Page last updated: 2024-09-03

pd 128483 and apomorphine

pd 128483 has been researched along with apomorphine in 2 studies

Compound Research Comparison

Studies
(pd 128483)
Trials
(pd 128483)
Recent Studies (post-2010)
(pd 128483)
Studies
(apomorphine)
Trials
(apomorphine)
Recent Studies (post-2010) (apomorphine)
5009,205287780

Protein Interaction Comparison

ProteinTaxonomypd 128483 (IC50)apomorphine (IC50)
Tryptophan 5-hydroxylase 1Rattus norvegicus (Norway rat)0.22
D(2) dopamine receptorHomo sapiens (human)0.0146
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.75
DRattus norvegicus (Norway rat)0.4744
D(3) dopamine receptorRattus norvegicus (Norway rat)0.1432
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.063
D(2) dopamine receptorBos taurus (cattle)0.3385
D(1A) dopamine receptorHomo sapiens (human)0.025
D(4) dopamine receptorHomo sapiens (human)0.025
D(1B) dopamine receptorHomo sapiens (human)0.025
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.063
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)7.75
D(1B) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(4) dopamine receptorRattus norvegicus (Norway rat)0.1432
D(3) dopamine receptorHomo sapiens (human)0.025
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.75
D(2) dopamine receptorRattus norvegicus (Norway rat)0.0813
E3 ubiquitin-protein ligase Mdm2Homo sapiens (human)0.205
5-hydroxytryptamine receptor 4 Rattus norvegicus (Norway rat)1.35
DBos taurus (cattle)0.3385

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lin, MY; Walters, DE1
Caprathe, BW; Christoffersen, CL; Corbin, AE; Jaen, JC; Meltzer, LT; Ninteman, FW; Pugsley, TA; Serpa, KA; Shih, YH; Whetzel, SZ1

Other Studies

2 other study(ies) available for pd 128483 and apomorphine

ArticleYear
Dopamine D2 autoreceptors in rats are behaviorally functional at 21 but not 10 days of age.
    Psychopharmacology, 1994, Volume: 114, Issue:2

    Topics: Aging; Aminoquinolines; Animals; Apomorphine; Azepines; Behavior, Animal; Benzothiazoles; Dopamine Agonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Male; Motor Activity; Piperidines; Pramipexole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Thiazoles

1994
Pharmacological profile of the dopamine partial agonist, (+/-)-PD 128483 and its enantiomers.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: 4-Butyrolactone; Aminoquinolines; Amphetamine; Animals; Apomorphine; Avoidance Learning; Behavior, Animal; Cebus; Dopamine; Dopamine Agents; Dose-Response Relationship, Drug; Extrapyramidal Tracts; Male; Mice; Motor Activity; Neurons; Norepinephrine; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Saimiri; Serotonin; Stereoisomerism; Stereotyped Behavior; Stimulation, Chemical; Thiazoles

1993