oxazoles has been researched along with yohimbine in 38 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 11 (28.95) | 18.7374 |
1990's | 19 (50.00) | 18.2507 |
2000's | 7 (18.42) | 29.6817 |
2010's | 1 (2.63) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Gundlach, AL; Jarrott, B; King, PR; Louis, WJ | 1 |
Coupry, I; Lachaud, V; Limon, I; Parini, A; Tesson, F | 1 |
Deckert, V; Elghozi, JL; Lachaud, V; Parini, A | 1 |
Bousquet, P; Feldman, J; Gonon, F; Mermet, C; Monassier, L; Tibiriça, E | 1 |
Belcourt, A; Bousquet, P; Bricca, G; Dontenwill, M; Feldman, J | 1 |
Hamilton, CA; Howie, CA; Jardine, E; Reid, JL; Yakubu, MA | 1 |
Belcourt, A; Bousquet, P; Bricca, G; Dontenwill, M; Feldman, J; Tibiriça, E | 1 |
Dresse, A; Scuvée-Moreau, J | 1 |
Coupry, I; Koenig, E; Lachaud, V; Parini, A; Podevin, RA | 2 |
Bidet, M; Coupry, I; Lachaud, V; Parini, A; Podevin, RA; Poujeol, P | 1 |
Carenzi, A; Chiarino, D; Napoletano, M; Reggiani, A; Sala, A; Sala, R | 1 |
Bourreau, JP; Tricoche, R | 1 |
Herman, AG; Jordaens, FH; Verbeuren, TJ; Zonnekeyn, LL | 1 |
Bourin, M; Colombel, MC; Creuzet, MH; Jarry, C | 1 |
de Jonge, A; Innemee, HC; Timmermans, PB; van Meel, JC; van Zwieten, PA | 1 |
Timmermans, PB; Van Zwieten, PA | 2 |
Szabo, B; Urban, R | 2 |
Starke, K; Szabo, B; Urban, R | 1 |
Hayashi, Y; Kamibayashi, T; Mammoto, T; Takada, K; Yamatodani, A; Yoshiya, I | 1 |
Boucher, M; Chapuy, E; Chassaing, C; Dubar, M | 1 |
Chayvialle, JA; Chéry-Croze, S; Détolle-Sarbach, S; Guez, D; Miampamba, M | 1 |
Boulanger, CM; Illiano, S; Marsault, R; Taddei, S; Vanhoutte, PM | 1 |
Chu, TC; Gluchowski, C; Hughes, BW; Potter, DE; Wong, W | 1 |
Avellar, MC; Markus, RP | 1 |
Bock, C; Niederhoffer, N; Szabo, B | 1 |
Bousquet, P; Brasili, L; Bruban, V; Dontenwill, M; Feldman, J; Giannella, M; Greney, H; Pigini, M | 1 |
Bock, C; Niederhoffer, N; Nordheim, U; Szabo, B | 1 |
Artigues-Varin, C; Mulder, P; Richard, V; Thuillez, C; Varin, R | 1 |
Ernsberger, P; Koletsky, RJ; Velliquette, RA | 1 |
Burgdorf, C; Engelhardt, A; Kurz, T; Raasch, W; Richardt, G; Schäfer, U | 1 |
Abelson, KS; Höglund, AU | 1 |
Merwid-Lad, A; Misiuk-Hojło, M; Pieśniewska, M; Szaliński, M; Trocha, M | 1 |
de Arruda Camargo, LA; Guarda, IF; Guarda, RS; Saad, WA; Simões, S | 1 |
Khansefid, N; Ladgevardi, MA; Sabetkasaie, M | 1 |
Goeders, NE; Runyon, SP; Schmoutz, CD; Zhang, Y | 1 |
38 other study(ies) available for oxazoles and yohimbine
Article | Year |
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Nature of [3H]rilmenidine binding to membranes of rat cerebral cortex.
Topics: Adrenergic alpha-Agonists; Amiloride; Animals; Binding Sites; Catecholamines; Cell Membrane; Cerebral Cortex; Guanidine; Guanidines; Imidazoles; Oxazoles; Prazosin; Rats; Receptors, Adrenergic; Rilmenidine; Tritium; Yohimbine | 1992 |
Characterization of imidazoline-guanidinium receptive sites in renal medulla from human kidney.
