Page last updated: 2024-08-21

oxazoles and rilmenidine

oxazoles has been researched along with rilmenidine in 341 studies

Research

Studies (341)

TimeframeStudies, this research(%)All Research%
pre-199061 (17.89)18.7374
1990's157 (46.04)18.2507
2000's99 (29.03)29.6817
2010's24 (7.04)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Guillet, C; Passeron, J1
Hamilton, CA; Howie, CA; Reid, JL; Yakubu, MA1
Berger, SB; Maiese, K; Pek, L; Reis, DJ1
Christen, O; Göthert, M; Michel, MC; Molderings, GJ; Schäfer, SG1
Belcourt, A; Bousquet, P; Bricca, G; Dontenwill, M; Feldman, J; Greney, H; Stutzmann, J; Tibirica, E1
Gundlach, AL; Jarrott, B; King, PR; Louis, WJ2
Harron, DW3
Laurent, S; Safar, M1
Barrès, C; Koenig-Bérard, E; Sannajust, F; Sassard, J1
Cerutti, C; Koenig-Bérard, E; Sannajust, F; Sassard, J1
Head, GA; Sannajust, F4
Bousquet, P; Gonon, F; Mermet, C; Suaud-Chagny, MF; Tibiriça, E1
Harron, DW; McKaigue, JP1
Macrae, IM; McAuley, MA; Reid, JL1
Berger, SB; Golanov, EV; Reis, DJ; Yamamoto, S1
Ernsberger, P; Feinland, G; Gomez, RE; Reis, DJ1
Beevers, DG; Bulpitt, CJ; Dollery, CT; Fletcher, AE; Wilkinson, R1
Bousquet, P; Feldman, J; Gonon, F; Mermet, C; Monassier, L; Tibiriça, E1
Bidet, M; Parini, A; Poujeol, P2
Frutoso, J; Geelen, G; Ghaemmaghami, F; Gharib, C; Ibanez, J; Vincent, M1
Burke, S; Head, GA1
Smits, JF; Struyker-Boudier, HA1
Frank, R; Grosgogeat, Y; Guillet, C; Jondeau, G; Poulain, F; Tonet, J; Vivet, P1
De Mey, JG; Eerdmans, PH; Struyker Boudier, HA1
Harron, DW; Spiers, JP; Wilson, R1
Belcourt, A; Bousquet, P; Bricca, G; Dontenwill, M; Feldman, J1
Hamilton, CA; Howie, CA; Jardine, E; Reid, JL; Yakubu, MA1
Dhib, M; Fillastre, JP1
Belcourt, A; Bousquet, P; Bricca, G; Dontenwill, M; Feldman, J; Tibiriça, E1
Dresse, A; Scuvée-Moreau, J1
Doyle, AE; Jarrott, B; Lewis, SJ2
Fillastre, JP1
Damase-Michel, C; Dard, B; Macquin-Mavier, I; Montastruc, JL; Tran, MA; Valet, P1
Corcoran, C; Mansy, S; Wilkinson, R1
Fiorentini, C; Guazzi, M; Guillet, C1
Pannier, B; Safar, M1
Safar, ME2
Callens-el Amrani, F; Paolaggi, F; Swynghedauw, B2
Belcourt, A; Bousquet, P; Bricca, G; Dontenwill, M; Feldman, J; Molines, A; Tibirica, E3
Coupry, I; Koenig, E; Lachaud, V; Parini, A; Podevin, RA2
Li, CG; Rand, MJ2
Damase-Michel, C; Koenig-Berard, E; Macquin-Mavier, I; Montastruc, JL; Tran, MA; Valet, P1
Dinh Xuan, AT; Lockhart, A1
Leary, WP1
Mahieux, F1
Barrès, C; Cerutti, C; Julien, C; Koenig-Bérard, E; Sannajust, F; Sassard, J1
Bidet, M; Coupry, I; Lachaud, V; Parini, A; Podevin, RA; Poujeol, P1
Bromet, N; Genissel, P1
Ketelslegers, JM; Lambert, AE; Mpoy, M; Vandeleene, B2
Dall, JL1
Brisgand, B; Daelemans, R; Dratwa, M; Lameire, N; Lins, RL; Sennesael, J; Verbeelen, D1
Ausiello, M; Brignoli, M; de Divitiis, O; Di Somma, S; Galderisi, M; Liguori, V; Magnotta, C; Natale, N; Petitto, M1
Davies, DS; Murray, S; Watson, D1
Ehrhardt, JD1
de Jonge, A; Jonkman, FA; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Al-Damluji, S; Besser, GM; Grossman, A; Turner, P; Weerasuriya, K1
Fourtillan, JB; Girault, J; Lefebvre, MA; Mignot, A; Ung, HL1
Beau, B; Delbarre, G; Koenig-Berard, E; Labrid, C; Lhoste, F; Tierney, C1
Dresse, A; Scuvée-Moreau, J; Seutin, V1
Koenig-Berard, E; Nadaud, D; Stinus, L; Tierney, C1
Doyle, AE; Jarrott, B; Lewis, SJ; Louis, WJ1
Clerici, C; Harf, A; Macquin-Mavier, I1
Albin, H; Bromet, N; Fourtillan, JB; Genissel, P; Mignot, A1
Ehrhardt, JD; Genissel, P; Pozet, N; Singlas, E; Zech, P1
Van Zwieten, PA4
Davies, DS; Dollery, CT; Duchier, J; Pannier, B; Safar, ME1
Aliot, E; Florentin, J; Gilgenkrantz, JM; Saulnier, JP; Zannad, F1
Levy, B; N'guyen van Cao, A; Slama, R1
Brisgand, B; Fillastre, JP; Ostermann, G; Schmitt, J1
Fillastre, JP; Galinier, F; Le Bihan, G; Letac, B; Schwartz, J1
Galley, P; Hessel, JL; Manciet, G; Michel, JP1
Beau, B; Brisgand, B; Laurin, S; Mahieux, F; Paraire, M; Vitou, P1
Bourreau, JP; Tricoche, R1
Advenier, C; Dinh Xuan, AT; Lockhart, A; Matran, R; Regnard, J; Vitou, P1
Anglade, F; Damase-Michel, C; Dang Tran, L; de Saint-Blanquat, G; Koenig-Berard, E; Montastruc, JL; Tran, MA; Valet, P1
Herman, AG; Jordaens, FH; Verbeuren, TJ; Zonnekeyn, LL1
Coupry, I; Dausse, JP; Koenig, E; Lachaud, V; Parini, A; Podevin, RA1
Beau, B; Begue, JM; Bromet, N; Du Vignaud, P; Genissel, P; Grislain, L; Guillouzo, A; Mocquard, MT; Ratanasavanh, D1
Shaw, E; Turner, P; Weerasuriya, K1
Dampney, RA; Li, YW1
Gregoire, JR; Sheps, SG1
Starke, K; Szabo, B; Urban, R3
Advenier, C; Biyah, K1
Jacob, R; Rupp, H1
Gundlach, AL; King, PR; Louis, WJ; Suzuki, S2
Bramwell, S; Regunathan, S; Reis, DJ1
Penner, SB; Smyth, DD3
Combes-George, M; Mory, G; Nechad, M; Parini, A; Tesson, F1
Head, GA2
Szabo, B; Urban, R2
Laragh, JH2
Elliott, HL; MacPhee, G; Panfilov, V; Reid, JL1
Chernobelski, M; Mayorov, D; Medvedev, O1
Gundlach, AL; King, PR; Louis, WJ2
Handley, SL; Jackson, HC; Jordan, S; Nutt, DJ1
Browne, SE; Macrae, IM2
García-Sevilla, JA; Pineda, J; Ugedo, L1
Hamilton, CA; Jardine, E; Reid, JL1
Gundlach, AL; King, PR; Louis, WJ; Nero, TL; Suzuki, S1
Godwin, SJ; Head, GA; Sannajust, F1
Cechetto, DF; Kline, RL; van der Mark, J1
Feinstein, DL; Golanov, EV; Regunathan, S; Reis, DJ1
DeLuca, N; Lorino, G; Rosiello, G; Rubattu, S; Sarno, D; Trimarco, B; Volpe, M1
Aparicio, M; Dratwa, M; el Esper, N; Fillastre, JP; Levaltier, B; Lins, R; Meyrier, A; Mignon, F; Ryckelynck, JP; Sennesael, J1
Corcoran, C; Coupez, G; Creytens, G; Opsomer, M; Pelemans, W; Van Dessel, A; Verhaeghe, J1
Codis, P; Fevrier, B; Pillion, G; Schutz, D1
Li, P; Penner, SB; Smyth, DD1
Christen, MO; Collins, LA; Dreshaj, I; Ernsberger, P; Graff, LM; Graves, ME; Grove, DL; Haxhiu, MA; Schäfer, SG1
Christen, O; Göthert, M; Molderings, GJ; Schäfer, SG1
Cechetto, DF; Kline, RL3
Janssen, BJ; Oosting, J; Struyker-Boudier, HA; Tyssen, CM1
Boucher, M; Chassaing, C; Dubar, M; Duchêne-Marullaz, P; Vivet, P1
Ambrosi, P; Lambert, M; Luccioni, R; Scemama, M1
Bousquet, P; Bricca, G; Dontenwill, M; Tibiriça, E1
Capuana, G; Guillet, C; Indovina, A; Licata, G; Lipari, R; Mazzola, G; Merlino, G; Parrinello, G; Scaglione, R1
Luccioni, R1
Anderson, WP; Evans, RG1
Elghozi, JL; Février, B; Girard, A1
Dabire, H; Levy, BI; Poitevin, P; Safar, ME1
Chan, CK; Head, GA; Sannajust, F1
Argenziano, L; De Luca, N; Iovino, G; Morisco, C; Russo, R; Sarno, D; Trimarco, B; Volpe, M1
Beucler, I; Dairou, F; Février, B; Scemama, M2
Hayashi, Y; Kamibayashi, T; Mammoto, T; Takada, K; Yamatodani, A; Yoshiya, I2
Donnelly, R; Morris, AD; Panfilov, V; Reid, JL1
Harron, DW; Hasson, B; King, DJ; McClelland, RJ; Regan, M1
Gargalidis-Moudanos, C; Parini, A1
Chudek, J; Nowicki, M; Wiecek, A1
Donnelly, R; Morris, AD; Panfilov, V; Reid, JL; Scemama, M1
Boucher, M; Chapuy, E; Chassaing, C; Dubar, M2
Fröhlich, R; Illes, P; Szabo, B1
Chan, CK; Head, GA1
Frishman, WH; Yu, A1
Boulanger, CM; Illiano, S; Marsault, R; Taddei, S; Vanhoutte, PM1
Chu, TC; Gluchowski, C; Hughes, BW; Potter, DE; Wong, W1
Johns, EJ; Zhang, T1
Bousquet, P; De Jong, W; Feldman, J; Monassier, L; Roegel, JC; Yannoulis, N1
Berthault, MF; Dubar, M; Ferré, P; Ktorza, A; Morin, J; Pénicaud, L2
Avellar, MC; Markus, RP1
Anderson, WP; Evans, RG; Fitzgerald, SM; Malpas, SC; Shweta, A1
Van den Buuse, M1
Hayashi, Y; Kamibayashi, T; Kitamura, S; Mammoto, T; Takada, K; Yamatodani, A; Yoshiya, I1
Lada, W1
Arrais, CA; Camargo, LA; Menani, JV; Renzi, A; Saad, R; Saad, WA; Silveira, JE1
Piletz, JE; Reis, DJ1
Cario-Toumaniantz, C; Loirand, G; Pacaud, P1
Kazaz, C; Sözmen, B; Sözmen, EY; Taşkiran, D; Tüzün, S1
Abdel-Rahman, AA; El-Mas, MM5
Arcade, B; Cribier, B; Grosshans, E; Michel, C1
Burke, SL; Chan, CK; Head, GA2
Bousquet, P; De Jong, W; Feldman, J; Roegel, JC; Yannoulis, N1
Bobik, A; Dilley, R; Kanellakis, P1
Balazovjech, I; Dubai, G; Dvorak, I; Januszewicz, W; Krupa-Wojciechowska, B; Kubasik, A; Kuch-Wocial, A; Polak, G; Sadowski, Z; Simon, K; Stejfa, M; Szwed, H1
Cechetto, DF; Dixon, SJ; Ozog, MA; Wilson, JX1
Ali, A; Cheng, HY; Ting, KN; Wilson, VG1
Burke, SL; Head, GA6
Gundlach, AL; Hosseini, AR; Iakovidis, D; Jackman, GP; King, PR; Louis, WJ; Nero, TL; Suzuki, S1
Gundlach, AL; Hosseini, AR; Jackman, GP; King, PR; Louis, WJ1
Kunduzova, OR; Medvedev, OS; Medvedeva, NA; Murashev, AN3
Burke, SL; Head, GA; Malpas, SC1
Burke, SL; Head, GA; Tritton, SB; van den Buuse, M1
Godwin, SJ; Head, GA; Parkin, ML; Tortelli, CF1
Amah, G1
Blue, DR; Dillon, MP; Eglen, RM; Jasper, JR; Lesnick, JD; MacLennan, SJ; Zhu, QM2
Bock, C; Niederhoffer, N; Szabo, B1
Hébert, CA; Kudo, LH; Rouch, AJ1
Drzewoski, J; Wiśniewska-Jarosińska, M1
Ducher, M; Fauvel, JP; Laville, M; Najem, R; Ryon, B1
Bousquet, P; Brasili, L; Bruban, V; Dontenwill, M; Feldman, J; Giannella, M; Greney, H; Pigini, M1
Bock, C; Niederhoffer, N; Nordheim, U; Szabo, B1
Peters, SL; Van Zwieten, PA1
Bousquet, P; Feldman, J; Pompermayer, K; Salgado, MC1
Masek, K; Sevcík, J1
Bousquet, P; Feldman, J1
Robles, NR1
Bauduceau, B; Dupuy, O; Mayaudon, H3
Castro Resende, AC; Leão, MC; Lima, AF; Mesquita Ferreira, AG; Moreira, CF; Nunes, FR; Sena, KM; Silveira, SS; Soares de Moura, RS1
Polónia, J1
Kourilsky, O1
Argengiano, L; de Luca, N; Guerrera, L; Iovino, GL; Izzo, R; Trimarco, B1
Bousquet, P2
Esler, M1
Reid, JL2
Bönisch, H; Brüss, M; Göthert, M; Likungu, J; Molderings, GJ1
Spinar, J; Vítovec, J1
Argenziano, L; De Luca, N; Fontana, D; Iovino, G; Izzo, R; Trimarco, B; Vecchione, C1
Schachter, M1
Bousquet, P; Bruban, V; Feldman, J; Sy, GY1
Burke, SL; Head, GA; Mayorov, DN1
Abdel-Rahman, AA; El-Mas, MM; Zhang, J1
Bousquet, P; Bruban, V; Ehrhardt, JD; Feldman, J; Pfeiffer, B; Pompermayer, K; Renard, P; Scalbert, E; Schann, S1
Cohen, AF; de Visser, SJ; Schoemaker, RC; van Gerven, JM1
Fritz, T; Szabo, B; Wedzony, K1
Burke, SL; Head, GA; Sannajust, FJ1
Head, GA; Janssen, BJ; Lukoshkova, EV1
Bousquet, P; Bruban, V; Ehrhardt, JD; Estato, V; Feldman, J; Monassier, L; Renard, P; Scalbert, E; Schann, S1
Nurminen, ML1
Kratochvíl'ová, H; Remková, A1
Abdel-Rahman, AA; Zhang, J4
Cohen, AF; de Visser, SJ; Nanhekhan, L; Schoemaker, RC; van der Post, JP; van Gerven, JM1
Choi, DH; Choi, SH; Chun, BG; Kim, DH; Park, YG1
Widimský, J1
Penner, SB; Pirnat, D; Smyth, DD1
Kourilsky, O; Meurin, P1
Bousquet, P; Catelli, M; Feldman, J; Tibirica, E1
Godwin, SJ; Head, GA; Parkin, ML1
Camilleri, G; Clerson, P; Portal, B; Quiniou, G1
Artigues-Varin, C; Mulder, P; Richard, V; Thuillez, C; Varin, R1
Khirmanov, VN1
Borbás, S; Dienes, BS; Farsang, C; Lengyel, M; Zorándi, A1
Bogdański, P; Bryl, W; Cymerys, M; Kujawska-Łuczak, M; Miczke, A; Pupek-Musialik, D1
Abdel-Rahman, AA; Li, G; Mao, L1
Koss, MC1
Ayan, F; Ikitimur, B; Koldas, L1
Buranakitjaroen, P; Kittipawong, P; Koanantakul, B; Piamsomboon, C; Prasassarakich, N; Silaraks, S; Sukonthasarn, A; Tiyapant, A1
Ernsberger, P; Koletsky, RJ; Velliquette, RA1
Burgdorf, C; Engelhardt, A; Kurz, T; Raasch, W; Richardt, G; Schäfer, U1
Bonisch, H; Bruss, M; Gothert, M; Molderings, GJ1
Forzley, B; Penner, SB; Pirnat, D; Smyth, DD1
Hefczyc, J; Konieczny, B; Kossmann, S; Szyguła, B; Szyguła, J1
Bousquet, P; Greney, H; Monassier, L; Thomas, L1
Abelson, KS; Höglund, AU1
Meredith, PA; Reid, JL1
Merwid-Lad, A; Misiuk-Hojło, M; Pieśniewska, M; Szaliński, M; Trocha, M1
Dardonville, C; Rozas, I1
de Arruda Camargo, LA; Guarda, IF; Guarda, RS; Saad, WA; Simões, S1
Esler, M; Hastings, J; Jennings, G; Lambert, G; Lux, A; Socratous, F1
Cohen, AF; de Visser, SJ; Schoemaker, RC; van der Post, JP; van Gerven, JM1
Celik, A; Kaya, D; Kerpeten, K; Kilit, C; Onrat, E1
Liebisch, B1
Araújo, CV; Bousquet, P; Estato, V; Tibiriçá, E1
Gerová, M; Matusková, J; Pecháòová, O; Török, J1
Anichkov, DA; Schastnaya, OV; Shostak, NA1
Abdel-Rahman, AA; Li, G; Wang, X2
Caillé, S; Georges, F; Le Moine, C; Stinus, L; Vouillac, C1
Adamczak, M; Nowak, Ł; Wiecek, A1
Briaud, S; Sannajust, F; Zhang, BL1
Kotanko, P1
Ernsberger, P; Kossover, R; Previs, SF; Velliquette, RA1
Bousquet, P; Feldman, J; Sy, GY1
Czarnecka, D; Jaworski, R; Kawecka-Jaszcz, K; Klocek, M; Kucharska, M; Pachocki, R; Zabojszcz, M1
Kasherininov, YR; Konrady, AO; Krutikov, AN; Shavarov, AA; Shavarova, EK; Shlyakhto, EV; Smirnova, EV; Vachrameeva, NV1
Cong, B; Li, F; Li, J; Lu, XQ; Su, RB; Wu, N; Xu, B; Zheng, JQ1
Catelli, MF; de Oliveira, MA; Moreira, PB; Nóbrega, AC; Rocha, NN; Teixeira de Castro, RR; Tibiriçá, E1
Sirotiaková, J; Widimský, J1
Alföldi, S; Elghozi, JL; Farsang, C; Finta, E; Laude, D1
Khansefid, N; Ladgevardi, MA; Sabetkasaie, M1
Abdel-Rahman, AA; Li, G1
Sica, DA1
Bousquet, PP; Monassier, LJ; Signolet, IL1
Hayashi, Y; Iwasaki, M; Kamibayashi, T; Mashimo, T; Yamatodani, A1
Avanza, AC; Mansur, AP; Ramires, JA1
Gyires, K; Zádori, Z1
Abdel-Rahman, AA; Bender, TS1
Dolezal, T; Krsiak, M; Soukupová, M2
Li, F; Li, J; Liu, Y; Lu, XQ; Su, RB; Wu, N1
Al-Khrasani, M; Gyires, K; Mátyus, P; Mózes, MM; Pap, B; Shujaa, N; Zádori, ZS1
Groenewoud, G; Meyer, B; Potgieter, L1
Burke, SL; Evans, RG; Head, GA2
Bousquet, P; Lessa, MA; Nascimento, AR; Sabino, B; Tibiriçá, E1
Acevedo-Arozena, A; Brown, SD; Corrochano, S; Menzies, FM; Renna, M; Rose, C; Rubinsztein, DC; Sadiq, O1
Chytil, L; Cvačka, J; Marešová, V; Slanař, O; Štícha, M; Štrauch, B; Widimský, J1
Hayashi, Y; Iwasaki, M; Kamibayashi, T; Mashimo, T; Yamanaka, H; Yamatodani, A1
Bakan, E; Borekci, B; Kumbasar, S; Kumtepe, Y; Salman, S; Suleyman, H; Yilmaz, M1
Chen, CT; Cheng, JT; Cheng, KC; Lin, KC; Niu, CS; Wu, HT1
Chen, CT; Cheng, JT; Chi, CW; Chung, HH; Wu, HT; Yang, PS; Yeh, CH1
Bellinger, DL; Ghamsary, M; Kozic, B; Lorton, D; Lubahn, CL; Molinaro, CA; Perez, SD; Thyagarajan, S1
Chen, MF; Cheng, JT; Chou, MT; Chung, HH; Yang, TT1
Agbaba, D; Gemovic, B; Nikolic, K; Srdic-Rajic, T; Veljkovic, N1
Al-Khrasani, M; Brancati, SB; Fehér, Á; Gyires, K; Hein, L; Lackó, E; Mátyus, P; Tóth, VE; Zádori, ZS1
Cheng, J; Chung, HH1
Davern, PJ; Head, GA; Jackson, KL; Nguyen-Huu, TP; Palma-Rigo, K1
Lin, F; Qin, ZH1
Eisenstein, M1
Bento, CF; Deretic, V; Rubinsztein, DC1
Cavic, M; Djokic, I; Gemovic, B; Nikolic, K; Perovic, V; Srdic-Rajic, T; Veljkovic, N1
Bousquet, P; Gomes, F; Gonçalves-de-Albuquerque, CF; Lessa, MA; Machado, MV; Nascimento, AR; Tibiriçá, E; Vieira, AB1
Agbaba, D; Azzali, E; Costantino, G; Glisic, S; Laurila, JM; Nikolic, K; Perovic, V; Pieroni, M; Radi, M; Scheinin, M; Srdic-Rajic, T; Tassini, S; Veljkovic, N; Vucicevic, J1
Burke, SL; Head, GA; Jackson, KL; Lim, K1
Beart, PM; Higgins, GC; Lau, CL; Lawrence, AJ; Mercer, LD1
Barker, RA; Green-Thompson, ZW; Griffin, J; Jones, PS; Lazic, SE; Mason, SL; Pugh, PJ; Rowe, JB; Rubinsztein, DC; Underwood, BR1

