Page last updated: 2024-08-21

oxazoles and diazepam

oxazoles has been researched along with diazepam in 55 studies

Research

Studies (55)

TimeframeStudies, this research(%)All Research%
pre-199049 (89.09)18.7374
1990's2 (3.64)18.2507
2000's0 (0.00)29.6817
2010's2 (3.64)24.3611
2020's2 (3.64)2.80

Authors

AuthorsStudies
Jobert, A; Soubrié, P; Thiébot, MH2
Costa, E; Guidotti, A; Naik, SR1
Biggio, G; Brodie, BB; Costa, E; Guidotti, A1
Longman, DA; Slater, P1
Risley, EA; Williams, M1
Maurer, R1
Anhut, H; Hertting, G; Steinhauer, HB1
Biggio, G; Casu, M; Corda, MG; Gessa, GL; Vernaleone, F1
Cheney, DL; Costa, E; Zsilla, G1
Cosi, C; Wood, PL1
Byberg, JR; Curtis, DR; Falch, E; Gynther, BD; Hjeds, H; Krogsgaard-Larsen, P; Labouta, IM1
Cavalla, D; Neff, NH1
Chuang, DM; Majewska, MD1
Löscher, W1
Hirate, K; Shinozaki, H1
Hailey, DM1
Ando, K; Yanagida, T1
Deguchi, T; Iwata, N; Mori, M; Nishijima, Y; Sakai, Y1
Millichap, JG1
Hooshmand, H; Suter, CG1
Borbély, F; Pasi, A; Velvart, J1
Mizutani, A1
Kamioka, T; Kobayashi, S; Suzuki, Y; Takagi, H1
Kaneto, H; Koida, M; Miyagawa, H; Tsuchie, F1
Kamioka, T; Kobayashi, S; Suzuki, Y; Tachikawa, R; Takagi, H1
Fromm, GH; Killian, JM; Sanchez, F1
Iwata, N; Mori, M; Nishijima, Y1
Hattori, K; Matsuda, K; Murata, H; Yasumura, A1
Ekstedt, J1
Clarke, DM1
Carrillo, L; de Bonnevaux, SC1
Hara, T; Iwata, N; Kobayashi, K; Shibata, T; Tonohiro, T1
Saano, V1
Ostrovskaia, RU1
Cananzi, AR; Costa, E; Guidotti, A1
Gardell, MA; Neale, JH; Shibla, DB1
Johnston, GA; Skerritt, JH1
Fukuda, H; Goto, M; Hasebe, Y; Kaneko, T; Kato, K1
Beani, L; Bianchi, C; Tanganelli, S1
Altmann, H; Dose, M; Emrich, HM; von Zerssen, D1
Bjørndal, N; Christensson, E; Gerlach, J1
Gomez-Ramos, P; Perez-Rico, C1
Macdonald, RL; Skerritt, JH1
Haddox, VG; Menon, MK; Vivonia, CA1
Back, KC; George, ME; Pinkerton, MK1
Cortese, I; Cuomo, V; Siro-Brigiani, G1
Fukuda, H; Kaneko, T; Ono, H1
Chieli, T; Cocchi, D; Fregnan, GB; Müller, EE1
Dixon, R; Hughes, AM; Kemp, JV; Nairn, K; Sellers, M; Yates, RA1
Hanson, GR; Jensen, M; Johnson, M; White, HS1
Chen, F; Chen, S; Liu, S; Peng, G; Zhang, C1
Cook, J; Golani, LK; Li, G; Moerke, MJ; Negus, SS1
Cerne, R; Cook, JM; Golani, LK; Jahan, R; Jin, X; Knutson, DE; Li, G; Mian, MY; Ping, X; Rashid, F; Sharmin, D; Smith, JL; Tiruveedhula, VVNPB; Witkin, JM1
Arnold, LA; Cerne, R; Cook, JM; Divović, B; Golani, LK; Jin, X; Lippa, A; Meyer, MJ; Mondal, P; Pandey, KP; Ping, X; Revanian, S; Savić, MM; Sharmin, D; Smith, JL; Witkin, JM; Zahn, NM1

Reviews

1 review(s) available for oxazoles and diazepam

ArticleYear
Chromatography of the 1,4-benzodiazepines.
    Journal of chromatography, 1974, Oct-30, Volume: 98, Issue:3

    Topics: Anti-Anxiety Agents; Chlordiazepoxide; Chromatography; Diazepam; Flurazepam; Humans; Methylation; Nitrazepam; Oxazepam; Oxazoles; Prazepam; Solvents; Spectrometry, Fluorescence; Temperature

1974

Trials

3 trial(s) available for oxazoles and diazepam

ArticleYear
Observations on the discrepancy between the clinical and the laboratory effects of anti-petit mal drugs.
    Transactions of the American Neurological Association, 1967, Volume: 92