Topics: Adrenergic alpha-Antagonists; Animals; Dioxanes; Guanidine; Guanidines; Humans; Idazoxan; Imidazoline Receptors; Indazoles; Kidney Medulla; Oxazoles; Rabbits; Receptors, Adrenergic; Receptors, Cell Surface; Receptors, Drug; Tritium; Yohimbine | 1992 |
Contribution of alpha 2-adrenoceptors to the central cardiovascular effects of clonidine and S 8350 in anaesthetized rats.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Cardiovascular System; Cerebral Cortex; Clonidine; Heart Rate; Male; Oxazoles; Rats; Receptors, Adrenergic, alpha; Yohimbine | 1991 |
Selectivity of rilmenidine for the nucleus reticularis lateralis, a ventrolateral medullary structure containing imidazoline-preferring receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Catecholamines; Clonidine; Dioxanes; Electrochemistry; Hemodynamics; Idazoxan; Imidazoline Receptors; Male; Medulla Oblongata; Neurons; Oxazoles; Piperoxan; Rats; Rats, Inbred WKY; Receptors, Drug; Reticular Formation; Rilmenidine; Stereotaxic Techniques; Yohimbine | 1991 |
[Selectivity of a new antihypertensive agent, rilmenidine, for imidazoline receptors in the human brain].
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Brain; Dioxanes; Humans; Idazoxan; Imidazoline Receptors; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Yohimbine | 1990 |
Desensitization and down-regulation of brain alpha 2-adrenoceptors by centrally acting antihypertensive drugs.
Topics: Animals; Antihypertensive Agents; Binding, Competitive; Brain; Central Nervous System; Clonidine; Down-Regulation; Guanabenz; Hemodynamics; In Vitro Techniques; Male; Oxazoles; Rabbits; Receptors, Adrenergic, alpha; Rilmenidine; Yohimbine | 1990 |
Evidence for the involvement of imidazoline receptors in the central hypotensive effect of rilmenidine in the rabbit.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Brain; Cisterna Magna; Dioxanes; Heart Rate; Hemodynamics; Idazoxan; Imidazoline Receptors; Injections; Injections, Intraventricular; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Tissue Extracts; Yohimbine | 1990 |
Influence of the alpha-2 agonist oxaminozoline (S3341) on firing rate of central noradrenergic and serotonergic neurons in the rat. Comparison with clonidine.
Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Electrophysiology; Iontophoresis; Locus Coeruleus; Male; Neurons; Norepinephrine; Oxazoles; Prazosin; Raphe Nuclei; Rats; Rilmenidine; Serotonin; Yohimbine | 1986 |
Different affinities of alpha 2-agonists for imidazoline and alpha 2-adrenergic receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Dioxanes; Guanfacine; Guanidine; Guanidines; Idazoxan; Imidazoline Receptors; Male; Oxazoles; Phenylacetates; Rabbits; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine; Yohimbine | 1989 |
[Selectivity of alpha 2-adrenergic agonists for the imidazoline-guanidine and alpha 2-adrenergic receptors].
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Guanfacine; Guanidines; Idazoxan; Kidney Tubules, Proximal; Male; Oxazoles; Phenylacetates; Rabbits; Receptors, Adrenergic, alpha; Rilmenidine; Yohimbine | 1989 |
[Interaction of rilmenidine with renal imidazoline-guanidine sites].
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Basement Membrane; Binding Sites; Dioxanes; Drug Interactions; Guanfacine; Guanidines; Idazoxan; Imidazoles; Imidazoline Receptors; Kidney; Male; Oxazoles; Phenylacetates; Rabbits; Receptors, Drug; Rilmenidine; Sodium Channels; Yohimbine | 1989 |
New isoxazole derivatives provided with antihypertensive activity.
Topics: Animals; Antihypertensive Agents; Aorta, Thoracic; Binding, Competitive; Chemical Phenomena; Chemistry; Clonidine; In Vitro Techniques; Isoxazoles; Magnetic Resonance Spectroscopy; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Vas Deferens; Yohimbine | 1989 |
Prejunctional alpha 2-adrenergic properties of S-3341 (dicyclopropylmethyl)amino-2-delta-2-oxazoline: a comparison with clonidine.
Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Oxazoles; Prazosin; Rats; Rats, Inbred WKY; Rilmenidine; Vas Deferens; Yohimbine | 1987 |
Effect of the amino-oxazoline derivative S-3341 on pre- and postjunctional alpha-adrenoceptors in isolated blood vessels.
