papaverine and cimetidine

papaverine has been researched along with cimetidine in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-199010 (45.45)18.7374
1990's2 (9.09)18.2507
2000's4 (18.18)29.6817
2010's6 (27.27)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Lombardo, F; Obach, RS; Waters, NJ1
Ahlin, G; Artursson, P; Bergström, CA; Gustavsson, L; Karlsson, J; Larsson, R; Matsson, P; Norinder, U; Pedersen, JM1
Chupka, J; El-Kattan, A; Feng, B; Miller, HR; Obach, RS; Troutman, MD; Varma, MV1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
García-Mera, X; González-Díaz, H; Prado-Prado, FJ1
Afshari, CA; Eschenberg, M; Hamadeh, HK; Lee, PH; Lightfoot-Dunn, R; Morgan, RE; Qualls, CW; Ramachandran, B; Trauner, M; van Staden, CJ1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Afshari, CA; Chen, Y; Dunn, RT; Hamadeh, HK; Kalanzi, J; Kalyanaraman, N; Morgan, RE; van Staden, CJ1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1
Bruggeman, TM; Davenport, HW; Wood, JG1
Bonfilio, AC; Gray, S; Jacoby, HI; Staus, A; Thomas, C1
Bevan, JA; Bevan, RD; Vorkapic, P1
Chiba, S; Haruta, K; Homma, N; Horiuchi, A; Iwatsuki, K; Yonekura, H1
Kitagawa, H; Kohei, H; Nishiwaki, H; Takeda, F1
Burbridge, BE; Irving, HD1
Dohi, Y; Tajima, T1
Clark, BG; Vestal, RE1
Davenport, HW; Wood, JG1
Ichikawa, T; Naito, Y; Nakazawa, S; Tsukamoto, Y1
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH1
Gründemann, D; Haag, C; Honold, C; Koschker, AC; Schömig, E; Zimmermann, T1

Reviews

1 review(s) available for papaverine and cimetidine

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

21 other study(ies) available for papaverine and cimetidine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Structural requirements for drug inhibition of the liver specific human organic cation transport protein 1.
    Journal of medicinal chemistry, 2008, Oct-09, Volume: 51, Issue:19

    Topics: Cell Line; Computer Simulation; Drug Design; Gene Expression Profiling; Humans; Hydrogen Bonding; Liver; Molecular Weight; Organic Cation Transporter 1; Pharmaceutical Preparations; Predictive Value of Tests; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Structure-Activity Relationship

2008
Physicochemical determinants of human renal clearance.
    Journal of medicinal chemistry, 2009, Aug-13, Volume: 52, Issue:15

    Topics: Humans; Hydrogen Bonding; Hydrogen-Ion Concentration; Hydrophobic and Hydrophilic Interactions; Kidney; Metabolic Clearance Rate; Molecular Weight

2009
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010
Multi-target spectral moment QSAR versus ANN for antiparasitic drugs against different parasite species.
    Bioorganic & medicinal chemistry, 2010, Mar-15, Volume: 18, Issue:6

    Topics: Antiparasitic Agents; Molecular Structure; Neural Networks, Computer; Parasitic Diseases; Quantitative Structure-Activity Relationship; Species Specificity; Thermodynamics

2010
Interference with bile salt export pump function is a susceptibility factor for human liver injury in drug development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2010, Volume: 118, Issue:2

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Assay; Biological Transport; Cell Line; Cell Membrane; Chemical and Drug Induced Liver Injury; Cytoplasmic Vesicles; Drug Evaluation, Preclinical; Humans; Liver; Rats; Reproducibility of Results; Spodoptera; Transfection; Xenobiotics

2010
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
A multifactorial approach to hepatobiliary transporter assessment enables improved therapeutic compound development.
    Toxicological sciences : an official journal of the Society of Toxicology, 2013, Volume: 136, Issue:1

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Biological Transport; Chemical and Drug Induced Liver Injury; Cluster Analysis; Drug-Related Side Effects and Adverse Reactions; Humans; Liver; Male; Multidrug Resistance-Associated Proteins; Pharmacokinetics; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Risk Assessment; Risk Factors; Toxicity Tests

2013
Local control of blood flow in the dog's stomach: vasodilatation caused by acid back-diffusion following topical application of salicylic acid.
    Gastroenterology, 1979, Volume: 77, Issue:4 Pt 1

    Topics: Animals; Atropine; Capillary Permeability; Cimetidine; Diffusion; Dogs; Histamine; Hydrochloric Acid; Hydrogen-Ion Concentration; Papaverine; Perfusion; Pyrilamine; Salicylates; Stomach; Vasodilation

1979
Antisecretory actions of aminophylline in the rat and dog.
    Digestion, 1979, Volume: 19, Issue:4

    Topics: Aminophylline; Animals; Cimetidine; Deoxyglucose; Dogs; Dose-Response Relationship, Drug; Female; Gastric Juice; Gastrins; Histamine; Imidazoles; Papaverine; Rats; Secretory Rate; Tetragastrin; Xanthines

