oxazoles has been researched along with diazepam in 55 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 49 (89.09) | 18.7374 |
1990's | 2 (3.64) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 2 (3.64) | 24.3611 |
2020's | 2 (3.64) | 2.80 |
Authors | Studies |
---|---|
Jobert, A; Soubrié, P; Thiébot, MH | 2 |
Costa, E; Guidotti, A; Naik, SR | 1 |
Biggio, G; Brodie, BB; Costa, E; Guidotti, A | 1 |
Longman, DA; Slater, P | 1 |
Risley, EA; Williams, M | 1 |
Maurer, R | 1 |
Anhut, H; Hertting, G; Steinhauer, HB | 1 |
Biggio, G; Casu, M; Corda, MG; Gessa, GL; Vernaleone, F | 1 |
Cheney, DL; Costa, E; Zsilla, G | 1 |
Cosi, C; Wood, PL | 1 |
Byberg, JR; Curtis, DR; Falch, E; Gynther, BD; Hjeds, H; Krogsgaard-Larsen, P; Labouta, IM | 1 |
Cavalla, D; Neff, NH | 1 |
Chuang, DM; Majewska, MD | 1 |
Löscher, W | 1 |
Hirate, K; Shinozaki, H | 1 |
Hailey, DM | 1 |
Ando, K; Yanagida, T | 1 |
Deguchi, T; Iwata, N; Mori, M; Nishijima, Y; Sakai, Y | 1 |
Millichap, JG | 1 |
Hooshmand, H; Suter, CG | 1 |
Borbély, F; Pasi, A; Velvart, J | 1 |
Mizutani, A | 1 |
Kamioka, T; Kobayashi, S; Suzuki, Y; Takagi, H | 1 |
Kaneto, H; Koida, M; Miyagawa, H; Tsuchie, F | 1 |
Kamioka, T; Kobayashi, S; Suzuki, Y; Tachikawa, R; Takagi, H | 1 |
Fromm, GH; Killian, JM; Sanchez, F | 1 |
Iwata, N; Mori, M; Nishijima, Y | 1 |
Hattori, K; Matsuda, K; Murata, H; Yasumura, A | 1 |
Ekstedt, J | 1 |
Clarke, DM | 1 |
Carrillo, L; de Bonnevaux, SC | 1 |
Hara, T; Iwata, N; Kobayashi, K; Shibata, T; Tonohiro, T | 1 |
Saano, V | 1 |
Ostrovskaia, RU | 1 |
Cananzi, AR; Costa, E; Guidotti, A | 1 |
Gardell, MA; Neale, JH; Shibla, DB | 1 |
Johnston, GA; Skerritt, JH | 1 |
Fukuda, H; Goto, M; Hasebe, Y; Kaneko, T; Kato, K | 1 |
Beani, L; Bianchi, C; Tanganelli, S | 1 |
Altmann, H; Dose, M; Emrich, HM; von Zerssen, D | 1 |
Bjørndal, N; Christensson, E; Gerlach, J | 1 |
Gomez-Ramos, P; Perez-Rico, C | 1 |
Macdonald, RL; Skerritt, JH | 1 |
Haddox, VG; Menon, MK; Vivonia, CA | 1 |
Back, KC; George, ME; Pinkerton, MK | 1 |
Cortese, I; Cuomo, V; Siro-Brigiani, G | 1 |
Fukuda, H; Kaneko, T; Ono, H | 1 |
Chieli, T; Cocchi, D; Fregnan, GB; Müller, EE | 1 |
Dixon, R; Hughes, AM; Kemp, JV; Nairn, K; Sellers, M; Yates, RA | 1 |
Hanson, GR; Jensen, M; Johnson, M; White, HS | 1 |
Chen, F; Chen, S; Liu, S; Peng, G; Zhang, C | 1 |
Cook, J; Golani, LK; Li, G; Moerke, MJ; Negus, SS | 1 |
Cerne, R; Cook, JM; Golani, LK; Jahan, R; Jin, X; Knutson, DE; Li, G; Mian, MY; Ping, X; Rashid, F; Sharmin, D; Smith, JL; Tiruveedhula, VVNPB; Witkin, JM | 1 |
Arnold, LA; Cerne, R; Cook, JM; Divović, B; Golani, LK; Jin, X; Lippa, A; Meyer, MJ; Mondal, P; Pandey, KP; Ping, X; Revanian, S; Savić, MM; Sharmin, D; Smith, JL; Witkin, JM; Zahn, NM | 1 |
1 review(s) available for oxazoles and diazepam
Article | Year |
---|---|
Chromatography of the 1,4-benzodiazepines.
