Page last updated: 2024-09-05

pd 140376 and sincalide

pd 140376 has been researched along with sincalide in 3 studies

Compound Research Comparison

Studies
(pd 140376)
Trials
(pd 140376)
Recent Studies (post-2010)
(pd 140376)
Studies
(sincalide)
Trials
(sincalide)
Recent Studies (post-2010) (sincalide)
5004,01572533

Protein Interaction Comparison

ProteinTaxonomypd 140376 (IC50)sincalide (IC50)
Cholecystokinin receptor type ARattus norvegicus (Norway rat)0.0006
Cholecystokinin receptor type AHomo sapiens (human)0.0006
Gastrin/cholecystokinin type B receptorHomo sapiens (human)0.001
Gastrin/cholecystokinin type B receptorMus musculus (house mouse)0.0008
Cholecystokinin receptor type ACavia porcellus (domestic guinea pig)0.0004

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dissanayake, VU; Hill, DR; Horwell, DC; Hughes, J; Hunter, JC; Kneen, CO; Meecham, KG; Pritchard, MC; Suman-Chauhan, N; Woodruff, GN1
Black, JW; Griffin, EP; Harper, EA; Shankley, NP1
Black, JW; Harper, EA; Shankley, NP1

Other Studies

3 other study(ies) available for pd 140376 and sincalide

ArticleYear
[3H]PD 140376: a novel and highly selective antagonist radioligand for the cholecystokininB/gastrin receptor in guinea pig cerebral cortex and gastric mucosa.
    Molecular pharmacology, 1993, Volume: 43, Issue:4

    Topics: Animals; Binding, Competitive; Bridged-Ring Compounds; Cerebral Cortex; Dipeptides; Gastric Mucosa; Gastrins; Guinea Pigs; In Vitro Techniques; Iodine Radioisotopes; Kinetics; Male; Peptoids; Radioligand Assay; Receptors, Cholecystokinin; Sincalide; Succinimides; Tritium

1993
Analysis of the behaviour of selected CCKB/gastrin receptor antagonists in radioligand binding assays performed in mouse and rat cerebral cortex.
    British journal of pharmacology, 1999, Volume: 126, Issue:6

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Bridged-Ring Compounds; Cerebral Cortex; Dipeptides; Guinea Pigs; Hormone Antagonists; Indoleacetic Acids; Indoles; Iodine Radioisotopes; Male; Meglumine; Mice; Pancreas; Phenylurea Compounds; Radioligand Assay; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Sincalide; Succinimides; Thiazoles; Tritium

1999
Characterization of the binding of a novel radioligand to CCKB/gastrin receptors in membranes from rat cerebral cortex.
    British journal of pharmacology, 1999, Volume: 126, Issue:6

    Topics: Animals; Benzodiazepines; Benzodiazepinones; Binding Sites; Binding, Competitive; Bridged-Ring Compounds; Cerebral Cortex; Dipeptides; Dose-Response Relationship, Drug; Hormone Antagonists; Indoles; Kinetics; Male; Meglumine; Membranes; Nootropic Agents; Pentagastrin; Phenylurea Compounds; Radioligand Assay; Rats; Rats, Wistar; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Sincalide; Tritium

1999