Reviews

49 review(s) available for oxazoles and rilmenidine

ArticleYear
[Imidazole receptors: site of action of a new generation of antihypertensive drugs. Current status and future prospects].
    Deutsche medizinische Wochenschrift (1946), 1992, Jan-10, Volume: 117, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Binding Sites; Cattle; Humans; Imidazoles; Oxazoles; Rats; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine

1992
Imidazoline receptors. A new concept in central regulation of the arterial blood pressure.
    American journal of hypertension, 1992, Volume: 5, Issue:4 Pt 2

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Clonidine; Hypertension; Imidazoline Receptors; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine

1992
Distinctive features of rilmenidine possibly related to its selectivity for imidazoline receptors.
    American journal of hypertension, 1992, Volume: 5, Issue:4 Pt 2

    Topics: Adrenergic alpha-Agonists; Animals; Chickens; Dogs; Humans; Hypertension; Imidazoline Receptors; Mice; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine

1992
Rilmenidine: a novel approach to first-line treatment of hypertension.
    American journal of hypertension, 1992, Volume: 5, Issue:4 Pt 2

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Oxazoles; Rilmenidine

1992
Clinical pharmacology of imidazolines and related compounds.
    Fundamental & clinical pharmacology, 1992, Volume: 6 Suppl 1

    Topics: Adrenergic alpha-Agonists; Humans; Imidazoles; Oxazoles; Rilmenidine

1992
[Current data on the pharmacology of rilmenidine].
    Archives des maladies du coeur et des vaisseaux, 1989, Volume: 82 Spec No 5

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Hypnotics and Sedatives; Oxazoles; Rilmenidine; Sympathetic Nervous System

1989
New concepts on the central regulation of blood pressure. Alpha 2-adrenoceptors and "imidazoline receptors".
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Adrenergic alpha-Agonists; Animals; Binding, Competitive; Blood Pressure; Brain; Clonidine; Humans; Imidazoles; Oxazoles; Receptors, Adrenergic, alpha; Rilmenidine

1989
Recent advances in the pharmacology of rilmenidine.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Brain; Hemodynamics; Oxazoles; Peripheral Nerves; Rilmenidine; Sympatholytics

1989
Rilmenidine: a novel antihypertensive agent.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Brain; Humans; Hypertension; Oxazoles; Rilmenidine; Wakefulness

1989
Bronchial effects of alpha 2-adrenoceptor agonists and of other antihypertensive agents in asthma.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Asthma; Bronchi; Calcium Channel Blockers; Clonidine; Humans; Hypertension; Oxazoles; Rilmenidine

1989
Rilmenidine and vigilance. Review of clinical studies.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Arousal; Blood Pressure; Double-Blind Method; Humans; Hypertension; Oxazoles; Random Allocation; Rilmenidine; Wakefulness

1989
Newer antihypertensive drugs.
    Current opinion in cardiology, 1995, Volume: 10, Issue:5

    Topics: Antihypertensive Agents; Dibenzothiepins; Humans; Imidazoles; Methionine; Oxazoles; Piperazines; Protease Inhibitors; Rilmenidine

1995
Importance of imidazoline receptors in the cardiovascular actions of centrally acting antihypertensive agents.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-2 Receptor Agonists; Agmatine; Animals; Antihypertensive Agents; Baroreflex; Female; Imidazoline Receptors; Kidney; Male; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

1995
Rilmenidine and the high risk hypertensive patient.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Animals; Antihypertensive Agents; Humans; Hypertension; Kidney; Oxazoles; Renin; Rilmenidine; Risk Factors; Sympathetic Nervous System

1995
Clinical pharmacology of drugs acting on imidazoline and adrenergic receptors. Studies with clonidine, moxonidine, rilmenidine, and atenolol.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Antihypertensive Agents; Atenolol; Clinical Trials as Topic; Clonidine; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Placebos; Receptors, Adrenergic; Receptors, Drug; Reference Values; Rilmenidine

1995
Protection of focal ischemic infarction by rilmenidine in the animal: evidence that interactions with central imidazoline receptors may be neuroprotective.
    The American journal of cardiology, 1994, Dec-22, Volume: 74, Issue:13

    Topics: Adrenergic alpha-Agonists; Animals; Brain Ischemia; Cerebral Infarction; Dioxanes; Idazoxan; Imidazoles; Imidazoline Receptors; Neurons; Neuroprotective Agents; Oxazoles; Receptors, Drug; Rilmenidine

1994
The high-risk hypertensive patient and the potential for brain imidazoline receptor binding by rilmenidine.
    The American journal of cardiology, 1994, Dec-22, Volume: 74, Issue:13

    Topics: Animals; Brain; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine; Risk Factors

1994
[Imidazole receptors and blood pressure regulation. High receptor selectivity of moxonidine].
    Deutsche medizinische Wochenschrift (1946), 1993, Jun-25, Volume: 118, Issue:25

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Blood Pressure; Cats; Clonidine; Humans; Hypertension; Imidazoles; Oxazoles; Rabbits; Rats; Receptors, Drug; Rilmenidine

1993
[The imidazoline receptor and the central regulation of arterial pressure].
    Pathologie-biologie, 1993, Volume: 41, Issue:7

    Topics: Blood Pressure; Catecholamines; Central Nervous System; Clonidine; Humans; Hypertension; Imidazoline Receptors; Oxazoles; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine

1993
[Imidazol receptor agonists--new possibilities for treating hypertension].
    Postepy higieny i medycyny doswiadczalnej, 1995, Volume: 49, Issue:5

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Hemodynamics; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1995
Imidazoline receptor agonist drugs: a new approach to the treatment of systemic hypertension.
    Journal of clinical pharmacology, 1996, Volume: 36, Issue:2

    Topics: Animals; Antihypertensive Agents; Clinical Trials as Topic; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1996
From alpha and beta to I1: an overview of sympathetic receptors involved in blood pressure control targets for drug treatment.
    Journal of cardiovascular pharmacology, 1996, Volume: 27 Suppl 3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Drug; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Rilmenidine

1996
[Imidazoline receptors and use of drug blocking receptors I1].
    Polski merkuriusz lekarski : organ Polskiego Towarzystwa Lekarskiego, 1996, Volume: 1, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Antihypertensive Agents; Arrhythmias, Cardiac; Cimetidine; Histamine H2 Antagonists; Humans; Hypertension; Imidazoles; Myocardial Infarction; Oxazoles; Rilmenidine

1996
The imidazoline receptor in control of blood pressure by clonidine and allied drugs.
    The American journal of physiology, 1997, Volume: 273, Issue:5

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Humans; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Neurons; Oxazoles; Receptors, Drug; Rilmenidine

1997
Central imidazoline (I1) receptors as targets of centrally acting antihypertensives: moxonidine and rilmenidine.
    Journal of hypertension, 1997, Volume: 15, Issue:2

    Topics: Animals; Antihypertensive Agents; Brain; Humans; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1997
Sympatho-adrenal mechanisms regulating cardiovascular hypertrophy in primary hypertension: a role for rilmenidine?
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1998, Volume: 16, Issue:3

    Topics: Adrenal Glands; Animals; Antihypertensive Agents; Blood Vessels; Cardiomegaly; Humans; Hypertension; Hypertrophy; Norepinephrine; Oxazoles; Rilmenidine; Sympathetic Nervous System

1998
[Clinical pharmacology of hypotensive drugs acting on central imidazoline receptors].
    Polskie Archiwum Medycyny Wewnetrznej, 1998, Volume: 100, Issue:6

    Topics: Antihypertensive Agents; Clonidine; Drug Interactions; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1998
Central I1-imidazoline receptors as targets of centrally acting antihypertensive drugs. Clinical pharmacology of moxonidine and rilmenidine.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Brain; Clinical Trials as Topic; Clonidine; Hemodynamics; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1999
[New, modern, centrally active antihypertensive agents in the treatment of essential hypertension].
    Casopis lekaru ceskych, 1999, Jun-07, Volume: 138, Issue:12

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Imidazoles; Medulla Oblongata; Oxazoles; Rilmenidine

1999
Drugs acting on imidazoline receptors: a review of their pharmacology, their use in blood pressure control and their potential interest in cardioprotection.
    Drugs, 1999, Volume: 58, Issue:5

    Topics: Animals; Antihypertensive Agents; Arrhythmias, Cardiac; Clinical Trials as Topic; Heart Failure; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1999
[New perspectives in the treatment of hypertension: the contribution of rilmenidine].
    Revista portuguesa de cardiologia : orgao oficial da Sociedade Portuguesa de Cardiologia = Portuguese journal of cardiology : an official journal of the Portuguese Society of Cardiology, 2000, Volume: 19 Suppl 2

    Topics: Antihypertensive Agents; Humans; Hypertension; Oxazoles; Rilmenidine

2000
Clinical benefits of rilmenidine.
    Revista portuguesa de cardiologia : orgao oficial da Sociedade Portuguesa de Cardiologia = Portuguese journal of cardiology : an official journal of the Portuguese Society of Cardiology, 2000, Volume: 19 Suppl 2

    Topics: Adult; Aged; Antihypertensive Agents; Clinical Trials as Topic; Humans; Hypertension; Insulin Resistance; Middle Aged; Multicenter Studies as Topic; Oxazoles; Rilmenidine

2000
The contribution of I1-selective agents in the management of syndrome X.
    Revista portuguesa de cardiologia : orgao oficial da Sociedade Portuguesa de Cardiologia = Portuguese journal of cardiology : an official journal of the Portuguese Society of Cardiology, 2000, Volume: 19 Suppl 2

    Topics: Antihypertensive Agents; Humans; Imidazoline Receptors; Insulin Resistance; Microvascular Angina; Oxazoles; Receptors, Drug; Rilmenidine

2000
Identification and characterization of I1 imidazoline receptors: their role in blood pressure regulation.
    American journal of hypertension, 2000, Volume: 13, Issue:6 Pt 2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Humans; Imidazoline Receptors; Oxazoles; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine

2000
I1 imidazoline receptors in cardiovascular regulation: the place of rilmenidine.
    American journal of hypertension, 2000, Volume: 13, Issue:6 Pt 2

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Cardiovascular Physiological Phenomena; Humans; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

2000
The sympathetic system and hypertension.
    American journal of hypertension, 2000, Volume: 13, Issue:6 Pt 2

    Topics: Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Norepinephrine; Oxazoles; Rilmenidine; Sympathetic Nervous System

2000
Rilmenidine: a clinical overview.
    American journal of hypertension, 2000, Volume: 13, Issue:6 Pt 2

    Topics: Albuminuria; Animals; Antihypertensive Agents; Diabetic Angiopathies; Humans; Hyperlipidemias; Hypertension; Hypertrophy, Left Ventricular; Insulin Resistance; Oxazoles; Rilmenidine; Treatment Outcome

2000
Efficacy of rilmenidine, a selective I1 imidazoline receptor binding agent in diabetic hypertensive patients.
    American journal of hypertension, 2000, Volume: 13, Issue:6 Pt 2

    Topics: Antihypertensive Agents; Clinical Trials as Topic; Diabetic Angiopathies; Humans; Hypertension; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

2000
Metabolic effects of moxonidine and other centrally acting antihypertensives.
    Diabetes, obesity & metabolism, 1999, Volume: 1, Issue:6

    Topics: Animals; Antihypertensive Agents; Diabetes Complications; Humans; Hypertension; Imidazoles; Insulin Resistance; Metabolism; Oxazoles; Rilmenidine; Sympathetic Nervous System; Sympatholytics; Syndrome

1999
I1 receptors, cardiovascular function, and metabolism.
    American journal of hypertension, 2001, Volume: 14, Issue:11 Pt 2

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Cardiovascular System; Clonidine; Humans; Hypertension; Imidazoline Receptors; Kidney; Oxazoles; Pancreas; Receptors, Drug; Rilmenidine; Treatment Outcome

2001
Update on rilmenidine: clinical benefits.
    American journal of hypertension, 2001, Volume: 14, Issue:11 Pt 2

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Humans; Hypertension; Oxazoles; Rilmenidine; Risk Factors; Treatment Outcome

2001
[Central nervous system as a target for the new antihypertensive agents].
    Duodecim; laaketieteellinen aikakauskirja, 1999, Volume: 115, Issue:20

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Autonomic Fibers, Preganglionic; Brain; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Oxazoles; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Sympatholytics

1999
[Albarel (rilmenidin)--a selective I1 imidazole receptor agonist. Pharmacologic properties and experience in clinical use].
    Terapevticheskii arkhiv, 2003, Volume: 75, Issue:2

    Topics: Antihypertensive Agents; Humans; Imidazoles; Oxazoles; Rilmenidine

2003
Centrally acting imidazoline I1-receptor agonists: do they have a place in the management of hypertension?
    American journal of cardiovascular drugs : drugs, devices, and other interventions, 2001, Volume: 1, Issue:5

    Topics: Animals; Antihypertensive Agents; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

2001
Imidazoline binding sites and their ligands: an overview of the different chemical structures.
    Medicinal research reviews, 2004, Volume: 24, Issue:5

    Topics: Amidines; Animals; Antihypertensive Agents; Binding Sites; Carbolines; Guanidines; Humans; Imidazoles; Imidazoline Receptors; Ligands; Oxazoles; Receptors, Drug; Rilmenidine; Structure-Activity Relationship

2004
Cause and consequences of sympathetic hyperactivity in chronic kidney disease.
    Blood purification, 2006, Volume: 24, Issue:1

    Topics: Adrenergic alpha-Agonists; Angiotensin II; Angiotensin II Type 1 Receptor Blockers; Arginine; Brain Stem; Humans; Hyperkinesis; Hypertension, Renal; Imidazoles; Kidney Failure, Chronic; Nitric Oxide Synthase; Oxazoles; Receptor, Angiotensin, Type 1; Renal Dialysis; Rilmenidine; Sympathetic Nervous System; Sympatholytics

2006
Centrally acting antihypertensive agents: an update.
    Journal of clinical hypertension (Greenwich, Conn.), 2007, Volume: 9, Issue:5

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Blood Pressure; Clonidine; Contraindications; Guanabenz; Guanfacine; Humans; Hypertension; Imidazoles; Methyldopa; Oxazoles; Rilmenidine

2007
Degradation of misfolded proteins by autophagy: is it a strategy for Huntington's disease treatment?
    Journal of Huntington's disease, 2013, Volume: 2, Issue:2

    Topics: Autophagy; Carbamazepine; Humans; Huntingtin Protein; Huntington Disease; Lithium; Mutant Proteins; Nerve Tissue Proteins; Oxazoles; Peptides; Rilmenidine; Sirolimus; Trehalose; Trinucleotide Repeat Expansion; Valproic Acid

2013
Therapeutic targeting of autophagy in neurodegenerative and infectious diseases.
    The Journal of experimental medicine, 2015, Jun-29, Volume: 212, Issue:7

    Topics: Autophagy; Communicable Diseases; Gene Expression Regulation; Humans; Models, Biological; Neurodegenerative Diseases; Oxazoles; Rilmenidine; Signal Transduction; Trehalose

2015

Trials

59 trial(s) available for oxazoles and rilmenidine

ArticleYear
[Treatment with rilmenidine 1 mg per day: time-lag to maximum response. A multicenter ambulatory study. Le Groupe Français d'étude Multicentrique d'Hyperium].
    Presse medicale (Paris, France : 1983), 1992, Dec-12, Volume: 21, Issue:43

    Topics: Adult; Aged; Aged, 80 and over; Antihypertensive Agents; Blood Pressure Determination; Female; Humans; Hypertension; Male; Middle Aged; Oxazoles; Placebos; Rilmenidine

1992
Clinical pharmacology of imidazolines and related compounds.
    Fundamental & clinical pharmacology, 1992, Volume: 6 Suppl 1

    Topics: Adrenergic alpha-Agonists; Humans; Imidazoles; Oxazoles; Rilmenidine

1992
The effects of two centrally-acting anti-hypertensive drugs on the quality of life.
    European journal of clinical pharmacology, 1991, Volume: 41, Issue:5

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Blood Pressure; Female; Humans; Hypertension; Male; Methyldopa; Middle Aged; Oxazoles; Quality of Life; Rilmenidine

1991
Antihypertensive drugs and baroreflex sensitivity. Effects of rilmenidine.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Adult; Antihypertensive Agents; Autonomic Nervous System; Blood Pressure; Double-Blind Method; Humans; Male; Nitroglycerin; Oxazoles; Phenylephrine; Pressoreceptors; Random Allocation; Reflex; Rilmenidine

1989
[Effects of rilmenidine on the central nervous system and kidney].
    Archives des maladies du coeur et des vaisseaux, 1989, Volume: 82 Spec No 5

    Topics: Antihypertensive Agents; Central Nervous System; Humans; Hypertension; Kidney; Oxazoles; Rilmenidine; Time Factors

1989
[Efficacy and acceptability of rilmenidine in mild to moderate arterial hypertension. A multicenter, randomized, double-blind trial, in comparison with methyldopa in 157 patients].
    Archives des maladies du coeur et des vaisseaux, 1989, Volume: 82 Spec No 5

    Topics: Adult; Antihypertensive Agents; Double-Blind Method; Female; Humans; Hypertension; Male; Methyldopa; Multicenter Studies as Topic; Oxazoles; Randomized Controlled Trials as Topic; Rilmenidine

1989
[Multicenter, double-blind study comparing rilmenidine 1 mg and hydrochlorothiazide 25 mg in 244 patients].
    Archives des maladies du coeur et des vaisseaux, 1989, Volume: 82 Spec No 5

    Topics: Adolescent; Adult; Aged; Antihypertensive Agents; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hydrochlorothiazide; Hypertension; Male; Middle Aged; Multicenter Studies as Topic; Oxazoles; Rilmenidine; Time Factors