Topics: Anti-Anxiety Agents; Chlordiazepoxide; Chromatography; Diazepam; Flurazepam; Humans; Methylation; Nitrazepam; Oxazepam; Oxazoles; Prazepam; Solvents; Spectrometry, Fluorescence; Temperature | 1974 |
3 trial(s) available for oxazoles and diazepam
Article | Year |
---|---|
Observations on the discrepancy between the clinical and the laboratory effects of anti-petit mal drugs.
Topics: Action Potentials; Anticonvulsants; Chloralose; Clinical Trials as Topic; Diazepam; Epilepsy, Absence; Humans; Oxazoles; Pentylenetetrazole; Trigeminal Nerve; Trimethadione | 1967 |
Therapeutic effects of GABA-ergic drugs in affective disorders. A preliminary report.
Topics: Adolescent; Adult; Analgesics; Anticonvulsants; Bipolar Disorder; Carbamazepine; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; gamma-Aminobutyric Acid; Humans; Isoxazoles; Male; Middle Aged; Mood Disorders; Oxazoles; Oxcarbazepine; Schizophrenia; Valproic Acid | 1983 |
Effects of the antimigraine compound zolmitriptan ('Zomig') on psychomotor performance alone and in combination with diazepam in healthy volunteers.
Topics: Adult; Cross-Over Studies; Diazepam; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hypnotics and Sedatives; Male; Middle Aged; Oxazoles; Oxazolidinones; Psychometrics; Psychomotor Performance; Reference Values; Serotonin Receptor Agonists; Tryptamines | 1998 |
51 other study(ies) available for oxazoles and diazepam
Article | Year |
---|---|
[Effects of muscimol and diazepam: a comparative study on behavioral inhibiton induced by novelty, punishment, and nonreward (author's transl)].
Topics: Animals; Behavior, Animal; Conditioning, Operant; Diazepam; Environment; Feeding Behavior; Male; Muscimol; Oxazoles; Punishment; Rats; Reward | 1979 |
Central GABA receptor agonists: comparison of muscimol and baclofen.
Topics: Aminobutyrates; Animals; Anticonvulsants; Baclofen; Cerebellum; Cyclic GMP; Diazepam; gamma-Aminobutyric Acid; Harmaline; Isoniazid; Male; Motor Activity; Muscle Tonus; Mycotoxins; Oxazoles; Phenobarbital; Quaternary Ammonium Compounds; Rats; Receptors, Drug; Strychnine; Substance P | 1976 |
Mechanisms by which diazepam, muscimol, and other drugs change the content of cGMP in cerebellar cortex.
Topics: Alkaloids; Animals; Cerebellar Cortex; Cyclic GMP; Diazepam; Haloperidol; Harmaline; Isoxazoles; Male; Morphine; Oxazoles; Purkinje Cells; Pyridines; Rats | 1977 |
Effects of diazepam and muscimol on GABA-mediated neurotransmission: interactions with inosine and nicotinamide.
Topics: Animals; Corpus Striatum; Diazepam; Drug Interactions; Female; gamma-Aminobutyric Acid; Globus Pallidus; Inosine; Muscimol; Niacinamide; Oxazoles; Rats; Synaptic Transmission; Time Factors | 1979 |
Enhancement of the binding of 3H-diazepam to rat brain membranes in vitro by SQ 20009, A novel anxiolytic, gamma-aminobutyric acid (GABA) and muscimol.
Topics: Animals; Bicuculline; Brain; Diazepam; Etazolate; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Membranes; Muscimol; Nicotinic Acids; Oxazoles; Picrotoxin; Rats; Stimulation, Chemical | 1979 |
The GABA agonist THIP a muscimol analogue, does not interfere with the benzodiazepine binding site on rats cortical membranes.
