Page last updated: 2024-09-03

pd 117302 and enkephalin, leucine-2-alanine

pd 117302 has been researched along with enkephalin, leucine-2-alanine in 2 studies

Compound Research Comparison

Studies
(pd 117302)
Trials
(pd 117302)
Recent Studies (post-2010)
(pd 117302)
Studies
(enkephalin, leucine-2-alanine)
Trials
(enkephalin, leucine-2-alanine)
Recent Studies (post-2010) (enkephalin, leucine-2-alanine)
48021,5812374

Protein Interaction Comparison

ProteinTaxonomypd 117302 (IC50)enkephalin, leucine-2-alanine (IC50)
Delta-type opioid receptorMus musculus (house mouse)0.0915
Delta-type opioid receptorRattus norvegicus (Norway rat)0.0017
Kappa-type opioid receptorMus musculus (house mouse)0.009
Mu-type opioid receptorRattus norvegicus (Norway rat)0.0419
Kappa-type opioid receptorCavia porcellus (domestic guinea pig)1.4691
Mu-type opioid receptorMus musculus (house mouse)0.009

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dissanayake, VU; Hill, RG; Hughes, J; Hunter, JC1
Magyar, A; Medzihradszky, K; RĂ³nai, AZ1

Other Studies

2 other study(ies) available for pd 117302 and enkephalin, leucine-2-alanine

ArticleYear
Characterization of kappa-opioid receptors in the guinea-pig ileum.
    European journal of pharmacology, 1990, Jun-21, Volume: 182, Issue:1

    Topics: Animals; Benzeneacetamides; Benzomorphans; Binding, Competitive; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle, Smooth; Naloxone; Pyrroles; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Thiophenes

1990
Kinetic parameters of antagonism by the delta opioid receptor selective peptide antagonist Boc-Tyr-Pro-Gly-Phe-Leu-Thr against selective and non-selective agonists in the mouse vas deferens.
    Neuropeptides, 1993, Volume: 25, Issue:2

    Topics: Analgesics; Animals; Anticonvulsants; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine-2-Alanine; Enkephalin, Methionine; Enkephalins; In Vitro Techniques; Kinetics; Male; Mice; Mice, Inbred Strains; Morphine Derivatives; Naltrexone; Oligopeptides; Pyrroles; Receptors, Opioid, delta; Thiophenes; Vas Deferens

1993