Page last updated: 2024-09-03

pd 117302 and metoclopramide

pd 117302 has been researched along with metoclopramide in 1 studies

Compound Research Comparison

Studies
(pd 117302)
Trials
(pd 117302)
Recent Studies (post-2010)
(pd 117302)
Studies
(metoclopramide)
Trials
(metoclopramide)
Recent Studies (post-2010) (metoclopramide)
48025,0441,216623

Protein Interaction Comparison

ProteinTaxonomypd 117302 (IC50)metoclopramide (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)2.383
MyeloperoxidaseHomo sapiens (human)0.35
Alpha-2A adrenergic receptorHomo sapiens (human)2.721
Cytochrome P450 2D6Homo sapiens (human)0.8
D(2) dopamine receptorHomo sapiens (human)0.127
Alpha-1B adrenergic receptorRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)7.8
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)7.7
Alpha-1D adrenergic receptorRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 2AHomo sapiens (human)3.675
5-hydroxytryptamine receptor 2CHomo sapiens (human)2.383
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1DRattus norvegicus (Norway rat)7.8
5-hydroxytryptamine receptor 1FRattus norvegicus (Norway rat)7.8
D(3) dopamine receptorHomo sapiens (human)0.2
5-hydroxytryptamine receptor 3ARattus norvegicus (Norway rat)0.88
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.63
Alpha-1A adrenergic receptorRattus norvegicus (Norway rat)7.8
D(2) dopamine receptorRattus norvegicus (Norway rat)0.6237
5-hydroxytryptamine receptor 3BRattus norvegicus (Norway rat)0.88

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baldwin, BA; Ebenezer, IS; Forsling, ML; Parrott, RF1

Other Studies

1 other study(ies) available for pd 117302 and metoclopramide

ArticleYear
Hormonal effects of apomorphine and cholecystokinin in pigs: modification of the response to cholecystokinin by a dopamine antagonist (metoclopramide) and a kappa opioid agonist (PD117302).
    Acta endocrinologica, 1991, Volume: 125, Issue:4

    Topics: Animals; Apomorphine; Cholecystokinin; Dopamine Antagonists; Feeding Behavior; Female; Hydrocortisone; Lypressin; Male; Metoclopramide; Pyrroles; Swine; Thiophenes

1991