Topics: Animals; Clonidine; Dogs; In Vitro Techniques; Norepinephrine; Oxazoles; Perfusion; Phenylephrine; Prazosin; Pulmonary Artery; Rabbits; Receptors, Adrenergic, alpha; Rilmenidine; Saphenous Vein; Vasoconstriction; Yohimbine | 1986 |
A 2-amino-2-oxazoline derivative as an antidepressant in mice.
Topics: 5-Hydroxytryptophan; Amphetamine; Animals; Antidepressive Agents; Apomorphine; Barbital; Drug Interactions; Helplessness, Learned; Male; Mice; Motor Activity; Oxazoles; Oxotremorine; Pentobarbital; Postural Balance; Reserpine; Yohimbine | 1988 |
The effect of selective alpha 1- and alpha 2-adrenoceptor stimulation on intraocular pressure in the conscious rabbit.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Female; Intraocular Pressure; Male; Oxazoles; Phenylephrine; Rabbits; Thiazoles; Yohimbine | 1981 |
Postsynaptic alpha 1- and alpha 2-adrenoceptors in the circulatory system of the pithed rat: selective stimulation of the alpha 2-type by B-HT 933.
Topics: Animals; Azepines; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Muscle, Smooth, Vascular; Oxazoles; Phentolamine; Phenylephrine; Prazosin; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Receptors, Neurotransmitter; Vasomotor System; Yohimbine | 1980 |
Vasoconstriction mediated by postsynaptic alpha 2-adrenoceptor stimulation.
Topics: Animals; Azepines; Blood Pressure; Dose-Response Relationship, Drug; Male; Oxazoles; Phenylephrine; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Vasoconstrictor Agents; Yohimbine | 1980 |
Mechanism of sympathoinhibition by imidazolines.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzazepines; Brimonidine Tartrate; Dioxanes; Hemodynamics; Idazoxan; Imidazoles; Oxazoles; Quinoxalines; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine | 1995 |
Sympathoinhibition by rilmenidine in conscious rabbits: involvement of alpha 2-adrenoceptors.
Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Catecholamines; Decerebrate State; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Electrodes, Implanted; Female; Heart Rate; Hemodynamics; Idazoxan; Kidney; Male; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine | 1993 |
Antiarrhythmic action of rilmenidine on adrenaline-induced arrhythmia via central imidazoline receptors in halothane-anaesthetized dogs.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Anesthetics, Inhalation; Animals; Arrhythmias, Cardiac; Blood Pressure; Dogs; Epinephrine; Female; Halothane; Heart Rate; Idazoxan; Imidazoline Receptors; Male; Oxazoles; Receptors, Drug; Rilmenidine; Yohimbine | 1996 |
Interactions of the cardiac chronotropic effects of rilmenidine with the autonomic nervous system in conscious dogs: comparison with clonidine.
Topics: Adrenergic beta-Antagonists; Animals; Antihypertensive Agents; Atropine; Blood Pressure; Chronic Disease; Clonidine; Depression, Chemical; Dogs; Female; Heart Block; Heart Rate; Male; Muscarinic Antagonists; Oxazoles; Phenoxybenzamine; Pindolol; Rilmenidine; Yohimbine | 1996 |
Antinociceptive effects of oral clonidine and S12813-4 in acute colon inflammation in rats.
Topics: Acute Disease; Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Clonidine; Colitis; Female; Formaldehyde; Idazoxan; Oxazoles; Rats; Rats, Sprague-Dawley; Yohimbine | 1996 |
Rilmenidine activates postjunctional alpha 1- and alpha 2-adrenoceptors in the canine saphenous vein.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dogs; Female; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isotope Labeling; Male; Medetomidine; Muscle Contraction; Muscle, Smooth; Osmolar Concentration; Oxazoles; Phenoxybenzamine; Prazosin; Protein Binding; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Tritium; Yohimbine | 1996 |
Rilmenidine-induced ocular hypotension: role of imidazoline1 and alpha 2 receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzofurans; Calcium; Ciliary Body; Cyclic AMP; Female; Imidazoles; Imidazoline Receptors; Intraocular Pressure; Iris; Male; Norepinephrine; Ocular Hypotension; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathectomy; Sympathetic Nervous System; Yohimbine | 1996 |
Are imidazoline receptors involved in sympathetic neurotransmission in rat vas deferens?
