pd 123177 has been researched along with saralasin in 14 studies
Studies (pd 123177) | Trials (pd 123177) | Recent Studies (post-2010) (pd 123177) | Studies (saralasin) | Trials (saralasin) | Recent Studies (post-2010) (saralasin) |
---|---|---|---|---|---|
142 | 0 | 2 | 1,497 | 13 | 16 |
Protein | Taxonomy | pd 123177 (IC50) | saralasin (IC50) |
---|---|---|---|
Type-1A angiotensin II receptor | Rattus norvegicus (Norway rat) | 0.0017 | |
Type-1B angiotensin II receptor | Rattus norvegicus (Norway rat) | 0.0017 | |
Type-1 angiotensin II receptor | Homo sapiens (human) | 0.0006 | |
Type-2 angiotensin II receptor | Homo sapiens (human) | 0.0008 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 14 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Absher, DR; Baisden, RH; Joyner, WL; Perez, RA; Rowe, BP; Saylor, DL; Woodruff, ML | 1 |
Christ, DD; Duncia, JV; Pierce, SK; Reilly, TM; Timmermans, PB | 1 |
Hart, SD; Timmermans, PB; Wong, PC | 1 |
Kunihara, M; Kushida, H; Morita, O | 1 |
Bornkessel, B | 1 |
Bihoreau, C; Clauser, E; Conchon, S; Corvol, P; Monnot, C; Sirieix, ME | 1 |
Heemskerk, FM; Michels, KM; Saavedra, JM | 1 |
Brown, JA; Cobb, CS | 1 |
Bensoussan, M; Mitchell, T; Reilly, T; Ronco, PM; Timmermans, PB; Verroust, PJ | 1 |
Barnes, JC; Clark, SA; Marshall, FH; Michel, AD | 1 |
Dagenais, P; Escher, E | 1 |
Barber, PC; Barnes, JM; Barnes, NM; Steward, LJ | 1 |
Baubonis, W; Benfield, P; Chiu, AT; Dunscomb, JH; McCall, DE; Sauer, B | 1 |
Barbera, F; Diamond, S; Gibson, RE; Herblin, WF; Timmermans, P | 1 |
1 review(s) available for pd 123177 and saralasin
Article | Year |
---|---|
[Angiotensin II receptor antagonists].
Topics: Amino Acid Sequence; Angiotensin II; Angiotensin Receptor Antagonists; Antihypertensive Agents; Biphenyl Compounds; Hemodynamics; Humans; Hypertension; Imidazoles; Losartan; Molecular Sequence Data; Pyridines; Receptors, Angiotensin; Renin-Angiotensin System; Saralasin; Tetrazoles | 1995 |
13 other study(ies) available for pd 123177 and saralasin
Article | Year |
---|---|
Angiotensin II binding sites in the hamster brain: localization and subtype distribution.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Brain; Cricetinae; Imidazoles; In Vitro Techniques; Mesencephalon; Mesocricetus; Prosencephalon; Pyridines; Receptors, Angiotensin; Rhombencephalon; Saralasin | 1992 |
Monoclonal antibodies to the nonpeptide angiotensin II receptor antagonist, losartan.
Topics: Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antibodies, Monoclonal; Antibody Specificity; Biphenyl Compounds; Cross Reactions; Enzyme-Linked Immunosorbent Assay; Imidazoles; Losartan; Mice; Mice, Inbred BALB C; Pyridines; Saralasin; Structure-Activity Relationship; Tetrazoles | 1992 |
Effect of angiotensin II antagonism on canine renal sympathetic nerve function.
Topics: Angiotensin II; Animals; Blood Pressure; Captopril; Dogs; Electric Stimulation; Female; Imidazoles; Kidney; Losartan; Male; Norepinephrine; Pyridines; Saralasin; Sympathetic Nervous System; Tetrazoles; Vascular Resistance; Vasoconstriction | 1991 |
Effects of U-97018 on pressor responses to intracerebroventricularly administered angiotensin II in conscious normotensive rats.
Topics: Administration, Oral; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Biphenyl Compounds; Blood Pressure; Disease Models, Animal; Dose-Response Relationship, Drug; Hypertension; Imidazoles; Injections, Intravenous; Injections, Intraventricular; Losartan; Male; Pyridazines; Pyridines; Rats; Rats, Inbred SHR; Rats, Sprague-Dawley; Saralasin; Tetrazoles | 1995 |
Synthetic cDNA encoding the rat AT1a receptor: a useful tool for structure-function relationship analysis.
