Page last updated: 2024-09-02

pd 123177 and saralasin

pd 123177 has been researched along with saralasin in 14 studies

Compound Research Comparison

Studies
(pd 123177)
Trials
(pd 123177)
Recent Studies (post-2010)
(pd 123177)
Studies
(saralasin)
Trials
(saralasin)
Recent Studies (post-2010) (saralasin)
142021,4971316

Protein Interaction Comparison

ProteinTaxonomypd 123177 (IC50)saralasin (IC50)
Type-1A angiotensin II receptor Rattus norvegicus (Norway rat)0.0017
Type-1B angiotensin II receptorRattus norvegicus (Norway rat)0.0017
Type-1 angiotensin II receptorHomo sapiens (human)0.0006
Type-2 angiotensin II receptorHomo sapiens (human)0.0008

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's14 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Absher, DR; Baisden, RH; Joyner, WL; Perez, RA; Rowe, BP; Saylor, DL; Woodruff, ML1
Christ, DD; Duncia, JV; Pierce, SK; Reilly, TM; Timmermans, PB1
Hart, SD; Timmermans, PB; Wong, PC1
Kunihara, M; Kushida, H; Morita, O1
Bornkessel, B1
Bihoreau, C; Clauser, E; Conchon, S; Corvol, P; Monnot, C; Sirieix, ME1
Heemskerk, FM; Michels, KM; Saavedra, JM1
Brown, JA; Cobb, CS1
Bensoussan, M; Mitchell, T; Reilly, T; Ronco, PM; Timmermans, PB; Verroust, PJ1
Barnes, JC; Clark, SA; Marshall, FH; Michel, AD1
Dagenais, P; Escher, E1
Barber, PC; Barnes, JM; Barnes, NM; Steward, LJ1
Baubonis, W; Benfield, P; Chiu, AT; Dunscomb, JH; McCall, DE; Sauer, B1
Barbera, F; Diamond, S; Gibson, RE; Herblin, WF; Timmermans, P1

Reviews

1 review(s) available for pd 123177 and saralasin

ArticleYear
[Angiotensin II receptor antagonists].
    Medizinische Monatsschrift fur Pharmazeuten, 1995, Volume: 18, Issue:6

    Topics: Amino Acid Sequence; Angiotensin II; Angiotensin Receptor Antagonists; Antihypertensive Agents; Biphenyl Compounds; Hemodynamics; Humans; Hypertension; Imidazoles; Losartan; Molecular Sequence Data; Pyridines; Receptors, Angiotensin; Renin-Angiotensin System; Saralasin; Tetrazoles

1995

Other Studies

13 other study(ies) available for pd 123177 and saralasin

ArticleYear
Angiotensin II binding sites in the hamster brain: localization and subtype distribution.
    Brain research, 1992, Nov-06, Volume: 595, Issue:1

    Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Brain; Cricetinae; Imidazoles; In Vitro Techniques; Mesencephalon; Mesocricetus; Prosencephalon; Pyridines; Receptors, Angiotensin; Rhombencephalon; Saralasin

1992
Monoclonal antibodies to the nonpeptide angiotensin II receptor antagonist, losartan.
    European journal of pharmacology, 1992, Jun-05, Volume: 226, Issue:2

    Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antibodies, Monoclonal; Antibody Specificity; Biphenyl Compounds; Cross Reactions; Enzyme-Linked Immunosorbent Assay; Imidazoles; Losartan; Mice; Mice, Inbred BALB C; Pyridines; Saralasin; Structure-Activity Relationship; Tetrazoles

1992
Effect of angiotensin II antagonism on canine renal sympathetic nerve function.
    Hypertension (Dallas, Tex. : 1979), 1991, Volume: 17, Issue:6 Pt 2

    Topics: Angiotensin II; Animals; Blood Pressure; Captopril; Dogs; Electric Stimulation; Female; Imidazoles; Kidney; Losartan; Male; Norepinephrine; Pyridines; Saralasin; Sympathetic Nervous System; Tetrazoles; Vascular Resistance; Vasoconstriction

1991
Effects of U-97018 on pressor responses to intracerebroventricularly administered angiotensin II in conscious normotensive rats.
    Journal of cardiovascular pharmacology, 1995, Volume: 25, Issue:6

    Topics: Administration, Oral; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Biphenyl Compounds; Blood Pressure; Disease Models, Animal; Dose-Response Relationship, Drug; Hypertension; Imidazoles; Injections, Intravenous; Injections, Intraventricular; Losartan; Male; Pyridazines; Pyridines; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Saralasin; Tetrazoles

1995
Synthetic cDNA encoding the rat AT1a receptor: a useful tool for structure-function relationship analysis.
    Biochemical and biophysical research communications, 1994, Mar-30, Volume: 199, Issue:3

