Page last updated: 2024-09-02

pd 123177 and avapro

pd 123177 has been researched along with avapro in 3 studies

Compound Research Comparison

Studies
(pd 123177)
Trials
(pd 123177)
Recent Studies (post-2010)
(pd 123177)
Studies
(avapro)
Trials
(avapro)
Recent Studies (post-2010) (avapro)
142021,369385495

Protein Interaction Comparison

ProteinTaxonomypd 123177 (IC50)avapro (IC50)
Bile salt export pumpHomo sapiens (human)7.3067
Type-1 angiotensin II receptorHomo sapiens (human)0.0099
Type-2 angiotensin II receptorHomo sapiens (human)0.003

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (66.67)18.2507
2000's1 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cazaubon, C; Chatelain, P; Delisée, C; Schaeffer, P1
García-Sáinz, JA; González-Espinosa, C; Martínez-Alfaro, M; Romero-Avila, MT1
Li, Q; Pfaffendorf, M; van Zwieten, PA1

Other Studies

3 other study(ies) available for pd 123177 and avapro

ArticleYear
Characterization of cardiac angiotensin AT1 receptors by [3H]SR 47436.
    European journal of pharmacology, 1993, Oct-15, Volume: 247, Issue:2

    Topics: Angiotensin I; Angiotensin Receptor Antagonists; Animals; Animals, Newborn; Biphenyl Compounds; Calcium; Cells, Cultured; Heart; Homeostasis; Imidazoles; Irbesartan; Kinetics; Losartan; Myocardium; Pyridines; Rats; Rats, Wistar; Receptors, Angiotensin; Tetrazoles

1993
Characterization of the AT1 angiotensin II receptor expressed in guinea pig liver.
    The Journal of endocrinology, 1997, Volume: 154, Issue:1

    Topics: Angiotensin I; Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Antihypertensive Agents; Binding, Competitive; Biphenyl Compounds; Enzyme Activation; Guinea Pigs; Imidazoles; Irbesartan; Liver; Losartan; Male; Polymerase Chain Reaction; Pyridines; Receptors, Angiotensin; RNA, Messenger; Tetrazoles

1997
Different types of antagonism by losartan and irbesartan on the effects of angiotensin II and its degradation products in rabbit arteries.
    Fundamental & clinical pharmacology, 2001, Volume: 15, Issue:2

    Topics: Angiotensin II; Angiotensin III; Angiotensin Receptor Antagonists; Animals; Anti-Bacterial Agents; Antihypertensive Agents; Biphenyl Compounds; Endothelium, Vascular; Femoral Artery; Imidazoles; In Vitro Techniques; Irbesartan; Leucine; Losartan; Male; Peptides; Protease Inhibitors; Pyridines; Rabbits; Receptor, Angiotensin, Type 1; Renal Artery; Tetrazoles; Vasoconstrictor Agents

2001