Page last updated: 2024-09-03

pd 128907 and apomorphine

pd 128907 has been researched along with apomorphine in 3 studies

Compound Research Comparison

Studies
(pd 128907)
Trials
(pd 128907)
Recent Studies (post-2010)
(pd 128907)
Studies
(apomorphine)
Trials
(apomorphine)
Recent Studies (post-2010) (apomorphine)
9049,205287780
16099,205287780

Protein Interaction Comparison

ProteinTaxonomypd 128907 (IC50)apomorphine (IC50)
Tryptophan 5-hydroxylase 1Rattus norvegicus (Norway rat)0.22
D(2) dopamine receptorHomo sapiens (human)0.0146
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.75
DRattus norvegicus (Norway rat)0.4744
D(3) dopamine receptorRattus norvegicus (Norway rat)0.1432
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.063
D(2) dopamine receptorBos taurus (cattle)0.3385
D(1A) dopamine receptorHomo sapiens (human)0.025
D(4) dopamine receptorHomo sapiens (human)0.025
D(1B) dopamine receptorHomo sapiens (human)0.025
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)7.75
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(4) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(3) dopamine receptorHomo sapiens (human)0.025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.75
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0813
E3 ubiquitin-protein ligase Mdm2Homo sapiens (human)0.205
5-hydroxytryptamine receptor 4 Rattus norvegicus (Norway rat)1.35
DBos taurus (cattle)0.3385

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19901 (33.33)18.7374
1990's2 (66.67)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
DeWald, HA; Heffner, TG; Jaen, JC; Lustgarten, DM; McPhail, AT; Meltzer, LT; Pugsley, TA; Wise, LD1
Griffon, N; Lévesque, D; Pilon, C; Sautel, F; Schwartz, JC; Sokoloff, P1
Dijkstra, D; Horn, AS; Mulder, TB; Rollema, H; Tepper, PG; Van der Weide, J1

Other Studies

3 other study(ies) available for pd 128907 and apomorphine

ArticleYear
Synthesis and dopamine agonist properties of (+-)-trans-3,4,4a,10b-tetrahydro-4-propyl-2H,5H-[1]benzopyrano [4,3-b]-1,4-oxazin-9-ol and its enantiomers.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:1

    Topics: Animals; Benzopyrans; Cell Membrane; Chemical Phenomena; Chemistry; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agents; Electrophysiology; Haloperidol; Male; Mice; Molecular Structure; Motor Activity; Neurons; Oxazines; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Stereoisomerism; Substantia Nigra

1990
A functional test identifies dopamine agonists selective for D3 versus D2 receptors.
    Neuroreport, 1995, Jan-26, Volume: 6, Issue:2

    Topics: Animals; CHO Cells; Cricetinae; Dopamine Agents; Humans; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D3

1995
Synthesis and pharmacology of trans-4-n-propyl-3,4,4a,10b-tetrahydro-2H,5H-1-benzopyrano[4,3-b ]-1,4-oxazin-7- and -9-ols: the significance of nitrogen pKa values for central dopamine receptor activation.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:11

    Topics: Animals; Benzopyrans; Binding Sites; Brain Chemistry; Cattle; Dopamine; Dopamine Agents; Nitrogen; Oxazines; Protons; Rats; Receptors, Dopamine

1988