    Topics: Action Potentials; Anticonvulsants; Chloralose; Clinical Trials as Topic; Diazepam; Epilepsy, Absence; Humans; Oxazoles; Pentylenetetrazole; Trigeminal Nerve; Trimethadione

1967
Therapeutic effects of GABA-ergic drugs in affective disorders. A preliminary report.
    Pharmacology, biochemistry, and behavior, 1983, Volume: 19, Issue:2

    Topics: Adolescent; Adult; Analgesics; Anticonvulsants; Bipolar Disorder; Carbamazepine; Clinical Trials as Topic; Diazepam; Double-Blind Method; Female; gamma-Aminobutyric Acid; Humans; Isoxazoles; Male; Middle Aged; Mood Disorders; Oxazoles; Oxcarbazepine; Schizophrenia; Valproic Acid

1983
Effects of the antimigraine compound zolmitriptan ('Zomig') on psychomotor performance alone and in combination with diazepam in healthy volunteers.
    Cephalalgia : an international journal of headache, 1998, Volume: 18, Issue:7

    Topics: Adult; Cross-Over Studies; Diazepam; Double-Blind Method; Drug Therapy, Combination; Female; Humans; Hypnotics and Sedatives; Male; Middle Aged; Oxazoles; Oxazolidinones; Psychometrics; Psychomotor Performance; Reference Values; Serotonin Receptor Agonists; Tryptamines

1998

Other Studies

51 other study(ies) available for oxazoles and diazepam

ArticleYear
[Effects of muscimol and diazepam: a comparative study on behavioral inhibiton induced by novelty, punishment, and nonreward (author's transl)].
    Psychopharmacology, 1979, Mar-14, Volume: 61, Issue:1

    Topics: Animals; Behavior, Animal; Conditioning, Operant; Diazepam; Environment; Feeding Behavior; Male; Muscimol; Oxazoles; Punishment; Rats; Reward

1979
Central GABA receptor agonists: comparison of muscimol and baclofen.
    Neuropharmacology, 1976, Volume: 15, Issue:8

    Topics: Aminobutyrates; Animals; Anticonvulsants; Baclofen; Cerebellum; Cyclic GMP; Diazepam; gamma-Aminobutyric Acid; Harmaline; Isoniazid; Male; Motor Activity; Muscle Tonus; Mycotoxins; Oxazoles; Phenobarbital; Quaternary Ammonium Compounds; Rats; Receptors, Drug; Strychnine; Substance P

1976
Mechanisms by which diazepam, muscimol, and other drugs change the content of cGMP in cerebellar cortex.
    Proceedings of the National Academy of Sciences of the United States of America, 1977, Volume: 74, Issue:8

    Topics: Alkaloids; Animals; Cerebellar Cortex; Cyclic GMP; Diazepam; Haloperidol; Harmaline; Isoxazoles; Male; Morphine; Oxazoles; Purkinje Cells; Pyridines; Rats

1977
Effects of diazepam and muscimol on GABA-mediated neurotransmission: interactions with inosine and nicotinamide.
    Life sciences, 1979, Dec-03, Volume: 25, Issue:23

    Topics: Animals; Corpus Striatum; Diazepam; Drug Interactions; Female; gamma-Aminobutyric Acid; Globus Pallidus; Inosine; Muscimol; Niacinamide; Oxazoles; Rats; Synaptic Transmission; Time Factors

1979
Enhancement of the binding of 3H-diazepam to rat brain membranes in vitro by SQ 20009, A novel anxiolytic, gamma-aminobutyric acid (GABA) and muscimol.
    Life sciences, 1979, Feb-26, Volume: 24, Issue:9

    Topics: Animals; Bicuculline; Brain; Diazepam; Etazolate; gamma-Aminobutyric Acid; In Vitro Techniques; Kinetics; Membranes; Muscimol; Nicotinic Acids; Oxazoles; Picrotoxin; Rats; Stimulation, Chemical

1979
The GABA agonist THIP a muscimol analogue, does not interfere with the benzodiazepine binding site on rats cortical membranes.
    Neuroscience letters, 1979, Volume: 12, Issue:1

    Topics: Animals; Cerebral Cortex; Diazepam; gamma-Aminobutyric Acid; Imidazoles; In Vitro Techniques; Isonicotinic Acids; Male; Muscimol; Oxazoles; Rats; Receptors, Drug; Taurine

1979
The synthesis of prostaglandins and thromboxane in the mouse brain in vivo. Influence of drug induced convulsions, hypoxia and the anticonvulsants trimethadione and diazepam.
    Naunyn-Schmiedeberg's archives of pharmacology, 1979, Volume: 310, Issue:1