1989
[Effects of rilmenidine on arterial parameters in essential arterial hypertension].
    Archives des maladies du coeur et des vaisseaux, 1989, Volume: 82 Spec No 5

    Topics: Antihypertensive Agents; Arm; Blood Pressure; Double-Blind Method; Hemodynamics; Humans; Hypertension; Middle Aged; Oxazoles; Pulsatile Flow; Randomized Controlled Trials as Topic; Rilmenidine; Vascular Resistance

1989
Renal excretory actions of antihypertensive agents. Effects of rilmenidine.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Adolescent; Adrenergic beta-Antagonists; Adult; Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Diuretics; Double-Blind Method; Drug Interactions; Electrolytes; Humans; Hydrochlorothiazide; Kidney; Male; Oxazoles; Rilmenidine; Vasodilator Agents

1989
Rilmenidine and vigilance. Review of clinical studies.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Arousal; Blood Pressure; Double-Blind Method; Humans; Hypertension; Oxazoles; Random Allocation; Rilmenidine; Wakefulness

1989
Effort blood pressure control in the course of antihypertensive treatment.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Adult; Antihypertensive Agents; Blood Pressure; Double-Blind Method; Exercise Test; Female; Humans; Hydrochlorothiazide; Hypertension; Male; Middle Aged; Oxazoles; Physical Exertion; Random Allocation; Rest; Rilmenidine

1989
Alpha 2-adrenoceptor agonists stimulate growth hormone secretion but have no acute effects on plasma cortisol under basal conditions.
    Hormone research, 1987, Volume: 25, Issue:2

    Topics: Adrenergic alpha-Agonists; Adult; Clonidine; Growth Hormone; Humans; Hydrocortisone; Male; Oxazoles; Rilmenidine

1987
Dose and concentration-effect relations for rilmenidine.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Administration, Oral; Adolescent; Adrenergic alpha-Agonists; Adult; Blood Pressure; Dose-Response Relationship, Drug; Female; Heart Rate; Humans; Hypertension; Hypnotics and Sedatives; Male; Oxazoles; Rilmenidine; Saliva; Secretory Rate; Xerostomia

1988
Efficacy and acceptability of rilmenidine for mild to moderate systemic hypertension.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic beta-Agonists; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Female; Humans; Hypertension; Male; Middle Aged; Oxazoles; Random Allocation; Rilmenidine; Xerostomia

1988
A multicenter double-blind comparative study of rilmenidine and clonidine in 333 hypertensive patients.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic beta-Agonists; Adult; Aged; Aged, 80 and over; Blood Pressure; Clinical Trials as Topic; Clonidine; Double-Blind Method; Female; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine

1988
Antihypertensive efficacy and acceptability of rilmenidine in elderly hypertensive patients.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic alpha-Agonists; Aged; Aged, 80 and over; Blood Pressure; Clinical Trials as Topic; Female; Humans; Hypertension; Male; Methyldopa; Oxazoles; Patient Compliance; Random Allocation; Rilmenidine; Supination

1988
Efficacy and safety of rilmenidine for arterial hypertension.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic alpha-Agonists; Adult; Aged; Aged, 80 and over; Blood Pressure; Clinical Trials as Topic; Double-Blind Method; Drug Therapy, Combination; Eye; Female; Glucose; Humans; Hypertension; Lipid Metabolism; Male; Middle Aged; Oxazoles; Random Allocation; Rilmenidine

1988
Comparative effects of rilmenidine and clonidine on bronchial responses to histamine in asthmatic subjects.
    British journal of clinical pharmacology, 1988, Volume: 26, Issue:6

    Topics: Adrenergic alpha-Agonists; Adult; Asthma; Bronchi; Clonidine; Female; Forced Expiratory Volume; Histamine; Humans; Male; Oxazoles; Rilmenidine

1988
Preliminary clinical pharmacological studies of S3341, a new hypotensive agent, and comparison with clonidine in normal males.
    European journal of clinical pharmacology, 1984, Volume: 27, Issue:3

    Topics: Adrenergic alpha-Agonists; Adult; Antihypertensive Agents; Blood Pressure; Central Nervous System; Clonidine; Dose-Response Relationship, Drug; Electrocardiography; Humans; Male; Oxazoles; Rilmenidine

1984
Effects of one-year treatment with rilmenidine on systemic hypertension-induced left ventricular hypertrophy in hypertensive patients.
    The American journal of cardiology, 1994, Dec-22, Volume: 74, Issue:13

    Topics: Antihypertensive Agents; Atrial Natriuretic Factor; Echocardiography; Female; Forearm; Humans; Hypertension; Hypertrophy, Left Ventricular; Male; Middle Aged; Oxazoles; Renin; Rilmenidine; Vascular Resistance

1994
Pharmacokinetics of rilmenidine in patients with chronic renal insufficiency and in hemodialysis patients.
    The American journal of cardiology, 1994, Dec-22, Volume: 74, Issue:13

    Topics: Adolescent; Adult; Aged; Antihypertensive Agents; Creatinine; Dialysis Solutions; Female; Humans; Hypertension; Kidney; Kidney Failure, Chronic; Male; Middle Aged; Oxazoles; Renal Dialysis; Rilmenidine; Single-Blind Method

1994
Efficacy and safety of rilmenidine in elderly patients--comparison with hydrochlorothiazide. The Belgian Multicentre Study Group.
    The American journal of cardiology, 1994, Dec-22, Volume: 74, Issue:13

    Topics: Aged; Aged, 80 and over; Antineoplastic Agents; Double-Blind Method; Female; Humans; Hydrochlorothiazide; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine

1994
Long-term control of blood pressure by rilmenidine in high-risk populations.
    The American journal of cardiology, 1994, Dec-22, Volume: 74, Issue:13

    Topics: Age Factors; Antihypertensive Agents; Blood Pressure; Female; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine; Risk Factors

1994
Dose-effect relationship of rilmenidine after chronic administration.
    European journal of clinical pharmacology, 1993, Volume: 45, Issue:2

    Topics: Antihypertensive Agents; Blood Pressure; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Heart Rate; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine; Supine Position

1993
Double-blind controlled study of rilmenidine versus hydrochlorothiazide in mild hypertension: clinical and renal haemodynamic evaluation.
    Journal of human hypertension, 1993, Volume: 7, Issue:2

    Topics: Adult; Antihypertensive Agents; Blood Pressure; Creatinine; Double-Blind Method; Female; Glomerular Filtration Rate; Hemodynamics; Humans; Hydrochlorothiazide; Hypertension; Iodine Radioisotopes; Kidney; Male; Middle Aged; Oxazoles; Regional Blood Flow; Rilmenidine; Time Factors; Vascular Resistance

1993
[Pharmaco-epidemiologic evaluation of rilmenidine in 18,235 hypertensive patients].
    Presse medicale (Paris, France : 1983), 1995, Dec-09, Volume: 24, Issue:38

    Topics: Adult; Aged; Antihypertensive Agents; Drug Administration Schedule; Female; Follow-Up Studies; Heart Rate; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine

1995
Cardiovascular variability after rilmenidine challenge: assessment of acute dosing effects by means of spectral analysis.
    Fundamental & clinical pharmacology, 1995, Volume: 9, Issue:4

    Topics: Adult; Analysis of Variance; Antihypertensive Agents; Blood Pressure; Blood Pressure Determination; Cross-Over Studies; Double-Blind Method; Female; Heart Rate; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine

1995
Rilmenidine in patients with left ventricular hypertrophy: beyond the reduction of left ventricular mass.
    Journal of cardiovascular pharmacology, 1995, Volume: 26 Suppl 2

    Topics: Antihypertensive Agents; Atrial Natriuretic Factor; Drug Administration Schedule; Electrolytes; Female; Heart Ventricles; Humans; Hypertension; Hypertrophy, Left Ventricular; Male; Middle Aged; Oxazoles; Renin; Rilmenidine

1995
Lipid profile and antihypertensive efficacy in hyperlipidemic hypertensive patients: comparison of rilmenidine and captopril.
    Journal of cardiovascular pharmacology, 1995, Volume: 26 Suppl 2

    Topics: Adrenergic alpha-Agonists; Adult; Aged; Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Captopril; Double-Blind Method; Female; Humans; Hyperlipoproteinemia Type II; Hypertension; Lipids; Male; Middle Aged; Oxazoles; Rilmenidine

1995
Comparative effects of rilmenidine and atenolol on tests of autonomic function and mental and dynamic exercise in patients with essential hypertension.
    Journal of cardiovascular pharmacology, 1995, Volume: 26 Suppl 2

    Topics: Adult; Anti-Arrhythmia Agents; Antihypertensive Agents; Atenolol; Autonomic Nervous System; Blood Pressure; Cross-Over Studies; Double-Blind Method; Exercise Test; Heart Rate; Humans; Hypertension; Male; Mental Processes; Middle Aged; Neurosecretory Systems; Oxazoles; Rilmenidine

1995
Effects of rilmenidine and clonidine on the electroencephalogram, saccadic eye movements, and psychomotor function.
    Journal of cardiovascular pharmacology, 1995, Volume: 26 Suppl 2

    Topics: Adult; Antihypertensive Agents; Blood Pressure; Clonidine; Cross-Over Studies; Double-Blind Method; Electroencephalography; Evoked Potentials, Auditory; Heart Rate; Humans; Male; Oxazoles; Placebos; Psychomotor Performance; Rilmenidine; Saccades

1995
The effects of rilmenidine and atenolol on mental stress, dynamic exercise and autonomic function in mild to moderate hypertension.
    British journal of clinical pharmacology, 1995, Volume: 40, Issue:6

    Topics: Adrenergic beta-Antagonists; Adult; Antihypertensive Agents; Atenolol; Blood Pressure; Cross-Over Studies; Double-Blind Method; Exercise; Heart Rate; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine; Stress, Psychological; Supine Position

1995
[Effects of rilmenidine (hyperium) on lipid balance in hyperlipidemic hypertensive patients. Randomized, controlled, double-blind 8-week study vs. captopril in parallel groups].
    Annales de cardiologie et d'angeiologie, 1996, Volume: 45, Issue:10

    Topics: Antihypertensive Agents; Captopril; Double-Blind Method; Female; Humans; Hypercholesterolemia; Hyperlipidemias; Hypertension; Lipids; Male; Middle Aged; Oxazoles; Rilmenidine; Time Factors

1996
Effect of N-dicyclopropylmethyl-amino-2-oxazoline (S-3341) on antioxidant status and nitric oxide in hypertensive patients.
    Current medical research and opinion, 1998, Volume: 14, Issue:2

    Topics: Adult; Aged; Antihypertensive Agents; Antioxidants; Blood Pressure; Catalase; Humans; Hypertension; Male; Malondialdehyde; Middle Aged; Nitrates; Nitric Oxide; Nitrites; Oxazoles; Rilmenidine; Vitamin E

1998
[Rilmenidine in rosacea: a double-blind study versus placebo].
    Annales de dermatologie et de venereologie, 1997, Volume: 124, Issue:10

    Topics: Adrenergic alpha-Agonists; Adult; Double-Blind Method; Drug Tolerance; Female; Flushing; Humans; Male; Middle Aged; Oxazoles; Placebos; Rilmenidine; Rosacea; Treatment Outcome

1997
Regression of left ventricular hypertrophy in hypertensive patients after 1 year of treatment with rilmenidine: a double-blind, randomized, controlled (versus nifedipine) study.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1998, Volume: 16, Issue:3

    Topics: Adult; Antihypertensive Agents; Blood Pressure; Calcium Channel Blockers; Diastole; Double-Blind Method; Echocardiography; Electrocardiography, Ambulatory; Female; Humans; Hypertension; Hypertrophy, Left Ventricular; Male; Middle Aged; Nifedipine; Oxazoles; Rilmenidine; Treatment Outcome

1998
[Essential arterial hypertension treated with rilmenidin : what dose for what patient?].
    Presse medicale (Paris, France : 1983), 1999, Jan-09, Volume: 28, Issue:1

    Topics: Antihypertensive Agents; Dose-Response Relationship, Drug; Humans; Hypertension; Oxazoles; Rilmenidine

1999
Effects of rilmenidine on stress-induced peak blood pressure and renal function.
    Journal of cardiovascular pharmacology, 1999, Volume: 34, Issue:1

    Topics: Adrenergic alpha-Agonists; Adult; Blood Pressure; Cardiovascular Diseases; Cross-Over Studies; Double-Blind Method; Exercise Test; Humans; Kidney; Kidney Function Tests; Lithium; Male; Oxazoles; Placebos; Rilmenidine; Sodium; Stress, Psychological; Time Factors

1999
Efficacy of rilmenidine versus captopril on microalbuminuria: a pilot study in hypertensive type 2 diabetics.
    Cardiovascular drugs and therapy, 1999, Volume: 13, Issue:6

    Topics: Albuminuria; Antihypertensive Agents; Captopril; Diabetes Mellitus, Type 2; Humans; Hypertension; Oxazoles; Pilot Projects; Random Allocation; Rilmenidine

1999
Rilmenidine in the hypertensive type-2 diabetic: a controlled pilot study versus captopril.
    Journal of cardiovascular risk, 2000, Volume: 7, Issue:1

    Topics: Aged; Albuminuria; Antihypertensive Agents; Blood Pressure Determination; Captopril; Diabetes Mellitus, Type 2; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Follow-Up Studies; Humans; Hypertension; Male; Middle Aged; Oxazoles; Pilot Projects; Rilmenidine

2000
Haemodynamic and metabolic effects of rilmenidine in hypertensive patients with metabolic syndrome X. A double-blind parallel study versus amlodipine.
    Journal of hypertension, 2000, Volume: 18, Issue:10

    Topics: Adult; Aged; Amlodipine; Antihypertensive Agents; Blood Glucose; Body Weight; Double-Blind Method; Female; Hemodynamics; Humans; Hypertension; Hypertriglyceridemia; Insulin; Male; Middle Aged; Oxazoles; Plasminogen Activator Inhibitor 1; Rilmenidine; Tissue Plasminogen Activator

2000
Concentration-effect relationships of two infusion rates of the imidazoline antihypertensive agent rilmenidine for blood pressure and development of side-effects in healthy subjects.
    British journal of clinical pharmacology, 2001, Volume: 51, Issue:5

    Topics: Adult; Antihypertensive Agents; Blood Pressure; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Electroencephalography; Female; Heart Rate; Humans; Infusions, Intravenous; Male; Oxazoles; Pain Measurement; Rilmenidine; Saccades; Salivary Glands

2001
Effect of the new centrally acting antihypertensive agent rilmenidine on endothelial and platelet function in essential hypertension.
    Journal of human hypertension, 2002, Volume: 16, Issue:8

    Topics: Adult; Aged; Antihypertensive Agents; Blood Platelets; Blood Pressure; Endothelium, Vascular; Female; Follow-Up Studies; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine; Time Factors; Treatment Outcome

2002
Concentration-effect relationships of two rilmenidine single-dose infusion rates in hypertensive patients.
    Clinical pharmacology and therapeutics, 2002, Volume: 72, Issue:4

    Topics: Adult; Aged; Analysis of Variance; Confidence Intervals; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Hemodynamics; Humans; Hypertension; Infusions, Intravenous; Least-Squares Analysis; Male; Middle Aged; Oxazoles; Rilmenidine; Salivation

2002
[Efficacy and tolerance of rilmenidine in patients with mild to moderate hypertension. Results of a Czech and Slovak 6-month multicenter study].
    Vnitrni lekarstvi, 2002, Volume: 48, Issue:8

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Blood Pressure; Female; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine; Risk Factors

2002
[Efficacy and acceptability of rilmenidine in a population of 2 738 hypertensive diabetic patients].
    Presse medicale (Paris, France : 1983), 2002, Nov-23, Volume: 31, Issue:39 Pt 1

    Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Body Mass Index; Diabetes Complications; Diastole; Female; Follow-Up Studies; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine; Risk Factors; Time Factors

2002
[Comparison of the antihypertensive efficacy of and tolerance to 2 imidazoline receptor agonists: moxonidine and rilmenidine in monotherapy].
    Annales de cardiologie et d'angeiologie, 2001, Volume: 50, Issue:3

    Topics: Antihypertensive Agents; Female; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Male; Middle Aged; Oxazoles; Receptors, Drug; Rilmenidine; Severity of Illness Index

2001
[The effect of analysed hypotensive drugs on certain metabolic parameters].
    Polskie Archiwum Medycyny Wewnetrznej, 2003, Volume: 109, Issue:3

    Topics: Adult; Antihypertensive Agents; Diabetes Mellitus, Type 2; Felodipine; Female; Humans; Hyperlipidemias; Hypertension; Hyperuricemia; Indoles; Male; Metabolic Syndrome; Middle Aged; Oxazoles; Rilmenidine

2003
Efficacy and safety of rilmenidine, a selective imidazoline I1 receptor binding ligand, in mild-to-moderate Thai hypertensive patients.
    Journal of the Medical Association of Thailand = Chotmaihet thangphaet, 2003, Volume: 86, Issue:10

    Topics: Adult; Antihypertensive Agents; Female; Humans; Hypertension; Imidazoline Receptors; Ligands; Male; Middle Aged; Oxazoles; Receptors, Drug; Rilmenidine; Thailand; Treatment Outcome

2003
Rilmenidine sympatholytic activity preserves mental stress, orthostatic sympathetic responses and adrenaline secretion.
    Journal of hypertension, 2004, Volume: 22, Issue:8

    Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Cross-Over Studies; Epinephrine; Female; Humans; Hypertension; Male; Middle Aged; Norepinephrine; Oxazoles; Posture; Rilmenidine; Stress, Psychological; Sympathetic Nervous System; Sympatholytics; Tilt-Table Test

2004
Pharmacokinetic/pharmacodynamic assessment of tolerance to central nervous system effects of a 3 mg sustained release tablet of rilmenidine in hypertensive patients.
    Journal of psychopharmacology (Oxford, England), 2004, Volume: 18, Issue:2

    Topics: Administration, Oral; Adult; Aged; Antihypertensive Agents; Delayed-Action Preparations; Drug Administration Schedule; Drug Tolerance; Female; Humans; Hypertension; Male; Middle Aged; Oxazoles; Pain Measurement; Psychometrics; Reaction Time; Rilmenidine; Saccades; Tablets; Time Factors

2004
[The effects of rilmenidine on cardiac autonomic function in healthy volunteers].
    Revista espanola de cardiologia, 2004, Volume: 57, Issue:8

    Topics: Adult; Antihypertensive Agents; Autonomic Nervous System; Cardiovascular Physiological Phenomena; Cross-Over Studies; Double-Blind Method; Heart Rate; Humans; Male; Oxazoles; Rilmenidine

2004
Comparison of rilmenidine and lisinopril on ambulatory blood pressure and plasma lipid and glucose levels in hypertensive women with metabolic syndrome.
    Current medical research and opinion, 2005, Volume: 21, Issue:1

    Topics: Adult; Aged; Analysis of Variance; Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Blood Glucose; Blood Pressure Monitoring, Ambulatory; Female; Heart Rate; Hemodynamics; Humans; Hypertension; Lisinopril; Metabolic Syndrome; Middle Aged; Oxazoles; Prospective Studies; Rilmenidine; Single-Blind Method; Statistics, Nonparametric; Treatment Outcome

2005
Blockade of sympathetic nervous system activity by rilmenidine increases plasma adiponectin concentration in patients with essential hypertension.
    American journal of hypertension, 2005, Volume: 18, Issue:11

    Topics: Adiponectin; Adult; Antihypertensive Agents; Blood Glucose; Blood Pressure; Female; Humans; Hypertension; Insulin; Male; Middle Aged; Oxazoles; Rilmenidine; Sympathetic Nervous System; Time Factors; Treatment Outcome

2005
Rilmenidine--its antihypertensive efficacy, safety and impact on quality of life in perimenopausal women with mild to moderate essential hypertension.
    Blood pressure, 2006, Volume: 15, Issue:1

    Topics: Antihypertensive Agents; Blood Pressure; Female; Heart Rate; Humans; Hypertension; Middle Aged; Oxazoles; Perimenopause; Prospective Studies; Quality of Life; Rilmenidine

