papaverine and prazosin

papaverine has been researched along with prazosin in 25 studies

Research

Studies (25)

TimeframeStudies, this research(%)All Research%
pre-19908 (32.00)18.7374
1990's4 (16.00)18.2507
2000's7 (28.00)29.6817
2010's6 (24.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Lombardo, F; Obach, RS; Waters, NJ1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Sen, S; Sinha, N1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Gomes da Silva, AC; Nigro, D; Scivoletto, R; Toledo, AJ1
Large, WA; Wang, Q1
Bevan, JA; Bevan, RD; Vorkapic, P1
Cohen, RA; Tesfamariam, B; Weisbrod, RM; Zitnay, KM1
Diecke, FP; Greenberg, S; Peevy, K; Tanaka, TP1
Andersson, KE; Forman, A; Kirkeby, HJ; Sørensen, S1
O'Hara, N; Ono, H1
Aramendía, P; Eisenschlos, CD; Márquez, MT1
Nakashima, M; Oguro, K; Ohguchi, S1
Estan, L; Martinez-Mir, I; Morales-Olivas, FJ; Rubio, E1
Advenier, C; Chulia, S; D'Ocon, P; Elorriaga, M; Ivorra, MD; Lugnier, C; Martinez, S; Noguera, MA; Valiente, M1
Abel, D; Danuser, H; Mettler, D; Scholtysik, G; Studer, UE; Walter, B; Weiss, R1
Hirouchi, M; Noda, K; Oka, M; Takebe, M; Toda, N; Ukai, Y1
Haslam, JL; Sotthivirat, S; Stella, VJ1
Guo, YM; Jin, QY; Liang, C; Zhang, YR1

Reviews

1 review(s) available for papaverine and prazosin

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

24 other study(ies) available for papaverine and prazosin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:2

    Topics: Computer Simulation; Ether-A-Go-Go Potassium Channels; Humans; Molecular Structure; Organic Chemicals; Quantitative Structure-Activity Relationship

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Mechanism of the hypotensive effect of prazosin.
    Archives internationales de pharmacodynamie et de therapie, 1976, Volume: 223, Issue:2

    Topics: Animals; Blood Pressure; Carotid Sinus; Depression, Chemical; Dogs; Drug Interactions; Electric Stimulation; Epinephrine; Female; Heart Rate; Male; Nitrates; Norepinephrine; Papaverine; Prazosin; Quinazolines; Time Factors; Venous Pressure

1976
Modulation of noradrenaline-induced membrane currents by papaverine in rabbit vascular smooth muscle cells.
    The Journal of physiology, 1991, Volume: 439

    Topics: Animals; Caffeine; Calcium; Chlorides; Dose-Response Relationship, Drug; Female; Ion Channels; Ionomycin; Male; Membrane Potentials; Muscle, Smooth, Vascular; Norepinephrine; Papaverine; Potassium Channels; Prazosin; Rabbits

1991
Pharmacologic irreversible narrowing in chronic cerebrovasospasm in rabbits is associated with functional damage.
    Stroke, 1990, Volume: 21, Issue:10

    Topics: Acetylcholine; Animals; Basilar Artery; Cimetidine; Epinephrine; Histamine; In Vitro Techniques; Ischemic Attack, Transient; Papaverine; Prazosin; Rabbits; Serotonin; Subarachnoid Hemorrhage; Tetrodotoxin; Vasoconstriction

1990
Influence of the endothelium on tone and the response of isolated pig coronary artery to norepinephrine.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:2

    Topics: Animals; Coronary Vessels; Dinoprost; Endothelium, Vascular; In Vitro Techniques; Nitroprusside; Norepinephrine; Papaverine; Prazosin; Prostaglandins F; Substance P; Swine; Vasoconstriction; Vasodilation

1988
The endothelium modulates adrenergic neurotransmission to canine pulmonary arteries and veins.
    European journal of pharmacology, 1989, Mar-14, Volume: 162, Issue:1

    Topics: Acetylcholine; Animals; Aorta, Thoracic; Biological Factors; Bretylium Compounds; Dogs; Electric Stimulation; Endothelium, Vascular; Epoprostenol; Female; In Vitro Techniques; Male; Muscle Contraction; Nitric Oxide; Norepinephrine; Papaverine; Prazosin; Pulmonary Artery; Pulmonary Veins; Sympathetic Nervous System; Synaptic Transmission; Tetrodotoxin