    Topics: Animals; Brain; Diazepam; In Vitro Techniques; Male; Mice; Oxazoles; Oxygen; Pentylenetetrazole; Picrotoxin; Prostaglandins; Seizures; Thromboxanes; Time Factors; Trimethadione

1979
A comparative study of the effects of muscimol and diazepam on the recall of noxious events.
    Experientia, 1979, Feb-15, Volume: 35, Issue:2

    Topics: Animals; Avoidance Learning; Diazepam; Dissociative Disorders; gamma-Aminobutyric Acid; Humans; Male; Memory; Mental Recall; Muscimol; Oxazoles; Rats

1979
Effect of muscimol, a GABA-mimetic agent, on dopamine metabolism in the mouse brain.
    Life sciences, 1977, Aug-15, Volume: 21, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Aminobutyrates; Animals; Brain; Caudate Nucleus; Diazepam; Dopamine; Dose-Response Relationship, Drug; Drug Synergism; gamma-Aminobutyric Acid; Homovanillic Acid; Isoxazoles; Male; Mice; Motor Activity; Oxazoles; Phenobarbital

1977
Regional changes in the rate of turnover of acetylcholine in rat brain following diazepam or muscimol.
    Naunyn-Schmiedeberg's archives of pharmacology, 1976, Volume: 294, Issue:3

    Topics: Acetylcholine; Animals; Brain; Cerebral Cortex; Corpus Striatum; Diazepam; gamma-Aminobutyric Acid; Hippocampus; Isoxazoles; Male; Oxazoles; Quaternary Ammonium Compounds; Rats; Receptors, Drug

1976
Lack of GABAergic modulation of acetylcholine turnover in the rat thalamus.
    Neuroscience letters, 1988, May-03, Volume: 87, Issue:3

    Topics: Acetylcholine; Animals; Brain Chemistry; Diazepam; gamma-Aminobutyric Acid; Isoxazoles; Male; Oxazoles; Rats; Rats, Inbred Strains; Receptors, GABA-A; Thalamus

1988
Synthesis and biological activity of a GABAA agonist which has no effect on benzodiazepine binding and of structurally related glycine antagonists.
    Drug design and delivery, 1987, Volume: 1, Issue:4

    Topics: Animals; Bicuculline; Brain Chemistry; Chemical Phenomena; Chemistry; Diazepam; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Isoxazoles; Oxazoles; Piperidines; Pyrrolidines; Rats; Receptors, GABA-A; Synaptic Membranes

1987
Photoaffinity labeling of the GABAA receptor with [3H]muscimol.
    Journal of neurochemistry, 1985, Volume: 44, Issue:3

    Topics: Affinity Labels; Animals; Baclofen; Diazepam; Glutamates; Glutamic Acid; Kinetics; Male; Molecular Weight; Muscimol; Oxazoles; Photochemistry; Rats; Rats, Inbred Strains; Receptors, GABA-A; Spectrophotometry, Ultraviolet

1985
Benzodiazepines enhance the muscimol-dependent activation of phospholipase A2 in glioma C6 cells.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 232, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Arachidonic Acid; Arachidonic Acids; Cell Line; Chromatography, High Pressure Liquid; Diazepam; Drug Interactions; Enzyme Activation; Glioma; Muscimol; Neuroglia; Oxazoles; Phospholipases; Phospholipases A; Phospholipases A2; Prostaglandin D2; Prostaglandins D; Rats; Receptors, GABA-A

1985
Development of tolerance to the anticonvulsant effect of GABAmimetic drugs in genetically epilepsy-prone gerbils.
    Pharmacology, biochemistry, and behavior, 1986, Volume: 24, Issue:4

    Topics: Acetates; Alkynes; Aminocaproates; Aminooxyacetic Acid; Animals; Anticonvulsants; Brain; Diazepam; Drug Tolerance; Epilepsy; Female; gamma-Aminobutyric Acid; Gerbillinae; Isoxazoles; Male; Oxazoles; Valproic Acid

1986
Depression of drug-induced tremor by a new isoxazol derivative in mice.
    Japanese journal of pharmacology, 1986, Volume: 41, Issue:1

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Harmaline; Isoxazoles; Male; Mice; Mice, Inbred ICR; Motor Activity; Oxazoles; Tremor; Tremorine

1986
[Effect of benzodiazepine derivatives on rats behavior pattern].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1974, Volume: 70, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Behavior, Animal; Chlordiazepoxide; Conditioning, Psychological; Diazepam; Dose-Response Relationship, Drug; Emotions; Escape Reaction; Lorazepam; Male; Oxazoles; Rats; Reinforcement Schedule

1974
[Neuropharmacological studies on the effects of a new psychotropic drug, "Oxazolam"].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1970, Volume: 66, Issue:6

