Page last updated: 2024-08-21

oxazoles and staurosporine

oxazoles has been researched along with staurosporine in 65 studies

Research

Studies (65)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's32 (49.23)18.2507
2000's30 (46.15)29.6817
2010's2 (3.08)24.3611
2020's1 (1.54)2.80

Authors

AuthorsStudies
Bitonti, AJ; Dumont, JA; Jones, WD1
Bize, I; Dunham, PB2
García-Sáinz, JA; González-Espinosa, C1
Henderson, LK; Matthews, N; Nemec, M; Southern, C; Thorp, KM; Wilkinson, PC1
Hunchuk, N; Li, XB; Wong, K1
Alverez, J; Garcia-Sancho, J; Montero, M1
Kawasaki, K; Shinohara, S1
Sakamoto, N; Shuntoh, H; Tanaka, C1
Brenner, HR; Britt, JC; Caroni, P; Rotzler, S1
Hosoi, K; Kurihara, K; Ueha, T1
Chock, PB; Huang, CY; Tekle, E; Zhu, DM1
Adragna, NC; Flatman, PW; Lauf, PK1
Cossins, AR; Weaver, YR1
Patzlaff, JS; Paulson, JR; Vallis, AJ1
Amieva, MR; Furthmayr, H; Hirota, C; Mizuno, Y; Nakamura, F1
Fukunaga, K; Kano, M; Konnerth, A1
Dunham, PB; Kelley, SJ1
Cesare, P; McNaughton, P1
Harris, RA; Huidobro-Toro, JP; Valenzuela, CF1
Gay, JC; Murray, JJ; Raddassi, K; Truett, AP1
Badwey, JA; Ding, J; Ellis, BA; Heyworth, PG; Robinson, JM1
Kramer, RH; Molokanova, E; Savchenko, A; Trivedi, B1
Datta, K; Deb, TB; Gupta, S; Rao, CM1
Isobe, M; Muto, S; Takahashi, K1
Lytle, C1
Harris, RA; Martinez, LD; Mascia, MP; Wick, MJ1
Fabre, S; Georget, V; Lobaccaro, JM; Lumbroso, S; Poujol, N; Sultan, C; Térouanne, B1
Cossins, AR; Gibson, JS; Muzyamba, MC1
Creanor, J; Flatman, PW1
Brender, C; Brockdorff, J; Christensen, ST; Engel, AM; Geisler, C; Kaltoft, K; Leick, V; Nielsen, M; Odum, N; Rygaard, J; Skov, S; Svejgaard, A; Woetmann, A1
Greger, R; Henger, A; Mundel, P; Nitschke, R; Pavenstädt, H; Rüdiger, F1
Bosch, RJ; Díez-Marqués, ML; García-Escribano, C; Rodríguez-Puyol, D; Rodríguez-Puyol, M; Torrecillas, G1
Dartt, DA; Hodges, RR; Sergheraert, C; Zoukhri, D1
Alcántara-Hernández, R; Gárcia-Sáinz, JA; Vázquez-Prado, J1
Albig, W; Doenecke, D; Hanecke, K; Kratzmeier, M1
Cossins, AR; Ellory, JC; Kiessling, K1
Dietrich, J; Geisler, C; Kastrup, J; Lauritsen, JP; Menné, C; Odum, N1
Crook, RB; Layne, J; Yip, S1
Hwang, JU; Lee, Y1
Adams, ME; Cardullo, RA; Kingan, TG1
Ellory, JC; Gibson, JS; Husain, F; Luckas, MC; Muzyamba, MC; Speake, PF1
Egger, T; Goti, D; Hammer, A; Malle, E; Sattler, W; Wintersperger, A1
Kurihara, K; Moore-Hoon, ML; Nakanishi, N; Turner, RJ1
Knight, H; Knight, MR; Wright, AJ1
Ramonell, K; Somerville, S; Stacey, G; Zhang, B1
Andrews, DA; Low, PS; Yang, L1
Brockdorff, J; Geisler, C; Leick, V; Lovato, P; Nielsen, M; Rieneck, K; Svejgaard, A; Woetmann, A; Ødum, N1
Dai, C; Liu, Y; Yang, J1
Chen, J; Chen, Q; Gu, L; Zhang, H1
Lee, S; Lee, Y; Park, J1
duBell, WH; Rogers, TB1
Dubery, IA; Gerber, IB1
Ebel, R; Edrada, RA; Proksch, P; Steube, K; Wray, V1
Blagden, S; de Bono, J1
Liu, L; Xu, J1
Flatman, PW; Hegney, KL; Matskevich, I1
Adragna, NC; Brown, TL; Lauf, PK; Warwar, R1
Chen, K; Chen, SR; Cheng, H; Obayashi, M; Shimoni, Y; Ter Keurs, H; Walsh, MP; Xiao, B; Yang, D; Zhong, G1
Bisschops, R; Cassiman, D; Fevery, J; Laleman, W; Nevens, F; Roskams, T; Severi, T; Van Landeghem, L; Van Pelt, J; Vander Elst, I; Zeegers, M1
Hoffmann, EK; Pedersen, SF1
Harrison, RA; Jebe, E; Petrunkina, AM; Töpfer-Petersen, E; Tsolova, M1
Cardullo, RA; Haimo, LT; Miyata, H; Thaler, CD1
Kim, BJ; Kim, JN1
Hu, L; Li, Y; Ruan, C; Wang, Q; Wang, S; Ye, M; Zhang, X1

Reviews

2 review(s) available for oxazoles and staurosporine

ArticleYear
Bioactive natural products from marine invertebrates and associated fungi.
    Progress in molecular and subcellular biology, 2003, Volume: 37