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Electric Stimulation; Idazoxan; Imidazoline Receptors; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Oxazoles; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Synaptic Transmission; Vas Deferens; Yohimbine | 1996 |
Role of I1 imidazoline receptors in the sympathoinhibition produced by intracisternally administered rilmenidine and moxonidine.
Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Cisterna Magna; Dose-Response Relationship, Drug; Female; Guanabenz; Heart Rate; Imidazoles; Imidazoline Receptors; Injections; Male; Norepinephrine; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Yohimbine | 1997 |
Analysis of the receptor involved in the central hypotensive effect of rilmenidine and moxonidine.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzazepines; Benzofurans; Blood Pressure; Dose-Response Relationship, Drug; Drug Interactions; Female; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Methyldopa; Norepinephrine; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Yohimbine | 1999 |
An unexpected central hypertensive effect of the new imidazoline compound benazoline.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension; Imidazoles; Imidazoline Receptors; Male; Nasal Decongestants; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Yohimbine | 1999 |
Mechanism of the sympathoinhibition produced by the clonidine-like drugs rilmenidine and moxonidine.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzazepines; Blood Pressure; Clonidine; Decerebrate State; Heart Rate; Imidazoles; Injections, Spinal; Medulla Oblongata; Microinjections; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine | 1999 |
Alpha2-adrenoceptor ligands inhibit alpha1-adrenoceptor-mediated contraction of isolated rat arteries.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Arteries; Azepines; Brimonidine Tartrate; Clonidine; Idazoxan; In Vitro Techniques; Ligands; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Oxazoles; Prostaglandins; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Rilmenidine; Yohimbine | 2002 |
The role of I(1)-imidazoline receptors and alpha(2)-adrenergic receptors in the modulation of glucose and lipid metabolism in the SHROB model of metabolic syndrome X.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Disease Models, Animal; Female; Glucagon; Glucose; Glucose Tolerance Test; Humans; Imidazoles; Imidazoline Receptors; Lipid Metabolism; Male; Metabolic Syndrome; Obesity; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Yohimbine | 2003 |
Moxonidine displays a presynaptic alpha-2-adrenoceptor-dependent synergistic sympathoinhibitory action at imidazoline-1 receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Benzofurans; Bridged Bicyclo Compounds; Brimonidine Tartrate; Drug Synergism; Heart; Heptanes; Imidazoles; Imidazoline Receptors; Norepinephrine; Oxazoles; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Sympatholytics; Yohimbine | 2003 |
The effects of the alpha2-adrenergic receptor agonists clonidine and rilmenidine, and antagonists yohimbine and efaroxan, on the spinal cholinergic receptor system in the rat.
Topics: Acetylcholine; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Benzofurans; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Injections, Spinal; Ligands; Male; Microdialysis; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Cholinergic; Rilmenidine; Spinal Cord; Time Factors; Yohimbine | 2004 |
[Effect of rilmenidine on intraocular pressure in rabbits, interaction with efaroxan and rauwolscine].
Topics: Administration, Topical; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzofurans; Drug Interactions; Glaucoma; Imidazoles; Intraocular Pressure; Male; Oxazoles; Rabbits; Rilmenidine; Time Factors; Yohimbine | 2004 |
Moxonidine and rilmenidine injected into the medial septal area reduces the salivation induced by pilocarpine.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Drug Interactions; Idazoxan; Imidazoles; Male; Muscarinic Agonists; Oxazoles; Pilocarpine; Rats; Rats, Sprague-Dawley; Rilmenidine; Salivation; Septum of Brain; Yohimbine | 2004 |
Possible role of NMDA receptors in antinociception induced by rilmenidine in mice in the formalin test.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analgesics; Animals; Benzofurans; Binding Sites; Binding, Competitive; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Imidazoles; Imidazoline Receptors; Male; Mice; Nervous System; Neurons, Afferent; Nociceptors; Oxazoles; Pain; Pain Measurement; Receptors, Drug; Receptors, N-Methyl-D-Aspartate; Rilmenidine; Yohimbine | 2007 |
Antagonism of the neuropeptide S receptor with RTI-118 decreases cocaine self-administration and cocaine-seeking behavior in rats.
Topics: Animals; Cocaine; Male; Motivation; Oxazoles; Pyrazines; Rats; Rats, Wistar; Receptors, Neuropeptide; Self Administration; Yohimbine | 2012 |