Compounds > oxophenylarsine

oxophenylarsine and pentamidine

oxophenylarsine has been researched along with pentamidine in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (10.00)18.2507
2000's2 (20.00)29.6817
2010's5 (50.00)24.3611
2020's2 (20.00)2.80

Authors

AuthorsStudies
Brun, R; de Koning, HP; Gould, M; Kaiser, M; Koomen, GJ; Rodenko, B; van der Burg, AM; Wanner, MJ1
Al-Salabi, MI; Ali, JA; de Koning, HP; El-Sabbagh, N; Ho, W; Ibrahim, HM; Koomen, GJ; Rodenko, B; Teka, IA; Wanner, MJ1
Alkorta, I; Dardonville, C; de Koning, HP; Ebiloma, GU; Nué Martínez, JJ; Ríos Martínez, CH1
Balogun, EO; Bruggeman, V; Dardonville, C; de Koning, HP; Donachie, A; Ebiloma, GU; Fueyo González, FJ; Harada, S; Inaoka, DK; Izquierdo García, C; Kita, K; Sánchez Villamañán, JM; Shiba, T1
Ayuga, TD; Balogun, EO; Dardonville, C; de Koning, HP; Donachie, A; Ebiloma, GU; Gil, LA; Harada, S; Herraiz, T; Inaoka, DK; Kaiser, M; Kita, K; Shiba, T1
Alhejely, AS; Arai, N; Balogun, EO; Cueto-Díaz, EJ; Dardonville, C; de Koning, HP; Ebiloma, GU; Harada, S; Martín-Domínguez, A; Martínez-Benayas, I; Matsui, M; Meco-Navas, A; Saito, M; Shiba, T1
Alfayez, IA; Cueto-Díaz, EJ; Dardonville, C; de Koning, HP; Ebiloma, GU; Fueyo-González, FJ; Giron, MD; González-García, MC; González-Vera, JA; Lemgruber, L; Orte, A; Ruedas Rama, MJ; Salto, R; Shiba, T; Ungogo, MA1
Aldfer, MM; Arai, N; Bernal-Fraile, T; Chevillard, R; Cisneros, D; Cueto-Díaz, EJ; Dardonville, C; de Koning, HP; Ebiloma, GU; Elati, HAA; Kojima, C; López-Sastre, R; Matsushiro, S; Medina-Gil, T; Otani, M; Shiba, T; Ungogo, MA1
Scott, AG; Tait, A; Turner, CM1
Barrett, MP; Brun, R; Burchmore, RJ; de Koning, HP; Enyaru, JC; Geiser, F; Kaminsky, R; Mäser, P; Matovu, E; Seebeck, T; Stewart, ML; Wallace, LJ1

Other Studies

10 other study(ies) available for oxophenylarsine and pentamidine

ArticleYear
2,N6-disubstituted adenosine analogs with antitrypanosomal and antimalarial activities.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:11

    Topics: Adenosine; Animals; Antimalarials; Dose-Response Relationship, Drug; Molecular Structure; Plasmodium falciparum; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma cruzi

2007
Synthesis of marine-derived 3-alkylpyridinium alkaloids with potent antiprotozoal activity.
    ACS medicinal chemistry letters, 2011, Dec-08, Volume: 2, Issue:12

    Topics:

2011
Lowering the pKa of a bisimidazoline lead with halogen atoms results in improved activity and selectivity against Trypanosoma brucei in vitro.
    European journal of medicinal chemistry, 2015, Aug-28, Volume: 101

    Topics: Cell Survival; Dose-Response Relationship, Drug; Halogens; HEK293 Cells; Humans; Hydrogen-Ion Concentration; Imidazolines; Molecular Structure; Parasitic Sensitivity Tests; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma cruzi

2015
Conjugates of 2,4-Dihydroxybenzoate and Salicylhydroxamate and Lipocations Display Potent Antiparasite Effects by Efficiently Targeting the Trypanosoma brucei and Trypanosoma congolense Mitochondrion.
    Journal of medicinal chemistry, 2017, 02-23, Volume: 60, Issue:4

    Topics: Cell Line; Drug Discovery; Humans; Hydroxybenzoates; Membrane Potential, Mitochondrial; Mitochondria; Salicylamides; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosoma congolense; Trypanosomiasis, African

2017
Inhibition of trypanosome alternative oxidase without its N-terminal mitochondrial targeting signal (ΔMTS-TAO) by cationic and non-cationic 4-hydroxybenzoate and 4-alkoxybenzaldehyde derivatives active against T. brucei and T. congolense.
    European journal of medicinal chemistry, 2018, Apr-25, Volume: 150

    Topics: Benzaldehydes; Cations; Dose-Response Relationship, Drug; Mitochondrial Proteins; Molecular Structure; Oxidoreductases; Parabens; Parasitic Sensitivity Tests; Plant Proteins; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma; Trypanosoma brucei brucei; Trypanosoma congolense

2018
SAR of 4-Alkoxybenzoic Acid Inhibitors of the Trypanosome Alternative Oxidase.
    ACS medicinal chemistry letters, 2018, Sep-13, Volume: 9, Issue:9

    Topics:

2018
Synthesis, biological, and photophysical studies of molecular rotor-based fluorescent inhibitors of the trypanosome alternative oxidase.
    European journal of medicinal chemistry, 2021, Aug-05, Volume: 220

    Topics: Cell Survival; Cells, Cultured; Density Functional Theory; Dose-Response Relationship, Drug; Enzyme Inhibitors; Fluorescent Dyes; HEK293 Cells; Humans; Microscopy, Fluorescence; Mitochondrial Proteins; Molecular Structure; Optical Imaging; Oxidoreductases; Plant Proteins; Structure-Activity Relationship; Trypanosoma; Trypanosoma brucei brucei

2021
Imidazoline- and Benzamidine-Based Trypanosome Alternative Oxidase Inhibitors: Synthesis and Structure-Activity Relationship Studies.
    ACS medicinal chemistry letters, 2022, Feb-10, Volume: 13, Issue:2

    Topics:

2022
Trypanosoma brucei: lack of cross-resistance to melarsoprol in vitro by cymelarsan-resistant parasites.
    Experimental parasitology, 1997, Volume: 86, Issue:3

    Topics: Adenine; Adenosine; Animals; Arsenicals; Diminazene; Dose-Response Relationship, Drug; Drug Resistance; Enzyme Inhibitors; Female; Inosine; Melarsoprol; Mice; Pentamidine; Trypanocidal Agents; Trypanosoma brucei brucei

1997
Mechanisms of arsenical and diamidine uptake and resistance in Trypanosoma brucei.
    Eukaryotic cell, 2003, Volume: 2, Issue:5

    Topics: Adenine; Adenosine; Animals; Arsenicals; Benzamidines; Cell Death; Cell Division; Diminazene; Drug Resistance; Female; Gene Silencing; Hypoxanthine; Inhibitory Concentration 50; Inosine; Melarsoprol; Mice; Mutation; Nucleoside Transport Proteins; Pentamidine; Stilbamidines; Trypanosoma brucei brucei

2003