papaverine and diazepam

papaverine has been researched along with diazepam in 35 studies

Research

Studies (35)

TimeframeStudies, this research(%)All Research%
pre-199022 (62.86)18.7374
1990's1 (2.86)18.2507
2000's7 (20.00)29.6817
2010's5 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Caron, G; Ermondi, G1
Lombardo, F; Obach, RS; Waters, NJ1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Ahman, M; Holmén, AG; Wan, H1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Buckle, P; Jameson, D1
Lehne, RA; Smith, PA; Weight, FF1
Chan, YH; Curtis-Prior, PB; Jenner, M; McColl, I1
Georgiev, V1
King, RD; Stoelting, RK1
Kirby, RS; Lees, W; Vale, JA1
Smedley, MJ; Stanisstreet, M1
Distler, A; Fiegel, P; Hecking, E; Köhler, H; Port, FK1
Bovill, JG; Coppel, DL; Dundee, JW1
Hall, GM; Morgan, M; Whitwam, JG1
Dundee, JW; Haslett, WH1
Ferrero, A; Marzullo, C; Salmoiraghi, ML1
Arora, MV; Carson, IW; Clarke, RS; Dundee, JW; McCaughey, W1
Bovill, JG; Clarke, RS; Dundee, JW; Moore, J; Pandit, SK1
Dundee, JW; Loan, WB; Morrison, JD1
Clarke, RS; Dundee, JW; Knox, JW1
Mosler, KH2
Bednarík, B; Cerný, E; Lupínek, Z; Mitová, M; Mitová, P1
Jarvis, SM; Young, JD1
Katsuragi, T; Su, C1
MOSLER, KH; SCHWALM, H1
Cankaya, H; Içli, M; Kiriş, M; Kutluhan, A1
Aruna, J; Kumar, P; Kumar, S; Malhotra, N; Roy, KK; Sharma, JB1

Reviews

2 review(s) available for papaverine and diazepam

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016
Nucleoside transport in animal cells.
    Bioscience reports, 1983, Volume: 3, Issue:4

    Topics: Animals; Biological Transport, Active; Diazepam; Dilazep; Dipyridamole; Erythrocyte Membrane; Erythrocytes; Humans; Inosine; Kinetics; Membrane Proteins; Models, Molecular; Nucleosides; Papaverine; Species Specificity; Thioinosine; Uridine

1983

Trials

4 trial(s) available for papaverine and diazepam

ArticleYear
The taming of ketamine.
    Anaesthesia, 1973, Volume: 28, Issue:3

    Topics: Adjuvants, Anesthesia; Adult; Anesthesia, Intravenous; Atropine; Delirium; Diazepam; Dreams; Droperidol; Female; Fentanyl; Humans; Ketamine; Male; Opium; Papaverine; Postoperative Complications; Preanesthetic Medication; Scopolamine

1973
Some respiratory effects of althesin.
    British journal of anaesthesia, 1973, Volume: 45, Issue:6

    Topics: Anesthesia, Intravenous; Anesthetics; Atropine; Depression, Chemical; Diazepam; Female; Humans; Ketones; Papaverine; Preanesthetic Medication; Pregnanes; Respiration; Scopolamine

1973
Studies of drugs given before anaesthesia. XIV. Two benzodiazepine derivatives--chlordiazepoxide and diazepam.
    British journal of anaesthesia, 1968, Volume: 40, Issue:4

    Topics: Chlordiazepoxide; Clinical Trials as Topic; Diazepam; Female; Humans; Injections, Intramuscular; Morphine; Papaverine; Placebos; Preanesthetic Medication; Promazine; Promethazine; Tranquilizing Agents

1968
Comparison of efficacy of oral drotaverine plus mefenamic acid with paracervical block and with intravenous sedation for pain relief during hysteroscopy and endometrial biopsy.
    Indian journal of medical sciences, 2009, Volume: 63, Issue:6

    Topics: Adjuvants, Anesthesia; Adult; Analgesics; Anesthesia, Intravenous; Anesthesia, Obstetrical; Anesthetics, Intravenous; Diazepam; Drug Therapy, Combination; Endometrium; Female; Humans; Hypnotics and Sedatives; Hysteroscopy; Mefenamic Acid; Middle Aged; Pain Measurement; Papaverine; Pentazocine; Treatment Outcome; Young Adult

2009

Other Studies

29 other study(ies) available for papaverine and diazepam

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).
    Journal of medicinal chemistry, 2005, May-05, Volume: 48, Issue:9

