Page last updated: 2024-09-03

pd 124816 and gatifloxacin

pd 124816 has been researched along with gatifloxacin in 2 studies

Compound Research Comparison

Studies
(pd 124816)
Trials
(pd 124816)
Recent Studies (post-2010)
(pd 124816)
Studies
(gatifloxacin)
Trials
(gatifloxacin)
Recent Studies (post-2010) (gatifloxacin)
10001,047131268

Protein Interaction Comparison

ProteinTaxonomypd 124816 (IC50)gatifloxacin (IC50)
DNA gyrase subunit AEscherichia coli K-120.5
DNA gyrase subunit BEscherichia coli K-120.5
DNA topoisomerase 4 subunit AStaphylococcus aureus1.2
DNA gyrase subunit AMycobacterium tuberculosis H37Rv9.4

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cohen, MA; Domagala, JM; Gogliotti, RD; Gracheck, SJ; Huband, MD; Sanchez, JP; Sesnie, JA; Shapiro, MA1
García-March, FJ; Jaén-Oltra, J; Pérez-Giménez, F; Salabert-Salvador, MT; Tomás-Vert, F1

Other Studies

2 other study(ies) available for pd 124816 and gatifloxacin

ArticleYear
The synthesis, structure-activity, and structure-side effect relationships of a series of 8-alkoxy- and 5-amino-8-alkoxyquinolone antibacterial agents.
    Journal of medicinal chemistry, 1995, Oct-27, Volume: 38, Issue:22

    Topics: Animals; Anti-Bacterial Agents; Bacteria; CHO Cells; Cricetinae; Dermatitis, Phototoxic; Drug Design; Female; Mice; Mice, Inbred Strains; Microbial Sensitivity Tests; Quinolones; Structure-Activity Relationship

1995
Artificial neural network applied to prediction of fluorquinolone antibacterial activity by topological methods.
    Journal of medicinal chemistry, 2000, Mar-23, Volume: 43, Issue:6

    Topics: Algorithms; Anti-Infective Agents; Fluoroquinolones; Microbial Sensitivity Tests; Neural Networks, Computer; Structure-Activity Relationship

2000