2006
How can we block sympathetic overactivity? Effects of rilmenidine and atenolol in overweight hypertensive patients.
    Journal of human hypertension, 2006, Volume: 20, Issue:6

    Topics: Adult; Analysis of Variance; Antihypertensive Agents; Area Under Curve; Atenolol; Brachial Artery; Echocardiography; Female; Glucose Tolerance Test; Humans; Hypertension; Lipids; Male; Middle Aged; Overweight; Oxazoles; Rilmenidine; Statistics, Nonparametric; Sympathetic Nervous System; Treatment Outcome

2006
Reduced hemodynamic responses to physical and mental stress under low-dose rilmenidine in healthy subjects.
    Cardiovascular drugs and therapy, 2006, Volume: 20, Issue:2

    Topics: Administration, Oral; Adult; Antihypertensive Agents; Blood Pressure; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Exercise; Exercise Test; Exercise Tolerance; Female; Heart Rate; Hemodynamics; Humans; Male; Middle Aged; Oxazoles; Physical Fitness; Rilmenidine; Stress, Psychological

2006
Efficacy of exercise, losartan, enalapril, atenolol and rilmenidine in subjects with blood pressure hyperreactivity at treadmill stress test and left ventricular hypertrophy.
    Journal of human hypertension, 2009, Volume: 23, Issue:4

    Topics: Adult; Antihypertensive Agents; Atenolol; Blood Pressure; Enalapril; Exercise Test; Exercise Therapy; Female; Humans; Hypertrophy, Left Ventricular; Losartan; Male; Oxazoles; Renin-Angiotensin System; Rilmenidine; Sympathetic Nervous System

2009
Bioequivalence evaluation of rilmenidine in healthy volunteers.
    Arzneimittel-Forschung, 2009, Volume: 59, Issue:5

    Topics: Adolescent; Adult; Antihypertensive Agents; Area Under Curve; Biological Availability; Chemistry, Pharmaceutical; Cross-Over Studies; Female; Humans; Male; Oxazoles; Rilmenidine; Therapeutic Equivalency; Young Adult

2009

Other Studies

235 other study(ies) available for oxazoles and rilmenidine

ArticleYear
Do centrally-acting antihypertensive drugs act at non-adrenergic as well as alpha-2 adrenoceptor sites?
    Clinical and experimental hypertension. Part A, Theory and practice, 1992, Volume: 14, Issue:5

    Topics: Animals; Antihypertensive Agents; Binding Sites; Blood Pressure; Brain; Cisterna Magna; Clonidine; Guanabenz; Heart Rate; Infusion Pumps; Injections; Male; Osmosis; Oxazoles; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha; Receptors, Cell Surface; Rilmenidine

1992
Reduction in focal cerebral ischemia by agents acting at imidazole receptors.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1992, Volume: 12, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzazepines; Brain; Dioxanes; Dose-Response Relationship, Drug; Idazoxan; Imidazoles; Ischemic Attack, Transient; Male; Neurons; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Drug; Rilmenidine

1992
Nature of [3H]rilmenidine binding to membranes of rat cerebral cortex.
    American journal of hypertension, 1992, Volume: 5, Issue:4 Pt 2

    Topics: Adrenergic alpha-Agonists; Amiloride; Animals; Binding Sites; Catecholamines; Cell Membrane; Cerebral Cortex; Guanidine; Guanidines; Imidazoles; Oxazoles; Prazosin; Rats; Receptors, Adrenergic; Rilmenidine; Tritium; Yohimbine

1992
Sympathoinhibitory effects of rilmenidine may be mediated by sites located below the brainstem.
    British journal of pharmacology, 1992, Volume: 105, Issue:3

    Topics: Adrenergic alpha-Agonists; Anesthesia; Animals; Blood Pressure; Brain Stem; Heart Rate; Injections, Intraventricular; Kidney; Male; Oxazoles; Pentobarbital; Rats; Rats, Inbred SHR; Rilmenidine; Spinal Cord; Sympathetic Nervous System; Sympatholytics

1992
Influence of anaesthesia on the cardiovascular effects of rilmenidine and clonidine in spontaneously hypertensive rats.
    British journal of pharmacology, 1992, Volume: 105, Issue:3

    Topics: Adrenergic alpha-Agonists; Anesthesia; Animals; Blood Pressure; Clonidine; Heart Rate; Hemodynamics; Injections, Intravenous; Injections, Intraventricular; Male; Oxazoles; Pentobarbital; Rats; Rats, Inbred SHR; Reflex; Rilmenidine; Sympathetic Nervous System

1992
Importance of imidazoline receptors in the cardiovascular responses to clonidine and rilmenidine in conscious rabbits.
    Fundamental & clinical pharmacology, 1992, Volume: 6 Suppl 1

    Topics: Adrenergic alpha-Agonists; Animals; Autonomic Nervous System; Biogenic Monoamines; Brain Stem; Cardiovascular System; Clonidine; Consciousness; Imidazoline Receptors; Neurotransmitter Agents; Oxazoles; Rabbits; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine

1992
Does rilmenidine act in vivo on central alpha 2-adrenoceptors modulating noradrenaline release?
    European journal of pharmacology, 1992, Mar-24, Volume: 213, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Hypothalamus; Norepinephrine; Oxazoles; Rats; Receptors, Adrenergic, alpha; Rilmenidine

1992
Alpha 2-adrenoceptor and catecholamine-insensitive binding sites for [3H]rilmenidine in membranes from rat cerebral cortex.
    European journal of pharmacology, 1992, Jul-21, Volume: 218, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Binding Sites; Catecholamines; Cerebral Cortex; In Vitro Techniques; Oxazoles; Rats; Receptors, Adrenergic, alpha; Rilmenidine

1992
The effects of rilmenidine on tests of autonomic function in humans.
    Clinical pharmacology and therapeutics, 1992, Volume: 52, Issue:5

    Topics: Adrenergic alpha-Agonists; Adult; Antihypertensive Agents; Autonomic Nervous System; Blood Pressure; Forearm; Heart Rate; Humans; Male; Oxazoles; Posture; Pressoreceptors; Reference Values; Regional Blood Flow; Rilmenidine; Valsalva Maneuver

1992
Central cardiovascular effects of rilmenidine and neuropeptide Y in the conscious spontaneously hypertensive rat: haemodynamic and biochemical evidence for a negative interaction.
    Journal of cardiovascular pharmacology, 1992, Volume: 19, Issue:6

    Topics: Adenylyl Cyclases; Adrenergic alpha-Agonists; Animals; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Hemodynamics; Hypertension; In Vitro Techniques; Male; Medulla Oblongata; Neuropeptide Y; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine

1992
Inhibition of nitric oxide synthesis increases focal ischemic infarction in rat.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1992, Volume: 12, Issue:5

    Topics: Amino Acid Oxidoreductases; Analysis of Variance; Animals; Antihypertensive Agents; Arginine; Cerebral Infarction; Ischemic Attack, Transient; Male; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Oxazoles; Phenylephrine; Rats; Rats, Inbred WKY; Rilmenidine

1992
Rilmenidine lowers arterial pressure via imidazole receptors in brainstem C1 area.
    European journal of pharmacology, 1991, Mar-26, Volume: 195, Issue:2

    Topics: Animals; Antihypertensive Agents; Benzazepines; Binding, Competitive; Blood Pressure; Brain Stem; Clonidine; Decerebrate State; Dose-Response Relationship, Drug; Heart Rate; Imidazoline Receptors; Male; Microinjections; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine

1991
Selectivity of rilmenidine for the nucleus reticularis lateralis, a ventrolateral medullary structure containing imidazoline-preferring receptors.
    European journal of pharmacology, 1991, Dec-17, Volume: 209, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Catecholamines; Clonidine; Dioxanes; Electrochemistry; Hemodynamics; Idazoxan; Imidazoline Receptors; Male; Medulla Oblongata; Neurons; Oxazoles; Piperoxan; Rats; Rats, Inbred WKY; Receptors, Drug; Reticular Formation; Rilmenidine; Stereotaxic Techniques; Yohimbine

1991
The imidazoline-guanidinium receptor site, a target for some alpha-2 adrenergic agonists, is involved in inhibition of Na(+)-H+ exchange in renal proximal tubule cells.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1991, Volume: 9, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Carrier Proteins; Dioxanes; Hydrogen; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Ion Exchange; Kidney Tubules, Proximal; Oxazoles; Quinoxalines; Rabbits; Receptors, Drug; Rilmenidine; Sodium; Sodium-Hydrogen Exchangers

1991
Effects of swim training alone and in combination with clonidine and rilmenidine on blood pressure, plasma electrolytes, vasopressin, and renin activity in spontaneously hypertensive rats.
    Journal of cardiovascular pharmacology, 1990, Volume: 15, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Body Weight; Clonidine; Electrolytes; Heart; Male; Organ Size; Oxazoles; Physical Conditioning, Animal; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Renin; Rilmenidine; Swimming; Vasopressins

1990
Importance of central noradrenergic and serotonergic pathways in the cardiovascular actions of rilmenidine and clonidine.
    Journal of cardiovascular pharmacology, 1991, Volume: 18, Issue:6

    Topics: 5,6-Dihydroxytryptamine; Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Blood Pressure; Brain; Clonidine; Dose-Response Relationship, Drug; Heart Rate; Male; Norepinephrine; Oxazoles; Oxidopamine; Rabbits; Rilmenidine; Serotonin

1991
Regional hemodynamic effects of rilmenidine and clonidine in the conscious spontaneously hypertensive rat.
    Fundamental & clinical pharmacology, 1991, Volume: 5, Issue:8

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Male; Oxazoles; Rats; Rats, Inbred SHR; Renal Circulation; Rilmenidine; Splanchnic Circulation

1991
Electrophysiological effects of intravenous rilmenidine in man.
    European journal of clinical pharmacology, 1991, Volume: 41, Issue:6

    Topics: Administration, Oral; Adult; Aged; Electrocardiography; Electrophysiology; Female; Heart Conduction System; Humans; Infusions, Intravenous; Male; Middle Aged; Oxazoles; Rilmenidine; Wolff-Parkinson-White Syndrome

1991
Contractile reactivity of isolated resistance arteries after 4 weeks of treatment with rilmenidine, clonidine or hydralazine in spontaneously hypertensive rats.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1991, Volume: 9, Issue:6

    Topics: Animals; Antihypertensive Agents; Arteries; Blood Pressure; Clonidine; Hydralazine; Hypertension; In Vitro Techniques; Male; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine; Time Factors; Vasoconstriction

1991
Acute and chronic effects of rilmenidine on baroreflex function in conscious dogs.
    European journal of pharmacology, 1990, Jun-08, Volume: 181, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Dogs; Female; Heart Rate; Male; Nitroglycerin; Oxazoles; Phenylephrine; Pressoreceptors; Reflex; Rilmenidine

1990
[Selectivity of a new antihypertensive agent, rilmenidine, for imidazoline receptors in the human brain].
    Archives des maladies du coeur et des vaisseaux, 1990, Volume: 83, Issue:8

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Brain; Dioxanes; Humans; Idazoxan; Imidazoline Receptors; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Yohimbine

1990
Desensitization and down-regulation of brain alpha 2-adrenoceptors by centrally acting antihypertensive drugs.
    British journal of clinical pharmacology, 1990, Volume: 30 Suppl 1

    Topics: Animals; Antihypertensive Agents; Binding, Competitive; Brain; Central Nervous System; Clonidine; Down-Regulation; Guanabenz; Hemodynamics; In Vitro Techniques; Male; Oxazoles; Rabbits; Receptors, Adrenergic, alpha; Rilmenidine; Yohimbine

1990
Effect of imidazolines on Na+ transport and intracellular pH in renal proximal tubule cells.
    Biochimica et biophysica acta, 1990, May-09, Volume: 1024, Issue:1

    Topics: Amiloride; Animals; Biological Transport; Brimonidine Tartrate; Cimetidine; Dioxanes; Dioxins; Hydrogen-Ion Concentration; Idazoxan; Imidazoles; In Vitro Techniques; Kidney Tubules, Proximal; Oxazoles; Quinoxalines; Rabbits; Rilmenidine; Sodium

1990
[The 1989 Bichat Conference. A new therapeutic orientation in arterial hypertension: the action of rilmenidine (Hyperium 1 mg) on the so-called imidazoline receptors].
    La Revue du praticien, 1990, Apr-11, Volume: 40, Issue:11

    Topics: Antihypertensive Agents; Humans; Hypertension; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1990
Evidence for the involvement of imidazoline receptors in the central hypotensive effect of rilmenidine in the rabbit.
    British journal of pharmacology, 1990, Volume: 100, Issue:3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Brain; Cisterna Magna; Dioxanes; Heart Rate; Hemodynamics; Idazoxan; Imidazoline Receptors; Injections; Injections, Intraventricular; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Tissue Extracts; Yohimbine

1990
Influence of the alpha-2 agonist oxaminozoline (S3341) on firing rate of central noradrenergic and serotonergic neurons in the rat. Comparison with clonidine.
    Archives internationales de physiologie et de biochimie, 1986, Volume: 94, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Electrophysiology; Iontophoresis; Locus Coeruleus; Male; Neurons; Norepinephrine; Oxazoles; Prazosin; Raphe Nuclei; Rats; Rilmenidine; Serotonin; Yohimbine

1986
Rapid eye movement sleep and the associated cardiovascular changes during and after continuous 10-day infusion of clonidine in normotensive rats: comparison with lofexidine and S3341.
    Journal of cardiovascular pharmacology, 1987, Volume: 9, Issue:6

    Topics: Animals; Blood Pressure; Cardiovascular System; Clonidine; Drug Administration Schedule; Female; Heart Rate; Infusions, Intravenous; Oxazoles; Rats; Rats, Inbred Strains; Rilmenidine; Sleep, REM; Time Factors

1987
[New discoveries in the regulation of arterial pressure: endazoline, rilmenidine and imidazoline receptors].
    Archives des maladies du coeur et des vaisseaux, 1989, Volume: 82 Spec No 5

    Topics: Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1989
[The heart in patients with hypertension: effects of rilmenidine on experimental cardiac hypertrophy of hypertensive origin in rats].
    Archives des maladies du coeur et des vaisseaux, 1989, Volume: 82 Spec No 5

    Topics: Animals; Antihypertensive Agents; Cardiomegaly; Collagen; Heart; Heart Failure; Hypertension; Nephrectomy; Oxazoles; Propranolol; Rats; Rats, Inbred Strains; Rilmenidine

1989
[From alpha 2-adrenergic to endazoline receptors].
    Archives des maladies du coeur et des vaisseaux, 1989, Volume: 82 Spec No 5

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Humans; Hypertension; Imidazoline Receptors; Oxazoles; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine

1989
Rilmenidine selectivity for imidazoline receptors in human brain.
    European journal of pharmacology, 1989, Apr-25, Volume: 163, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Brain; Humans; Imidazoline Receptors; In Vitro Techniques; Nerve Tissue Proteins; Oxazoles; Receptors, Drug; Rilmenidine

1989
Different affinities of alpha 2-agonists for imidazoline and alpha 2-adrenergic receptors.
    American journal of hypertension, 1989, Volume: 2, Issue:6 Pt 1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Dioxanes; Guanfacine; Guanidine; Guanidines; Idazoxan; Imidazoline Receptors; Male; Oxazoles; Phenylacetates; Rabbits; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine; Yohimbine

1989
Rilmenidine differs from clonidine in that it lacks histamine-like activity.
    The Journal of pharmacy and pharmacology, 1989, Volume: 41, Issue:7

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Female; Guinea Pigs; Heart; Heart Rate; Histamine; In Vitro Techniques; Male; Myocardium; Oxazoles; Potassium Chloride; Rats; Rats, Inbred Strains; Receptors, Histamine H2; Rilmenidine; Uterine Contraction; Uterus

1989
[Selectivity of alpha 2-adrenergic agonists for the imidazoline-guanidine and alpha 2-adrenergic receptors].
    Archives des maladies du coeur et des vaisseaux, 1989, Volume: 82, Issue:7

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Guanfacine; Guanidines; Idazoxan; Kidney Tubules, Proximal; Male; Oxazoles; Phenylacetates; Rabbits; Receptors, Adrenergic, alpha; Rilmenidine; Yohimbine

1989
Cardiovascular effects of rilmenidine, a new alpha 2-adrenoceptor agonist, and clonidine in conscious spontaneously hypertensive rats.
    Clinical and experimental pharmacology & physiology, 1989, Volume: 16, Issue:11

    Topics: Administration, Oral; Adrenergic alpha-Agonists; Animals; Blood Pressure; Catecholamines; Clonidine; Heart Rate; Hemodynamics; Injections, Intravenous; Male; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine

1989
Remodelling of the heart in DOCA-salt hypertensive rats by propranolol and by an alpha-2 agonist, rilmenidine.
    Journal of hypertension, 1989, Volume: 7, Issue:12

    Topics: Adrenergic alpha-Agonists; Analysis of Variance; Animals; Antihypertensive Agents; Blood Pressure; Cardiomegaly; Desoxycorticosterone; Disease Models, Animal; Heart; Heart Rate; Hypertension; Male; Oxazoles; Propranolol; Rats; Rats, Inbred Strains; Rilmenidine; Sodium Chloride

1989
[Interaction of rilmenidine with renal imidazoline-guanidine sites].
    Archives des maladies du coeur et des vaisseaux, 1989, Volume: 82 Spec No 5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Basement Membrane; Binding Sites; Dioxanes; Drug Interactions; Guanfacine; Guanidines; Idazoxan; Imidazoles; Imidazoline Receptors; Kidney; Male; Oxazoles; Phenylacetates; Rabbits; Receptors, Drug; Rilmenidine; Sodium Channels; Yohimbine

1989
Second International Symposium on Rilmenidine. Paris, March 11, 1988. Proceedings.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Animals; Antihypertensive Agents; Humans; Hypertension; Oxazoles; Rilmenidine

1989
Pharmacokinetics of rilmenidine.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Adult; Antihypertensive Agents; Biological Availability; Capsules; Carbon Radioisotopes; Female; Food; Humans; Male; Oxazoles; Rilmenidine; Solutions; Tablets

1989
Treatment of hypertension in diabetic patients.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Antihypertensive Agents; Blood Glucose; Diabetes Complications; Diabetes Mellitus; Diuretics; Drug Therapy, Combination; Female; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine

1989
Hypertension in the elderly.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Aged; Aged, 80 and over; Antihypertensive Agents; Humans; Hypertension; Oxazoles; Rilmenidine

1989
Acceptability of rilmenidine and long-term surveillance of plasma concentrations in hypertensive patients with renal insufficiency.
    The American journal of medicine, 1989, Sep-18, Volume: 87, Issue:3C

    Topics: Adult; Aged; Antihypertensive Agents; Blood Pressure; Drug Therapy, Combination; Heart Rate; Humans; Hypertension, Renal; Kidney; Kidney Failure, Chronic; Middle Aged; Oxazoles; Rilmenidine

1989
Bistrifluoromethylaryl derivatives for drug analysis by gas chromatography electron capture negative ion chemical ionization mass spectrometry. Application to the measurement of (N-dicyclopropylmethyl)amino-2-oxazoline in plasma.
    Biomedical mass spectrometry, 1985, Volume: 12, Issue:5

    Topics: Adrenergic alpha-Agonists; Chemical Phenomena; Chemistry; Fluorobenzenes; Gas Chromatography-Mass Spectrometry; Humans; Oxazoles; Rilmenidine

1985
Gas chromatographic negative ion mass spectrometric assay of 2-dicyclopropylmethylamino-2-oxazoline (S-3341), a new antihypertensive drug.
    Biomedical mass spectrometry, 1985, Volume: 12, Issue:10

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Chemical Phenomena; Chemistry; Gas Chromatography-Mass Spectrometry; Humans; Kinetics; Oxazoles; Rilmenidine

1985
Central and peripheral effects of S 3341 [(N-dicyclopropylmethyl)-amino-2-oxazoline] in animal models.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 279, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cats; Clonidine; Decerebrate State; Female; Heart Rate; Hexobarbital; In Vitro Techniques; Male; Mice; Oxazoles; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rilmenidine; Sleep; Time Factors

1986
Quantitative analysis of S3341 in human plasma and urine by combined gas chromatography-negative ion chemical ionization mass spectrometry: 15 month inter-day precision and accuracy validation.
    Biomedical & environmental mass spectrometry, 1987, Volume: 14, Issue:6