Topics: Animals; Cerebral Cortex; Diazepam; gamma-Aminobutyric Acid; Imidazoles; In Vitro Techniques; Isonicotinic Acids; Male; Muscimol; Oxazoles; Rats; Receptors, Drug; Taurine | 1979 |
The synthesis of prostaglandins and thromboxane in the mouse brain in vivo. Influence of drug induced convulsions, hypoxia and the anticonvulsants trimethadione and diazepam.
Topics: Animals; Brain; Diazepam; In Vitro Techniques; Male; Mice; Oxazoles; Oxygen; Pentylenetetrazole; Picrotoxin; Prostaglandins; Seizures; Thromboxanes; Time Factors; Trimethadione | 1979 |
A comparative study of the effects of muscimol and diazepam on the recall of noxious events.
Topics: Animals; Avoidance Learning; Diazepam; Dissociative Disorders; gamma-Aminobutyric Acid; Humans; Male; Memory; Mental Recall; Muscimol; Oxazoles; Rats | 1979 |
Effect of muscimol, a GABA-mimetic agent, on dopamine metabolism in the mouse brain.
Topics: 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Aminobutyrates; Animals; Brain; Caudate Nucleus; Diazepam; Dopamine; Dose-Response Relationship, Drug; Drug Synergism; gamma-Aminobutyric Acid; Homovanillic Acid; Isoxazoles; Male; Mice; Motor Activity; Oxazoles; Phenobarbital | 1977 |
Regional changes in the rate of turnover of acetylcholine in rat brain following diazepam or muscimol.
Topics: Acetylcholine; Animals; Brain; Cerebral Cortex; Corpus Striatum; Diazepam; gamma-Aminobutyric Acid; Hippocampus; Isoxazoles; Male; Oxazoles; Quaternary Ammonium Compounds; Rats; Receptors, Drug | 1976 |
Lack of GABAergic modulation of acetylcholine turnover in the rat thalamus.
Topics: Acetylcholine; Animals; Brain Chemistry; Diazepam; gamma-Aminobutyric Acid; Isoxazoles; Male; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Thalamus | 1988 |
Synthesis and biological activity of a GABAA agonist which has no effect on benzodiazepine binding and of structurally related glycine antagonists.
Topics: Animals; Bicuculline; Brain Chemistry; Chemical Phenomena; Chemistry; Diazepam; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Isoxazoles; Oxazoles; Piperidines; Pyrrolidines; Rats; Receptors, GABA-A; Synaptic Membranes | 1987 |
Photoaffinity labeling of the GABAA receptor with [3H]muscimol.
Topics: Affinity Labels; Animals; Baclofen; Diazepam; Glutamates; Glutamic Acid; Kinetics; Male; Molecular Weight; Muscimol; Oxazoles; Photochemistry; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spectrophotometry, Ultraviolet | 1985 |
Benzodiazepines enhance the muscimol-dependent activation of phospholipase A2 in glioma C6 cells.
Topics: Animals; Anti-Anxiety Agents; Arachidonic Acid; Arachidonic Acids; Cell Line; Chromatography, High Pressure Liquid; Diazepam; Drug Interactions; Enzyme Activation; Glioma; Muscimol; Neuroglia; Oxazoles; Phospholipases; Phospholipases A; Phospholipases A2; Prostaglandin D2; Prostaglandins D; Rats; Receptors, GABA-A | 1985 |
Development of tolerance to the anticonvulsant effect of GABAmimetic drugs in genetically epilepsy-prone gerbils.
Topics: Acetates; Alkynes; Aminocaproates; Aminooxyacetic Acid; Animals; Anticonvulsants; Brain; Diazepam; Drug Tolerance; Epilepsy; Female; gamma-Aminobutyric Acid; Gerbillinae; Isoxazoles; Male; Oxazoles; Valproic Acid | 1986 |
Depression of drug-induced tremor by a new isoxazol derivative in mice.
Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Harmaline; Isoxazoles; Male; Mice; Mice, Inbred ICR; Motor Activity; Oxazoles; Tremor; Tremorine | 1986 |
[Effect of benzodiazepine derivatives on rats behavior pattern].
Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Chlordiazepoxide; Conditioning, Psychological; Diazepam; Dose-Response Relationship, Drug; Emotions; Escape Reaction; Lorazepam; Male; Oxazoles; Rats; Reinforcement Schedule | 1974 |
[Neuropharmacological studies on the effects of a new psychotropic drug, "Oxazolam"].
