Page last updated: 2024-09-03

pak 104p and verlukast

pak 104p has been researched along with verlukast in 4 studies

Compound Research Comparison

Studies
(pak 104p)
Trials
(pak 104p)
Recent Studies (post-2010)
(pak 104p)
Studies
(verlukast)
Trials
(verlukast)
Recent Studies (post-2010) (verlukast)
160039614115

Protein Interaction Comparison

ProteinTaxonomypak 104p (IC50)verlukast (IC50)
Multidrug resistance-associated protein 1 Homo sapiens (human)2.8

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (50.00)18.2507
2000's2 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Akiyama, SI; Chen, ZS; Furukawa, T; Ono, K; Seto, K; Sumizawa, T; Ueda, K1
Akiyama, SI; Aoki, S; Chen, ZS; Furukawa, T; Kawabe, T; Kuwano, M; Ono, M; Sumizawa, T; Uchiumi, T; Wada, M1
Garnier-Suillerot, A; Salerno, M1
Garnier-Suillerot, A; Loechariyakul, P; Saengkhae, C; Salerno, M1

Other Studies

4 other study(ies) available for pak 104p and verlukast

ArticleYear
ATP-Dependent efflux of CPT-11 and SN-38 by the multidrug resistance protein (MRP) and its inhibition by PAK-104P.
    Molecular pharmacology, 1999, Volume: 55, Issue:5

    Topics: Adenosine Triphosphate; Anion Transport Proteins; Antineoplastic Agents, Phytogenic; ATP-Binding Cassette Transporters; Biological Transport; Buthionine Sulfoximine; Camptothecin; Carrier Proteins; Cell Line; Cell Survival; Culture Media; Cyclic P-Oxides; DNA Topoisomerases, Type I; Drug Resistance, Multiple; Glutathione S-Transferase pi; Glutathione Transferase; Humans; Irinotecan; Isoenzymes; KB Cells; Multidrug Resistance-Associated Proteins; Nicotinic Acids; Propionates; Quinolines

1999
Effect of multidrug resistance-reversing agents on transporting activity of human canalicular multispecific organic anion transporter.
    Molecular pharmacology, 1999, Volume: 56, Issue:6

    Topics: Adenosine Triphosphate; Animals; Anion Transport Proteins; Antineoplastic Agents; Biological Transport; Carrier Proteins; Cells, Cultured; Cyclic P-Oxides; Cyclosporine; Drug Interactions; Drug Resistance, Multiple; Glutathione; Humans; Kinetics; Leukotriene C4; Nicotinic Acids; Osmolar Concentration; Propionates; Quinolines; Swine; Transfection; Tritium; Vincristine

1999
Kinetics of glutathione and daunorubicin efflux from multidrug resistance protein overexpressing small-cell lung cancer cells.
    European journal of pharmacology, 2001, Jun-01, Volume: 421, Issue:1

    Topics: ATP-Binding Cassette Transporters; Biological Transport; Carcinoma, Small Cell; Cyclic P-Oxides; Daunorubicin; Dose-Response Relationship, Drug; Extracellular Space; Gene Expression Regulation, Neoplastic; Glutathione; Humans; K562 Cells; Kinetics; Lung Neoplasms; Multidrug Resistance-Associated Proteins; Nicotinic Acids; Propionates; Quinolines; Time Factors; Tumor Cells, Cultured; Vinblastine

2001
Relation between the ability of some compounds to modulate the MRP1-mediated efflux of glutathione and to inhibit the MRPl-mediated efflux of daunorubicin.
    Biochemical pharmacology, 2004, Dec-01, Volume: 68, Issue:11

    Topics: Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cyclic P-Oxides; Daunorubicin; Glutathione; Humans; Nicotinic Acids; Propionates; Quinolines; Tumor Cells, Cultured; Verapamil

2004