    Topics: Adrenergic alpha-Agonists; Gas Chromatography-Mass Spectrometry; Humans; Oxazoles; Quality Control; Rilmenidine

1987
A symposium: Rilmenidine--a novel alpha2 agonist antihypertensive agent.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Humans; Oxazoles; Rilmenidine

1988
Cardiovascular and central nervous system effects of rilmenidine (S 3341) in rats.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenalectomy; Adrenergic alpha-Agonists; Anesthesia; Animals; Blood Pressure; Catecholamines; Central Nervous System; Chickens; Clonidine; Decerebrate State; Electric Stimulation; Heart Rate; Hemodynamics; Male; Motor Activity; Oxazoles; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Reflex; Rilmenidine; Sleep

1988
Action of rilmenidine on locus ceruleus and dorsal raphe cells in vivo and in vitro.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Action Potentials; Adrenergic alpha-Agonists; Animals; Clonidine; In Vitro Techniques; Infusions, Intravenous; Iontophoresis; Locus Coeruleus; Lysergic Acid Diethylamide; Male; Oxazoles; Prazosin; Raphe Nuclei; Rats; Rats, Inbred Strains; Rilmenidine

1988
Effects of two alpha 2 agonists, rilmenidine and clonidine, on the morphine withdrawal syndrome and their potential addictive properties in rats.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic alpha-Agonists; Animals; Behavior, Animal; Clonidine; Male; Morphine; Oxazoles; Rats; Rats, Inbred Strains; Rilmenidine; Substance Withdrawal Syndrome; Substance-Related Disorders

1988
Effects of continuous infusions (10 days) and cessation of infusions of clonidine and rilmenidine (S 3341) on cardiovascular and behavioral parameters of spontaneously hypertensive rats.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic alpha-Agonists; Animals; Behavior, Animal; Blood Pressure; Clonidine; Female; Heart Rate; Infusion Pumps; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine; Sleep, REM; Time Factors

1988
Effects of rilmenidine on bronchomotor responses in the guinea pig.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic alpha-Agonists; Animals; Bronchi; Clonidine; Compliance; Drug Synergism; Guinea Pigs; Histamine; Male; Oxazoles; Rilmenidine

1988
Pharmacokinetics of rilmenidine in healthy subjects.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Absorption; Administration, Oral; Adrenergic beta-Agonists; Biological Availability; Carbon Radioisotopes; Drug Administration Schedule; Eating; Female; Half-Life; Humans; Injections, Intravenous; Male; Oxazoles; Rilmenidine

1988
Pharmacokinetics of rilmenidine.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Absorption; Administration, Oral; Adrenergic beta-Agonists; Adult; Aged; Aged, 80 and over; Female; Humans; Hypertension; Kidney Failure, Chronic; Liver Diseases; Male; Middle Aged; Oxazoles; Rilmenidine

1988
Pharmacology of the alpha 2-adrenoceptor agonist rilmenidine.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Central Nervous System; Chemical Phenomena; Chemistry; Clonidine; Dose-Response Relationship, Drug; Hexobarbital; Humans; Hypnotics and Sedatives; Mice; Oxazoles; Rats; Rilmenidine; Sleep

1988
Hemodynamic and electrophysiologic effects of a new alpha 2-adrenoceptor agonist, rilmenidine, for systemic hypertension.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic beta-Agonists; Adult; Blood Pressure; Cardiac Output; Cardiac Pacing, Artificial; Electrocardiography; Electrophysiology; Female; Heart Conduction System; Heart Rate; Hemodynamics; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine; Stroke Volume; Time Factors

1988
Noninvasive study of cardiac structure and function after rilmenidine for essential hypertension.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic alpha-Agonists; Adult; Aged; Blood Pressure; Echocardiography; Female; Heart; Hemodynamics; Humans; Hypertension; Male; Middle Aged; Myocardium; Oxazoles; Rilmenidine; Stroke Volume; Time Factors; Vascular Resistance

1988
Treatment of systemic hypertension in insulin-treated diabetes mellitus with rilmenidine.
    The American journal of cardiology, 1988, Feb-24, Volume: 61, Issue:7

    Topics: Adrenergic beta-Agonists; Adult; Aged; Albuminuria; Blood Pressure; Diabetes Mellitus, Type 1; Electrocardiography; Female; Glucose; Humans; Hypertension; Lipid Metabolism; Male; Middle Aged; Oxazoles; Proteinuria; Rilmenidine

1988
Prejunctional alpha 2-adrenergic properties of S-3341 (dicyclopropylmethyl)amino-2-delta-2-oxazoline: a comparison with clonidine.
    Canadian journal of physiology and pharmacology, 1987, Volume: 65, Issue:12

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Oxazoles; Prazosin; Rats; Rats, Inbred WKY; Rilmenidine; Vas Deferens; Yohimbine

1987
Rilmenidine (S 3341) and the sympathoadrenal system: adrenoreceptors, plasma and adrenal catecholamines in dogs.
    Journal of autonomic pharmacology, 1988, Volume: 8, Issue:4

    Topics: Adrenal Medulla; Adrenergic alpha-Agonists; Animals; Blood Flow Velocity; Blood Platelets; Blood Pressure; Catecholamines; Dogs; Heart Rate; Leukocytes; Oxazoles; Rilmenidine; Sympathetic Nervous System

1988
Rilmenidine acts as a partial agonist at prejunctional alpha 2-adrenoceptors in guinea-pig atria.
    Clinical and experimental pharmacology & physiology, 1988, Volume: 15, Issue:10

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Atrial Function; Electric Stimulation; Female; Guinea Pigs; Male; Norepinephrine; Oxazoles; Receptors, Adrenergic, alpha; Rilmenidine

1988
Effect of the amino-oxazoline derivative S-3341 on pre- and postjunctional alpha-adrenoceptors in isolated blood vessels.
    Archives internationales de pharmacodynamie et de therapie, 1986, Volume: 284, Issue:1

    Topics: Animals; Clonidine; Dogs; In Vitro Techniques; Norepinephrine; Oxazoles; Perfusion; Phenylephrine; Prazosin; Pulmonary Artery; Rabbits; Receptors, Adrenergic, alpha; Rilmenidine; Saphenous Vein; Vasoconstriction; Yohimbine

1986
Interaction of clonidine and rilmenidine with imidazoline-preferring receptors.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1988, Volume: 6, Issue:4

    Topics: Animals; Binding, Competitive; Clonidine; Imidazoline Receptors; In Vitro Techniques; Kidney Tubules, Proximal; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine

1988
Use of hepatocyte cultures for preliminary metabolism and cytotoxicity studies of a new anti-hypertensive agent, oxaminozoline.
    Xenobiotica; the fate of foreign compounds in biological systems, 1988, Volume: 18, Issue:6

    Topics: Animals; Antihypertensive Agents; Biotransformation; Cells, Cultured; Clonidine; Drug Evaluation, Preclinical; Endothelium; L-Lactate Dehydrogenase; Liver; Oxazoles; Rats; Rats, Inbred Strains; Rilmenidine; Serum Albumin

1988
Rapid eye movement (REM)-sleep during and after continuous infusion of the oxazoline derivate S3341: a comparison with clonidine.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1984, Volume: 2, Issue:3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Female; Oxazoles; Rats; Rats, Inbred WKY; Rilmenidine; Sleep, REM; Time Factors

1984
Clonidine and rilmenidine suppress hypotension-induced Fos expression in the lower brainstem of the conscious rabbit.
    Neuroscience, 1995, Volume: 66, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Brain Stem; Clonidine; Consciousness; Female; Heart Rate; Hypotension; Immunohistochemistry; Male; Oxazoles; Proto-Oncogene Proteins c-fos; Rabbits; Rats; Rilmenidine; Tyrosine 3-Monooxygenase

1995
Involvement of peripheral presynaptic inhibition in the reduction of sympathetic tone by moxonidine, rilmenidine and UK 14304.
    European journal of pharmacology, 1995, Aug-25, Volume: 282, Issue:1-3

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Antihypertensive Agents; Brimonidine Tartrate; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Female; Imidazoles; Male; Neural Inhibition; Oxazoles; Peripheral Nervous System; Presynaptic Terminals; Quinoxalines; Rabbits; Rilmenidine; Sympathetic Nervous System; Vasoconstrictor Agents

1995
Rilmenidine-induced hypotension in conscious rabbits involves imidazoline-preferring receptors.
    Journal of cardiovascular pharmacology, 1994, Volume: 23, Issue:1

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Blood Pressure; Dioxanes; Dose-Response Relationship, Drug; Female; Heart Rate; Hypotension; Idazoxan; Imidazoline Receptors; Male; Methyldopa; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine

1994
Effects of three alpha 2-adrenoceptor agonists, rilmenidine, UK 14304 and clonidine on bradykinin- and substance P-induced airway microvascular leakage in guinea-pigs.
    Neuropeptides, 1995, Volume: 28, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Bradykinin; Brimonidine Tartrate; Capillaries; Capillary Permeability; Clonidine; Dioxanes; Extravascular Lung Water; Guinea Pigs; Idazoxan; Oxazoles; Prazosin; Quinoxalines; Rilmenidine; Substance P; Trachea

1995
Excess catecholamines and the metabolic syndrome: should central imidazoline receptors be a therapeutic target?
    Medical hypotheses, 1995, Volume: 44, Issue:3

    Topics: Animals; Antihypertensive Agents; Cardiovascular Diseases; Catecholamines; Energy Intake; Energy Metabolism; Humans; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Models, Biological; Neurons; Obesity; Oxazoles; Receptors, Drug; Rilmenidine; Social Conditions; Stress, Psychological; Sympathetic Nervous System

1995
Distribution of nonadrenergic [3H]rilmenidine binding in rat brain and kidney.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autoradiography; Binding Sites; Brain; Dioxanes; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kidney; Male; Oxazoles; Radioligand Assay; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Tritium

1995
Effects of rilmenidine on signal transduction mechanisms associated with alpha 2-adrenergic and imidazoline receptors in brain.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Brain Stem; Calcium; Cerebral Cortex; Cyclic AMP; Cyclic GMP; Imidazoline Receptors; In Vitro Techniques; Ion Transport; Oxazoles; Phosphatidylinositols; Rats; Receptors, Drug; Rilmenidine; Rubidium; Signal Transduction

1995
Rilmenidine alters renal function when administered intracerebroventricularly or intrarenally.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Drug Administration Routes; Imidazoline Receptors; Kidney; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Drug; Renal Artery; Rilmenidine

1995
Evidence for a role for imidazoline I1 binding site in rat brown adipocytes.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adipose Tissue, Brown; Animals; Carrier Proteins; Clonidine; Imidazoline Receptors; Ion Channels; Isoproterenol; Membrane Proteins; Mitochondria; Mitochondrial Proteins; Oxazoles; Oxygen; Rats; Rats, Wistar; Receptors, Drug; Rilmenidine; Uncoupling Protein 1

1995
Mechanism of sympathoinhibition by imidazolines.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzazepines; Brimonidine Tartrate; Dioxanes; Hemodynamics; Idazoxan; Imidazoles; Oxazoles; Quinoxalines; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine

1995
Sympathoinhibitory action of rilmenidine in conscious sinoaortically denervated rats.
    Journal of cardiovascular pharmacology, 1993, Volume: 22, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cisterna Magna; Denervation; Dioxanes; Heart Rate; Idazoxan; Infusions, Intravenous; Injections; Injections, Intra-Arterial; Kidney; Male; Oxazoles; Phenylephrine; Rats; Rats, Wistar; Rilmenidine; Sinoatrial Node; Sympatholytics

1993
Quantitative autoradiographic localization in rat brain of alpha 2-adrenergic and non-adrenergic I-receptor binding sites labelled by [3H]rilmenidine.
    Brain research, 1995, Mar-27, Volume: 675, Issue:1-2

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Autoradiography; Binding Sites; Brain; Brain Chemistry; Clonidine; Epinephrine; Imidazoline Receptors; Male; Oxazoles; Radioligand Assay; Rats; Rats, Inbred WKY; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

1995
Central alpha-2 adrenoceptors are responsible for a clonidine-induced cue in a rat drug discrimination paradigm.
    Psychopharmacology, 1993, Volume: 110, Issue:1-2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Clonidine; Conditioning, Operant; Cues; Discrimination, Psychological; Male; Oxazoles; Rats; Receptors, Adrenergic, alpha-2; Reinforcement Schedule; Reward; Rilmenidine

1993
Differential patterns of local cerebral glucose utilisation associated with rilmenidine- or B-HT 933-induced hypotension.
    Brain research, 1994, Dec-15, Volume: 666, Issue:2

    Topics: Animals; Antihypertensive Agents; Autoradiography; Azepines; Brain; Glucose; Hypotension; Male; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine; Tissue Distribution

1994
Stimulatory effects of clonidine, cirazoline and rilmenidine on locus coeruleus noradrenergic neurones: possible involvement of imidazoline-preferring receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 348, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Dose-Response Relationship, Drug; Imidazoles; Imidazoline Receptors; Locus Coeruleus; Male; Membrane Potentials; Neurons; Norepinephrine; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

1993
Down-regulation of imidazoline sites in rabbit kidney.
    European journal of pharmacology, 1993, Oct-12, Volume: 243, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Down-Regulation; Guanabenz; Idazoxan; Imidazoline Receptors; Kidney; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine

1993
Sympathoinhibition by rilmenidine in conscious rabbits: involvement of alpha 2-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 348, Issue:6

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Catecholamines; Decerebrate State; Dioxanes; Dose-Response Relationship, Drug; Electric Stimulation; Electrodes, Implanted; Female; Heart Rate; Hemodynamics; Idazoxan; Kidney; Male; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine

1993
Molecular studies of alpha-2-adrenoceptor and catecholamine-insensitive imidazoline-receptor binding sites using [3H]-rilmenidine in rat brain and kidney.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1993, Volume: 11, Issue:5

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Binding Sites; Brain; Catecholamines; Imidazoline Receptors; In Vitro Techniques; Kidney; Oxazoles; Rats; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Tissue Distribution

1993
Differential receptors involved in the cardiovascular effects of clonidine and rilmenidine in conscious rabbits.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1993, Volume: 11, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cardiovascular Physiological Phenomena; Cardiovascular System; Clonidine; Dioxanes; Female; Idazoxan; Imidazoline Receptors; Male; Methyldopa; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

1993
Effect of rilmenidine on baroreflex control of renal sympathetic nerve activity.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1993, Volume: 11, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Baroreflex; Blood Pressure; Dioxanes; Female; Idazoxan; Imidazoline Receptors; Kidney; Male; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System

1993
Is the sympathoinhibitory effect of rilmenidine mediated by alpha-2 adrenoceptors or imidazoline receptors?
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzazepines; Blood Pressure; Brimonidine Tartrate; Dose-Response Relationship, Drug; Heart Rate; Imidazoline Receptors; Kidney; Oxazoles; Quinoxalines; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System

1994
Imidazoline Receptors: A Novel Approach to Hypertension--the Contribution of Rilmenidine. Symposium proceedings. Milan, Italy, June 8, 1993.
    The American journal of cardiology, 1994, Dec-22, Volume: 74, Issue:13

    Topics: Animals; Antihypertensive Agents; Humans; Hypertension; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1994
Natriuretic effect of rilmenidine in anesthetized rats.
    The American journal of cardiology, 1994, Dec-22, Volume: 74, Issue:13

    Topics: Adrenergic alpha-Agonists; Adrenergic Fibers; Animals; Hemodynamics; Kidney; Natriuresis; Oxazoles; Rats; Rats, Wistar; Rilmenidine; Sodium; Thiopental

1994
Involvement of imidazoline-preferring receptors in regulation of sympathetic tone.
    The American journal of cardiology, 1994, Dec-22, Volume: 74, Issue:13

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Central Nervous System; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Female; Hemodynamics; Hypertension; Idazoxan; Imidazoles; Imidazoline Receptors; Male; Oxazoles; Rabbits; Rats; Rats, Inbred SHR; Receptors, Drug; Rilmenidine

1994
Attenuated renal response to moxonidine and rilmenidine in one kidney-one clip hypertensive rats.
    British journal of pharmacology, 1994, Volume: 112, Issue:1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Hemodynamics; Hypertension, Renovascular; Imidazoles; Infusions, Intra-Arterial; Kidney; Male; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Renal Circulation; Rilmenidine; Sodium; Urodynamics

1994
A novel mechanism of action for hypertension control: moxonidine as a selective I1-imidazoline agonist.
    Cardiovascular drugs and therapy, 1994, Volume: 8 Suppl 1

    Topics: Adrenal Medulla; Animals; Antihypertensive Agents; Autoradiography; Binding Sites; Blood Pressure; Cattle; Cells, Cultured; Clonidine; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine

1994
Renal effects of rilmenidine in anesthetized rats: importance of renal nerves.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: Adrenergic alpha-Agonists; Anesthesia; Animals; Hemodynamics; Kidney; Male; Oxazoles; Rats; Rats, Wistar; Renal Circulation; Rilmenidine; Sympathectomy; Sympathetic Nervous System

1993
Time-dependent efficacy of antihypertensive agents in spontaneously hypertensive rats.
    Chronobiology international, 1993, Volume: 10, Issue:6

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Captopril; Circadian Rhythm; Clonidine; Felodipine; Heart Rate; Hypertension; Labetalol; Male; Metoprolol; Oxazoles; Prazosin; Propanolamines; Propranolol; Rats; Rats, Inbred SHR; Rilmenidine; Thiophenes

1993
Cardiac electrophysiological effects of rilmenidine, a novel antihypertensive agent, in the conscious dog: comparison with clonidine.
    Life sciences, 1994, Volume: 54, Issue:22

    Topics: Animals; Antihypertensive Agents; Atrial Function; Blood Pressure; Clonidine; Dogs; Electrocardiography; Electrophysiology; Female; Heart; Heart Atria; Male; Oxazoles; Rilmenidine; Sinoatrial Node

1994
Differential characteristics and localisation of [3H]oxazoline and [3H]imidazoline binding sites in rat kidney.
    European journal of pharmacology, 1995, Aug-15, Volume: 281, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Autoradiography; Binding Sites; Dioxanes; Idazoxan; Imidazoles; Kidney; Male; Oxazoles; Radioligand Assay; Rats; Rats, Inbred WKY; Rilmenidine

1995
Renal effects of infusion of rilmenidine and guanabenz in conscious dogs: contribution of peripheral and central nervous system alpha 2-adrenoceptors.
    British journal of pharmacology, 1995, Volume: 116, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Autonomic Nerve Block; Binding Sites; Blood Pressure; Central Nervous System; Consciousness; Dioxanes; Dogs; Dose-Response Relationship, Drug; Ganglia, Autonomic; Guanabenz; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Kidney; Male; Oxazoles; Peripheral Nervous System; Receptors, Adrenergic, alpha-2; Receptors, Drug; Renal Circulation; Rilmenidine

1995
Carotid arterial changes produced by a centrally mediated antihypertensive agent in hypertensive rats.
    Journal of cardiovascular pharmacology, 1995, Volume: 26, Issue:4

    Topics: Analysis of Variance; Animals; Antihypertensive Agents; Blood Pressure; Cardiac Output; Carotid Arteries; Disease Models, Animal; Heart Rate; Hypertension; Injections, Intravenous; Oxazoles; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Rilmenidine; Vascular Resistance

1995
Role of imidazoline receptors in the cardiovascular actions of moxonidine, rilmenidine and clonidine in conscious rabbits.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 276, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Female; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

1996
Imidazoline Receptors in a Comprehensive Approach to Hypertension. Proceedings of an international symposium. Berlin, Germany, September 10, 1994.
    Journal of cardiovascular pharmacology, 1995, Volume: 26 Suppl 2

    Topics: Animals; Antihypertensive Agents; Humans; Hypertension; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

1995
Rilmenidine prevents epinephrine-induced arrhythmias in halothane-anesthetized dogs.
    Journal of cardiovascular pharmacology, 1995, Volume: 26 Suppl 2

    Topics: Adrenergic alpha-Agonists; Anesthesia, Inhalation; Anesthetics, Inhalation; Animals; Antihypertensive Agents; Arrhythmias, Cardiac; Dogs; Dose-Response Relationship, Drug; Epinephrine; Female; Halothane; Imidazoline Receptors; Male; Oxazoles; Receptors, Drug; Rilmenidine