Topics: Action Potentials; Amines; Animals; Azepines; Behavior, Animal; Cats; Chlordiazepoxide; Diazepam; Electroencephalography; In Vitro Techniques; Male; Membrane Potentials; Mice; Muscles; Oxazoles; Rabbits; Rats; Reflex; Sympathetic Nervous System; Synaptic Transmission; Tranquilizing Agents | 1970 |
Drug treatment of convulsive disorders.
Topics: Acetazolamide; Adrenocorticotropic Hormone; Adult; Anticonvulsants; Barbiturates; Child; Diazepam; Epilepsy; Epilepsy, Absence; Epilepsy, Tonic-Clonic; Ethosuximide; Humans; Infant; Myoclonus; Oxazoles; Phenobarbital; Phenytoin; Primidone; Pyrrolidinones; Seizures; Trimethadione | 1972 |
Classification and treatment of seizure disorders in children.
Topics: Acetazolamide; Adolescent; Adrenocorticotropic Hormone; Anticonvulsants; Barbiturates; Child; Child, Preschool; Diazepam; Electroencephalography; Epilepsy, Absence; Epilepsy, Temporal Lobe; Epilepsy, Tonic-Clonic; Ethosuximide; Humans; Infant; Infant, Newborn; Male; Nitrazepam; Oxazoles; Phenytoin; Seizures; Succinimides; Trimethadione | 1970 |
[Acute peroral intoxication with 2-amino-5-phenyl-oxazoline fumarate in humans, based upon 30 observed cases].
Topics: Appetite Depressants; Blood Pressure; Central Nervous System; Chlorpromazine; Diazepam; Erythema; Fumarates; Gastric Lavage; Humans; Ipecac; Oxazoles; Phenobarbital; Psychomotor Disorders; Pupil; Respiration; Tachycardia | 1970 |
[Research on fluctuating states of accommodation disorders. 2. PEAG study on effects of several drugs on accommodative function].
Topics: Accommodation, Ocular; Adolescent; Adult; Asthenopia; Chlordiazepoxide; Diazepam; Humans; Male; Mydriatics; Oxazoles; Pilocarpine; Psychotropic Drugs | 1974 |
Pharmacological studies on 10-chloro-11b-(2-chlorophenyl)-2,3,5,6,7,11b-hexahydrobenzo-(6,7)-1,4-diazepino(5,4-b)-oxazol-6-one (CS-370), a new psychosedative agent.
Topics: Aggression; Animals; Anxiety; Avoidance Learning; Behavior, Animal; Benzazepines; Cats; Conditioning, Psychological; Cricetinae; Diazepam; Dogs; Female; Haplorhini; Humans; Ketones; Male; Mice; Motor Activity; Oxazoles; Rats; Seizures; Tranquilizing Agents | 1972 |
[Screening procedure for barbital type physical dependence liability of psychotropic drugs in mice].
Topics: Amitriptyline; Animals; Barbiturates; Behavior, Animal; Benzazepines; Benzodiazepinones; Body Weight; Carboxylic Acids; Chlordiazepoxide; Chlorpromazine; Diazepam; Doxepin; Dronabinol; Humans; Imines; Isoquinolines; Male; Mice; Morphine; Nitrazepam; Oxazoles; Substance Withdrawal Syndrome; Substance-Related Disorders; Tranquilizing Agents | 1973 |
[Pharmacological studies of oxazolazepam, a new psychotropic agent. I. Actions on the central nervous system, especially on the behavioral aspect].
Topics: Adaptation, Biological; Analgesics; Anesthesia; Animals; Anticonvulsants; Apomorphine; Avoidance Learning; Azepines; Behavior, Animal; Central Nervous System; Chlordiazepoxide; Chlorpromazine; Cricetinae; Diazepam; Dogs; Drug Synergism; Drug Tolerance; Electric Stimulation; Female; Guinea Pigs; Haplorhini; Male; Mice; Morphine; Oxazoles; Rats; Seizures; Thiopental; Tranquilizing Agents; Tremorine | 1970 |
[Central action of a new tranquilizing agent, CS-370 (10-chloro-11b-(2-chlorophenyl)-2,3,5,6,7,11b-hexahydrobenzo(6,7)-1, 4-diazepino(5,4b) oxazol-6-one)].
