Page last updated: 2024-08-23

paroxetine and ketanserin

paroxetine has been researched along with ketanserin in 35 studies

Research

Studies (35)

TimeframeStudies, this research(%)All Research%
pre-19905 (14.29)18.7374
1990's19 (54.29)18.2507
2000's7 (20.00)29.6817
2010's4 (11.43)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Betti, L; Caputo, F; Clerici, F; Fabbrini, L; Gelmi, ML; Giannaccini, G; Lucacchini, A; Palego, L; Pellegrino, S; Schmid, L1
Lombardo, F; Obach, RS; Waters, NJ1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Cleves, AE; Jain, AN; Kirshner, D; Langham, JJ; Spitzer, R1
Barnes, JC; Bradley, P; Day, NC; Fourches, D; Reed, JZ; Tropsha, A1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Dalvie, D; Loi, CM; Smith, DA1
Emilsson, K; Hardebo, JE; Nystedt, S; Owman, C; Szabò, C1
Karnovsky, ML; Polanski, M1
Arora, RC; Meltzer, HY; Nash, JF; Schreiber, MA1
Bird, ED; Crino, PB; Plager, MD; Vogt, BA1
Bertocci, B; Cesura, AM; Da Prada, M1
Brunello, N; Galimberti, R; Racagni, G; Riva, M; Rovescalli, AC1
Koshikawa, N; Maruyama, Y; Stephenson, JD1
Laruelle, M; Maloteaux, JM; Vanisberg, MA1
Kobayashi, M; Koshikawa, N; Maruyama, Y; Mori, E; Nomura, H; Oka, K; Stephenson, JD1
Koshikawa, N; Smokcum, RW; Stephenson, JD1
Abi-Dargham, A; Casanova, MF; Kleinman, JE; Laruelle, M; Toti, R; Weinberger, DR1
Hrdina, PD; Vu, TB1
Battaglia, G; Pinto, W1
Demeter, E; Hrdina, PD; Palkovits, M; Sótónyi, P; Vu, TB1
Cadogan, AK; Kendall, DA; Marsden, CA; Tulloch, I1
Arranz, B; Eriksson, A; Marcusson, J; Mellerup, E; Plenge, P1
Abe, S; Baba, A; Hori, T; Moroji, T; Shiraishi, H; Suzuki, T; Yamamoto, T1
Copolov, DL; Dean, B; Hayes, W; Hill, C; Keks, N; Naylor, L; Opeskin, K; Pavey, G1
Egashira, T; Goto, S; Takayama, F; Wada, Y; Yamanaka, Y1
Choi, DS; Launay, JM; Maroteaux, L; Messaddeq, N; Ward, SJ1
Alder, JT; Bray, L; Chen, CP; Foster, OJ; Francis, PT; Kingsbury, AE1
Abe, S; Baba, A; Hori, T; Shiraishi, H; Suzuki, T; Yamamoto, T1
Fujiseki, Y; Inagaki, C; Kinoshita, T; Okugawa, G; Omori, K; Suzukawa, J1
Akagawa, Y; Hishikawa, Y; Maruyama, A; Masuda, Y; Shimizu, T1
Duman, EN; Erciyes, N; Kadioglu, M; Kalyoncu, NI; Kesim, M; Yaris, E1
Imanishi, T; Matsushima, T; Miyara, T; Yamauchi, M1
Bell, W; Deng, C; du Bois, TM; Huang, XF1
Maraschin, M; Rodrigues, AL; Tasca, CI; Zeni, AL; Zomkowski, AD1

Other Studies

35 other study(ies) available for paroxetine and ketanserin

ArticleYear
1-Aminocyclopentane-1,2,4-tricarboxylic acids screening on glutamatergic and serotonergic systems.
    Bioorganic & medicinal chemistry, 2007, Dec-15, Volume: 15, Issue:24

    Topics: Animals; Cells, Cultured; Cyclopentanes; Drug Evaluation, Preclinical; Humans; Molecular Structure; Rats; Receptors, Glutamate; Receptors, Serotonin; Serotonin Receptor Agonists; Stereoisomerism; Tricarboxylic Acids

2007
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physical binding pocket induction for affinity prediction.
    Journal of medicinal chemistry, 2009, Oct-08, Volume: 52, Issue:19

    Topics: Binding Sites; Ligands; Models, Molecular; Neural Networks, Computer; Peptide Fragments; Protein Binding; Receptor, Serotonin, 5-HT1A

2009
Cheminformatics analysis of assertions mined from literature that describe drug-induced liver injury in different species.
    Chemical research in toxicology, 2010, Volume: 23, Issue:1