1995
Brain structures involved in the hypotensive effects of rilmenidine: evaluation by [14C]2-deoxyglucose autoradiography.
    Journal of cardiovascular pharmacology, 1995, Volume: 26 Suppl 2

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Autoradiography; Azepines; Blood Pressure; Brain; Carbon Radioisotopes; Deoxyglucose; Glucose; Hypertension; Imidazoline Receptors; Male; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

1995
Selectivity of rilmenidine for I1-imidazoline-binding sites in rabbit proximal tubule cells.
    Journal of cardiovascular pharmacology, 1995, Volume: 26 Suppl 2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Binding Sites; Binding, Competitive; Cells, Cultured; Clonidine; Dioxanes; Idazoxan; Imidazoles; Imidazoline Receptors; Kidney Tubules, Proximal; Kinetics; Male; Oxazoles; Rabbits; Radioligand Assay; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Tritium

1995
Renal I1-imidazoline receptor-selective compounds mediate natriuresis in the rat.
    Journal of cardiovascular pharmacology, 1995, Volume: 26 Suppl 2

    Topics: Adrenergic alpha-Agonists; Agmatine; Animals; Antihypertensive Agents; Imidazoline Receptors; Kidney; Male; Natriuresis; Oxazoles; Rats; Receptors, Drug; Rilmenidine; Urodynamics

1995
Antiarrhythmic action of rilmenidine on adrenaline-induced arrhythmia via central imidazoline receptors in halothane-anaesthetized dogs.
    British journal of pharmacology, 1996, Volume: 117, Issue:8

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Anesthetics, Inhalation; Animals; Arrhythmias, Cardiac; Blood Pressure; Dogs; Epinephrine; Female; Halothane; Heart Rate; Idazoxan; Imidazoline Receptors; Male; Oxazoles; Receptors, Drug; Rilmenidine; Yohimbine

1996
Interactions of the cardiac chronotropic effects of rilmenidine with the autonomic nervous system in conscious dogs: comparison with clonidine.
    Journal of autonomic pharmacology, 1996, Volume: 16, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Antihypertensive Agents; Atropine; Blood Pressure; Chronic Disease; Clonidine; Depression, Chemical; Dogs; Female; Heart Block; Heart Rate; Male; Muscarinic Antagonists; Oxazoles; Phenoxybenzamine; Pindolol; Rilmenidine; Yohimbine

1996
No evidence for functional imidazoline receptors on locus coeruleus neurons.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzazepines; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Imidazoles; Imidazoline Receptors; Injections, Intravenous; Locus Coeruleus; Male; Microelectrodes; Neurons; Oxazoles; Quinolines; Rats; Rats, Wistar; Receptors, Drug; Rilmenidine

1996
Relative importance of central imidazoline receptors for the antihypertensive effects of moxonidine and rilmenidine.
    Journal of hypertension, 1996, Volume: 14, Issue:7

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Cardiac Catheterization; Clonidine; Dose-Response Relationship, Drug; Female; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Injections, Intravenous; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Time Factors

1996
Rilmenidine activates postjunctional alpha 1- and alpha 2-adrenoceptors in the canine saphenous vein.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:4

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dogs; Female; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isotope Labeling; Male; Medetomidine; Muscle Contraction; Muscle, Smooth; Osmolar Concentration; Oxazoles; Phenoxybenzamine; Prazosin; Protein Binding; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Tritium; Yohimbine

1996
Rilmenidine-induced ocular hypotension: role of imidazoline1 and alpha 2 receptors.
    Current eye research, 1996, Volume: 15, Issue:9

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzofurans; Calcium; Ciliary Body; Cyclic AMP; Female; Imidazoles; Imidazoline Receptors; Intraocular Pressure; Iris; Male; Norepinephrine; Ocular Hypotension; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathectomy; Sympathetic Nervous System; Yohimbine

1996
Rilmenidine and reflex renal sympathetic nerve activation in Wistar and hypertensive rats.
    British journal of pharmacology, 1996, Volume: 119, Issue:6

    Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Imidazoline Receptors; Kidney; Male; Oxazoles; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Drug; Reflex; Rilmenidine; Sympathetic Nervous System

1996
Inhibition of centrally induced ventricular arrhythmias by rilmenidine and idazoxan in rabbits.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 354, Issue:5

    Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Antihypertensive Agents; Arrhythmias, Cardiac; Bicuculline; Blood Pressure; Dose-Response Relationship, Drug; GABA Antagonists; Heart Rate; Idazoxan; Injections, Intravenous; Male; Oxazoles; Rabbits; Rilmenidine

1996
[Effects of rilmenidine on rats made insulin resistant and hypertensive by a high fructose diet].
    Archives des maladies du coeur et des vaisseaux, 1996, Volume: 89, Issue:8

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Blood Glucose; Blood Pressure; Diabetes Mellitus, Experimental; Dietary Carbohydrates; Disease Models, Animal; Fructose; Hypertension; Insulin; Insulin Resistance; Oxazoles; Rats; Rats, Wistar; Rilmenidine

1996
Are imidazoline receptors involved in sympathetic neurotransmission in rat vas deferens?
    General pharmacology, 1996, Volume: 27, Issue:7

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Electric Stimulation; Idazoxan; Imidazoline Receptors; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Oxazoles; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Synaptic Transmission; Vas Deferens; Yohimbine

1996
Renal effects of rilmenidine in volume-loaded anaesthetized dogs.
    Clinical and experimental pharmacology & physiology, 1997, Volume: 24, Issue:1

    Topics: Anesthesia; Animals; Antihypertensive Agents; Blood Volume; Diuresis; Dogs; Hematocrit; Kidney; Male; Natriuresis; Oxazoles; Pentobarbital; Plasma Volume; Rilmenidine

1997
Pretreatment with quinpirole inhibits the central antihypertensive effects of rilmenidine and alpha-methyldopa in conscious rats.
    European journal of pharmacology, 1997, Mar-19, Volume: 322, Issue:2-3

    Topics: Animals; Antihypertensive Agents; Domperidone; Dopamine Agonists; Male; Methyldopa; Oxazoles; Quinpirole; Rats; Rats, Inbred SHR; Rilmenidine; Species Specificity; Vasopressins

1997
The involvement of pertussis toxin-sensitive G proteins in the post receptor mechanism of central I1-imidazoline receptors.
    British journal of pharmacology, 1997, Volume: 120, Issue:8

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Animals; GTP-Binding Proteins; Imidazoles; Imidazoline Receptors; Male; Medetomidine; Oxazoles; Pertussis Toxin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Signal Transduction; Virulence Factors, Bordetella

1997
Renal denervation altered the hemodynamic and renal effects following intracerebroventricular administration of the I1-imidazoline receptor agonist, rilmenidine, in pentobarbital anaesthetized rats.
    Neurochemistry international, 1997, Volume: 30, Issue:1

    Topics: Anesthesia; Animals; Blood Pressure; Denervation; Dose-Response Relationship, Drug; Heart Rate; Hemodynamics; Imidazoline Receptors; Injections, Intraventricular; Kidney; Natriuresis; Osmolar Concentration; Oxazoles; Pentobarbital; Rats; Rats, Sprague-Dawley; Receptors, Drug; Rilmenidine

1997
Effect of rilmenidine on arterial pressure and urinary output in the spontaneously hypertensive rat.
    European journal of pharmacology, 1997, Apr-23, Volume: 325, Issue:1

    Topics: Administration, Oral; Animals; Antihypertensive Agents; Blood Pressure; Food Preferences; Heart Rate; Hypertension; Kidney; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine; Sodium Chloride; Urine

1997
Cardiac vagal effects of rilmenidine in the dog: comparison with clonidine.
    Journal of autonomic pharmacology, 1997, Volume: 17, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Clonidine; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Electrocardiography; Female; Heart; Heart Rate; In Vitro Techniques; Male; Oxazoles; Rilmenidine; Vagus Nerve

1997
Effect of rilmenidine injection into the paraventricular nucleus of the hypothalamus on the water intake induced by application of angiotensin II to the subfornical organ.
    Journal of physiology, Paris, 1997, Volume: 91, Issue:2

    Topics: Angiotensin II; Animals; Drinking; Idazoxan; Imidazoles; Injections; Male; Oxazoles; Paraventricular Hypothalamic Nucleus; Rats; Rats, Sprague-Dawley; Rilmenidine; Subfornical Organ

1997
Role of I1 imidazoline receptors in the sympathoinhibition produced by intracisternally administered rilmenidine and moxonidine.
    Arzneimittel-Forschung, 1997, Volume: 47, Issue:9

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Cisterna Magna; Dose-Response Relationship, Drug; Female; Guanabenz; Heart Rate; Imidazoles; Imidazoline Receptors; Injections; Male; Norepinephrine; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Yohimbine

1997
Antagonism of alpha1-adrenoceptor agonist-induced responses by rilmenidine in vascular smooth muscle.
    European journal of pharmacology, 1998, Jan-12, Volume: 341, Issue:2-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Calcium; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Phenylephrine; Portal Vein; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Rilmenidine

1998
Ethanol selectively counteracts hypotension evoked by central I(1)-imidazoline but not alpha2-adrenergic receptor activation in spontaneously hypertensive rats.
    Journal of cardiovascular pharmacology, 1998, Volume: 32, Issue:3

    Topics: Animals; Blood Pressure; Brain; Clonidine; Ethanol; Heart Rate; Hypertension; Imidazoline Receptors; Male; Nordefrin; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

1998
Site and receptors involved in the sympathoinhibitory actions of rilmenidine.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1998, Volume: 16, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Female; Imidazoline Receptors; Injections, Intraventricular; Kidney; Male; Neural Inhibition; Oxazoles; Rabbits; Receptors, Adrenergic, alpha; Receptors, Drug; Rilmenidine; Sympathetic Nervous System

1998
Complementary antihypertensive action of rilmenidine on the pressure-natriuresis relationship and sodium preference in spontaneously hypertensive rats.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1998, Volume: 16, Issue:3

    Topics: Animals; Antihypertensive Agents; Appetite; Blood Pressure; Hypertension; Natriuresis; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine; Sodium Chloride

1998
Preventive effect of rilmenidine on the occurrence of neurogenic ventricular arrhythmias in rabbits.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1998, Volume: 16, Issue:3

    Topics: Animals; Antihypertensive Agents; Bicuculline; Cardiac Complexes, Premature; GABA Antagonists; Hemodynamics; Idazoxan; Injections, Intravenous; Injections, Intraventricular; Male; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Tachycardia, Ventricular

1998
Rilmenidine normalizes fructose-induced insulin resistance and hypertension in rats.
    Journal of hypertension. Supplement : official journal of the International Society of Hypertension, 1998, Volume: 16, Issue:3

    Topics: Animals; Antihypertensive Agents; Blood Glucose; Blood Pressure; Fructose; Hypertension; Insulin Resistance; Kinetics; Lipids; Male; Oxazoles; Rats; Rats, Wistar; Reference Values; Rilmenidine

1998
Rilmenidine elevates cytosolic free calcium concentration in suspended cerebral astrocytes.
    Journal of neurochemistry, 1998, Volume: 71, Issue:4

    Topics: Adenosine Triphosphate; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Astrocytes; Calcium; Cells, Cultured; Cerebral Cortex; Cytosol; Endoplasmic Reticulum; Imidazoles; Oxazoles; Rats; Receptors, Adrenergic, alpha-2; Rilmenidine

1998
Rilmenidine reveals differences in the pharmacological characteristics of prejunctional alpha2-adrenoceptors in the guinea-pig, rat and pig.
    British journal of pharmacology, 1998, Volume: 125, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Arteries; Brimonidine Tartrate; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Ileum; Male; Muscle Contraction; Oxazoles; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Rilmenidine; Species Specificity; Swine; Vas Deferens

1998
Relative importance of medullary brain nuclei for the sympatho-inhibitory actions of rilmenidine in the anaesthetized rabbit.
    Journal of hypertension, 1998, Volume: 16, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Baroreflex; Hypotension; Imidazoline Receptors; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Solitary Nucleus; Sympathetic Nervous System

1998
[3H]Rilmenidine-labelled imidazoline-receptor binding sites co-localize with [3H]2-(benzofuranyl)-2-imidazoline-labelled imidazoline-receptor binding sites and monoamine oxidase-B in rabbit, but not rat, kidney.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Animals; Autoradiography; Benzofurans; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isoenzymes; Kidney; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Rabbits; Rats; Rats, Inbred WKY; Receptors, Drug; Rilmenidine; Species Specificity; Thiazoles

1998
Pharmacology and subcellular distribution of [3H]rilmenidine binding sites in rat brain.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Animals; Binding Sites; Brain; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Membranes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Radioligand Assay; Rats; Rats, Inbred WKY; Receptors, Drug; Rilmenidine; Subcellular Fractions; Thiazoles

1998
Chronopharmacological dependence of antihypertensive effects of the imidazoline-like drugs in stroke-prone spontaneously hypertensive rats.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cerebrovascular Disorders; Circadian Rhythm; Clonidine; Dose-Response Relationship, Drug; Heart Rate; Hypertension; Imidazoles; Male; Motor Activity; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine

1998
Effect of rilmenidine on the cadiovascular responses to stress in the conscious rabbit.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Female; Heart Rate; Hemodynamics; Kidney; Male; Noise; Oxazoles; Rabbits; Rilmenidine; Stress, Psychological; Sympathetic Nervous System

1998
Interaction of the dopamine D2 receptor agonist quinpirole with sympathetic vasomotor tone and the central action of rilmenidine in conscious rabbits.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Dopamine Agonists; Dose-Response Relationship, Drug; Female; Heart Rate; Kidney; Male; Muscle Tonus; Muscle, Smooth, Vascular; Oxazoles; Quinpirole; Rabbits; Receptors, Dopamine D2; Rilmenidine; Sympathetic Nervous System

1998
Comparison of the baroreceptor-heart rate reflex effects of moxonidine, rilmenidine and clonidine in conscious rabbits.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Adrenergic alpha-Agonists; Algorithms; Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Clonidine; Female; Heart Rate; Imidazoles; Injections, Intraventricular; Male; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Vagus Nerve

1998
Influence of sino-aortic barodenervation on the cardiovascular effects of imidazoline-like drugs.
    Journal of the autonomic nervous system, 1998, Oct-15, Volume: 72, Issue:2-3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Circadian Rhythm; Clonidine; Denervation; Heart Rate; Imidazoles; Injections, Intravenous; Male; Motor Activity; Oxazoles; Pressoreceptors; Rats; Rats, Wistar; Rilmenidine; Sinus of Valsalva; Telemetry

1998
Ethanol counteraction of I1-imidazoline but not alpha-2 adrenergic receptor-mediated reduction in vascular resistance in conscious spontaneously hypertensive rats.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 288, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Cardiac Output; Central Nervous System Depressants; Drug Interactions; Ethanol; Heart Rate; Imidazoline Receptors; Male; Nordefrin; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Vascular Resistance; Vasoconstrictor Agents

1999
Cardiovascular effects of rilmenidine, moxonidine and clonidine in conscious wild-type and D79N alpha2A-adrenoceptor transgenic mice.
    British journal of pharmacology, 1999, Volume: 126, Issue:6

    Topics: Adrenergic alpha-Antagonists; Amino Acid Substitution; Animals; Binding, Competitive; Blood Pressure; Cardiovascular Agents; Cell Line; Clonidine; Consciousness; Dogs; Heart Rate; Humans; Imidazoles; In Vitro Techniques; Isoquinolines; Male; Mice; Mice, Inbred Strains; Mice, Transgenic; Mutation; Naphthyridines; Oxazoles; Quinolizines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Rilmenidine; Saphenous Vein; Tritium

1999
Analysis of the receptor involved in the central hypotensive effect of rilmenidine and moxonidine.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 359, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzazepines; Benzofurans; Blood Pressure; Dose-Response Relationship, Drug; Drug Interactions; Female; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Methyldopa; Norepinephrine; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Yohimbine

1999
Inhibition of water permeability in the rat collecting duct: effect of imidazoline and alpha-2 compounds.
    Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine (New York, N.Y.), 1999, Volume: 221, Issue:2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Arginine Vasopressin; Clonidine; Cyclic AMP; Dose-Response Relationship, Drug; Imidazoles; Kidney Tubules, Collecting; Medetomidine; Oxazoles; Oxymetazoline; Permeability; Rats; Rats, Wistar; Rilmenidine; Water

1999
An unexpected central hypertensive effect of the new imidazoline compound benazoline.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypertension; Imidazoles; Imidazoline Receptors; Male; Nasal Decongestants; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Yohimbine

1999
Identification of imidazoline-receptor binding sites in cortex and medulla of the bovine adrenal gland. Colocalization with MAO-A and MAO-B.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Adrenal Cortex; Adrenal Medulla; Adrenergic beta-Agonists; Animals; Autoradiography; Benzofurans; Binding Sites; Cattle; Clonidine; Imidazoles; Imidazoline Receptors; Isoenzymes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Rats; Receptors, Drug; Rilmenidine; Thiazoles; Tritium

1999
Mechanism of the sympathoinhibition produced by the clonidine-like drugs rilmenidine and moxonidine.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzazepines; Blood Pressure; Clonidine; Decerebrate State; Heart Rate; Imidazoles; Injections, Spinal; Medulla Oblongata; Microinjections; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Yohimbine

1999
Central imidazoline- and alpha 2-receptors involved in the cardiovascular actions of centrally acting antihypertensive agents.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Microinjections; Models, Neurological; Norepinephrine; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Serotonin; Sympathetic Nervous System

1999
alpha 2A-adrenoceptors, not I1-imidazoline receptors, mediate the hypotensive effects of rilmenidine and moxonidine in conscious mice. In vivo and in vitro studies.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cell Line; Dogs; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hypotension; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Quinolizines; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Transfection

1999
Influence of sinoaortic barodenervation on the hypotensive effects of imidazoline-like drugs in stroke-prone spontaneously hypertensive rats.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cerebrovascular Disorders; Circadian Rhythm; Clonidine; Denervation; Heart Rate; Hypotension; Imidazoles; Male; Oxazoles; Pressoreceptors; Rats; Rats, Inbred SHR; Rilmenidine; Sinus of Valsalva; Time Factors

1999
Cardiovascular effects of clonidine-like drugs in pithed rabbits.
    Hypertension (Dallas, Tex. : 1979), 1999, Volume: 34, Issue:4 Pt 2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cardiovascular Physiological Phenomena; Clonidine; Electric Stimulation; Heart Rate; Imidazoles; Male; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System; Synaptic Transmission

1999
[New central agents in the treatment of arterial hypertension].
    Anales de medicina interna (Madrid, Spain : 1984), 1999, Volume: 16, Issue:10

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Antagonists; Adrenergic Uptake Inhibitors; Adult; Antihypertensive Agents; Atenolol; Calcium Channel Blockers; Clonidine; Diabetes Complications; Humans; Hypertension; Imidazoles; Nifedipine; Oxazoles; Renin-Angiotensin System; Reserpine; Rilmenidine; Risk Factors; Sympathetic Nervous System; Vasodilator Agents

1999
Actions of L-NAME and methylene blue on the hypotensive effects of clonidine and rilmenidine in the anesthetized rat.
    Journal of cardiovascular pharmacology, 2000, Volume: 35, Issue:5

    Topics: Anesthesia; Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Cyclic GMP; Drug Interactions; Enzyme Inhibitors; Hypotension; Male; Methylene Blue; NG-Nitroarginine Methyl Ester; Nitric Oxide; Oxazoles; Rats; Rats, Wistar; Rilmenidine

2000
Species-specific pharmacological properties of human alpha(2A)-adrenoceptors.
    Hypertension (Dallas, Tex. : 1979), 2000, Volume: 36, Issue:3

    Topics: Adrenergic alpha-Agonists; Adult; Aged; Amino Acid Sequence; Animals; Antihypertensive Agents; Female; Heart Atria; Humans; Imidazoles; Male; Middle Aged; Molecular Sequence Data; Norepinephrine; Oxazoles; Oxymetazoline; Pulmonary Artery; Rabbits; Receptors, Adrenergic, alpha-2; Rilmenidine; Species Specificity; Tritium

