pd 117302 has been researched along with substance p in 2 studies
Studies (pd 117302) | Trials (pd 117302) | Recent Studies (post-2010) (pd 117302) | Studies (substance p) | Trials (substance p) | Recent Studies (post-2010) (substance p) |
---|---|---|---|---|---|
48 | 0 | 2 | 17,289 | 277 | 2,010 |
Protein | Taxonomy | pd 117302 (IC50) | substance p (IC50) |
---|---|---|---|
Substance-P receptor | Rattus norvegicus (Norway rat) | 0.0005 | |
Substance-K receptor | Rattus norvegicus (Norway rat) | 0.2 | |
Substance-K receptor | Homo sapiens (human) | 0.2455 | |
Substance-P receptor | Homo sapiens (human) | 0.0011 | |
Neuromedin-K receptor | Homo sapiens (human) | 0.125 | |
Substance-K receptor | Mesocricetus auratus (golden hamster) | 0.148 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Blanchard, JC; Carruette, A; Garret, C; Laduron, PM; Montier, F; Moussaoui, SM | 1 |
Carruette, A; Garret, C; Moussaoui, S | 1 |
2 other study(ies) available for pd 117302 and substance p
Article | Year |
---|---|
A non-peptide NK1-receptor antagonist, RP 67580, inhibits neurogenic inflammation postsynaptically.
Topics: Animals; Animals, Newborn; Anti-Inflammatory Agents, Non-Steroidal; Anticonvulsants; Capsaicin; Electric Stimulation; Indoles; Inflammation; Injections, Intravenous; Isoindoles; Male; Morphine; Mucus; Nasal Mucosa; Pyrroles; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Neurotransmitter; Substance P; Synapses; Thiophenes; Xylenes | 1993 |
Further evidence that substance P is a mediator of both neurogenic inflammation and pain: two phenomena inhibited either by postsynaptic blockade of NK1 receptors or by presynaptic action of opioid receptor agonists.
Topics: Analgesics; Animals; Anticonvulsants; Electric Stimulation; Formaldehyde; Indoles; Inflammation; Isoindoles; Male; Mice; Mice, Inbred Strains; Morphine; Pain; Peripheral Nerves; Pyrroles; Rats; Rats, Sprague-Dawley; Substance P; Thiophenes | 1993 |