Page last updated: 2024-08-23

paclitaxel and vx680

paclitaxel has been researched along with vx680 in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (20.00)29.6817
2010's4 (80.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Morioka, M1
Benigno, BB; Laycock, N; Logani, S; McDonald, JF; Moreno, CS; Osunkoya, AO; Scharer, CD1
Bak, A; Bush, TL; Cee, VJ; Chung, G; Deak, HL; Dussault, I; Eden, P; Geuns-Meyer, S; Hodous, BL; Kendall, RL; McElroy, P; Nguyen, HN; Olivieri, PR; Patel, VF; Payton, M; Radinsky, R; Romero, K; Ross, S; Schenkel, LB; Stanton, M; Ziegler, B1
Deng, X; Gray, N; Huang, HC; Kwiatkowski, N; Mitchison, T; Musacchio, A; Santaguida, S; Tan, L; Villa, F; Wang, J1
Huang, D; Murray, GF; Reed, J; Roy, IJ; Teitell, MA; Zangle, TA1

Other Studies

5 other study(ies) available for paclitaxel and vx680

ArticleYear
3-Cyano-6-(5-methyl-3-pyrazoloamino) pyridines (Part 2): A dual inhibitor of Aurora kinase and tubulin polymerization.
    Bioorganic & medicinal chemistry letters, 2016, 12-15, Volume: 26, Issue:24

    Topics: Aminopyridines; Animals; Antineoplastic Agents; Aurora Kinases; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; HCT116 Cells; Humans; Mice; Molecular Structure; Neoplasms, Experimental; Polymerization; Protein Kinase Inhibitors; Pyrazoles; Structure-Activity Relationship; Tubulin

2016
Aurora kinase inhibitors synergize with paclitaxel to induce apoptosis in ovarian cancer cells.
    Journal of translational medicine, 2008, Dec-11, Volume: 6

    Topics: Aged; Animals; Antineoplastic Agents, Phytogenic; Apoptosis; Aurora Kinases; Cell Line, Tumor; Drug Resistance, Neoplasm; Drug Synergism; Drug Therapy, Combination; Female; Gene Expression Profiling; Humans; Middle Aged; Oligonucleotide Array Sequence Analysis; Ovarian Neoplasms; Paclitaxel; Piperazines; Protein Serine-Threonine Kinases

2008
Preclinical evaluation of AMG 900, a novel potent and highly selective pan-aurora kinase inhibitor with activity in taxane-resistant tumor cell lines.
    Cancer research, 2010, Dec-01, Volume: 70, Issue:23

    Topics: Adult; Animals; Aurora Kinase A; Aurora Kinase B; Aurora Kinases; Benzamides; Cell Line, Tumor; Cell Proliferation; Clinical Trials as Topic; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Resistance, Neoplasm; Female; HCT116 Cells; HeLa Cells; Histones; Humans; Mice; Mice, Nude; Mutation; Neoplasms; Organophosphates; Paclitaxel; Phosphorylation; Phthalazines; Piperazines; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyrazoles; Quinazolines; Xenograft Model Antitumor Assays

2010
Selective aurora kinase inhibitors identified using a taxol-induced checkpoint sensitivity screen.
    ACS chemical biology, 2012, Jan-20, Volume: 7, Issue:1

    Topics: Animals; Antineoplastic Agents, Phytogenic; Antineoplastic Combined Chemotherapy Protocols; Aurora Kinase B; Aurora Kinases; Benzazepines; Cell Line, Tumor; Cell Survival; Crystallography, X-Ray; High-Throughput Screening Assays; Humans; Inhibitory Concentration 50; Isoenzymes; M Phase Cell Cycle Checkpoints; Models, Molecular; Organophosphates; Paclitaxel; Piperazines; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Pyrimidines; Quinazolines; Structure-Activity Relationship; Xenopus laevis

2012
Identifying fates of cancer cells exposed to mitotic inhibitors by quantitative phase imaging.
    The Analyst, 2019, Dec-16, Volume: 145, Issue:1

    Topics: Antineoplastic Agents; Aurora Kinase A; Cell Line, Tumor; Colchicine; Humans; Mitosis; Paclitaxel; Piperazines; Proof of Concept Study; Protein Kinase Inhibitors; Tubulin Modulators

2019
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