1989
Alpha-adrenoceptor function in isolated penile circumflex veins from potent and impotent men.
    The Journal of urology, 1989, Volume: 142, Issue:5

    Topics: Adult; Aged; Erectile Dysfunction; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Norepinephrine; Papaverine; Penile Erection; Penis; Phentolamine; Phenylephrine; Potassium; Prazosin; Receptors, Adrenergic, alpha; Veins; Yohimbine

1989
Papaverine inhibits binding of [3H]-prazosin and [3H]-yohimbine to rat renal cortical membranes.
    Research communications in chemical pathology and pharmacology, 1986, Volume: 54, Issue:2

    Topics: Animals; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Kidney Cortex; Kinetics; Male; Norepinephrine; Papaverine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tritium; Verapamil; Yohimbine

1986
Antagonism and supersensitivity to phenylephrine-induced chronotropic responses.
    Acta physiologica latino americana, 1983, Volume: 33, Issue:3

    Topics: Animals; Calcium; Female; Heart Rate; In Vitro Techniques; Myocardium; Papaverine; Phentolamine; Phenylephrine; Prazosin; Quinazolines; Rats

1983
Induction of opposite response of hindlimb vasculature to adrenergic agents in hypothyroid rats.
    Archives internationales de pharmacodynamie et de therapie, 1984, Volume: 268, Issue:2

    Topics: Acetylcholine; Animals; Blood Pressure; Clonidine; Heart Rate; Hindlimb; Hypothyroidism; In Vitro Techniques; Isoproterenol; Male; Muscle, Smooth, Vascular; Papaverine; Prazosin; Rats; Rats, Inbred Strains; Regional Blood Flow; Sympathomimetics

1984
No evidence for dopamine-induced relaxation in isolated human mesenteric arterial strips from elderly patients.
    General pharmacology, 1995, Volume: 26, Issue:8

    Topics: Aged; Aged, 80 and over; Dopamine; Epinephrine; Fenoldopam; Humans; In Vitro Techniques; Mesenteric Arteries; Middle Aged; Papaverine; Prazosin; Vasodilation

1995
Relationships between structure and vascular activity in a series of benzylisoquinolines.
    British journal of pharmacology, 1997, Volume: 122, Issue:3

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Aorta; Diltiazem; Female; In Vitro Techniques; Inositol Phosphates; Isoquinolines; Male; Muscle Contraction; Muscle, Smooth, Vascular; Papaverine; Parasympatholytics; Prazosin; Radioligand Assay; Rats; Structure-Activity Relationship

1997
Systemic and topical drug administration in the pig ureter: effect of phosphodiesterase inhibitors alpha1, beta and beta2-adrenergic receptor agonists and antagonists on the frequency and amplitude of ureteral contractions.
    The Journal of urology, 2001, Volume: 166, Issue:2

    Topics: Administration, Topical; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Female; Fenoterol; Injections, Intravenous; Isoproterenol; Male; Muscle Contraction; Papaverine; Phenylephrine; Phosphodiesterase Inhibitors; Prazosin; Propranolol; Rolipram; Swine; Ureter

2001
Functional role of inhibitory and excitatory nerves in the porcine lower urinary tract.
    European journal of pharmacology, 2002, Dec-05, Volume: 456, Issue:1-3

    Topics: Adrenergic alpha-Antagonists; Animals; Arginine; Atropine; Cyclic GMP; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Papaverine; Prazosin; Swine; Tetrodotoxin; Urethra; Urinary Bladder; Urinary Tract; Vasodilator Agents; Yohimbine

2002
Evaluation of various properties of alternative salt forms of sulfobutylether-beta-cyclodextrin, (SBE)7M-beta-CD.
    International journal of pharmaceutics, 2007, Feb-07, Volume: 330, Issue:1-2

    Topics: beta-Cyclodextrins; Calcium; Delayed-Action Preparations; Diffusion; Drug Delivery Systems; Ethylenediamines; Osmolar Concentration; Papaverine; Potassium; Prazosin; Prednisolone; Sodium; Solubility; Testosterone; Viscosity

2007
[Analysis of 37 drugs in whole blood by HPLC after solid phase extraction].
    Fa yi xue za zhi, 2006, Oct-15, Volume: 22, Issue:5

    Topics: Chromatography, High Pressure Liquid; Doxapram; Doxepin; Estazolam; Forensic Medicine; Humans; Morphine; Papaverine; Pharmaceutical Preparations; Prazosin; Procaine; Reproducibility of Results; Sensitivity and Specificity; Solid Phase Extraction; Solvents

2006