    Topics: Animals; Chemical and Drug Induced Liver Injury; Cluster Analysis; Databases, Factual; Humans; MEDLINE; Mice; Models, Chemical; Molecular Conformation; Quantitative Structure-Activity Relationship

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Which metabolites circulate?
    Drug metabolism and disposition: the biological fate of chemicals, 2013, Volume: 41, Issue:5

    Topics: Humans; Metabolic Clearance Rate; Pharmaceutical Preparations

2013
Uptake and release of serotonin in rat cerebrovascular nerves after subarachnoid hemorrhage.
    Stroke, 1992, Volume: 23, Issue:1

    Topics: Animals; Basilar Artery; Electric Stimulation; Ischemic Attack, Transient; Ketanserin; Male; Oxidopamine; Paroxetine; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Subarachnoid Hemorrhage; Sympathetic Nervous System; Tetrodotoxin; Vasoconstriction

1992
Serotonergic aspects of the response of human platelets to immune-adjuvant muramyl dipeptide.
    Journal of neuroimmunology, 1992, Volume: 37, Issue:1-2

    Topics: Acetylmuramyl-Alanyl-Isoglutamine; Adenosine Diphosphate; Adjuvants, Immunologic; Blood Platelets; Carrier Proteins; Humans; Imipramine; Ketanserin; Lysergic Acid Diethylamide; Paroxetine; Piperidines; Platelet Aggregation; Platelet Aggregation Inhibitors; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1992
Effect of 3,4-methylenedioxymethamphetamine on [3H]paroxetine binding in the frontal cortex and blood platelets of rats.
    Biochemical pharmacology, 1991, Jan-01, Volume: 41, Issue:1

    Topics: 3,4-Methylenedioxyamphetamine; Animals; Blood Platelets; Frontal Lobe; Hydroxyindoleacetic Acid; Ketanserin; Kinetics; Male; N-Methyl-3,4-methylenedioxyamphetamine; Paroxetine; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Serotonin Antagonists; Time Factors; Tritium

1991
Laminar distributions of muscarinic acetylcholine, serotonin, GABA and opioid receptors in human posterior cingulate cortex.
    Neuroscience, 1990, Volume: 36, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aged; Autoradiography; Cerebral Cortex; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Humans; Iodocyanopindolol; Ketanserin; Male; Middle Aged; Oxotremorine; Paroxetine; Pindolol; Piperidines; Pirenzepine; Receptors, Cell Surface; Receptors, Cholinergic; Receptors, GABA-A; Receptors, Muscarinic; Receptors, Opioid; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes

1990
Binding of [3H]dihydrotetrabenazine and [125I]azidoiodoketanserin photoaffinity labeling of the monoamine transporter of platelet 5-HT organelles.
    European journal of pharmacology, 1990, Sep-04, Volume: 186, Issue:1

    Topics: Affinity Labels; Animals; Azides; Biogenic Monoamines; Blood Platelets; Blood Proteins; Cell Membrane; Guinea Pigs; Humans; In Vitro Techniques; Iodine Radioisotopes; Ketanserin; Paroxetine; Photochemistry; Piperidines; Rabbits; Rats; Receptors, Serotonin; Subcellular Fractions; Tetrabenazine

1990
Age-related changes in rat serotonergic and adrenergic systems and in receptor responsiveness to subchronic desipramine treatment.
    Pharmacology & toxicology, 1988, Volume: 63, Issue:3

    Topics: Aging; Animals; Brain; Clonidine; Desipramine; Dihydroalprenolol; Hydroxyindoleacetic Acid; Imipramine; Ketanserin; Kinetics; Male; Paroxetine; Piperidines; Prazosin; Proteins; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Serotonin; Serotonin; Time Factors

1988
Production of wet-dog shakes in rats and down-regulation of spinal 5-HT2 receptors.
    European journal of pharmacology, 1989, May-30, Volume: 164, Issue:3

    Topics: Animals; Behavior, Animal; Brain Stem; Ketanserin; Male; Paroxetine; Phenelzine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Spinal Cord

1989
Regional and subcellular localization in human brain of [3H]paroxetine binding, a marker of serotonin uptake sites.
    Biological psychiatry, 1988, Volume: 24, Issue:3

    Topics: Adult; Aged; Animals; Binding, Competitive; Brain; Brain Mapping; Cerebral Cortex; Corpus Striatum; Humans; Ketanserin; Male; Middle Aged; Paroxetine; Piperidines; Putamen; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin Antagonists; Subcellular Fractions; Synaptosomes

