papaverine and glyburide

papaverine has been researched along with glyburide in 20 studies

Research

Studies (20)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's5 (25.00)18.2507
2000's9 (45.00)29.6817
2010's6 (30.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Sen, S; Sinha, N1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Hatake, K; Hishida, S; Wakabayashi, I1
Halama, A; Korolkiewicz, KZ; Korolkiewicz, R; Rekowski, P; Sliwiński, W1
Faraci, FM; Sobey, CG2
Deka, DK; Mishra, SK; Raviprakash, V1
García de Boto, MJ; Hidalgo, A; Martínez, C; Sánchez, M1
Bosnjak, JJ; Gutterman, DD; Miura, H; Miura, M; Ning, G; Saito, T1
Clancy, JP; Cobb, BR; Fan, L; Kovacs, TE; Sorscher, EJ1
Antunes, E; de Miranda Cará, A; De Nucci, G; Fregonesi, A; Rodrigues Netto, N1
Fujimoto, S; Kunimatsu, M; Mori, M; Tsushima, H1
Colantuoni, A; Lapi, D; Marchiafava, PL1

Reviews

1 review(s) available for papaverine and glyburide

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

19 other study(ies) available for papaverine and glyburide

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Predicting hERG activities of compounds from their 3D structures: development and evaluation of a global descriptors based QSAR model.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:2

    Topics: Computer Simulation; Ether-A-Go-Go Potassium Channels; Humans; Molecular Structure; Organic Chemicals; Quantitative Structure-Activity Relationship

2011
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Endothelium-dependent relaxation resistant to NG-nitro-L-arginine in rat aorta.
    European journal of pharmacology, 1995, Feb-14, Volume: 274, Issue:1-3

    Topics: Acetylcholine; Analysis of Variance; Animals; Aorta, Thoracic; Arginine; Atropine; Biological Factors; Cyclic GMP; Endothelium, Vascular; Glyburide; Indomethacin; Isometric Contraction; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroarginine; Norepinephrine; Oxyhemoglobins; Papaverine; Potassium Channel Blockers; Rats; Rats, Wistar; Tetraethylammonium; Tetraethylammonium Compounds

1995
Actions of galanin and some of its analogues on rat isolated gastric fundus.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:5

    Topics: Analysis of Variance; Animals; Bucladesine; Calcium Channel Blockers; Dibenzylchlorethamine; Diltiazem; Dimethyl Sulfoxide; Dose-Response Relationship, Drug; Female; Galanin; Gastric Fundus; Glyburide; Lethal Dose 50; Male; Muscle Contraction; Muscle, Smooth; Papaverine; Parasympatholytics; Rats; Rats, Wistar; Substance P

1996
Effect of nitric oxide and potassium channel agonists and inhibitors on basilar artery diameter.
    The American journal of physiology, 1997, Volume: 272, Issue:1 Pt 2

    Topics: Animals; Basilar Artery; Enzyme Inhibitors; Glyburide; Male; Nitric Oxide; Nitroarginine; Nitroprusside; Papaverine; Peptides; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Tetraethylammonium; Tetraethylammonium Compounds; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

1997
Basal nitric oxide release differentially modulates vasodilations by pinacidil and levcromakalim in goat coronary artery.
    European journal of pharmacology, 1998, May-01, Volume: 348, Issue:1

    Topics: Animals; Coronary Vessels; Cromakalim; Endothelium, Vascular; Enzyme Inhibitors; Glyburide; Goats; Guanidines; Hypoglycemic Agents; In Vitro Techniques; Methylene Blue; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Papaverine; Pinacidil; Potassium Channels; Vasodilation; Vasodilator Agents

1998
Inhibitory effect of 4-aminopyridine on responses of the basilar artery to nitric oxide.
    British journal of pharmacology, 1999, Volume: 126, Issue:6

    Topics: 4-Aminopyridine; Acetylcholine; Adenosine Triphosphate; Animals; Basilar Artery; Cromakalim; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Guanylate Cyclase; Male; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Oxadiazoles; Papaverine; Potassium Channel Blockers; Quinoxalines; Rats; Rats, Sprague-Dawley; Vasodilation; Vasodilator Agents