    Topics: Alkaloids; Animals; Biodiversity; Biological Products; Biotechnology; Fungal Proteins; Fungi; Marine Biology; Marine Toxins; Models, Chemical; Oxazoles; Porifera; Staurosporine; Urochordata

2003
Drugging cell cycle kinases in cancer therapy.
    Current drug targets, 2005, Volume: 6, Issue:3

    Topics: Adenosine Triphosphate; Animals; Antineoplastic Agents; Binding Sites; Cyclin-Dependent Kinases; Flavonoids; Humans; Neoplasms; Oxazoles; Piperidines; Protein Kinase Inhibitors; Purines; Roscovitine; Staurosporine; Sulfonamides; Thiazoles

2005

Other Studies

63 other study(ies) available for oxazoles and staurosporine

ArticleYear
Inhibition of experimental metastasis and cell adhesion of B16F1 melanoma cells by inhibitors of protein kinase C.
    Cancer research, 1992, Mar-01, Volume: 52, Issue:5

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Animals; Cell Adhesion; Isoquinolines; Lung Neoplasms; Melanoma, Experimental; Membrane Proteins; Mice; Mice, Inbred C57BL; Neoplasm Metastasis; Oxazoles; Oxazolone; Phosphorylation; Piperazines; Protein Kinase C; Pyridines; Staurosporine; Time Factors

1992
H2O2 activates red blood cell K-Cl cotransport via stimulation of a phosphatase.
    The American journal of physiology, 1995, Volume: 269, Issue:4 Pt 1

    Topics: Alkaloids; Animals; Carrier Proteins; Catalase; Erythrocytes; Ethylmaleimide; Hydrogen Peroxide; Intracellular Membranes; K Cl- Cotransporters; Marine Toxins; Oxazoles; Phosphoprotein Phosphatases; Phosphoric Monoester Hydrolases; Potassium; Sheep; Staurosporine; Symporters

1995
Protein kinases and phosphatases modulate c-fos expression in rat hepatocytes. Effects of angiotensin II and phorbol myristate acetate.
    Life sciences, 1995, Volume: 56, Issue:10

    Topics: Alkaloids; Angiotensin II; Animals; Ethers, Cyclic; Female; Gene Expression; Genes, fos; Genistein; Isoflavones; Marine Toxins; Microcystins; Naphthalenes; Okadaic Acid; Oxazoles; Peptides, Cyclic; Phosphoprotein Phosphatases; Phosphorylation; Polycyclic Compounds; Protein Kinase Inhibitors; Protein Kinases; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Rats; Rats, Wistar; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate

1995
Inhibition of protein kinase C results in a switch from a non-motile to a motile phenotype in diverse human lymphocyte populations.
    Immunology, 1995, Volume: 84, Issue:2

    Topics: Alkaloids; B-Lymphocytes; Blotting, Western; Cell Line; Cell Movement; Cells, Cultured; Enzyme Activation; Humans; Indoles; Lymphocytes; Maleimides; Marine Toxins; Oxazoles; Phenotype; Phosphoprotein Phosphatases; Protein Kinase C; Staurosporine; T-Lymphocytes

1995
N-acetylsphingosine (C2-ceramide) inhibited neutrophil superoxide formation and calcium influx.
    The Journal of biological chemistry, 1995, Feb-17, Volume: 270, Issue:7

    Topics: Alkaloids; Biological Transport, Active; Blood Proteins; Calcium; Enzyme Activation; Humans; In Vitro Techniques; Kinetics; Marine Toxins; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Oxazoles; Phosphoprotein Phosphatases; Phosphoproteins; Phosphorylation; Protein Kinase C; Spectrometry, Fluorescence; Sphingosine; Staurosporine; Superoxides

1995
Chemotactic peptide down-regulation of calcium mobilization induced by platelet-activating factor and by leukotriene B4 in human neutrophils is uncovered by protein phosphatase inhibitors.
    The Biochemical journal, 1994, Oct-15, Volume: 303 ( Pt 2)

    Topics: Alkaloids; Calcium; Down-Regulation; Ethers, Cyclic; Humans; Indoles; Leukotriene B4; Marine Toxins; N-Formylmethionine Leucyl-Phenylalanine; Neutrophils; Okadaic Acid; Oxazoles; Phorbol 12,13-Dibutyrate; Phosphoprotein Phosphatases; Phosphorylation; Platelet Activating Factor; Protein Kinase C; Signal Transduction; Staurosporine

1994
Desensitization of cholecystokininB receptors in GH3 cells.
    Journal of neurochemistry, 1994, Volume: 62, Issue:4

    Topics: Alkaloids; Calcium; Drug Tolerance; Enzyme Activation; Inositol 1,4,5-Trisphosphate; Marine Toxins; Oxazoles; Phorbol 12,13-Dibutyrate; Phosphoric Monoester Hydrolases; Pituitary Neoplasms; Protein Kinase C; Receptors, Cholecystokinin; Sincalide; Staurosporine; Thyrotropin-Releasing Hormone; Tumor Cells, Cultured

1994
Staurosporine, a protein kinase inhibitor, activates K-Cl cotransport in LK sheep erythrocytes.
    The American journal of physiology, 1994, Volume: 266, Issue:3 Pt 1

    Topics: Alkaloids; Animals; Carrier Proteins; Erythrocytes; K Cl- Cotransporters; Magnesium; Marine Toxins; Osmolar Concentration; Oxazoles; Oxidation-Reduction; Phosphoprotein Phosphatases; Potassium; Protein Kinase Inhibitors; Sheep; Staurosporine; Symporters; Tetradecanoylphorbol Acetate; Time Factors

1994
Protein phosphatase inhibitors induce the release of serotonin from rat basophilic leukemia cells (RBL-2H3).
    Biochimica et biophysica acta, 1994, Apr-28, Volume: 1221, Issue:3