2000
Comparison of renal sympathetic baroreflex effects of rilmenidine and alpha-methylnoradrenaline in the ventrolateral medulla of the rabbit.
    Journal of hypertension, 2000, Volume: 18, Issue:9

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Dose-Response Relationship, Drug; Female; Idazoxan; Kidney; Male; Medulla Oblongata; Nordefrin; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Rilmenidine; Sympathetic Nervous System; Vasoconstrictor Agents

2000
[Imidazole receptor agonists--a new advance in the treatment of hypertension?].
    Vnitrni lekarstvi, 2000, Volume: 46, Issue:2

    Topics: Antihypertensive Agents; Humans; Hypertension; Imidazoles; Imidazoline Receptors; Oxazoles; Receptors, Drug; Rilmenidine

2000
Nitric oxide and central antihypertensive drugs: one more difference between catecholamines and imidazolines.
    Hypertension (Dallas, Tex. : 1979), 2001, Volume: 37, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cardiovascular System; Catecholamines; Clonidine; Heart Rate; Hypotension; Imidazoles; Male; Nitric Oxide; Nitroarginine; Nordefrin; Oxazoles; Rabbits; Rilmenidine

2001
Relative importance of rostral ventrolateral medulla in sympathoinhibitory action of rilmenidine in conscious and anesthetized rabbits.
    Journal of cardiovascular pharmacology, 2001, Volume: 37, Issue:3

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Female; Kidney; Male; Medulla Oblongata; Microinjections; Oxazoles; Pressoreceptors; Rabbits; Reflex; Rilmenidine; Sympathetic Nervous System

2001
Imidazoline I(1) receptor-induced activation of phosphatidylcholine-specific phospholipase C elicits mitogen-activated protein kinase phosphorylation in PC12 cells.
    European journal of pharmacology, 2001, Volume: 415, Issue:2-3

    Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzofurans; Choline; Diglycerides; Enzyme Activation; Imidazoles; Imidazoline Receptors; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nerve Growth Factor; Oxazoles; PC12 Cells; Phosphorylation; Phosphorylcholine; Rats; Receptors, Drug; Rilmenidine; Signal Transduction; Type C Phospholipases

2001
Synthesis and biological evaluation of pyrrolinic isosteres of rilmenidine. Discovery of cis-/trans-dicyclopropylmethyl-(4,5-dimethyl-4,5-dihydro-3H-pyrrol-2-yl)-amine (LNP 509), an I1 imidazoline receptor selective ligand with hypotensive activity.
    Journal of medicinal chemistry, 2001, May-10, Volume: 44, Issue:10

    Topics: Adrenal Medulla; Animals; Antihypertensive Agents; Binding Sites; Blood Pressure; Cattle; Cyclopropanes; Frontal Lobe; Imidazoline Receptors; In Vitro Techniques; Kidney Cortex; Ligands; Male; Oxazoles; Pyrroles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Stereoisomerism; Structure-Activity Relationship

2001
Effects of imidazoline antihypertensive drugs on sympathetic tone and noradrenaline release in the prefrontal cortex.
    British journal of pharmacology, 2001, Volume: 134, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Guanabenz; Heart Rate; Imidazoles; Male; Microdialysis; Norepinephrine; Oxazoles; Prefrontal Cortex; Rats; Rats, Wistar; Rilmenidine; Sympathetic Nervous System

2001
Involvement of imidazoline receptors in the baroreflex effects of rilmenidine in conscious rabbits.
    Journal of hypertension, 2001, Volume: 19, Issue:9

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Fourth Ventricle; Heart Rate; Imidazoline Receptors; Injections, Intraventricular; Methyldopa; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine

2001
Sympathetic modulation of renal blood flow by rilmenidine and captopril: central vs. peripheral effects.
    American journal of physiology. Renal physiology, 2002, Volume: 282, Issue:1

    Topics: Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Captopril; Feedback; Female; Kidney Glomerulus; Male; Oxazoles; Rabbits; Renal Circulation; Rilmenidine; Sympathetic Nervous System

2002
Evidence for synergy between alpha(2)-adrenergic and nonadrenergic mechanisms in central blood pressure regulation.
    Circulation, 2002, Mar-05, Volume: 105, Issue:9

    Topics: Adrenergic Agonists; Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Blood Pressure; Brain Stem; Cardiovascular System; Cyclopropanes; Drug Synergism; Guanosine 5'-O-(3-Thiotriphosphate); Hypotension; Imidazoles; Injections, Intraventricular; Mice; Mice, Transgenic; Microinjections; Nordefrin; Oxazoles; Pyrroles; Rabbits; Receptors, Adrenergic; Receptors, Adrenergic, alpha-2; Rilmenidine; Sympathetic Nervous System

2002
The hypotensive action of rilmenidine is dependent on functional N-methyl-D-aspartate receptor in the rostral ventrolateral medulla of conscious spontaneously hypertensive rats.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Animals; Antihypertensive Agents; Dose-Response Relationship, Drug; Hemodynamics; Hypertension; Male; Medulla Oblongata; Microinjections; N-Methylaspartate; Oxazoles; Rats; Rats, Inbred SHR; Receptors, N-Methyl-D-Aspartate; Rilmenidine

2002
Protective effects of rilmenidine and AGN 192403 on oxidative cytotoxicity and mitochondrial inhibitor-induced cytotoxicity in astrocytes.
    Free radical biology & medicine, 2002, Nov-15, Volume: 33, Issue:10

    Topics: Animals; Animals, Newborn; Antihypertensive Agents; Antimycin A; Astrocytes; Bridged Bicyclo Compounds; Caspase 9; Caspases; Cell Death; Cytochrome c Group; Dose-Response Relationship, Drug; Free Radicals; Heptanes; Lysosomes; Membrane Potentials; Mitochondria; Models, Chemical; Naphthoquinones; Neuroglia; Oxazoles; Oxidative Stress; Oxygen; Rats; Rats, Sprague-Dawley; Reactive Oxygen Species; Rilmenidine; Time Factors

2002
Effects of rilmenidine and guanfacine in acute renal denervated rats.
    Proceedings of the Western Pharmacology Society, 2002, Volume: 45

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Denervation; Guanfacine; Heart Rate; Kidney; Male; Natriuresis; Oxazoles; Rats; Rats, Sprague-Dawley; Rilmenidine

2002
Protective effects of centrally acting sympathomodulatory drugs on myocardial ischemia induced by sympathetic overactivity in rabbits.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 2003, Volume: 36, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Electrocardiography; Female; Glutamic Acid; Heart Rate; Hemodynamics; Male; Myocardial Ischemia; NG-Nitroarginine Methyl Ester; Oxazoles; Propranolol; Rabbits; Rilmenidine; Sympathetic Nervous System

2003
Importance of imidazoline-preferring receptors in the cardiovascular actions of chronically administered moxonidine, rilmenidine and clonidine in conscious rabbits.
    Journal of hypertension, 2003, Volume: 21, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Cardiovascular System; Clonidine; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Fourth Ventricle; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Injections, Intraventricular; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine

2003
Alpha2-adrenoceptor ligands inhibit alpha1-adrenoceptor-mediated contraction of isolated rat arteries.
    Fundamental & clinical pharmacology, 2002, Volume: 16, Issue:4

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Arteries; Azepines; Brimonidine Tartrate; Clonidine; Idazoxan; In Vitro Techniques; Ligands; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Oxazoles; Prostaglandins; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Rilmenidine; Yohimbine

2002
Value of rilmenidine therapy and its combination with perindopril on blood pressure and left ventricular hypertrophy in patients with essential hypertension (VERITAS).
    Current medical research and opinion, 2003, Volume: 19, Issue:3

    Topics: Adrenergic alpha-Agonists; Adult; Aged; Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Blood Pressure; Drug Therapy, Combination; Echocardiography; Humans; Hypertension; Hypertrophy, Left Ventricular; Male; Middle Aged; Oxazoles; Perindopril; Rilmenidine

2003
Effect of ethanol on reductions in norepinephrine electrochemical signal in the rostral ventrolateral medulla and hypotension elicited by I1-receptor activation in spontaneously hypertensive rats.
    Alcoholism, clinical and experimental research, 2003, Volume: 27, Issue:9

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Electrochemistry; Ethanol; Hypotension; Imidazoline Receptors; Male; Medulla Oblongata; Microdialysis; Norepinephrine; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Drug; Rilmenidine; Sympatholytics

2003
Rilmenidine produces mydriasis in cats by stimulation of CNS alpha 2-adrenoceptors.
    Autonomic & autacoid pharmacology, 2003, Volume: 23, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Cats; Central Nervous System; Dose-Response Relationship, Drug; Female; Male; Mydriatics; Oxazoles; Pupil; Receptors, Adrenergic, alpha-2; Rilmenidine

2003
Short-term effects of rilmenidine on left ventricular hypertrophy and systolic and diastolic function in patients with essential hypertension: comparison with an angiotensin converting enzyme inhibitor and a calcium antagonist.
    Japanese heart journal, 2003, Volume: 44, Issue:5

    Topics: Aged; Angiotensin-Converting Enzyme Inhibitors; Antihypertensive Agents; Calcium Channel Blockers; Diastole; Female; Humans; Hypertension; Hypertrophy, Left Ventricular; Male; Middle Aged; Oxazoles; Rilmenidine; Systole; Ventricular Function, Left

2003
Sympathetic responses to stress and rilmenidine in 2K1C rabbits: evidence of enhanced nonvascular effector mechanism.
    Hypertension (Dallas, Tex. : 1979), 2004, Volume: 43, Issue:3

    Topics: Animals; Blood Pressure; Female; Heart Rate; Hypertension, Renovascular; Kidney; Male; Organ Size; Oxazoles; Rabbits; Rilmenidine; Stress, Physiological; Sympathetic Nervous System

2004
Chronic ethanol administration attenuates imidazoline I1 receptor- or alpha 2-adrenoceptor-mediated reductions in blood pressure and hemodynamic variability in hypertensive rats.
    European journal of pharmacology, 2004, Feb-06, Volume: 485, Issue:1-3

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Blood Pressure; Dose-Response Relationship, Drug; Ethanol; Hemodynamics; Hypertension; Imidazoline Receptors; Male; Methyldopa; Motor Activity; Oxazoles; Protein Subunits; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

2004
Are centrally acting imidazoline agents appropriate therapy for renovascular hypertension?
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Humans; Hypertension, Renovascular; Kidney; Oxazoles; Rabbits; Renin; Rilmenidine; Sympathetic Nervous System

2003
The role of I(1)-imidazoline receptors and alpha(2)-adrenergic receptors in the modulation of glucose and lipid metabolism in the SHROB model of metabolic syndrome X.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Disease Models, Animal; Female; Glucagon; Glucose; Glucose Tolerance Test; Humans; Imidazoles; Imidazoline Receptors; Lipid Metabolism; Male; Metabolic Syndrome; Obesity; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Yohimbine

2003
Moxonidine displays a presynaptic alpha-2-adrenoceptor-dependent synergistic sympathoinhibitory action at imidazoline-1 receptors.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Benzofurans; Bridged Bicyclo Compounds; Brimonidine Tartrate; Drug Synergism; Heart; Heptanes; Imidazoles; Imidazoline Receptors; Norepinephrine; Oxazoles; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Sympatholytics; Yohimbine

2003
Alpha(2A)-adrenergic versus imidazoline receptor controversy in rilmenidine's action: alpha(2A)-antagonism in humans versus alpha(2A)-agonism in rabbits.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Antihypertensive Agents; Humans; Imidazoline Receptors; Molecular Sequence Data; Oxazoles; Oxymetazoline; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sequence Alignment

2003
Apparent absence of direct renal effect of imidazoline receptor agonists.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Diuretics; Furosemide; Imidazoles; Imidazoline Receptors; Kidney; Male; Natriuresis; Nephrectomy; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Drug; Rilmenidine

2003
[Effect of Rilmenidine(Tenaxum) on the activity of the autonomic nervous system in patients with hypertension and asthma].
    Wiadomosci lekarskie (Warsaw, Poland : 1960), 2003, Volume: 56, Issue:11-12

    Topics: Adrenergic alpha-Agonists; Antihypertensive Agents; Asthma; Autonomic Nervous System; Female; Heart Rate; Humans; Hypertension; Oxazoles; Rilmenidine

2003
Chronic treatment with rilmenidine in spontaneously hypertensive rats: differences between two schedules of administration.
    Journal of cardiovascular pharmacology, 2004, Volume: 43, Issue:3

    Topics: Analysis of Variance; Animals; Antihypertensive Agents; Heart Rate; Hypertension; Infusion Pumps; Injections, Intraperitoneal; Male; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine

2004
The effects of the alpha2-adrenergic receptor agonists clonidine and rilmenidine, and antagonists yohimbine and efaroxan, on the spinal cholinergic receptor system in the rat.
    Basic & clinical pharmacology & toxicology, 2004, Volume: 94, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Benzofurans; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Injections, Spinal; Ligands; Male; Microdialysis; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Cholinergic; Rilmenidine; Spinal Cord; Time Factors; Yohimbine

2004
Efficacy and tolerability of long-term rilmenidine treatment in hypertensive diabetic patients. A retrospective analysis of a general practice study.
    American journal of cardiovascular drugs : drugs, devices, and other interventions, 2004, Volume: 4, Issue:3

    Topics: Adult; Aged; Antihypertensive Agents; Biomarkers; Blood Pressure; Creatinine; Diabetes Mellitus; Diastole; Drug Therapy, Combination; Family Practice; Female; Humans; Hypertension; Incidence; Male; Middle Aged; Oxazoles; Retrospective Studies; Rilmenidine; Systole; Time; Treatment Outcome; Triglycerides

2004
Differential modulation by estrogen of alpha2-adrenergic and I1-imidazoline receptor-mediated hypotension in female rats.
    Journal of applied physiology (Bethesda, Md. : 1985), 2004, Volume: 97, Issue:4

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Behavior, Animal; Blood Pressure; Estrogens; Female; Heart Rate; Hormone Replacement Therapy; Hypotension; Imidazoline Receptors; Methyldopa; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

2004
[Effect of rilmenidine on intraocular pressure in rabbits, interaction with efaroxan and rauwolscine].
    Klinika oczna, 2004, Volume: 106, Issue:1-2

    Topics: Administration, Topical; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzofurans; Drug Interactions; Glaucoma; Imidazoles; Intraocular Pressure; Male; Oxazoles; Rabbits; Rilmenidine; Time Factors; Yohimbine

2004
Moxonidine and rilmenidine injected into the medial septal area reduces the salivation induced by pilocarpine.
    Autonomic neuroscience : basic & clinical, 2004, May-31, Volume: 112, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Drug Interactions; Idazoxan; Imidazoles; Male; Muscarinic Agonists; Oxazoles; Pilocarpine; Rats; Rats, Sprague-Dawley; Rilmenidine; Salivation; Septum of Brain; Yohimbine

2004
[Case report: hypertension after stroke].
    Wiener medizinische Wochenschrift (1946), 2004, Volume: 154 Spec No 1, Issue:1

    Topics: Aged; Aged, 80 and over; Amlodipine; Antihypertensive Agents; Basal Ganglia Cerebrovascular Disease; Blood Pressure Monitoring, Ambulatory; Blood Urea Nitrogen; Body Weight; Cerebral Infarction; Circadian Rhythm; Dose-Response Relationship, Drug; Drug Therapy, Combination; Follow-Up Studies; Glycated Hemoglobin; Humans; Hypertension; Internal Capsule; Male; Oxazoles; Prognosis; Ramipril; Rilmenidine; Sympathetic Nervous System

2004
Effects of centrally acting antihypertensive drugs on the microcirculation of spontaneously hypertensive rats.
    Brazilian journal of medical and biological research = Revista brasileira de pesquisas medicas e biologicas, 2004, Volume: 37, Issue:10

    Topics: Animals; Antihypertensive Agents; Clonidine; Cyclopropanes; Imidazoline Receptors; Microcirculation; Oxazoles; Pyrroles; Rats; Rats, Inbred SHR; Receptors, Drug; Rilmenidine; Splanchnic Circulation; Sympathetic Nervous System; Vasodilation

2004
Rilmenidine prevents blood pressure increase in rats with compromised nitric oxide production.
    Acta pharmacologica Sinica, 2004, Volume: 25, Issue:12

    Topics: Animals; Antihypertensive Agents; Aorta, Thoracic; Blood Pressure; Brain; Endothelium, Vascular; Heart Ventricles; Hypertension; Imidazoline Receptors; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Oxazoles; Rats; Rats, Wistar; Receptors, Drug; Rilmenidine

2004
Mitogen-activated protein kinase phosphorylation in the rostral ventrolateral medulla plays a key role in imidazoline (i1)-receptor-mediated hypotension.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:3

    Topics: Animals; Benzofurans; Blood Pressure; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Medulla Oblongata; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Oxazoles; Phosphorylation; Rats; Rats, Sprague-Dawley; Receptors, Drug; Rilmenidine; Signal Transduction

2005
Site-dependent inhibition of neuronal c-jun in the brainstem elicited by imidazoline I1 receptor activation: role in rilmenidine-evoked hypotension.
    European journal of pharmacology, 2005, May-09, Volume: 514, Issue:2-3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzazepines; Benzofurans; Blood Pressure; Brain Stem; Cerebrospinal Fluid; Clonidine; Consciousness; Gene Expression; Heart Rate; Hydralazine; Hypotension; Imidazoles; Imidazoline Receptors; Immunohistochemistry; Male; Medulla Oblongata; Neurons; Nordefrin; Oxazoles; Proto-Oncogene Proteins c-jun; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; RNA, Messenger; Time Factors; Vasoconstrictor Agents; Vasodilator Agents

2005
Neuronal norepinephrine responses of the rostral ventrolateral medulla and nucleus tractus solitarius neurons distinguish the I1- from the alpha2-receptor-mediated hypotension in conscious SHRs.
    Journal of cardiovascular pharmacology, 2005, Volume: 46, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Area Postrema; Benzazepines; Benzofurans; Blood Pressure; Clonidine; Consciousness; Heart Rate; Hypotension; Imidazoles; Interleukin-1; Male; Motor Activity; Neurons; Nordefrin; Norepinephrine; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Rilmenidine; Solitary Nucleus

2005
Role of imidazoline receptors in the anti-aversive properties of clonidine during opiate withdrawal in rats.
    The European journal of neuroscience, 2005, Volume: 22, Issue:7

    Topics: Adrenergic alpha-Agonists; Animals; Avoidance Learning; Behavior, Animal; Clonidine; Conditioning, Operant; Dose-Response Relationship, Drug; Drug Interactions; Imidazoline Receptors; Male; Morphine Dependence; Naloxone; Narcotic Antagonists; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Drug; Rilmenidine; Statistics, Nonparametric; Substance Withdrawal Syndrome

2005
Central actions of agmatine in conscious spontaneously hypertensive rats.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 2005, Volume: 27, Issue:8

    Topics: Agmatine; Animals; Antihypertensive Agents; Blood Pressure; Brain; Cardiovascular System; Clonidine; Consciousness; Dose-Response Relationship, Drug; Drug Interactions; Heart Rate; Hypertension; Injections, Intraventricular; Male; Movement; Oxazoles; Rats; Rats, Inbred SHR; Rilmenidine

2005
Lipid-lowering actions of imidazoline antihypertensive agents in metabolic syndrome X.
    Naunyn-Schmiedeberg's archives of pharmacology, 2006, Volume: 372, Issue:4

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Cell Membrane; Cholesterol; Clonidine; Disease Models, Animal; Female; Guanabenz; Hyperlipidemias; Imidazoles; Imidazoline Receptors; Liver; Male; Metabolic Syndrome; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Drug; Rilmenidine; Triglycerides

2006
Opposite to alpha2-adrenergic agonists, an imidazoline I1 selective compound does not influence reflex bradycardia in rabbits.
    Autonomic neuroscience : basic & clinical, 2006, Jul-30, Volume: 128, Issue:1-2

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Autonomic Nervous System; Baroreflex; Blood Pressure; Bradycardia; Brain Stem; Cyclopropanes; Dexmedetomidine; Drug Interactions; Drug Synergism; Enzyme Inhibitors; Heart; Heart Rate; Imidazoline Receptors; Male; Nitric Oxide; Nitric Oxide Synthase; Oxazoles; Phenylephrine; Pyrroles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Reticular Formation; Rilmenidine; Solitary Nucleus