1999
Involvement of K(ATP) channels in diethylstilbestrol-induced relaxation in rat aorta.
    European journal of pharmacology, 2001, Feb-09, Volume: 413, Issue:1

    Topics: Animals; Aorta; Colforsin; Cyclic AMP; Diazoxide; Diethylstilbestrol; Dose-Response Relationship, Drug; Eflornithine; Glyburide; In Vitro Techniques; Indoles; Male; Muscle, Smooth, Vascular; Norepinephrine; Papaverine; Potassium Channels; Rats; Rats, Wistar; Spermine; Tamoxifen; Tetraethylammonium; Vasoconstriction; Vasodilation; Vasodilator Agents

2001
Role for hydrogen peroxide in flow-induced dilation of human coronary arterioles.
    Circulation research, 2003, Feb-07, Volume: 92, Issue:2

    Topics: Apamin; Arterioles; Catalase; Cerium; Coronary Vessels; Enzyme Inhibitors; Fluorescent Dyes; Glyburide; Humans; Hydrogen Peroxide; In Vitro Techniques; Iron Chelating Agents; Membrane Potentials; Microscopy, Confocal; Microscopy, Electron; Microscopy, Video; Muscle, Smooth, Vascular; Oxidants; Papaverine; Potassium Channel Blockers; Stress, Mechanical; Vasodilation; Vasodilator Agents

2003
Adenosine receptors and phosphodiesterase inhibitors stimulate Cl- secretion in Calu-3 cells.
    American journal of respiratory cell and molecular biology, 2003, Volume: 29, Issue:3 Pt 1

    Topics: Adenosine Deaminase; Anions; Cell Line; Chlorine; Cilostazol; Colforsin; Cyclic AMP; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Electrophysiology; Epithelium; Glyburide; Humans; Hypoglycemic Agents; Milrinone; Mutation; Papaverine; Phosphodiesterase Inhibitors; Piperazines; Purines; Receptors, Purinergic P1; Rolipram; Sildenafil Citrate; Sulfones; Tetrazoles; Time Factors

2003
Role of adenosine triphosphate-dependent potassium channels in canine penile erection.
    Urology, 2004, Volume: 64, Issue:3

    Topics: Adenosine Triphosphate; Animals; Arginine; Cromakalim; Dogs; Electric Stimulation; Glyburide; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Papaverine; Penile Erection; Potassium Channel Blockers; Potassium Channels; Pressure; Receptors, Drug

2004
Capsaicin-induced, capsazepine-insensitive relaxation of the guinea-pig ileum.
    European journal of pharmacology, 2006, Jan-13, Volume: 530, Issue:1-2

    Topics: 4-Aminopyridine; Acetylcholine; Animals; Apamin; Barium; Benzopyrans; Caffeine; Calcitonin Gene-Related Peptide; Calcium; Capsaicin; Charybdotoxin; Diclofenac; Dimethyl Sulfoxide; Diterpenes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glyburide; Guanethidine; Guinea Pigs; Ileum; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Muscle Relaxation; Muscle, Smooth; Myosin Light Chains; Nitroarginine; Papaverine; Peptide Fragments; Phosphodiesterase Inhibitors; Phosphorylation; Piperidines; Potassium Channel Blockers; Potassium Channels; Potassium Chloride; Protein Serine-Threonine Kinases; Pyrazoles; Receptor, Cannabinoid, CB1; rho-Associated Kinases; Tetraethylammonium; Vasodilator Agents

2006
Pial microvascular responses to transient bilateral common carotid artery occlusion: effects of hypertonic glycerol.
    Journal of vascular research, 2008, Volume: 45, Issue:2

    Topics: Animals; Blood Flow Velocity; Capillary Permeability; Carotid Artery, Common; Carotid Stenosis; Cell Adhesion; Cerebrovascular Circulation; Chemotaxis, Leukocyte; Disease Models, Animal; Glyburide; Glycerol; Hypertonic Solutions; Infusions, Intravenous; KATP Channels; Ligation; Male; Microcirculation; Microscopy, Fluorescence; Neuroprotective Agents; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Papaverine; Pia Mater; Potassium Channel Blockers; Rats; Rats, Wistar; Regional Blood Flow; Vasodilation; Vasodilator Agents

2008