    Topics: Alkaloids; Animals; Calcium; Ethers, Cyclic; Leukemia, Basophilic, Acute; Marine Toxins; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase Inhibitors; Rats; Serotonin; Staurosporine; Tumor Cells, Cultured

1994
Calcium influx and protein phosphorylation mediate the metabolic stabilization of synaptic acetylcholine receptors in muscle.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:3

    Topics: Alkaloids; Animals; Bucladesine; Calcium; Calcium Channels; Cyclic AMP; Dibutyryl Cyclic GMP; Dihydropyridines; Electric Stimulation; Ethers, Cyclic; Kinetics; Male; Marine Toxins; Motor Endplate; Muscle Denervation; Muscles; Okadaic Acid; Organ Culture Techniques; Oxazoles; Phosphoprotein Phosphatases; Phosphoproteins; Phosphorylation; Potassium Chloride; Protein Kinase Inhibitors; Protein Kinases; Rats; Rats, Sprague-Dawley; Receptors, Cholinergic; Staurosporine; Synapses; Tetrodotoxin; Time Factors

1993
Bradykinin-stimulated transient modulation of epidermal growth factor receptors in A-431 human epidermoid carcinoma cells.
    Journal of cellular physiology, 1993, Volume: 157, Issue:1

    Topics: Alkaloids; Binding, Competitive; Bradykinin; Carcinoma, Squamous Cell; ErbB Receptors; Humans; Marine Toxins; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase C; Staurosporine; Tumor Cells, Cultured

1993
Reversible phosphorylation as a controlling factor for sustaining calcium oscillations in HeLa cells: Involvement of calmodulin-dependent kinase II and a calyculin A-inhibitable phosphatase.
    Biochemistry, 1996, Jun-04, Volume: 35, Issue:22

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Amino Acid Sequence; Binding Sites; Calcium; Calcium Channels; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Calcium-Transporting ATPases; Enzyme Inhibitors; Ethers, Cyclic; HeLa Cells; Histamine; Humans; Indoles; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Isoquinolines; Maleimides; Marine Toxins; Molecular Sequence Data; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Piperazines; Protein Kinase C; Receptors, Cytoplasmic and Nuclear; Ryanodine; Spectrometry, Fluorescence; Staurosporine; Sulfonamides

1996
Role of protein kinases in regulating sheep erythrocyte K-Cl cotransport.
    The American journal of physiology, 1996, Volume: 271, Issue:1 Pt 1

    Topics: Adenosine Triphosphate; Animals; Benzylidene Compounds; Carrier Proteins; Erythrocytes; Ethylmaleimide; Genistein; Isoflavones; K Cl- Cotransporters; Marine Toxins; Nitriles; Oxazoles; Protein Kinases; Sheep; Staurosporine; Symporters; Tyrphostins

1996
Protein tyrosine phosphorylation and the regulation of KCl cotransport in trout erythrocytes.
    Pflugers Archiv : European journal of physiology, 1996, Volume: 432, Issue:4

    Topics: Animals; Carrier Proteins; Dose-Response Relationship, Drug; Enzyme Inhibitors; Erythrocytes; Genistein; Isoflavones; Isoproterenol; K Cl- Cotransporters; Marine Toxins; Oncorhynchus mykiss; Oxazoles; Phosphorylation; Potassium Chloride; Protein-Tyrosine Kinases; Staurosporine; Symporters; Tyrosine; Vanadates

1996
Evidence that the endogenous histone H1 phosphatase in HeLa mitotic chromosomes is protein phosphatase 1, not protein phosphatase 2A.
    Journal of cell science, 1996, Volume: 109 ( Pt 6)

    Topics: Cell Nucleus; Chromatin; Enzyme Inhibitors; HeLa Cells; Histones; Humans; Kinetin; Marine Toxins; Metaphase; Microcystins; Mitosis; Okadaic Acid; Oxazoles; Peptides, Cyclic; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase Inhibitors; Protein Phosphatase 1; Protein Phosphatase 2; Purines; Staurosporine

1996
Phosphorylation of 558T of moesin detected by site-specific antibodies in RAW264.7 macrophages.
    Biochemical and biophysical research communications, 1996, Sep-24, Volume: 226, Issue:3

    Topics: Amino Acid Sequence; Animals; Antibodies; Antibody Specificity; Antigen-Antibody Complex; Blotting, Western; Cell Line; Cytochalasin B; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Macrophages; Marine Toxins; Microfilament Proteins; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Phosphothreonine; Proteins; Rabbits; Staurosporine; Threonine

1996
Ca(2+)-induced rebound potentiation of gamma-aminobutyric acid-mediated currents requires activation of Ca2+/calmodulin-dependent kinase II.
    Proceedings of the National Academy of Sciences of the United States of America, 1996, Nov-12, Volume: 93, Issue:23

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Cerebellum; Drug Synergism; Enzyme Activation; Enzyme Inhibitors; gamma-Aminobutyric Acid; Imidazoles; In Vitro Techniques; Kinetics; Marine Toxins; Membrane Potentials; Nerve Fibers; Oxazoles; Purkinje Cells; Rats; Receptors, GABA-A; Signal Transduction; Staurosporine

1996
Mechanism of swelling activation of K-Cl cotransport in inside-out vesicles of LK sheep erythrocyte membranes.
    The American journal of physiology, 1996, Volume: 270, Issue:4 Pt 1

    Topics: Adenosine Triphosphate; Animals; Body Fluids; Carrier Proteins; Chlorides; Erythrocyte Membrane; Ethylmaleimide; Homeostasis; K Cl- Cotransporters; Kinetics; Magnesium; Marine Toxins; Oxazoles; Phenotype; Phosphorylation; Potassium; Sheep; Staurosporine; Symporters; Time Factors