Topics: Animals; Benzazepines; Cats; Central Nervous System; Diazepam; Electric Stimulation; Electroencephalography; Evoked Potentials; Female; Hippocampus; Hypothalamus; Ketones; Male; Mesencephalon; Motor Cortex; Motor Neurons; Nictitating Membrane; Oxazoles; Rabbits; Reflex; Reticular Formation; Spinal Cord; Thalamic Nuclei; Tranquilizing Agents | 1972 |
Studies on the metabolism of oxazolam. II. Isolation and identification of the metabolites of oxazolam in rats.
Topics: Animals; Benzazepines; Benzophenones; Bile; Brain; Chromatography, Thin Layer; Diazepam; Feces; Glucuronates; Kidney; Liver; Male; Oxazepam; Oxazoles; Rats; Spectrum Analysis; Ultraviolet Rays | 1971 |
[Anticonvulsants. 2. Pharmacodynamics].
Topics: Anticonvulsants; Barbiturates; Carbamazepine; Diazepam; Epilepsy; Humans; Hydantoins; Oxazoles; Primidone; Pyrrolidines | 1971 |
Granuloma disciformis (Miescher).
Topics: Diazepam; Female; Granuloma; Humans; Middle Aged; Oxazoles; Skin Diseases; Trifluoperazine | 1969 |
Autonomic response to pentamethylenetetrazol following trimetadione and benzodiazepines administration.
Topics: Animals; Anticonvulsants; Autonomic Nervous System; Blood Glucose; Blood Pressure; Chlordiazepoxide; Curare; Diazepam; Drug Antagonism; Female; Hyperglycemia; Male; Oxazoles; Pentylenetetrazole; Pupil; Rabbits; Trimethadione | 1968 |
Effects of CS-386 and diazepam upon the gastric contraction and excitation of lumbar gamma-motoneurons following stimulation of the hypothalamus in the cat.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Cats; Diazepam; Electric Stimulation; Gastrointestinal Motility; Hypothalamus; Lumbosacral Region; Male; Motor Neurons; Motor Neurons, Gamma; Oxazoles; Vagus Nerve | 1980 |
Tofizopam affects binding of [3H]muscimol to gamma-amino-butyric acid receptors in rat and mouse brains.
Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Binding, Competitive; Brain; Diazepam; Kinetics; Male; Mice; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter | 1982 |
[Differences in the mechanism of the antihypoxic action of benzodiazepine receptor agonists and muscimol].
Topics: Animals; Anti-Anxiety Agents; Diazepam; Drug Evaluation, Preclinical; gamma-Aminobutyric Acid; Hypoxia; Ligands; Mice; Muscimol; Oxazoles; Receptors, GABA-A | 1984 |
Potentiation by intraventricular muscimol of the anticonflict effect of benzodiazepines.
Topics: Animals; Conditioning, Operant; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Drinking; Eating; Fear; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats; Receptors, Neurotransmitter | 1980 |
The insensitivity of developing benzodiazepine receptors to chronic treatment with diazepam, GABA and muscimol in brain cell cultures.
Topics: Animals; Brain; Cell Membrane; Cells, Cultured; Diazepam; Female; Fetus; gamma-Aminobutyric Acid; Kinetics; Mice; Mice, Inbred C57BL; Muscimol; Oxazoles; Pregnancy; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter | 1981 |
Diazepam stimulates the binding of GABA and muscimol but not THIP to rat brain membranes.
Topics: Analgesics; Animals; Brain; Diazepam; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A | 1983 |
Effects of valproic acid on spinal reflexes and [3H]muscimol and [3H]diazepam binding in brain membranes in rats.
Topics: Animals; Brain; Diazepam; Male; Membranes; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Reflex; Spinal Cord; Valproic Acid | 1983 |
Diazepam antagonizes GABA- and muscimol-induced changes of acetylcholine release in slices of guinea-pig cerebral cortex.
Topics: Acetylcholine; Animals; Benzodiazepinones; Cerebral Cortex; Diazepam; Flumazenil; GABA Antagonists; Guinea Pigs; In Vitro Techniques; Muscimol; Oxazoles | 1983 |
Methylphenidate, apomorphine, THIP, and diazepam in monkeys: dopamine-GABA behavior related to psychoses and tardive dyskinesia.