1988
Changes in cortical 5-HT2 receptors following 5-HTP and paroxetine administration in rats.
    The Journal of Nihon University School of Dentistry, 1988, Volume: 30, Issue:3

    Topics: Animals; Carbidopa; Cerebral Cortex; Ketanserin; Male; Paroxetine; Phenelzine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin

1988
Is waning of a 5-hydroxytryptamine (5-HT)-mediated syndrome due to 5-HT2 receptor down-regulation?
    Neuroscience letters, 1985, Apr-19, Volume: 55, Issue:3

    Topics: Animals; Cerebral Cortex; Ketanserin; Male; Myoclonus; Paroxetine; Phenelzine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Syndrome; Time Factors; Tritium

1985
Selective abnormalities of prefrontal serotonergic receptors in schizophrenia. A postmortem study.
    Archives of general psychiatry, 1993, Volume: 50, Issue:10

    Topics: Adult; Diagnosis, Differential; Down-Regulation; Female; Frontal Lobe; Humans; Ketanserin; Male; Middle Aged; Occipital Lobe; Paroxetine; Psychotic Disorders; Receptors, Serotonin; Schizophrenia; Suicide; Tritium

1993
Chronic fluoxetine treatment upregulates 5-HT uptake sites and 5-HT2 receptors in rat brain: an autoradiographic study.
    Synapse (New York, N.Y.), 1993, Volume: 14, Issue:4

    Topics: Animals; Autoradiography; Brain Chemistry; Fluoxetine; Image Processing, Computer-Assisted; Ketanserin; Male; Mianserin; Paroxetine; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Up-Regulation

1993
In vivo EEDQ dose-dependently inactivates rat brain 5-HT receptors but not 5-HT uptake sites.
    Neuroreport, 1993, Oct-25, Volume: 5, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Analysis of Variance; Animals; Brain; Carrier Proteins; Cerebral Cortex; Dose-Response Relationship, Drug; Iodocyanopindolol; Ketanserin; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Paroxetine; Pindolol; Quinolines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins

1993
5-HT uptake sites and 5-HT2 receptors in brain of antidepressant-free suicide victims/depressives: increase in 5-HT2 sites in cortex and amygdala.
    Brain research, 1993, Jun-18, Volume: 614, Issue:1-2

    Topics: Adult; Aged; Amygdala; Binding, Competitive; Cerebral Cortex; Depressive Disorder; Female; Humans; In Vitro Techniques; Ketanserin; Male; Middle Aged; Nerve Tissue Proteins; Paroxetine; Protein Binding; Receptors, Serotonin; Suicide

1993
Evidence that chronic administration of paroxetine or fluoxetine enhances 5-HT2 receptor function in the brain of the guinea pig.
    Neuropharmacology, 1993, Volume: 32, Issue:3

    Topics: Amitriptyline; Animals; Brain Chemistry; Calcimycin; Calcium; Cerebral Cortex; Female; Fluoxetine; Guinea Pigs; In Vitro Techniques; Inositol; Ketanserin; Male; Paroxetine; Phosphatidylinositols; Receptors, Serotonin; Serotonin; Serotonin Antagonists

1993
Effect of aging in human cortical pre- and postsynaptic serotonin binding sites.
    Brain research, 1993, Aug-20, Volume: 620, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adolescent; Adult; Aged; Aging; Binding Sites; Female; Frontal Lobe; Humans; Ketanserin; Male; Middle Aged; Paroxetine; Radioligand Assay; Serotonin; Synapses

1993
Effects of phencyclidine metabolites on serotonin uptake in rat brain.
    Neuroscience letters, 1996, May-17, Volume: 209, Issue:3

    Topics: Animals; Brain; Ketanserin; Male; Paroxetine; Phencyclidine; Rats; Rats, Wistar; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin

1996
Serotonin2 receptors and the serotonin transporter in the schizophrenic brain.
    Behavioural brain research, 1996, Volume: 73, Issue:1-2

    Topics: Adolescent; Adult; Aged; Brain Chemistry; Carrier Proteins; Caudate Nucleus; Female; Hippocampus; Humans; In Vitro Techniques; Ketanserin; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Membranes; Middle Aged; Nerve Tissue Proteins; Paroxetine; Prefrontal Cortex; Receptors, Serotonin; Schizophrenia; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins

1996
Effect of fluvoxamine on 5-hydroxytryptamine uptake, paroxetine binding sites and ketanserin binding sites in the Japanese monkey brain and platelets, in vivo and in vitro.
    Japanese journal of pharmacology, 1996, Volume: 71, Issue:4

