papaverine has been researched along with pf-2545920 in 8 studies
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 0 (0.00) | 29.6817 |
| 2010's | 8 (100.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Brandon, NJ; Egerland, U; Grunwald, C; Hage, T; Harrison, BL; Höfgen, N; Kronbach, T; Langen, B; Lankau, HJ; Malamas, MS; Marquis, KL; Pangalos, MN; Schindler, R; Stange, H; Tremmel, P | 1 |
| Bundgaard, C; Christoffersen, CT; Farah, MM; Kehler, J; Kilburn, JP; Langgård, M; Nielsen, J; Petersen, SL; Ritzen, A | 1 |
| Lu, X; Mach, RH; Rothfuss, J; Tu, Z; Xu, J; Zhang, Z | 1 |
| Chappie, TA; Helal, CJ; Hou, X | 1 |
| Christoffersen, CT; Erichsen, MN; Kehler, J; Kilburn, JP; Langgård, M; Larsen, M; Leth-Petersen, S; Nielsen, J | 1 |
| Fan, J; Flores, HP; Jin, H; Jones, LA; Li, J; Padakanti, PK; Perlmutter, JS; Su, Y; Tu, Z; Zhang, X | 1 |
| Jin, H; Li, J; Murigi, FN; Tu, Z; Wang, Z; Yang, H | 1 |
| Chen, Y; Guo, L; Huang, YY; Li, Z; Luo, HB; Wu, D; Wu, Y; Yu, YF; Zhang, C; Zhou, Q; Zhou, S | 1 |
8 other study(ies) available for papaverine and pf-2545920
| Article | Year |
|---|---|
Discovery of imidazo[1,5-a]pyrido[3,2-e]pyrazines as a new class of phosphodiesterase 10A inhibitiors.
Topics: Animals; Drug Discovery; Female; Humans; Models, Molecular; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Protein Conformation; Pyrazines; Quantitative Structure-Activity Relationship; Rats; Rats, Wistar | 2010 |
Triazoloquinazolines as a novel class of phosphodiesterase 10A (PDE10A) inhibitors.
Topics: Animals; Benzimidazoles; Crystallography, X-Ray; Enzyme Activation; Inhibitory Concentration 50; Models, Molecular; Molecular Structure; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Protein Binding; Quinazolines; Rats | 2011 |
Synthesis and in vitro evaluation of new analogues as inhibitors for phosphodiesterase 10A.
Topics: Drug Evaluation, Preclinical; Humans; Inhibitory Concentration 50; Magnetic Resonance Spectroscopy; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases | 2011 |
Current landscape of phosphodiesterase 10A (PDE10A) inhibition.
Topics: Animals; Cyclic AMP; Cyclic GMP; Humans; Hydrolysis; Mice; Models, Molecular; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Rats | 2012 |
N-Methylanilide and N-methylbenzamide derivatives as phosphodiesterase 10A (PDE10A) inhibitors.
Topics: Anilides; Benzamides; Crystallography, X-Ray; Enzyme Activation; Humans; Inhibitory Concentration 50; Molecular Structure; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Structure-Activity Relationship | 2013 |
Radiosyntheses and in vivo evaluation of carbon-11 PET tracers for PDE10A in the brain of rodent and nonhuman primate.
Topics: Animals; Brain; Carbon Radioisotopes; Macaca fascicularis; Male; Phosphoric Diester Hydrolases; Positron-Emission Tomography; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Tissue Distribution | 2014 |
Synthesis and in vitro characterization of cinnoline and benzimidazole analogues as phosphodiesterase 10A inhibitors.
Topics: Benzimidazoles; Heterocyclic Compounds, 2-Ring; Humans; In Vitro Techniques; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases | 2015 |
Validation of Phosphodiesterase-10 as a Novel Target for Pulmonary Arterial Hypertension via Highly Selective and Subnanomolar Inhibitors.
Topics: Animals; Crystallography, X-Ray; Humans; Hypertension, Pulmonary; Male; Molecular Dynamics Simulation; Muscle, Smooth; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Platelet-Derived Growth Factor; Protein Binding; Protein Conformation; Rats | 2019 |