Topics: Animals; Apomorphine; Chlorocebus aethiops; Diazepam; Dopamine; Drug Interactions; Dyskinesia, Drug-Induced; Female; gamma-Aminobutyric Acid; Hallucinations; Humans; Isoxazoles; Male; Methylphenidate; Motor Activity; Oxazoles; Psychoses, Substance-Induced | 1984 |
Histological study of ibotenic acid-induced modifications of rat retina and their attenuation by diazepam.
Topics: Animals; Diazepam; Drug Interactions; Ibotenic Acid; Oxazoles; Rats; Rats, Inbred Strains; Retina; Time Factors | 1984 |
Diazepam enhances the action but not the binding of the GABA analog, THIP.
Topics: Animals; Brain; Chlorides; Culture Techniques; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Ganglia, Spinal; Isoxazoles; Membrane Potentials; Mice; Oxazoles; Rats; Spinal Cord | 1984 |
A new method for the evaluation of benzodiazepines based on their ability to block muscimol-induced myoclonic jerks in mice.
Topics: Animals; Benzodiazepines; Diazepam; Drug Evaluation; Flunitrazepam; Male; Mice; Muscimol; Myoclonus; Oxazoles; Spinal Cord | 1981 |
Therapeutics of monomethylhydrazine intoxication.
Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Drug Therapy, Combination; Male; Methylhydrazines; Mice; Mice, Inbred ICR; Monomethylhydrazine; Muscimol; Oxazoles; Pyridoxine; Seizures | 1982 |
Effects of muscimol alone and in combination with diazepam on shuttle-box performance in rats.
Topics: Animals; Avoidance Learning; Bicuculline; Diazepam; Drug Interactions; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains | 1981 |
Decrease in effects of muscimol on the dorsal root after repeated administration of diazepam in rats.
Topics: Animals; Bicuculline; Diazepam; gamma-Aminobutyric Acid; Male; Membrane Potentials; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Spinal Nerve Roots; Time Factors | 1981 |
Neuroleptic-induced prolactin rise: influence of pharmacological alterations of different neurotransmitter system.
Topics: Animals; Apomorphine; Diazepam; Diphenhydramine; Haloperidol; Kinetics; Male; Metergoline; Muscimol; Oxazoles; Piperazines; Prolactin; Rats | 1980 |
Distinct features of seizures induced by cocaine and amphetamine analogs.
Topics: Animals; Central Nervous System Agents; Central Nervous System Stimulants; Diazepam; Dose-Response Relationship, Drug; Flunarizine; Hallucinogens; Male; Methamphetamine; Mice; N-Methyl-3,4-methylenedioxyamphetamine; Oxazoles; Rats; Rats, Sprague-Dawley; Seizures; Time Factors; Valproic Acid | 1999 |
Effects of lorazepam and WAY-200070 in larval zebrafish light/dark choice test.
Topics: Animals; Anti-Anxiety Agents; Anxiety; Boron Compounds; Choice Behavior; Diazepam; Estradiol; Estrogen Receptor beta; Habenula; Hypothalamus; Larva; Light; Lorazepam; Models, Animal; Neuropsychological Tests; Oxazoles; Phenols; Phenylalanine; Proto-Oncogene Proteins c-fos; Pyrazoles; Pyrimidines; Visual Perception; Zebrafish; Zebrafish Proteins | 2015 |
Effects of the α2/α3-subtype-selective GABAA receptor positive allosteric modulator KRM-II-81 on pain-depressed behavior in rats: comparison with ketorolac and diazepam.
Topics: Analgesics; Animals; Behavior, Animal; Conditioning, Operant; Diazepam; Electric Stimulation; Ketorolac; Male; Oxazoles; Pain; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Self Stimulation | 2019 |
Imidazodiazepine Anticonvulsant, KRM-II-81, Produces Novel, Non-diazepam-like Antiseizure Effects.
Topics: Animals; Anticonvulsants; Diazepam; Humans; Mice; Oxazoles; Receptors, GABA-A | 2020 |
Comparative anticonvulsant activity of the GABAkine KRM-II-81 and a deuterated analog.
Topics: Animals; Anticonvulsants; Diazepam; Mice; Oxazoles; Seizures | 2023 |