2006
Involvement of phosphatidylcholine-selective phospholipase C in activation of mitogen-activated protein kinase pathways in imidazoline receptor antisera-selected protein.
    Journal of cellular biochemistry, 2006, Aug-15, Volume: 98, Issue:6

    Topics: Animals; Cell Membrane; CHO Cells; Cricetinae; Diglycerides; Dose-Response Relationship, Drug; Extracellular Signal-Regulated MAP Kinases; Guanosine Triphosphate; Imidazoles; Imidazoline Receptors; Intracellular Signaling Peptides and Proteins; Ligands; MAP Kinase Signaling System; Oxazoles; Rilmenidine; Signal Transduction; Type C Phospholipases

2006
Nischarin as a functional imidazoline (I1) receptor.
    FEBS letters, 2006, May-29, Volume: 580, Issue:13

    Topics: Adrenergic alpha-Agonists; Animals; Antibodies; Imidazoline Receptors; Intracellular Signaling Peptides and Proteins; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; NIH 3T3 Cells; Oligodeoxyribonucleotides, Antisense; Oxazoles; PC12 Cells; Rats; Receptors, Drug; Rilmenidine

2006
Efficacy and tolerability of rilmenidine compared with isradipine in hypertensive patients with features of metabolic syndrome.
    Current medical research and opinion, 2006, Volume: 22, Issue:7

    Topics: Adult; Aged; Antihypertensive Agents; Blood Glucose; Blood Pressure; Double-Blind Method; Drug Tolerance; Female; Humans; Hypertension; Insulin; Isradipine; Lipids; Male; Metabolic Syndrome; Middle Aged; Oxazoles; Rilmenidine

2006
Effects of rilmenidine on 24-h rhythmicity of blood pressure and spontaneous baroreflex sensitivity in essential hypertensive subjects.
    Journal of hypertension, 2006, Volume: 24, Issue:8

    Topics: Adult; Analysis of Variance; Antihypertensive Agents; Baroreflex; Blood Pressure; Circadian Rhythm; Confounding Factors, Epidemiologic; Female; Heart Rate; Humans; Hypertension; Male; Middle Aged; Oxazoles; Rilmenidine; Severity of Illness Index; Time Factors; Treatment Outcome

2006
Possible role of NMDA receptors in antinociception induced by rilmenidine in mice in the formalin test.
    European journal of pain (London, England), 2007, Volume: 11, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analgesics; Animals; Benzofurans; Binding Sites; Binding, Competitive; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Imidazoles; Imidazoline Receptors; Male; Mice; Nervous System; Neurons, Afferent; Nociceptors; Oxazoles; Pain; Pain Measurement; Receptors, Drug; Receptors, N-Methyl-D-Aspartate; Rilmenidine; Yohimbine

2007
Contribution of imidazoline receptors and alpha2-adrenoceptors in the rostral ventrolateral medulla to sympathetic baroreflex inhibition by systemic rilmenidine.
    Journal of hypertension, 2007, Volume: 25, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Dose-Response Relationship, Drug; Idazoxan; Imidazoline Receptors; Injections, Intravenous; Kidney; Medulla Oblongata; Neural Inhibition; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System

2007
Direct evidence for imidazoline (I1) receptor modulation of ethanol action on norepinephrine-containing neurons in the rostral ventrolateral medulla in conscious spontaneously hypertensive rats.
    Alcoholism, clinical and experimental research, 2007, Volume: 31, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Central Nervous System Depressants; Clonidine; Dose-Response Relationship, Drug; Electrochemistry; Ethanol; Heart Rate; Imidazoline Receptors; Male; Medulla Oblongata; Microinjections; Neurons; Nordefrin; Norepinephrine; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

2007
Inhibition of nischarin expression attenuates rilmenidine-evoked hypotension and phosphorylated extracellular signal-regulated kinase 1/2 production in the rostral ventrolateral medulla of rats.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 324, Issue:1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Heart Rate; Hypotension; Intracellular Signaling Peptides and Proteins; Male; Medulla Oblongata; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Oligodeoxyribonucleotides, Antisense; Oxazoles; Phosphorylation; Rats; Rats, Sprague-Dawley; Rilmenidine

2008
Improvement of cardiac diastolic function by long-term centrally mediated sympathetic inhibition in one-kidney, one-clip hypertensive rabbits.
    American journal of hypertension, 2008, Volume: 21, Issue:1

    Topics: Adrenergic beta-Antagonists; Animals; Antihypertensive Agents; Blood Pressure; Cardiomyopathies; Diastole; Disease Models, Animal; Heart Rate; Hypertension, Renovascular; Hypertrophy, Left Ventricular; Ligation; Male; Metoprolol; Myocardial Contraction; Nephrectomy; Oxazoles; Rabbits; Renal Artery; Rilmenidine; Sympathetic Nervous System; Systole; Time Factors; Ultrasonography; Ventricular Function; Ventricular Remodeling

2008
The antiarrhythmic effect of centrally administered rilmenidine involves muscarinic receptors, protein kinase C and mitochondrial signalling pathways.
    British journal of pharmacology, 2008, Volume: 153, Issue:8

    Topics: Adrenergic alpha-Agonists; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Epinephrine; KATP Channels; Male; Mitochondrial Membrane Transport Proteins; Mitochondrial Permeability Transition Pore; Oxazoles; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Rilmenidine

2008
[Analysis of central mechanisms involved in gastric mucosal integrity].
    Neuropsychopharmacologia Hungarica : a Magyar Pszichofarmakologiai Egyesulet lapja = official journal of the Hungarian Association of Psychopharmacology, 2008, Volume: 10, Issue:3

    Topics: Animals; Arachidonic Acids; beta-Endorphin; Clonidine; Endocannabinoids; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Ethanol; Excitatory Amino Acids; Gastric Mucosa; Injections, Intraventricular; Male; Naloxone; Naltrexone; Narcotic Antagonists; Neurotransmitter Agents; Nociceptin; Oligopeptides; Opioid Peptides; Oxazoles; Polyunsaturated Alkamides; Rats; Rats, Wistar; Receptors, Opioid; Rilmenidine; Stomach Ulcer

2008
Chronic ethanol attenuates centrally-mediated hypotension elicited via alpha(2)-adrenergic, but not I(1)-imidazoline, receptor activation in female rats.
    Life sciences, 2009, Jan-16, Volume: 84, Issue:3-4

    Topics: Animals; Area Under Curve; Blood Pressure; Ethanol; Female; Heart Rate; Imidazoline Receptors; Methyldopa; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Rilmenidine

2009
Alpha 2A-adrenergic receptor signaling underlies synergistic enhancement of ethanol-induced behavioral impairment by clonidine.
    Alcoholism, clinical and experimental research, 2009, Volume: 33, Issue:3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Behavior, Animal; Central Nervous System Depressants; Cerebellum; Clonidine; Drug Synergism; Ethanol; Imidazoline Receptors; Locus Coeruleus; Male; Motor Activity; Oxazoles; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Reflex; Rilmenidine; Rotarod Performance Test

2009
Cardiac and renal baroreflex control during stress in conscious renovascular hypertensive rabbits: effect of rilmenidine.
    Journal of hypertension, 2009, Volume: 27, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Female; Heart Rate; Hypertension, Renovascular; Kidney; Male; Oxazoles; Rabbits; Renin; Rilmenidine; Stress, Psychological; Sympathetic Nervous System

2009
The synergistic interaction between rilmenidine and paracetamol in the writhing test in mice.
    Naunyn-Schmiedeberg's archives of pharmacology, 2009, Volume: 379, Issue:6

    Topics: Acetaminophen; Animals; Dose-Response Relationship, Drug; Drug Interactions; Drug Synergism; Drug Therapy, Combination; Male; Mice; Oxazoles; Pain; Pain Measurement; Rilmenidine; Rotarod Performance Test

2009
Comparison of agmatine with moxonidine and rilmenidine in morphine dependence in vitro: role of imidazoline I(1) receptors.
    European journal of pharmacology, 2009, Jun-10, Volume: 612, Issue:1-3

    Topics: Agmatine; Animals; Antihypertensive Agents; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Dose-Response Relationship, Drug; Imidazoles; Imidazoline Receptors; Morphine Dependence; Oxazoles; Rilmenidine; RNA, Messenger; RNA, Small Interfering; Time Factors; Transfection

2009
Pharmacological analysis of alpha(2)-adrenoceptor subtypes mediating analgesic, anti-inflammatory and gastroprotective actions.
    Inflammopharmacology, 2009, Volume: 17, Issue:3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Analgesics; Animals; Anti-Inflammatory Agents; Anti-Ulcer Agents; Clonidine; Disease Models, Animal; Edema; Gastrointestinal Motility; Hyperalgesia; Male; Oxazoles; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Rilmenidine; Stomach Ulcer

2009
Synergistic interaction between rilmenidine and ibuprofen in the writhing test in mice.
    Neuro endocrinology letters, 2009, Volume: 30, Issue:2

    Topics: Acetic Acid; Adrenergic alpha-Agonists; Analgesics, Non-Narcotic; Analysis of Variance; Animals; Dose-Response Relationship, Drug; Drug Synergism; Ibuprofen; Male; Mice; Motor Activity; Oxazoles; Pain; Pain Measurement; Rilmenidine; Rotarod Performance Test

2009
Effects of chronic sympatho-inhibition on reflex control of renal blood flow and plasma renin activity in renovascular hypertension.
    British journal of pharmacology, 2010, Jan-01, Volume: 159, Issue:2

    Topics: Animals; Antihypertensive Agents; Baroreflex; Blood Pressure; Female; Hypertension, Renovascular; Kidney; Male; Oxazoles; Rabbits; Renal Circulation; Renin; Rilmenidine; Sympathetic Nervous System

2010
Microvascular effects of centrally acting antihypertensive drugs in spontaneously hypertensive rats.
    Journal of cardiovascular pharmacology, 2010, Volume: 55, Issue:3

    Topics: Administration, Oral; Animals; Antihypertensive Agents; Blood Pressure; Capillaries; Clonidine; Disease Models, Animal; Hypertension; Imidazoles; Male; Microcirculation; Microscopy, Video; Muscle, Skeletal; Oxazoles; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Rilmenidine; Skin; Time Factors

2010
Rilmenidine attenuates toxicity of polyglutamine expansions in a mouse model of Huntington's disease.
    Human molecular genetics, 2010, Jun-01, Volume: 19, Issue:11

    Topics: Animals; Autophagy; Cells, Cultured; Huntingtin Protein; Huntington Disease; Mice; Mice, Transgenic; Nerve Tissue Proteins; Neurons; Nuclear Proteins; Oxazoles; Peptides; Rilmenidine; Rotarod Performance Test

2010
Development of a fast LC-MS/MS method for quantification of rilmenidine in human serum: elucidation of fragmentation pathways by HRMS.
    Journal of mass spectrometry : JMS, 2010, Volume: 45, Issue:10

    Topics: Antihypertensive Agents; Chromatography, Liquid; Drug Stability; Humans; Least-Squares Analysis; Oxazoles; Reproducibility of Results; Rilmenidine; Sensitivity and Specificity; Solid Phase Extraction; Tandem Mass Spectrometry

2010
Activation of phosphatidylinositol 3-kinase/Akt signaling pathway and endogenous nitric oxide are needed for the antiarrhythmic effect of centrally administered rilmenidine.
    European journal of pharmacology, 2010, Nov-25, Volume: 647, Issue:1-3

    Topics: Androstadienes; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Epinephrine; Halothane; Male; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Oxazoles; Phosphatidylinositol 3-Kinase; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Rilmenidine; Signal Transduction; Sympathomimetics; Wortmannin

2010
Investigation of the effects of the chronic administration of some antihypertensive drugs on enzymatic and non-enzymatic oxidant/antioxidant parameters in rat ovarian tissue.
    Gynecological endocrinology : the official journal of the International Society of Gynecological Endocrinology, 2011, Volume: 27, Issue:11

    Topics: Amlodipine; Animals; Antihypertensive Agents; Antioxidants; Clonidine; Female; Glutathione; Glutathione Peroxidase; Glutathione Reductase; Glutathione Transferase; Methyldopa; Ovary; Oxazoles; Oxidants; Ramipril; Rats; Rats, Wistar; Rilmenidine; Superoxide Dismutase

2011
Effects of chronic sympatho-inhibition on renal excretory function in renovascular hypertension.
    Journal of hypertension, 2011, Volume: 29, Issue:5

    Topics: Animals; Antihypertensive Agents; Female; Hypertension, Renovascular; Kidney; Male; Oxazoles; Rabbits; Rilmenidine; Sympathetic Nervous System

2011
A novel mechanism for decreasing plasma lipid level from imidazoline I-1 receptor activation in high fat diet-fed mice.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 2011, Volume: 43, Issue:7

    Topics: Animals; Dietary Fats; Feeding Behavior; Gene Expression Regulation; Hep G2 Cells; Humans; Hyperlipidemias; Imidazoline Receptors; Intracellular Signaling Peptides and Proteins; Lipids; Liver; Male; Mice; Mice, Inbred C57BL; Oxazoles; Oxidation-Reduction; Receptors, Cytoplasmic and Nuclear; Rilmenidine; Signal Transduction

2011
Rilmenidine improves hepatic steatosis through p38-dependent pathway to higher the expression of farnesoid X receptor.
    Naunyn-Schmiedeberg's archives of pharmacology, 2012, Volume: 385, Issue:1

    Topics: Animals; Calcium; Cell Line, Tumor; Diet, High-Fat; Egtazic Acid; Fatty Liver; Humans; Imidazoline Receptors; Lipid Metabolism; Male; MAP Kinase Signaling System; Mice; Mice, Inbred C57BL; Oleic Acid; Oxazoles; Receptors, Cytoplasmic and Nuclear; Rilmenidine

2012
Chronically lowering sympathetic activity protects sympathetic nerves in spleens from aging F344 rats.
    Journal of neuroimmunology, 2012, Jun-15, Volume: 247, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Aging; Analysis of Variance; Animals; Body Weight; Catecholamines; Chromatography, High Pressure Liquid; Cyclic AMP; Dose-Response Relationship, Drug; Male; Norepinephrine; Organ Size; Oxazoles; Propanolamines; Protein Binding; Random Allocation; Rats; Rats, Inbred F344; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Rilmenidine; Spleen; Sympathetic Nervous System; Time Factors

2012
Improvement of hyperphagia by activation of cerebral I(1)-imidazoline receptors in streptozotocin-induced diabetic mice.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 2012, Volume: 44, Issue:9

    Topics: Animals; Benzofurans; Cerebrum; Diabetes Mellitus, Type 1; Disease Models, Animal; Eating; Female; Humans; Hyperphagia; Hypothalamus; Imidazoles; Imidazoline Receptors; Male; Mice; Mice, Inbred BALB C; Neuropeptide Y; Oxazoles; Rilmenidine; Streptozocin

2012
Imidazoline-1 receptor ligands as apoptotic agents: pharmacophore modeling and virtual docking study.
    Combinatorial chemistry & high throughput screening, 2013, Volume: 16, Issue:4

    Topics: Antineoplastic Agents; Apoptosis; Benzofurans; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Imidazoles; Imidazoline Receptors; K562 Cells; Ligands; Models, Molecular; Molecular Docking Simulation; Oxazoles; Quantitative Structure-Activity Relationship; Rilmenidine; Tumor Cells, Cultured

2013
Imidazoline versus alpha₂-adrenoceptors in the control of gastric motility in mice.
    European journal of pharmacology, 2013, Apr-05, Volume: 705, Issue:1-3

    Topics: Agmatine; Animals; Electric Stimulation; Female; Gastric Emptying; Harmine; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isoquinolines; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Oxazoles; Piperazines; Receptors, Adrenergic, alpha-2; Rilmenidine; Stomach

2013
Improvement of obesity by activation of I1-imidazoline receptors in high fat diet-fed mice.
    Hormone and metabolic research = Hormon- und Stoffwechselforschung = Hormones et metabolisme, 2013, Volume: 45, Issue:8

    Topics: Adipose Tissue, White; Animals; Body Weight; Diet, High-Fat; Energy Intake; Humans; Imidazoline Receptors; Male; Mice; Mice, Inbred C57BL; Obesity; Oxazoles; Rilmenidine

2013
Actions of rilmenidine on neurogenic hypertension in BPH/2J genetically hypertensive mice.
    Journal of hypertension, 2014, Volume: 32, Issue:3

    Topics: Administration, Oral; Animals; Antihypertensive Agents; Atropine; Baroreflex; Blood Pressure; Circadian Rhythm; Heart Rate; Hypertension; Infusions, Intraventricular; Infusions, Subcutaneous; Injections, Intraperitoneal; Male; Medulla Oblongata; Mice; Motor Activity; Oxazoles; Restraint, Physical; Rilmenidine; Stress, Physiological; Sympathetic Nervous System; Sympathomimetics

2014
Molecular biology: Remove, reuse, recycle.
    Nature, 2014, Oct-16, Volume: 514, Issue:7522

    Topics: Aging; Alzheimer Disease; Autophagy; Biomedical Research; Caloric Restriction; HIV; Humans; Longevity; Neoplasms; Oxazoles; Parkinson Disease; Phagosomes; Rilmenidine

2014
Rilmenidine suppresses proliferation and promotes apoptosis via the mitochondrial pathway in human leukemic K562 cells.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2016, Jan-01, Volume: 81

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents; Apoptosis; bcl-2-Associated X Protein; Caspase 3; Cell Cycle; Cell Proliferation; Cyclin B1; Doxorubicin; Humans; Imidazoline Receptors; K562 Cells; Leukemia; Mitochondria; Mitogen-Activated Protein Kinases; Oxazoles; Rilmenidine; RNA, Messenger

2016
Central Sympathetic Modulation Reverses Microvascular Alterations in a Rat Model of High-Fat Diet-Induced Metabolic Syndrome.
    Microcirculation (New York, N.Y. : 1994), 2016, Volume: 23, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Diet, High-Fat; Intravital Microscopy; Male; Metabolic Syndrome; Microcirculation; Microvessels; Muscle, Skeletal; Oxazoles; Rats; Rats, Wistar; Rilmenidine; Sodium Chloride, Dietary; Sympathetic Nervous System; Sympatholytics

2016
A combined ligand- and structure-based approach for the identification of rilmenidine-derived compounds which synergize the antitumor effects of doxorubicin.
    Bioorganic & medicinal chemistry, 2016, 07-15, Volume: 24, Issue:14

    Topics: Adrenergic alpha-Agonists; Antibiotics, Antineoplastic; Apoptosis; Doxorubicin; Drug Synergism; Humans; K562 Cells; Ligands; Molecular Structure; Oxazoles; Receptors, Adrenergic, alpha-2; Rilmenidine

2016
The Effects of Rilmenidine and Perindopril on Arousal Blood Pressure during 24 Hour Recordings in SHR.
    PloS one, 2016, Volume: 11, Issue:12

    Topics: Administration, Oral; Animals; Antihypertensive Agents; Blood Pressure; Blood Pressure Monitoring, Ambulatory; Heart Rate; Logistic Models; Male; Oxazoles; Perindopril; Rats; Rats, Inbred SHR; Rilmenidine; Telemetry

2016
MDMA-induced neurotoxicity of serotonin neurons involves autophagy and rilmenidine is protective against its pathobiology.
    Neurochemistry international, 2017, Volume: 105

    Topics: Adrenergic alpha-Agonists; Animals; Autophagy; Cell Survival; Cells, Cultured; Dose-Response Relationship, Drug; Female; Male; Mice; Mice, Inbred C57BL; N-Methyl-3,4-methylenedioxyamphetamine; Neuroprotective Agents; Oxazoles; Pregnancy; Rilmenidine; Serotonergic Neurons; Serotonin Agents

2017
An open-label study to assess the feasibility and tolerability of rilmenidine for the treatment of Huntington's disease.
    Journal of neurology, 2017, Volume: 264, Issue:12

    Topics: Adolescent; Adrenergic alpha-Agonists; Adult; Aged; Brain; Female; Humans; Huntington Disease; Longitudinal Studies; Magnetic Resonance Imaging; Male; Metabolomics; Middle Aged; Neuropsychological Tests; Oxazoles; Retrospective Studies; Rilmenidine; Time Factors; Treatment Outcome; Young Adult

2017