Topics: Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Base Sequence; Biphenyl Compounds; CHO Cells; Codon; Cricetinae; DNA, Complementary; Imidazoles; Kinetics; Losartan; Molecular Sequence Data; Mutagenesis, Site-Directed; Oligodeoxyribonucleotides; Oligopeptides; Open Reading Frames; Pyridines; Rats; Receptors, Angiotensin; Restriction Mapping; Saralasin; Signal Transduction; Structure-Activity Relationship; Tetrazoles; Transfection | 1994 |
Selective changes in angiotensin II AT1 and AT2 receptor subtypes in the rat superior colliculus following eye enucleation.
Topics: Angiotensin I; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Autoradiography; Biphenyl Compounds; Eye Enucleation; Geniculate Bodies; Imidazoles; Iodine Radioisotopes; Losartan; Male; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Angiotensin; Retina; Saralasin; Subcellular Fractions; Superior Colliculi; Suprachiasmatic Nucleus; Synapses; Tetrazoles; Visual Pathways | 1994 |
Characterization of putative glomerular receptors for angiotensin II in the rainbow trout Oncorhynchus mykiss using the antagonists Losartan, PD 123177, and saralasin.
Topics: Analysis of Variance; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Biphenyl Compounds; Imidazoles; Iodine Radioisotopes; Kidney Glomerulus; Kinetics; Losartan; Oncorhynchus mykiss; Pyridines; Receptors, Angiotensin; Saralasin; Tetrazoles | 1993 |
Immunological reactivity of angiotensin II receptor antagonists: possible implications for receptor binding sites.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antibodies, Monoclonal; Antihypertensive Agents; Biphenyl Compounds; Imidazoles; In Vitro Techniques; Indicators and Reagents; Iodine Radioisotopes; Losartan; Molecular Conformation; Oligopeptides; Pyridines; Rats; Receptors, Angiotensin; Saralasin; Tetrazoles | 1993 |
Binding of angiotensin antagonists to rat liver and brain membranes measured ex vivo.
Topics: 1-Sarcosine-8-Isoleucine Angiotensin II; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Binding, Competitive; Biphenyl Compounds; Blood-Brain Barrier; Brain; Imidazoles; In Vitro Techniques; Iodine Radioisotopes; Liver; Losartan; Male; Membranes; Nicotinic Acids; Pyridines; Rats; Receptors, Angiotensin; Saralasin; Tetrazoles | 1993 |
Anti-angiotensin antibodies cross-reactive with nonpeptide angiotensin antagonists as angiotensin receptor model.
Topics: Adrenocorticotropic Hormone; Amino Acid Sequence; Angiotensin II; Angiotensin Receptor Antagonists; Animals; Antibodies; Biphenyl Compounds; Cross Reactions; Enzyme-Linked Immunosorbent Assay; Imidazoles; Losartan; Mice; Mice, Inbred BALB C; Molecular Sequence Data; Naloxone; Pyridines; Saralasin; Structure-Activity Relationship; Tetrazoles | 1993 |
Identification and characterisation of angiotensin II receptor subtypes in human brain.
Topics: Aged; Angiotensin II; Angiotensin Receptor Antagonists; Autoradiography; Binding, Competitive; Biphenyl Compounds; Brain Chemistry; Female; Humans; Imidazoles; In Vitro Techniques; Iodine Radioisotopes; Losartan; Male; Middle Aged; Pyridines; Radioligand Assay; Receptors, Angiotensin; Saralasin; Tetrazoles | 1993 |
Characterization of angiotensin AT1A receptor isoform by its ligand binding signature.
Topics: Adrenal Cortex; Angiotensin I; Angiotensin III; Animals; Base Sequence; Binding, Competitive; Biphenyl Compounds; CHO Cells; Cricetinae; Guanosine 5'-O-(3-Thiotriphosphate); Imidazoles; Losartan; Molecular Sequence Data; Muscle, Smooth, Vascular; Nicotinic Acids; Pyridines; Rats; Receptors, Angiotensin; Recombinant Proteins; Saralasin; Tetrazoles; Transfection | 1993 |
A novel angiotensin II binding site in murine tissues.
Topics: Amino Acid Sequence; Angiotensin II; Animals; Autoradiography; Binding Sites; Humans; Imidazoles; Losartan; Mice; Mice, Inbred C57BL; Mice, Nude; Pyridines; Saralasin; Tumor Cells, Cultured | 1998 |