    Topics: 1-Octanol; Alkanes; Hydrogen-Ion Concentration; Least-Squares Analysis; Mathematics; Models, Chemical; Models, Molecular; Solvents; Water

2005
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Relationship between brain tissue partitioning and microemulsion retention factors of CNS drugs.
    Journal of medicinal chemistry, 2009, Mar-26, Volume: 52, Issue:6

    Topics: Brain; Central Nervous System; Chromatography, Liquid; Emulsions; Mass Spectrometry

2009
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
A comparison of anti-inflammatory and other compounds on the spontaneously contracting pregnant rat uterus.
    The Journal of pharmacy and pharmacology, 1977, Volume: 29, Issue:2

    Topics: Animals; Anti-Inflammatory Agents; Chlorpromazine; Desipramine; Diazepam; Female; In Vitro Techniques; Ketamine; Muscle, Smooth; Papaverine; Pregnancy; Pregnancy, Animal; Rats; Uterine Contraction

1977
Potentiation of Ca2+-dependent K+ activation by theophylline is independent of cyclic nucleotide elevation.
    Nature, 1979, Aug-02, Volume: 280, Issue:5721

    Topics: Action Potentials; Animals; Anura; Bucladesine; Calcium; Diazepam; Dibutyryl Cyclic GMP; Methacholine Compounds; Nucleotides, Cyclic; Papaverine; Potassium; Rana catesbeiana; Sympathetic Nervous System; Theophylline

1979
Effects of several preoperative medications on fat cell lipolysis, and activity of adipose tissue cyclic AMP phosphodiesterase.
    Experientia, 1979, Nov-15, Volume: 35, Issue:11

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adipose Tissue; Animals; Atropine; Diazepam; Lipid Mobilization; Male; Meperidine; Papaverine; Promethazine; Rats; Scopolamine

1979
[Effects of imidazole, papaverine and theophylline on the picrotoxin convulsion-seizure threshold. The correlation with gamma-aminobutyric acid (GABA) and diazepam].
    Eksperimentalna meditsina i morfologiia, 1978, Volume: 17, Issue:3

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Drug Antagonism; Drug Interactions; gamma-Aminobutyric Acid; Imidazoles; Male; Mice; Papaverine; Picrotoxin; Seizures; Theophylline; Time Factors

1978
Aortocoronary vein graft flow in response to peripheral venous administration of sodium nitroprusside or diazepam.
    The Annals of thoracic surgery, 1977, Volume: 24, Issue:1

    Topics: Blood Pressure; Cardiopulmonary Bypass; Coronary Circulation; Diazepam; Ferricyanides; Humans; Male; Nitroprusside; Papaverine; Transplantation, Autologous; Veins

1977
Papaverine, benzodiazepines, and prolonged erections.
    Lancet (London, England), 1991, Jun-22, Volume: 337, Issue:8756

    Topics: Anxiety; Diazepam; Drug Interactions; Humans; Male; Middle Aged; Papaverine; Penile Erection; Priapism; Time Factors

1991
Calcium and neurulation in mammalian embryos. II. Effects of cytoskeletal inhibitors and calcium antagonists on the neural folds of rat embryos.
    Journal of embryology and experimental morphology, 1986, Volume: 93

    Topics: Animals; Benzimidazoles; Calcium; Calcium Channel Blockers; Cells, Cultured; Colchicine; Cytochalasin B; Diazepam; Embryo, Mammalian; Gallic Acid; Microscopy, Electron, Scanning; Nervous System; Nocodazole; Papaverine; Rats

1986
Priapism during regular haemodialysis.
    Lancet (London, England), 1974, Nov-30, Volume: 2, Issue:7892

    Topics: Adult; Chronic Disease; Diazepam; Glomerulonephritis; Heparin; Home Care Services; Humans; Infusions, Parenteral; Kidney Diseases; Male; Papaverine; Priapism; Pyelonephritis; Renal Dialysis; Saphenous Vein; Streptokinase; Time Factors; Tuberculosis, Renal

1974
[Intensive therapy of gestoses. Our experience in the years 1969-1971].
    Annali di ostetricia, ginecologia, medicina perinatale, 1971, Volume: 92, Issue:12

    Topics: Betamethasone; Brain Edema; Diazepam; Ergoloid Mesylates; Female; Furosemide; Humans; Mannitol; Papaverine; Phytotherapy; Plants, Medicinal; Pre-Eclampsia; Pregnancy; Rauwolfia; Thiopental

