Page last updated: 2024-09-03

pd 135158 and l 365260

pd 135158 has been researched along with l 365260 in 7 studies

Compound Research Comparison

Studies
(pd 135158)
Trials
(pd 135158)
Recent Studies (post-2010)
(pd 135158)
Studies
(l 365260)
Trials
(l 365260)
Recent Studies (post-2010) (l 365260)
5100422108

Protein Interaction Comparison

ProteinTaxonomypd 135158 (IC50)l 365260 (IC50)
5-hydroxytryptamine receptor 2CRattus norvegicus (Norway rat)0.0081
5-hydroxytryptamine receptor 2ARattus norvegicus (Norway rat)0.0081
Cholecystokinin receptor type ARattus norvegicus (Norway rat)0.4981
Gastrin/cholecystokinin type B receptorRattus norvegicus (Norway rat)0.039
5-hydroxytryptamine receptor 2BRattus norvegicus (Norway rat)0.0081
Histamine H1 receptorCavia porcellus (domestic guinea pig)5
Cholecystokinin receptor type AHomo sapiens (human)0.1585
Gastrin/cholecystokinin type B receptorHomo sapiens (human)0.0079
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)5
Cholecystokinin receptor type ACavia porcellus (domestic guinea pig)0.044
Cysteinyl leukotriene receptor 2Homo sapiens (human)5
Cysteinyl leukotriene receptor 1Homo sapiens (human)5

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's7 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, D; Ding, XQ; Håkanson, R1
Dickenson, AH; Hewett, K; Sullivan, AF1
Fuxe, K; Hernandez-Gómez, AM; Méndez-Franco, J; Pérez de la Mora, M1
Blackmore, M; Doherty, E; Hirst, BH; Manning, JE1
Colombo, S; Letari, O; Makovec, F; Mennuni, L; Revel, L1
Bradwejn, J; Frankland, PW; Josselyn, SA; Vaccarino, FJ; Yeomans, JS1
Dorré, D; Smith, GP1

Other Studies

7 other study(ies) available for pd 135158 and l 365260

ArticleYear
Cholecystokinin-B receptor ligands of the dipeptoid series act as agonists on rat stomach histidine decarboxylase.
    Gastroenterology, 1995, Volume: 109, Issue:4

    Topics: Animals; Benzodiazepinones; Devazepide; Enzyme Activation; Gastrins; Histidine Decarboxylase; Indoles; Ligands; Male; Meglumine; Phenethylamines; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Sincalide; Stomach

1995
Differential modulation of alpha 2-adrenergic and opioid spinal antinociception by cholecystokinin and cholecystokinin antagonists in the rat dorsal horn: an electrophysiological study.
    Brain research, 1994, Oct-31, Volume: 662, Issue:1-2

    Topics: Analgesics; Analgesics, Non-Narcotic; Animals; Anti-Anxiety Agents; Benzodiazepinones; Cholecystokinin; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Imidazoles; Indoles; Injections, Spinal; Male; Medetomidine; Meglumine; Morphine; Nerve Fibers; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Cholecystokinin; Receptors, Opioid; Spinal Cord

1994
Cholecystokinin-8 increases K(+)-evoked [3H] gamma-aminobutyric acid release in slices from various brain areas.
    European journal of pharmacology, 1993, Dec-21, Volume: 250, Issue:3

    Topics: Animals; Benzodiazepinones; beta-Alanine; Brain; Calcium; Devazepide; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Indoles; Male; Meglumine; Phenylurea Compounds; Potassium; Rats; Rats, Wistar; Receptors, Cholecystokinin; Sincalide

1993
Autocrine growth stimulation of human renal Wilms' tumour G401 cells by a gastrin-like peptide.
    International journal of cancer, 1994, May-01, Volume: 57, Issue:3

    Topics: Benzamides; Benzodiazepinones; Cell Division; Devazepide; Gastrins; Humans; Indoles; Kidney Neoplasms; Meglumine; Phenylurea Compounds; Proglumide; Receptors, Cholecystokinin; Tumor Cells, Cultured; Wilms Tumor

1994
Cytosolic Ca2+ evaluation in rabbit parietal cells: a novel method to screen gastrin receptor antagonists.
    European journal of pharmacology, 1996, Jun-13, Volume: 306, Issue:1-3

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Benzodiazepinones; Calcium; Devazepide; Dose-Response Relationship, Drug; Fura-2; Gastrins; Hormone Antagonists; Humans; Indoles; Male; Meglumine; Parietal Cells, Gastric; Phenylurea Compounds; Rabbits; Receptors, Cholecystokinin; Sincalide

1996
Activation of amygdala cholecystokininB receptors potentiates the acoustic startle response in the rat.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Mar-01, Volume: 17, Issue:5

    Topics: Acoustic Stimulation; Amygdala; Animals; Anti-Anxiety Agents; Anxiety; Benzodiazepinones; Corpus Striatum; Fear; Indoles; Injections, Intraperitoneal; Injections, Intraventricular; Meglumine; Nucleus Accumbens; Pentagastrin; Phenylurea Compounds; Rats; Rats, Wistar; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Reflex, Startle

1997
CholecystokininB receptor antagonist increases food intake in rats.
    Physiology & behavior, 1998, Volume: 65, Issue:1

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepinones; Brain Chemistry; Dose-Response Relationship, Drug; Eating; Indoles; Injections, Intraventricular; Male; Meglumine; Phenylurea Compounds; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin B; Receptors, Cholecystokinin; Stereoisomerism

1998