1996
A novel heat-activated current in nociceptive neurons and its sensitization by bradykinin.
    Proceedings of the National Academy of Sciences of the United States of America, 1996, Dec-24, Volume: 93, Issue:26

    Topics: Animals; Animals, Newborn; Bradykinin; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Ganglia, Spinal; Hot Temperature; Kinetics; Marine Toxins; Membrane Potentials; Neurons; Neurons, Afferent; Nociceptors; Oxazoles; Pain; Protein Kinase C; Protein Tyrosine Phosphatases; Rats; Rats, Wistar; Staurosporine; Tetradecanoylphorbol Acetate; Time Factors

1996
Modulation of GABAA receptor function by G protein-coupled 5-HT2C receptors.
    Neuropharmacology, 1996, Volume: 35, Issue:9-10

    Topics: Animals; Chelating Agents; Chloride Channels; Egtazic Acid; Enzyme Inhibitors; GTP-Binding Proteins; Humans; Marine Toxins; Oocytes; Oxazoles; Phosphoprotein Phosphatases; Receptors, GABA-A; Receptors, Serotonin; RNA, Messenger; Staurosporine; Transcription, Genetic; Xenopus laevis

1996
Phosphatase activity regulates superoxide anion generation and intracellular signaling in human neutrophils.
    Biochimica et biophysica acta, 1997, Aug-29, Volume: 1336, Issue:2

    Topics: Adult; Humans; Marine Toxins; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; Neutrophils; Oxazoles; Phosphatidic Acids; Phospholipase D; Phosphoric Monoester Hydrolases; Phosphorylation; Protein Kinase C; Staurosporine; Superoxides; Tetradecanoylphorbol Acetate

1997
Cofilin undergoes rapid dephosphorylation in stimulated neutrophils and translocates to ruffled membranes enriched in products of the NADPH oxidase complex. Evidence for a novel cycle of phosphorylation and dephosphorylation.
    Histochemistry and cell biology, 1997, Volume: 108, Issue:3

    Topics: Actin Depolymerizing Factors; Actins; Amino Acid Sequence; Animals; Calcimycin; Cell Membrane; Diglycerides; Diterpenes; Guinea Pigs; Humans; Hydrogen Peroxide; Immunoblotting; Marine Toxins; Microfilament Proteins; Molecular Sequence Data; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; Neutrophil Activation; Neutrophils; Okadaic Acid; Oxazoles; Oxides; Phosphorylation; Staurosporine; Terpenes; Tetradecanoylphorbol Acetate

1997
Modulation of rod photoreceptor cyclic nucleotide-gated channels by tyrosine phosphorylation.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Dec-01, Volume: 17, Issue:23

    Topics: Adenosine Triphosphate; Animals; Cyclic GMP; Enzyme Inhibitors; Eye Proteins; Hydroquinones; Ion Channel Gating; Marine Toxins; Microcystins; Okadaic Acid; Oocytes; Oxazoles; Patch-Clamp Techniques; Peptides, Cyclic; Phenols; Phosphorylation; Protein Processing, Post-Translational; Protein Tyrosine Phosphatases; Rod Cell Outer Segment; Staurosporine; Vanadates; Xenopus laevis

1997
Regulation of cellular phosphorylation of hyaluronan binding protein and its role in the formation of second messenger.
    Biochimica et biophysica acta, 1997, Oct-20, Volume: 1336, Issue:3

    Topics: Animals; Cell Line; Cell Line, Transformed; Cell Membrane; Enzyme Inhibitors; Hyaluronan Receptors; Hyaluronic Acid; Immunoblotting; Inositol 1,4,5-Trisphosphate; Isoenzymes; Kinetics; Marine Toxins; Oxazoles; Phospholipase C gamma; Phosphorylation; Polyomavirus; Protein Kinase Inhibitors; Protein Kinases; Rats; Second Messenger Systems; Skin; Staurosporine; Tetradecanoylphorbol Acetate; Type C Phospholipases

1997
Mastoparan induces an increase in cytosolic calcium ion concentration and subsequent activation of protein kinases in tobacco suspension culture cells.
    Biochimica et biophysica acta, 1998, Mar-05, Volume: 1401, Issue:3

    Topics: Aequorin; Apoproteins; Calcium; Calcium Channel Blockers; Cells, Cultured; Cytosol; Enzyme Activation; Enzyme Inhibitors; Gallic Acid; Hydrogen Peroxide; Intercellular Signaling Peptides and Proteins; Marine Toxins; Neomycin; Nicotiana; Oxazoles; Oxidation-Reduction; Peptides; Phosphoprotein Phosphatases; Plants, Genetically Modified; Plants, Toxic; Protein Kinase Inhibitors; Protein Kinases; Recombinant Proteins; Signal Transduction; Staurosporine; Wasp Venoms

1998
A volume-sensitive protein kinase regulates the Na-K-2Cl cotransporter in duck red blood cells.
    The American journal of physiology, 1998, Volume: 274, Issue:4

    Topics: Animals; Carrier Proteins; Ducks; Enzyme Inhibitors; Erythrocytes; Ethylmaleimide; Female; Kinetics; Marine Toxins; Oxazoles; Phosphorylation; Protein Kinases; Sodium-Potassium-Chloride Symporters; Staurosporine

1998
Enhancement of glycine receptor function by ethanol: role of phosphorylation.
    British journal of pharmacology, 1998, Volume: 125, Issue:2