1971
Clinical studies of induction agents. XL. Althesin with various premedicants.
    British journal of anaesthesia, 1972, Volume: 44, Issue:8

    Topics: Anesthesia, Intravenous; Anesthetics; Atropine; Diazepam; Female; Humans; Hypotension; Ketones; Meperidine; Methohexital; Morphine; Movement; Nausea; Papaverine; Preanesthetic Medication; Pregnanes; Respiration; Respiratory Insufficiency; Scopolamine; Vomiting

1972
Clinical studies of induction agents. 38. Effect of premedicants and supplements on ketamine anaesthesia.
    British journal of anaesthesia, 1971, Volume: 43, Issue:6

    Topics: Adult; Analgesics; Anesthesia; Atropine; Benperidol; Blood Pressure; Cyclohexanes; Diazepam; Dreams; Female; Fentanyl; Heart Rate; Humans; Hypertension; Ketamine; Meperidine; Papaverine; Pentobarbital; Preanesthetic Medication; Promethazine; Scopolamine; Surgical Procedures, Operative

1971
Studies of drugs given before anaesthesia. XIX. The opiates.
    British journal of anaesthesia, 1970, Volume: 42, Issue:1

    Topics: Analgesics; Diazepam; Female; Fentanyl; Heroin; Humans; Levorphanol; Male; Meperidine; Methadone; Morphine; Papaverine; Phenazocine; Preanesthetic Medication; Vomiting

1970
The effect of dosage and premedication on the action of ketamine.
    British journal of anaesthesia, 1970, Volume: 42, Issue:9

    Topics: Analgesics; Anesthesia, General; Anesthetics; Atropine; Blood Pressure; Cyclohexanes; Delirium; Diazepam; Humans; Ketamine; Muscle Tonus; Papaverine; Preanesthetic Medication; Scopolamine

1970
[Problems of labor pain inhibition by pharmacological agents].
    Medizinische Klinik, 1969, Jan-24, Volume: 64, Issue:4

    Topics: Bronchodilator Agents; Chlordiazepoxide; Diazepam; Female; Halothane; Humans; Infant Mortality; Isoproterenol; Metaproterenol; Obstetric Labor, Premature; Papaverine; Phenethylamines; Pregnancy; Progesterone; Resorcinols; Sympathomimetics; Uterus; Vasodilator Agents

1969
Tocolysis.
    Bibliotheca gynaecologica, 1966, Volume: 42

    Topics: Animals; Chlordiazepoxide; Diazepam; Female; Guinea Pigs; Humans; In Vitro Techniques; Muscle Contraction; Papaverine; Pregnancy; Rats; Uterus; Vasodilator Agents

1966
[The effect of analgesics and psychopharmaceuticals on myocardial injury].
    Ceskoslovenska patologie, 1984, Volume: 20, Issue:4

    Topics: Aminopyrine; Animals; Barbiturates; Diazepam; Drug Combinations; Heart; Isoproterenol; Male; Morphine; Myocardium; Papaverine; Plant Extracts; Rats; Rats, Inbred Strains

1984
Possible selective inhibition of [3H]adenosine uptake by papaverine in vascular adrenergic nerves.
    European journal of pharmacology, 1982, Apr-08, Volume: 79, Issue:1-2

    Topics: Adenosine; Animals; Blood Vessels; Diazepam; Dipyridamole; Epinephrine; Male; Papaverine; Potassium Chloride; Pulmonary Artery; Rabbits; Sympathetic Nervous System

1982
[COMPARATIVE INVESTIGATIONS OF TOCOLYTIC AND RELAXANT SUBSTANCES IN THE ISOLATED UTERUS].
    Zentralblatt fur Gynakologie, 1965, May-01, Volume: 87

    Topics: Chlordiazepoxide; Diazepam; Female; Humans; Papaverine; Pharmacology; Rats; Research; Tocolytic Agents; Uterus; Vasodilator Agents

1965
Retrospective analysis of our cases with sudden hearing loss.
    The Journal of otolaryngology, 2003, Volume: 32, Issue:6

    Topics: Adolescent; Adult; Aged; Anti-Anxiety Agents; Anticoagulants; Audiometry, Pure-Tone; Auditory Threshold; Child; Dextrans; Diazepam; Drug Therapy, Combination; Female; Glucocorticoids; Hearing Loss, Sudden; Humans; Male; Methylprednisolone; Middle Aged; Papaverine; Pentoxifylline; Prognosis; Retrospective Studies; Risk Factors; Treatment Outcome; Vasodilator Agents

2003