1979
Pharmacologic irreversible narrowing in chronic cerebrovasospasm in rabbits is associated with functional damage.
    Stroke, 1990, Volume: 21, Issue:10

    Topics: Acetylcholine; Animals; Basilar Artery; Cimetidine; Epinephrine; Histamine; In Vitro Techniques; Ischemic Attack, Transient; Papaverine; Prazosin; Rabbits; Serotonin; Subarachnoid Hemorrhage; Tetrodotoxin; Vasoconstriction

1990
Effects of DN-9693, a synthesized phosphodiesterase inhibitor, on pancreatic exocrine secretion in dogs.
    Japanese journal of pharmacology, 1989, Volume: 49, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Atropine; Cholecystokinin; Cimetidine; Dogs; Dose-Response Relationship, Drug; Female; Male; Pancreas; Pancreatic Juice; Papaverine; Phentolamine; Phosphodiesterase Inhibitors; Propranolol; Quinazolines; Secretin; Sulpiride; Theophylline

1989
Roles of gastric acid secretion and motility in gastric mucosal lesion formation induced by water-immersion stress in rats.
    Scandinavian journal of gastroenterology. Supplement, 1989, Volume: 162

    Topics: Animals; Cimetidine; Gastric Acid; Gastric Mucosa; Gastrointestinal Motility; Immersion; Male; Papaverine; Rats; Rats, Inbred Strains; Stress, Physiological

1989
Incompatibility of contrast agents with intravascular medications. Work in progress.
    Radiology, 1989, Volume: 173, Issue:1

    Topics: Chemical Precipitation; Cimetidine; Contrast Media; Diatrizoate Meglumine; Diphenhydramine; Drug Incompatibility; Gentamicins; In Vitro Techniques; Infusions, Intravenous; Iohexol; Iopamidol; Iothalamate Meglumine; Ioxaglic Acid; Papaverine; Pharmaceutical Preparations; Protamines; Spectrophotometry

1989
Histamine induced or enhanced delayed afterdepolarization and triggered activity in guinea-pig papillary muscles. A preliminary study.
    Japanese heart journal, 1985, Volume: 26, Issue:6

    Topics: Action Potentials; Animals; Cimetidine; Cyclic AMP; Diphenhydramine; Electrophysiology; Guinea Pigs; Histamine; Histamine Antagonists; Imidazoles; In Vitro Techniques; Microelectrodes; Papaverine; Papillary Muscles; Receptors, Histamine H2

1985
Adverse drug reactions in the elderly: case studies.
    Geriatrics, 1984, Volume: 39, Issue:12

    Topics: Acetazolamide; Aged; Anemia, Hemolytic; Bromocriptine; Captopril; Chlorpropamide; Cimetidine; Clonidine; Dienestrol; Drug-Related Side Effects and Adverse Reactions; Female; Humans; Hydralazine; Lung Diseases; Male; Middle Aged; Nitrofurantoin; Pancreatitis; Papaverine; Peripheral Nervous System Diseases; Procainamide; Propranolol; Sulindac; Theophylline; Timolol

1984
Measurement of canine gastric vascular permeability to plasma proteins in the normal and protein-losing states.
    Gastroenterology, 1982, Volume: 82, Issue:4

    Topics: Animals; Blood Proteins; Capillary Permeability; Cimetidine; Dithiothreitol; Dogs; Fibrinogen; Gastric Mucosa; Histamine; Histamine Antagonists; Papaverine; Protein-Losing Enteropathies; Pyrilamine; Salicylates; Salicylic Acid; Serum Albumin, Radio-Iodinated

1982
Effect of histamine on the gastric smooth muscles of guinea pig.
    Digestion, 1981, Volume: 22, Issue:4

    Topics: Acetylcholine; Animals; Cimetidine; Guinea Pigs; Histamine; Male; Muscle Contraction; Muscle, Smooth; Papaverine; Pyrilamine; Receptors, Histamine H1; Receptors, Histamine H2; Stomach

1981
Characterization and function of histamine receptors in corpus cavernosum.
    The Journal of urology, 1995, Volume: 153, Issue:2

    Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles

1995
Activation of the extraneuronal monoamine transporter (EMT) from rat expressed in 293 cells.
    British journal of pharmacology, 2002, Volume: 137, Issue:6

    Topics: 1-Methyl-4-phenylpyridinium; Animals; Biological Transport; Cell Line; Cimetidine; Cloning, Molecular; Corticosterone; Dose-Response Relationship, Drug; Gene Expression; Genetic Vectors; Humans; Imidazoles; Kinetics; Mice; Norepinephrine; Organic Cation Transport Proteins; Papaverine; Piperidines; Quinolines; Rats; Thiourea; Transfection; Tritium

2002