    Topics: Animals; Cloning, Molecular; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ethanol; Female; Glycine; Glycine Agents; Halothane; Humans; Indoles; Maleimides; Marine Toxins; Oocytes; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Propofol; Protein Kinase C; Receptors, Glycine; Staurosporine; Strychnine; Xenopus laevis

1998
Transcriptional interferences between normal or mutant androgen receptors and the activator protein 1--dissection of the androgen receptor functional domains.
    Endocrinology, 1999, Volume: 140, Issue:1

    Topics: Aldehyde Reductase; Androgens; Animals; Breast Neoplasms, Male; COS Cells; DNA; Enzyme Inhibitors; Genes, Reporter; Genetic Engineering; Humans; Luciferases; Male; Marine Toxins; Mice; Mutation; Okadaic Acid; Oxazoles; Proteins; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; Receptors, Androgen; Staurosporine; Structure-Activity Relationship; Tetradecanoylphorbol Acetate; Transcription Factor AP-1; Transcription, Genetic; Transfection

1999
Regulation of Na+-K+-2Cl- cotransport in turkey red cells: the role of oxygen tension and protein phosphorylation.
    The Journal of physiology, 1999, Jun-01, Volume: 517 ( Pt 2)

    Topics: Adrenergic beta-Agonists; Animals; Carrier Proteins; Dithiothreitol; Drug Interactions; Enzyme Inhibitors; Erythrocytes; Ethylmaleimide; Isoproterenol; Marine Toxins; Oxazoles; Oxygen; Partial Pressure; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase Inhibitors; Sodium-Potassium-Chloride Symporters; Staurosporine; Turkeys

1999
Regulation of Na+-K+-2Cl- cotransport by protein phosphorylation in ferret erythrocytes.
    The Journal of physiology, 1999, Jun-15, Volume: 517 ( Pt 3)

    Topics: Animals; Blood Proteins; Carrier Proteins; Chlorides; Enzyme Inhibitors; Erythrocytes; Ferrets; Homeostasis; Kinetics; Magnesium; Marine Toxins; Models, Biological; Oxazoles; Phosphorylation; Potassium; Pyrazoles; Pyrimidines; Rubidium; Sodium; Sodium-Potassium-Chloride Symporters; Staurosporine

1999
Inhibition of protein phosphatase 2A induces serine/threonine phosphorylation, subcellular redistribution, and functional inhibition of STAT3.
    Proceedings of the National Academy of Sciences of the United States of America, 1999, Sep-14, Volume: 96, Issue:19

    Topics: Calcineurin Inhibitors; CD4-Positive T-Lymphocytes; Cell Nucleus; Cyclosporine; Cytoplasm; DNA-Binding Proteins; Enzyme Inhibitors; Humans; Marine Toxins; Microscopy, Confocal; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Phosphatase 2; Serine; Signal Transduction; STAT3 Transcription Factor; Staurosporine; Threonine; Trans-Activators; Tumor Cells, Cultured

1999
Polycations induce calcium signaling in glomerular podocytes.
    Kidney international, 1999, Volume: 56, Issue:5

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 3T3 Cells; Animals; Benzoquinones; Calcium Signaling; Cells, Cultured; DEAE-Dextran; Heparin; Kidney Glomerulus; Lactams, Macrocyclic; Marine Toxins; Mice; Muramidase; Oxazoles; Protamines; Quinones; Rifabutin; Staurosporine; Thapsigargin

1999
Mechanisms of cGMP-dependent mesangial-cell relaxation: a role for myosin light-chain phosphatase activation.
    The Biochemical journal, 2000, Feb-15, Volume: 346 Pt 1

    Topics: Angiotensin II; Animals; Azepines; Calcium; Calcium Signaling; Cell Size; Cells, Cultured; Dibutyryl Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Activation; Glomerular Mesangium; Marine Toxins; Myosin Light Chains; Myosin-Light-Chain Kinase; Myosin-Light-Chain Phosphatase; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase C; Rats; Rats, Wistar; Staurosporine; Tetradecanoylphorbol Acetate

2000
Cholinergic-induced Ca2+ elevation in rat lacrimal gland acini is negatively modulated by PKCdelta and PKCepsilon.
    Investigative ophthalmology & visual science, 2000, Volume: 41, Issue:2

    Topics: Animals; Calcium; Carbachol; Cholinergic Agonists; Enzyme Activation; Enzyme Inhibitors; Fura-2; Isoenzymes; Lacrimal Apparatus; Male; Marine Toxins; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase C; Protein Kinase C-delta; Protein Kinase C-epsilon; Rats; Rats, Wistar; Staurosporine; Tetradecanoylphorbol Acetate; Thapsigargin

2000
Protein phosphatase-protein kinase interplay modulates alpha 1b-adrenoceptor phosphorylation: effects of okadaic acid.
    British journal of pharmacology, 2000, Volume: 129, Issue:4

    Topics: Animals; Antifungal Agents; Dose-Response Relationship, Drug; Enzyme Inhibitors; Indoles; Kinetics; Marine Toxins; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase C; Pyrans; Pyrethrins; Rats; Receptors, Adrenergic, alpha-1; Spiro Compounds; Staurosporine; Tetradecanoylphorbol Acetate

2000
Rapid dephosphorylation of H1 histones after apoptosis induction.
    The Journal of biological chemistry, 2000, Sep-29, Volume: 275, Issue:39

    Topics: Apoptosis; Deoxyribonucleases; DNA Fragmentation; DNA, Neoplasm; Enzyme Activation; Histones; HL-60 Cells; Humans; Marine Toxins; Nucleosomes; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate; Topotecan

2000
The relationship between hypotonically-induced taurine and K fluxes in trout red blood cells.
    Pflugers Archiv : European journal of physiology, 2000, Volume: 440, Issue:3

