Compounds > pd 151242
Page last updated: 2024-09-04

pd 151242 and bq 123

pd 151242 has been researched along with bq 123 in 4 studies

Compound Research Comparison

Studies
(pd 151242)		Trials
(pd 151242)		Recent Studies (post-2010)
(pd 151242)		Studies
(bq 123)		Trials
(bq 123)		Recent Studies (post-2010) (bq 123)
21001,39163152

Protein Interaction Comparison

ProteinTaxonomypd 151242 (IC50)bq 123 (IC50)
Endothelin-1 receptorHomo sapiens (human)0.017
Endothelin-1 receptorRattus norvegicus (Norway rat)0.014

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (75.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Godfraind, T1
Bacon, CR; Cameron, IT; Davenport, AP; Morrison, JJ; O'Reilly, G1
Berryman, K; Davenport, AP; Doherty, AM; Fitzgerald, F; Kuc, RE; Maguire, JJ1
Harada, N; Himeno, A; Niwa, M; Shigematsu, K; Sumikawa, K1

Other Studies

4 other study(ies) available for pd 151242 and bq 123

ArticleYear
Endothelin receptors in human coronary arteries.
    Trends in pharmacological sciences, 1994, Volume: 15, Issue:5

    Topics: Animals; Azepines; Coronary Vessels; Endothelin Receptor Antagonists; Endothelins; Humans; In Vitro Techniques; Indoles; Oligopeptides; Peptides, Cyclic; Receptors, Endothelin; Xenopus laevis

1994
ETA and ETB endothelin receptors in human myometrium characterized by the subtype selective ligands BQ123, BQ3020, FR139317 and PD151242.
    The Journal of endocrinology, 1995, Volume: 144, Issue:1

    Topics: Azepines; Base Sequence; DNA Primers; Endothelin Receptor Antagonists; Endothelins; Female; Humans; Indoles; Ligands; Molecular Sequence Data; Myometrium; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Polymerase Chain Reaction; Receptors, Endothelin

1995
[125I]-PD151242: a selective radioligand for human ETA receptors.
    British journal of pharmacology, 1994, Volume: 111, Issue:1

    Topics: Adult; Amino Acid Sequence; Aorta; Arteries; Azepines; Binding, Competitive; Coronary Vessels; Endothelin Receptor Antagonists; Endothelins; Humans; In Vitro Techniques; Indoles; Iodine Radioisotopes; Middle Aged; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Pulmonary Artery; Radioligand Assay; Receptors, Endothelin

1994
Endothelin-1 binding to endothelin receptors in the rat anterior pituitary gland: possible formation of an ETA-ETB receptor heterodimer.
    Cellular and molecular neurobiology, 2002, Volume: 22, Issue:2

    Topics: Animals; Azepines; Binding Sites; Cell Membrane; Dimerization; Endothelin-1; Endothelins; Epithelial Cells; Iodine Radioisotopes; Kinetics; Ligands; Male; Oligopeptides; Peptide Fragments; Peptides, Cyclic; Pituitary Gland, Anterior; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Receptor, Endothelin A; Receptor, Endothelin B; Receptors, Endothelin; RNA, Messenger; Viper Venoms

2002