective radioligand for human ETA receptors.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: Adult; Amino Acid Sequence; Aorta; Arteries; Azepines; Binding, Competitive; Coronary Vessels; Endothelin Receptor Antagonists; Endothelins; Humans; In Vitro Techniques; Indoles; Iodine Radioisotopes; Middle Aged; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Pulmonary Artery; Radioligand Assay; Receptors, Endothelin

1994
Endothelin ETA receptor expression in human cerebrovascular smooth muscle cells.
    British journal of pharmacology, 1995, Volume: 116, Issue:5

    Topics: Aged; Autoradiography; Azepines; Base Sequence; Binding, Competitive; Cells, Cultured; Cerebrovascular Circulation; Endothelin Receptor Antagonists; Endothelin-1; Endothelins; Female; Humans; Kinetics; Male; Middle Aged; Molecular Sequence Data; Muscle, Smooth, Vascular; Oligopeptides; Peptide Fragments; Polymerase Chain Reaction; Protein Precursors; Radioimmunoassay; Receptors, Endothelin; RNA, Messenger

1995
Characterization of endothelin receptors in human brain cortex, gliomas, and meningiomas.
    Journal of cardiovascular pharmacology, 1995, Volume: 26 Suppl 3

    Topics: Autoradiography; Azepines; Cerebral Cortex; Endothelins; Glioma; Humans; Meningeal Neoplasms; Meningioma; Oligopeptides; Peptide Fragments; Receptors, Endothelin

1995
Endothelin receptor subtypes and their functional relevance in human small coronary arteries.
    British journal of pharmacology, 1998, Volume: 124, Issue:3

    Topics: Autoradiography; Azepines; Coronary Vessels; Dioxoles; Endothelin Receptor Antagonists; Endothelins; Female; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth, Vascular; Oligopeptides; Peptide Fragments; Receptors, Endothelin

1998
Upregulation of endothelin A receptor sites in the rabbit diabetic kidney: potential relevance to the early pathogenesis of diabetic nephropathy.
    Nephron, 1999, Volume: 83, Issue:3

    Topics: Alloxan; Animals; Autoradiography; Azepines; Blood Glucose; Blood Urea Nitrogen; Body Weight; Diabetes Mellitus, Experimental; Diabetic Nephropathies; Disease Models, Animal; Endothelin-1; Endothelins; Immunoenzyme Techniques; Iodine Radioisotopes; Kidney; Male; Oligopeptides; Peptide Fragments; Potassium; Rabbits; Radioligand Assay; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin; Sodium; Up-Regulation

1999
Stobadine is a potent modulator of endogenous endothelin-1 in human fibroblasts.
    Life sciences, 1999, Volume: 65, Issue:18-19

    Topics: Antioxidants; Azepines; Carbolines; Cells, Cultured; Chloroquine; Endothelin Receptor Antagonists; Endothelin-1; Endothelins; Enzyme Inhibitors; Fibroblasts; Humans; Iodine Radioisotopes; Lysosomes; Mitogens; Oligopeptides; Peptide Fragments; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin

1999
Endothelin-1[1-31], acting as an ETA-receptor selective agonist, stimulates proliferation of cultured rat zona glomerulosa cells.
    FEBS letters, 2000, Dec-29, Volume: 487, Issue:2

    Topics: Animals; Azepines; Cell Division; Cells, Cultured; Endothelin Receptor Antagonists; Endothelin-1; Endothelins; Iodine Radioisotopes; Kinetics; Male; Mitogen-Activated Protein Kinases; Oligopeptides; Peptide Fragments; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Receptors, Endothelin; Thymidine Kinase; Zona Glomerulosa

2000
Comparison of endothelin-A and endothelin-B receptor distribution visualized by radioligand binding versus immunocytochemical localization using subtype selective antisera.
    Journal of cardiovascular pharmacology, 2004, Volume: 44 Suppl 1

    Topics: Autoradiography; Azepines; Endothelins; Humans; Immune Sera; Immunohistochemistry; Iodine Radioisotopes; Kidney Cortex; Kidney Medulla; Ligands; Oligopeptides; Peptide Fragments; Radioligand Assay; Radiopharmaceuticals; Receptor, Endothelin A; Receptor, Endothelin B

2004