    Topics: Animals; Biological Transport; Cell Size; Chlorides; Enzyme Inhibitors; Erythrocytes; Ethylmaleimide; Hypotonic Solutions; Marine Toxins; Oncorhynchus mykiss; Osmolar Concentration; Oxazoles; Potassium; Sodium; Staurosporine; Taurine

2000
beta2-adaptin is constitutively de-phosphorylated by serine/threonine protein phosphatase PP2A and phosphorylated by a staurosporine-sensitive kinase.
    Biochimica et biophysica acta, 2000, Sep-20, Volume: 1497, Issue:3

    Topics: Adaptor Protein Complex beta Subunits; Antifungal Agents; Cell Membrane; Cells, Cultured; Endocytosis; Enzyme Inhibitors; Humans; Jurkat Cells; Marine Toxins; Membrane Proteins; Microscopy, Confocal; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinases; Protein Phosphatase 2; Pyrans; Spiro Compounds; Staurosporine

2000
Down-regulation of Na-K-Cl cotransport by protein kinase C is mediated by protein phosphatase 1 in pigmented ciliary epithelial cells.
    Experimental eye research, 2001, Volume: 72, Issue:4

    Topics: Carcinogens; Cells, Cultured; Chloride Channels; Ciliary Body; Down-Regulation; Enzyme Inhibitors; Humans; Indoles; Maleimides; Marine Toxins; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Pigment Epithelium of Eye; Potassium Channels; Protein Kinase C; Protein Phosphatase 1; Rubidium Radioisotopes; Sodium Channels; Staurosporine; Tetradecanoylphorbol Acetate

2001
Abscisic acid-induced actin reorganization in guard cells of dayflower is mediated by cytosolic calcium levels and by protein kinase and protein phosphatase activities.
    Plant physiology, 2001, Volume: 125, Issue:4

    Topics: Abscisic Acid; Actins; Calcium; Calcium Chloride; Cytosol; Enzyme Inhibitors; Kinetics; Magnoliopsida; Marine Toxins; Oxazoles; Phosphoprotein Phosphatases; Plant Growth Regulators; Protein Kinases; Staurosporine

2001
Signal transduction in eclosion hormone-induced secretion of ecdysis-triggering hormone.
    The Journal of biological chemistry, 2001, Jul-06, Volume: 276, Issue:27

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cyclic GMP; Egtazic Acid; Insect Hormones; Manduca; Marine Toxins; Oxazoles; Signal Transduction; Staurosporine; Thapsigargin

2001
K(+) transport in red blood cells from human umbilical cord.
    Biochimica et biophysica acta, 2001, Jun-06, Volume: 1512, Issue:2

    Topics: Acetates; Biological Transport; Bumetanide; Carrier Proteins; Chlorides; Erythrocyte Membrane; Erythrocytes; Ethylmaleimide; Female; Fetal Blood; Fetal Hemoglobin; Fetus; Humans; Indenes; Infant, Newborn; K Cl- Cotransporters; Kinetics; Labor, Obstetric; Marine Toxins; Ouabain; Oxazoles; Oxygen; Potassium; Pregnancy; Sodium-Potassium-Exchanging ATPase; Staurosporine; Symporters; Urea

2001
Modulation of microglial superoxide production by alpha-tocopherol in vitro: attenuation of p67(phox) translocation by a protein phosphatase-dependent pathway.
    Journal of neurochemistry, 2001, Volume: 79, Issue:6

    Topics: alpha-Tocopherol; Animals; Antioxidants; Cell Membrane; Cells, Cultured; Cytosol; Dose-Response Relationship, Drug; Enzyme Inhibitors; Marine Toxins; Mice; Microglia; NADH, NADPH Oxidoreductases; NADPH Oxidases; Nerve Tissue Proteins; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Phosphoproteins; Phosphorylation; Protein Kinase C; Protein Processing, Post-Translational; Protein Transport; Rats; Respiratory Burst; Staurosporine; Superoxides; Swine

2001
Phosphorylation of the salivary Na(+)-K(+)-2Cl(-) cotransporter.
    American journal of physiology. Cell physiology, 2002, Volume: 282, Issue:4

    Topics: Adenosine Triphosphate; Animals; Carbazoles; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Indole Alkaloids; Indoles; Isoproterenol; Isoquinolines; Maleimides; Marine Toxins; Microcystins; Okadaic Acid; Oxazoles; Parotid Gland; Peptides, Cyclic; Phenols; Phosphorus Radioisotopes; Phosphorylation; Rats; Sodium-Potassium-Chloride Symporters; Solute Carrier Family 12, Member 2; Staurosporine; Sulfonamides; Sympathomimetics; Vanadates

2002
Mechanically stimulated TCH3 gene expression in Arabidopsis involves protein phosphorylation and EIN6 downstream of calcium.
    Plant physiology, 2002, Volume: 128, Issue:4

    Topics: Arabidopsis; Arabidopsis Proteins; Calcium; Calcium-Binding Proteins; Dimethyl Sulfoxide; Gene Expression Regulation, Plant; Marine Toxins; Mutation; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Plant Proteins; Protein Kinase Inhibitors; Receptors, Cell Surface; Signal Transduction; Staurosporine; Stress, Mechanical

2002
Characterization of early, chitin-induced gene expression in Arabidopsis.
    Molecular plant-microbe interactions : MPMI, 2002, Volume: 15, Issue:9

    Topics: Arabidopsis; Arabidopsis Proteins; Carbazoles; Chitin; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gene Expression Regulation, Plant; Indole Alkaloids; Lectins; Marine Toxins; Mitogen-Activated Protein Kinase Kinases; Okadaic Acid; Oligosaccharides; Oxazoles; Phosphorylation; Plant Proteins; RNA, Messenger; Signal Transduction; Staurosporine; Transcriptional Activation; Zinc Fingers