    Topics: Animals; Binding, Competitive; Blood Platelets; Brain; Cerebral Cortex; Fluvoxamine; In Vitro Techniques; Ketanserin; Macaca; Male; Paroxetine; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin

1996
5-HT2B receptor-mediated serotonin morphogenetic functions in mouse cranial neural crest and myocardiac cells.
    Development (Cambridge, England), 1997, Volume: 124, Issue:9

    Topics: Animals; Binding Sites; Brain; Cell Differentiation; DNA Primers; Embryo, Mammalian; Embryonic and Fetal Development; Embryonic Induction; Gene Expression Regulation, Developmental; Heart; Humans; In Situ Hybridization; Ketanserin; Methysergide; Mice; Microscopy, Electron, Scanning; Morphogenesis; Neural Crest; Organ Culture Techniques; Paroxetine; Polymerase Chain Reaction; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Ritanserin; RNA, Messenger; Serotonin; Serotonin Antagonists; Signal Transduction; Transcription, Genetic

1997
Post-synaptic 5-HT1A and 5-HT2A receptors are increased in Parkinson's disease neocortex.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Humans; Ketanserin; Kinetics; Neocortex; Parkinson Disease; Paroxetine; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Reference Values

1998
Effects of chronic administration of interferon alpha A/D on serotonergic receptors in rat brain.
    Neurochemical research, 1999, Volume: 24, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Carrier Proteins; Cell Membrane; Cerebral Cortex; Hippocampus; Interferon Type I; Ketanserin; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Paroxetine; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Recombinant Proteins; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Tritium

1999
Long-term treatment with antidepressants increases glucocorticoid receptor binding and gene expression in cultured rat hippocampal neurones.
    Journal of neuroendocrinology, 1999, Volume: 11, Issue:11

    Topics: Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Cells, Cultured; Desipramine; Dexamethasone; Gene Expression Regulation; Haloperidol; Hippocampus; Ketanserin; Mianserin; Neurons; Paroxetine; Phentolamine; Propranolol; Radioligand Assay; Rats; Receptors, Glucocorticoid; Receptors, Mineralocorticoid; RNA, Messenger; Sulpiride; Transcription, Genetic; Tritium

1999
Effects of repeated selective serotonin reuptake inhibitor paroxetine treatments on mouse forced swimming.
    Methods and findings in experimental and clinical pharmacology, 1999, Volume: 21, Issue:9

    Topics: Animals; Drug Evaluation, Preclinical; Drug Interactions; Indazoles; Ketanserin; Male; Mice; Paroxetine; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Swimming; Time Factors; Tropanes

1999
The different roles of 5-HT(2) and 5-HT(3) receptors on antinociceptive effect of paroxetine in chemical stimuli in mice.
    Journal of pharmacological sciences, 2005, Volume: 97, Issue:1

    Topics: Abdominal Pain; Acetic Acid; Analgesia; Analgesics; Animals; Dose-Response Relationship, Drug; Drug Synergism; Female; Injections, Intraperitoneal; Ketanserin; Male; Mice; Mice, Inbred BALB C; Morphine; Naloxone; Ondansetron; Pain Measurement; Paroxetine; Receptors, Serotonin, 5-HT2; Receptors, Serotonin, 5-HT3

2005
Desensitization of 5-HT2A receptor function by chronic administration of selective serotonin reuptake inhibitors.
    Brain research, 2006, Jan-05, Volume: 1067, Issue:1

    Topics: Animals; Corticosterone; Fluvoxamine; Ketanserin; Paroxetine; Rats; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors

2006
Fatty acids differentially affect serotonin receptor and transporter binding in the rat brain.
    Neuroscience, 2006, Volume: 139, Issue:4

    Topics: Analysis of Variance; Animals; Brain; Ergolines; Fatty Acids; Ketanserin; Male; Paroxetine; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins

2006
Ferulic acid exerts antidepressant-like effect in the tail suspension test in mice: evidence for the involvement of the serotonergic system.
    European journal of pharmacology, 2012, Mar-15, Volume: 679, Issue:1-3

    Topics: Animals; Antidepressive Agents; Coumaric Acids; Dose-Response Relationship, Drug; Drug Interactions; Fluoxetine; Immobility Response, Tonic; Ketanserin; Male; Mice; Motor Activity; Paroxetine; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT2A; Selective Serotonin Reuptake Inhibitors; Serotonin 5-HT1 Receptor Antagonists; Serotonin 5-HT2 Receptor Antagonists; Sertraline

2012