Page last updated: 2024-09-03

pagoclone and flumazenil

pagoclone has been researched along with flumazenil in 3 studies

Compound Research Comparison

Studies
(pagoclone)
Trials
(pagoclone)
Recent Studies (post-2010)
(pagoclone)
Studies
(flumazenil)
Trials
(flumazenil)
Recent Studies (post-2010) (flumazenil)
13444,673426981

Protein Interaction Comparison

ProteinTaxonomypagoclone (IC50)flumazenil (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-1Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit beta-1Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit alpha-2Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit alpha-3Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-4Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit gamma-2Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0038
GABA theta subunitRattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0038

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (33.33)18.2507
2000's2 (66.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Jackson, HC; Nutt, DJ; Ramsay, E1
Feeney, A; Grasby, PG; Lingford-Hughes, A; Nutt, DJ; Wilson, SJ1
Atack, JR; Blackaby, WP; Cook, SM; Dawson, GR; Goodacre, SC; Lewis, RT; Lincoln, R; Marshall, G; McKernan, RM; Pike, A; Reynolds, DS; Stanley, J; Wafford, KA1

Trials

1 trial(s) available for pagoclone and flumazenil

ArticleYear
A proof-of-concept study using [11C]flumazenil PET to demonstrate that pagoclone is a partial agonist.
    Psychopharmacology, 2005, Volume: 180, Issue:4

    Topics: Area Under Curve; Brain; Carbon Isotopes; Drug Interactions; Flumazenil; GABA Modulators; Humans; Isoindoles; Lorazepam; Male; Naphthyridines; Positron-Emission Tomography

2005

Other Studies

2 other study(ies) available for pagoclone and flumazenil

ArticleYear
Effect of the cyclopyrrolones suriclone and RP 59037 on body temperature in mice.
    European journal of pharmacology, 1992, May-27, Volume: 216, Issue:1

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Benzodiazepines; Body Temperature; Carbolines; Drug Interactions; Flumazenil; Indoles; Isoindoles; Male; Mice; Naphthyridines; Piperazines; Receptors, GABA-A; Sulfur Compounds

1992
The in vivo properties of pagoclone in rat are most likely mediated by 5'-hydroxy pagoclone.
    Neuropharmacology, 2006, Volume: 50, Issue:6

    Topics: Animals; Behavior, Animal; Binding Sites; Brain; Cell Line; Dose-Response Relationship, Drug; Fibroblasts; Flumazenil; GABA Modulators; Humans; Indoles; Isoindoles; Isomerism; Male; Maze Learning; Mice; Motor Activity; Naphthyridines; Protein Subunits; Psychomotor Performance; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Time Factors; Tritium

2006