2002
Phorbol ester stimulates a protein kinase C-mediated agatoxin-TK-sensitive calcium permeability pathway in human red blood cells.
    Blood, 2002, Nov-01, Volume: 100, Issue:9

    Topics: Adult; Agatoxins; Alkaloids; Benzophenanthridines; Calcimycin; Calcium; Calcium Channel Blockers; Calcium Channels, N-Type; Calcium Signaling; Cell Size; Diglycerides; Dimethyl Sulfoxide; Enzyme Inhibitors; Erythrocytes; Humans; Ion Transport; Ionophores; Marine Toxins; Okadaic Acid; Osmotic Fragility; Oxazoles; Phenanthridines; Phosphoprotein Phosphatases; Protein Kinase C; Spider Venoms; Staurosporine; Tetradecanoylphorbol Acetate

2002
Protein phosphatase 2A (PP2A) regulates interleukin-4-mediated STAT6 signaling.
    The Journal of biological chemistry, 2003, Jan-31, Volume: 278, Issue:5

    Topics: Base Sequence; CD4-Positive T-Lymphocytes; Cell Line; Enzyme Inhibitors; Humans; Interleukin-4; Jurkat Cells; Marine Toxins; Molecular Sequence Data; Oligodeoxyribonucleotides; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Promoter Regions, Genetic; Protein Phosphatase 2; Recombinant Proteins; Signal Transduction; STAT6 Transcription Factor; Staurosporine; Trans-Activators; Transfection

2003
Transforming growth factor-beta1 potentiates renal tubular epithelial cell death by a mechanism independent of Smad signaling.
    The Journal of biological chemistry, 2003, Apr-04, Volume: 278, Issue:14

    Topics: Caspase 3; Caspase 9; Caspases; Cell Death; Cells, Cultured; DNA-Binding Proteins; Enzyme Inhibitors; Enzyme Precursors; Epithelial Cells; Humans; Kidney Tubules, Proximal; Mitogen-Activated Protein Kinases; Oxazoles; p38 Mitogen-Activated Protein Kinases; Pyridines; Signal Transduction; Smad2 Protein; Smad7 Protein; Staurosporine; Trans-Activators; Transforming Growth Factor beta; Transforming Growth Factor beta1

2003
Calyculin A-induced actin phosphorylation and depolymerization in renal epithelial cells.
    Cell motility and the cytoskeleton, 2003, Volume: 54, Issue:4

    Topics: Actin Cytoskeleton; Adenosine Triphosphate; Animals; Cell Line; Enzyme Inhibitors; Epithelial Cells; Kidney Tubules, Proximal; Marine Toxins; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Polymers; Protein Serine-Threonine Kinases; Serine; Staurosporine

2003
Phosphatidic acid induces actin polymerization by activating protein kinases in soybean cells.
    Molecules and cells, 2003, Jun-30, Volume: 15, Issue:3

    Topics: Actin Cytoskeleton; Actins; Cells, Cultured; Egtazic Acid; Enzyme Activation; Enzyme Inhibitors; Glycine max; Marine Toxins; Naphthalenes; Oxazoles; Phosphatidic Acids; Plant Proteins; Polymers; Protein Kinase Inhibitors; Protein Kinases; Repressor Proteins; Staurosporine

2003
Protein phosphatase 1 and an opposing protein kinase regulate steady-state L-type Ca2+ current in mouse cardiac myocytes.
    The Journal of physiology, 2004, Apr-01, Volume: 556, Issue:Pt 1

    Topics: Animals; Biophysical Phenomena; Biophysics; Buffers; Calcium Channels, L-Type; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Egtazic Acid; Electric Conductivity; Enzyme Inhibitors; Homeostasis; Isoenzymes; Male; Marine Toxins; Mice; Mice, Inbred Strains; Myocytes, Cardiac; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Protein Kinase C; Protein Phosphatase 1; Staurosporine; Thionucleotides

2004
Protein phosphorylation in Nicotiana tabacum cells in response to perception of lipopolysaccharides from Burkholderia cepacia.
    Phytochemistry, 2004, Volume: 65, Issue:22

    Topics: Burkholderia cepacia; Cells, Cultured; Lipopolysaccharides; Marine Toxins; Nicotiana; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Plant Proteins; Protein Kinase Inhibitors; Protein Processing, Post-Translational; Receptors, Cell Surface; Respiratory Burst; Signal Transduction; Staurosporine

2004
The role of calcium desensitization in vascular hyporeactivity and its regulation after hemorrhagic shock in the rat.
    Shock (Augusta, Ga.), 2005, Volume: 23, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Blood Vessels; Calcium; Carbazoles; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Indoles; Insulin; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Phosphatase; Oxazoles; Perfusion; Protein Kinase Inhibitors; Rats; Rats, Wistar; Shock, Hemorrhagic; Staurosporine; Tetradecanoylphorbol Acetate

2005
Regulation of erythrocyte Na-K-2Cl cotransport by threonine phosphorylation.
    Biochimica et biophysica acta, 2005, Aug-01, Volume: 1714, Issue:1

    Topics: Animals; Erythrocytes; Ferrets; Genistein; Magnesium; Marine Toxins; Microcystins; Molecular Weight; Oxazoles; Peptides, Cyclic; Phosphoprotein Phosphatases; Phosphorylation; Phosphothreonine; Protein Phosphatase 1; Pyrazoles; Pyrimidines; Sodium Potassium Chloride Symporter Inhibitors; Sodium-Potassium-Chloride Symporters; Staurosporine; Threonine

2005
Regulation of potassium transport in human lens epithelial cells.
    Experimental eye research, 2006, Volume: 82, Issue:1

