pak 104p has been researched along with verlukast in 4 studies
Studies (pak 104p) | Trials (pak 104p) | Recent Studies (post-2010) (pak 104p) | Studies (verlukast) | Trials (verlukast) | Recent Studies (post-2010) (verlukast) |
---|---|---|---|---|---|
16 | 0 | 0 | 396 | 14 | 115 |
Protein | Taxonomy | pak 104p (IC50) | verlukast (IC50) |
---|---|---|---|
Multidrug resistance-associated protein 1 | Homo sapiens (human) | 2.8 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 2 (50.00) | 18.2507 |
2000's | 2 (50.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Akiyama, SI; Chen, ZS; Furukawa, T; Ono, K; Seto, K; Sumizawa, T; Ueda, K | 1 |
Akiyama, SI; Aoki, S; Chen, ZS; Furukawa, T; Kawabe, T; Kuwano, M; Ono, M; Sumizawa, T; Uchiumi, T; Wada, M | 1 |
Garnier-Suillerot, A; Salerno, M | 1 |
Garnier-Suillerot, A; Loechariyakul, P; Saengkhae, C; Salerno, M | 1 |
4 other study(ies) available for pak 104p and verlukast
Article | Year |
---|---|
ATP-Dependent efflux of CPT-11 and SN-38 by the multidrug resistance protein (MRP) and its inhibition by PAK-104P.
Topics: Adenosine Triphosphate; Anion Transport Proteins; Antineoplastic Agents, Phytogenic; ATP-Binding Cassette Transporters; Biological Transport; Buthionine Sulfoximine; Camptothecin; Carrier Proteins; Cell Line; Cell Survival; Culture Media; Cyclic P-Oxides; DNA Topoisomerases, Type I; Drug Resistance, Multiple; Glutathione S-Transferase pi; Glutathione Transferase; Humans; Irinotecan; Isoenzymes; KB Cells; Multidrug Resistance-Associated Proteins; Nicotinic Acids; Propionates; Quinolines | 1999 |
Effect of multidrug resistance-reversing agents on transporting activity of human canalicular multispecific organic anion transporter.
Topics: Adenosine Triphosphate; Animals; Anion Transport Proteins; Antineoplastic Agents; Biological Transport; Carrier Proteins; Cells, Cultured; Cyclic P-Oxides; Cyclosporine; Drug Interactions; Drug Resistance, Multiple; Glutathione; Humans; Kinetics; Leukotriene C4; Nicotinic Acids; Osmolar Concentration; Propionates; Quinolines; Swine; Transfection; Tritium; Vincristine | 1999 |
Kinetics of glutathione and daunorubicin efflux from multidrug resistance protein overexpressing small-cell lung cancer cells.
Topics: ATP-Binding Cassette Transporters; Biological Transport; Carcinoma, Small Cell; Cyclic P-Oxides; Daunorubicin; Dose-Response Relationship, Drug; Extracellular Space; Gene Expression Regulation, Neoplastic; Glutathione; Humans; K562 Cells; Kinetics; Lung Neoplasms; Multidrug Resistance-Associated Proteins; Nicotinic Acids; Propionates; Quinolines; Time Factors; Tumor Cells, Cultured; Vinblastine | 2001 |
Relation between the ability of some compounds to modulate the MRP1-mediated efflux of glutathione and to inhibit the MRPl-mediated efflux of daunorubicin.
Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cyclic P-Oxides; Daunorubicin; Glutathione; Humans; Nicotinic Acids; Propionates; Quinolines; Tumor Cells, Cultured; Verapamil | 2004 |