Page last updated: 2024-08-23

paclitaxel and pi103

paclitaxel has been researched along with pi103 in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (20.00)29.6817
2010's3 (60.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Hayakawa, M; Kaizawa, H; Kawaguchi, K; Koizumi, T; Ohishi, T; Ohta, M; Okada, M; Parker, P; Raynaud, FI; Tsukamoto, S; Waterfield, MD; Workman, P; Yamano, M1
Chen, Y; Han, J; Liu, T; Song, Y; Wang, M; Xu, H; Yang, C; Zhang, L; Zheng, C; Zhu, J1
Dilasser, F; Dubreuil, D; Le Gall, E; Le Guével, R; Lebreton, J; Léonel, E; Loirand, G; Martens, T; Pipelier, M; Rousselle, M; Sauzeau, V; Sengmany, S; Sitter, M1
Gu, D; Hu, Y; Ma, X; Sheng, R; Wang, C; Wei, J1
Hou, Y; Kuang, W; Min, W; Sun, C; Wang, L; Wang, X; Wang, Y; Xia, F; Yang, P; Yuan, K; Zhang, F; Zhang, H; Zhu, Y1

Other Studies

5 other study(ies) available for paclitaxel and pi103

ArticleYear
Synthesis and biological evaluation of sulfonylhydrazone-substituted imidazo[1,2-a]pyridines as novel PI3 kinase p110alpha inhibitors.
    Bioorganic & medicinal chemistry, 2007, Sep-01, Volume: 15, Issue:17

    Topics: Animals; Cell Line, Tumor; Cell Proliferation; Enzyme Activation; Humans; Hydrazones; Imidazoles; Inhibitory Concentration 50; Isoenzymes; Mice; Molecular Structure; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase Inhibitors; Protein Subunits; Pyridines; Structure-Activity Relationship; Sulfur; Temperature; Xenograft Model Antitumor Assays

2007
Structure-based optimization leads to the discovery of NSC765844, a highly potent, less toxic and orally efficacious dual PI3K/mTOR inhibitor.
    European journal of medicinal chemistry, 2016, Oct-21, Volume: 122

    Topics: Administration, Oral; Amino Acid Sequence; Animals; Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Drug Design; Enzyme Inhibitors; Humans; Male; Models, Molecular; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Conformation; Rats; Signal Transduction; Structure-Activity Relationship; Sulfonamides; TOR Serine-Threonine Kinases; Xenograft Model Antitumor Assays

2016
Synthesis and biological evaluation of 3-amino-, 3-alkoxy- and 3-aryloxy-6-(hetero)arylpyridazines as potent antitumor agents.
    Bioorganic & medicinal chemistry letters, 2019, 03-01, Volume: 29, Issue:5

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Drug Screening Assays, Antitumor; Humans; Pyridazines

2019
Design, synthesis and biological evaluation of novel benzothiadiazine derivatives as potent PI3Kδ-selective inhibitors for treating B-cell-mediated malignancies.
    European journal of medicinal chemistry, 2019, May-15, Volume: 170

    Topics: Administration, Oral; Animals; Antineoplastic Agents; B-Lymphocytes; Benzothiadiazines; Cell Line, Tumor; Cell Proliferation; Class I Phosphatidylinositol 3-Kinases; Drug Design; Lymphoma, B-Cell; Molecular Docking Simulation; Protein Kinase Inhibitors; Rats, Sprague-Dawley

2019
Discovery of Novel Phosphoinositide-3-Kinase α Inhibitors with High Selectivity, Excellent Bioavailability, and Long-Acting Efficacy for Gastric Cancer.
    Journal of medicinal chemistry, 2022, 07-28, Volume: 65, Issue:14

    Topics: Antineoplastic Agents; Biological Availability; Cell Line, Tumor; Cell Proliferation; Humans; Phosphatidylinositol 3-Kinases; Phosphatidylinositols; Phosphoinositide-3 Kinase Inhibitors; Stomach Neoplasms; Structure-Activity Relationship

2022