    Topics: Bumetanide; Cell Line; Diuretics; Enzyme Inhibitors; Epithelial Cells; Ethylmaleimide; Furosemide; Genistein; Humans; Ion Transport; K Cl- Cotransporters; Lens, Crystalline; Marine Toxins; Ouabain; Oxazoles; Phosphoprotein Phosphatases; Potassium; Protein Kinase C; Protein Phosphatase 1; Protein-Tyrosine Kinases; Rubidium; Sodium-Potassium-Chloride Symporters; Sodium-Potassium-Exchanging ATPase; Staurosporine; Symporters

2006
Ser-2030, but not Ser-2808, is the major phosphorylation site in cardiac ryanodine receptors responding to protein kinase A activation upon beta-adrenergic stimulation in normal and failing hearts.
    The Biochemical journal, 2006, May-15, Volume: 396, Issue:1

    Topics: Adrenergic beta-Agonists; Animals; Arrhythmias, Cardiac; Benzylamines; Blotting, Western; Calcium Signaling; Carrier Proteins; Cell Line; Cyclic AMP-Dependent Protein Kinases; Heart Failure; Humans; Ion Channel Gating; Ion Transport; Isoproterenol; Kidney; Marine Toxins; Mice; Myocytes, Cardiac; Oxazoles; Peptide Fragments; Phosphoprotein Phosphatases; Phosphorylation; Phosphoserine; Protein Processing, Post-Translational; Protein Serine-Threonine Kinases; Rabbits; Rats; Recombinant Fusion Proteins; Ryanodine Receptor Calcium Release Channel; Sodium-Calcium Exchanger; Staurosporine; Structure-Activity Relationship; Sulfonamides; Transfection

2006
Both Ca2+ -dependent and -independent pathways are involved in rat hepatic stellate cell contraction and intrahepatic hyperresponsiveness to methoxamine.
    American journal of physiology. Gastrointestinal and liver physiology, 2007, Volume: 292, Issue:2

    Topics: Actomyosin; Amides; Animals; Calcimycin; Calcium; Cell Shape; Cells, Cultured; Diacetyl; Enzyme Inhibitors; Liver; Male; Marine Toxins; Methoxamine; Myocytes, Cardiac; Myocytes, Smooth Muscle; Myosin-Light-Chain Kinase; Oxazoles; Protein Kinase Inhibitors; Pyridines; Rats; Rats, Wistar; Signal Transduction; Staurosporine; Sulfonamides; Vasoconstrictor Agents

2007
Shrinkage insensitivity of NKCC1 in myosin II-depleted cytoplasts from Ehrlich ascites tumor cells.
    American journal of physiology. Cell physiology, 2007, Volume: 292, Issue:5

    Topics: Actins; Animals; Bumetanide; Carcinoma, Ehrlich Tumor; Cell Membrane; Cell Size; Cell-Free System; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Female; Hypertonic Solutions; Isoquinolines; Marine Toxins; Mice; Myosin Type II; Myosin-Light-Chain Kinase; Oxazoles; p38 Mitogen-Activated Protein Kinases; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Rubidium Radioisotopes; Sodium Potassium Chloride Symporter Inhibitors; Sodium-Potassium-Chloride Symporters; Solute Carrier Family 12, Member 2; Staurosporine; Sulfonamides

2007
Signalling pathways involved in the control of sperm cell volume.
    Reproduction (Cambridge, England), 2007, Volume: 133, Issue:1

    Topics: Animals; Cell Size; Cells, Cultured; Chloride Channels; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Indoles; Ion Channels; Male; Maleimides; Marine Toxins; Okadaic Acid; Osmosis; Oxazoles; Papaverine; Phosphoprotein Phosphatases; Protein Kinase C; Signal Transduction; Spermatozoa; Staurosporine; Swine

2007
Protease activation and the signal transduction pathway regulating motility in sperm from the water strider Aquarius remigis.
    Cytoskeleton (Hoboken, N.J.), 2012, Volume: 69, Issue:4

    Topics: Animals; Calcium; Egtazic Acid; Heteroptera; Male; MAP Kinase Signaling System; Marine Toxins; Oxazoles; Phosphorylation; Protein Kinase Inhibitors; Protein Kinases; Receptor, PAR-2; Signal Transduction; Sperm Motility; Spermatozoa; Staurosporine; Thapsigargin; Trypsin

2012
The Mechanism of Action of Ghrelin and Motilin in the Pacemaker Potentials of Interstitial Cells of Cajal from the Murine Small Intestine.
    Molecules and cells, 2019, Jun-30, Volume: 42, Issue:6

    Topics: Acetophenones; Amides; Animals; Benzopyrans; Boron Compounds; Calcium; Carbazoles; Gastrointestinal Motility; Ghrelin; Inositol 1,4,5-Trisphosphate Receptors; Interstitial Cells of Cajal; Intestine, Small; Macrocyclic Compounds; Membrane Potentials; Mice; Mice, Inbred ICR; Motilin; Oligopeptides; Oxazoles; Protein Kinase C; Pyridines; Receptors, Ghrelin; rho-Associated Kinases; Signal Transduction; Staurosporine; Thapsigargin

2019
Solvent-Induced Protein Precipitation for Drug Target Discovery on the Proteomic Scale.
    Analytical chemistry, 2020, 01-07, Volume: 92, Issue:1

    Topics: Acetic Acid; Acetone; Cells, Cultured; Drug Discovery; Drug Evaluation, Preclinical; Ethanol; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; HSP90 Heat-Shock Proteins; Humans; Methotrexate; NADH Dehydrogenase; Oxazoles; Proteomics; Solvents; Staurosporine; Thiazoles

2020