    Topics: Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Base Sequence; Biphenyl Compounds; CHO Cells; Codon; Cricetinae; DNA, Complementary; Imidazoles; Kinetics; Losartan; Molecular Sequence Data; Mutagenesis, Site-Directed; Oligodeoxyribonucleotides; Oligopeptides; Open Reading Frames; Pyridines; Rats; Receptors, Angiotensin; Restriction Mapping; Saralasin; Signal Transduction; Structure-Activity Relationship; Tetrazoles; Transfection

1994
Selective changes in angiotensin II AT1 and AT2 receptor subtypes in the rat superior colliculus following eye enucleation.
    Neuroscience, 1994, Volume: 58, Issue:4

    Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Biphenyl Compounds; Eye Enucleation; Geniculate Bodies; Imidazoles; Iodine Radioisotopes; Losartan; Male; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Retina; Saralasin; Subcellular Fractions; Superior Colliculi; Suprachiasmatic Nucleus; Synapses; Tetrazoles; Visual Pathways

1994
Characterization of putative glomerular receptors for angiotensin II in the rainbow trout Oncorhynchus mykiss using the antagonists Losartan, PD 123177, and saralasin.
    General and comparative endocrinology, 1993, Volume: 92, Issue:1

    Topics: Analysis of Variance; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Imidazoles; Iodine Radioisotopes; Kidney Glomerulus; Kinetics; Losartan; Oncorhynchus mykiss; Pyridines; Receptors, Angiotensin; Saralasin; Tetrazoles

1993
Immunological reactivity of angiotensin II receptor antagonists: possible implications for receptor binding sites.
    European journal of pharmacology, 1993, Oct-15, Volume: 247, Issue:2

    Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antibodies, Monoclonal; Antihypertensive Agents; Biphenyl Compounds; Imidazoles; In Vitro Techniques; Indicators and Reagents; Iodine Radioisotopes; Losartan; Molecular Conformation; Oligopeptides; Pyridines; Rats; Receptors, Angiotensin; Saralasin; Tetrazoles

1993
Binding of angiotensin antagonists to rat liver and brain membranes measured ex vivo.
    British journal of pharmacology, 1993, Volume: 109, Issue:3

    Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Binding, Competitive; Biphenyl Compounds; Blood-Brain Barrier; Brain; Imidazoles; In Vitro Techniques; Iodine Radioisotopes; Liver; Losartan; Male; Membranes; Nicotinic Acids; Pyridines; Rats; Receptors, Angiotensin; Saralasin; Tetrazoles

1993
Anti-angiotensin antibodies cross-reactive with nonpeptide angiotensin antagonists as angiotensin receptor model.
    Regulatory peptides, 1993, Mar-19, Volume: 44, Issue:2

    Topics: Adrenocorticotropic Hormone; Amino Acid Sequence; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antibodies; Biphenyl Compounds; Cross Reactions; Enzyme-Linked Immunosorbent Assay; Imidazoles; Losartan; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Naloxone; Pyridines; Saralasin; Structure-Activity Relationship; Tetrazoles

1993
Identification and characterisation of angiotensin II receptor subtypes in human brain.
    European journal of pharmacology, 1993, Jan-19, Volume: 230, Issue:3

    Topics: Aged; Angiotensin II; Angiotensin Receptor Antagonists; Autoradiography; Binding, Competitive; Biphenyl Compounds; Brain Chemistry; Female; Humans; Imidazoles; In Vitro Techniques; Iodine Radioisotopes; Losartan; Male; Middle Aged; Pyridines; Radioligand Assay; Receptors, Angiotensin; Saralasin; Tetrazoles

1993
Characterization of angiotensin AT1A receptor isoform by its ligand binding signature.
    Regulatory peptides, 1993, Mar-19, Volume: 44, Issue:2

    Topics: Adrenal Cortex; Angiotensin I; Angiotensin III; Animals; Base Sequence; Binding, Competitive; Biphenyl Compounds; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Imidazoles; Losartan; Molecular Sequence Data; Muscle, Smooth, Vascular; Nicotinic Acids; Pyridines; Rats; Receptors, Angiotensin; Recombinant Proteins; Saralasin; Tetrazoles; Transfection

1993
A novel angiotensin II binding site in murine tissues.
    Life sciences, 1998, Volume: 63, Issue:3

    Topics: Amino Acid Sequence; Angiotensin II; Animals; Autoradiography; Binding Sites; Humans; Imidazoles; Losartan; Mice; Mice, Inbred C57BL; Mice, Nude; Pyridines; Saralasin; Tumor Cells, Cultured

1998