    Topics: Action Potentials; Amines; Animals; Azepines; Behavior, Animal; Cats; Chlordiazepoxide; Diazepam; Electroencephalography; In Vitro Techniques; Male; Membrane Potentials; Mice; Muscles; Oxazoles; Rabbits; Rats; Reflex; Sympathetic Nervous System; Synaptic Transmission; Tranquilizing Agents

1970
Drug treatment of convulsive disorders.
    The New England journal of medicine, 1972, Mar-02, Volume: 286, Issue:9

    Topics: Acetazolamide; Adrenocorticotropic Hormone; Adult; Anticonvulsants; Barbiturates; Child; Diazepam; Epilepsy; Epilepsy, Absence; Epilepsy, Tonic-Clonic; Ethosuximide; Humans; Infant; Myoclonus; Oxazoles; Phenobarbital; Phenytoin; Primidone; Pyrrolidinones; Seizures; Trimethadione

1972
Classification and treatment of seizure disorders in children.
    Virginia medical monthly, 1970, Volume: 97, Issue:2

    Topics: Acetazolamide; Adolescent; Adrenocorticotropic Hormone; Anticonvulsants; Barbiturates; Child; Child, Preschool; Diazepam; Electroencephalography; Epilepsy, Absence; Epilepsy, Temporal Lobe; Epilepsy, Tonic-Clonic; Ethosuximide; Humans; Infant; Infant, Newborn; Male; Nitrazepam; Oxazoles; Phenytoin; Seizures; Succinimides; Trimethadione

1970
[Acute peroral intoxication with 2-amino-5-phenyl-oxazoline fumarate in humans, based upon 30 observed cases].
    Archiv fur Toxikologie, 1970, Volume: 26, Issue:2

    Topics: Appetite Depressants; Blood Pressure; Central Nervous System; Chlorpromazine; Diazepam; Erythema; Fumarates; Gastric Lavage; Humans; Ipecac; Oxazoles; Phenobarbital; Psychomotor Disorders; Pupil; Respiration; Tachycardia

1970
[Research on fluctuating states of accommodation disorders. 2. PEAG study on effects of several drugs on accommodative function].
    Nippon Ganka Gakkai zasshi, 1974, Nov-10, Volume: 78, Issue:11

    Topics: Accommodation, Ocular; Adolescent; Adult; Asthenopia; Chlordiazepoxide; Diazepam; Humans; Male; Mydriatics; Oxazoles; Pilocarpine; Psychotropic Drugs

1974
Pharmacological studies on 10-chloro-11b-(2-chlorophenyl)-2,3,5,6,7,11b-hexahydrobenzo-(6,7)-1,4-diazepino(5,4-b)-oxazol-6-one (CS-370), a new psychosedative agent.
    Arzneimittel-Forschung, 1972, Volume: 22, Issue:5

    Topics: Aggression; Animals; Anxiety; Avoidance Learning; Behavior, Animal; Benzazepines; Cats; Conditioning, Psychological; Cricetinae; Diazepam; Dogs; Female; Haplorhini; Humans; Ketones; Male; Mice; Motor Activity; Oxazoles; Rats; Seizures; Tranquilizing Agents

1972
[Screening procedure for barbital type physical dependence liability of psychotropic drugs in mice].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1973, Volume: 69, Issue:5

    Topics: Amitriptyline; Animals; Barbiturates; Behavior, Animal; Benzazepines; Benzodiazepinones; Body Weight; Carboxylic Acids; Chlordiazepoxide; Chlorpromazine; Diazepam; Doxepin; Dronabinol; Humans; Imines; Isoquinolines; Male; Mice; Morphine; Nitrazepam; Oxazoles; Substance Withdrawal Syndrome; Substance-Related Disorders; Tranquilizing Agents

1973
[Pharmacological studies of oxazolazepam, a new psychotropic agent. I. Actions on the central nervous system, especially on the behavioral aspect].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1970, Volume: 66, Issue:1

    Topics: Adaptation, Biological; Analgesics; Anesthesia; Animals; Anticonvulsants; Apomorphine; Avoidance Learning; Azepines; Behavior, Animal; Central Nervous System; Chlordiazepoxide; Chlorpromazine; Cricetinae; Diazepam; Dogs; Drug Synergism; Drug Tolerance; Electric Stimulation; Female; Guinea Pigs; Haplorhini; Male; Mice; Morphine; Oxazoles; Rats; Seizures; Thiopental; Tranquilizing Agents; Tremorine

1970
[Central action of a new tranquilizing agent, CS-370 (10-chloro-11b-(2-chlorophenyl)-2,3,5,6,7,11b-hexahydrobenzo(6,7)-1, 4-diazepino(5,4b) oxazol-6-one)].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1972, Volume: 68, Issue:3

    Topics: Animals; Benzazepines; Cats; Central Nervous System; Diazepam; Electric Stimulation; Electroencephalography; Evoked Potentials; Female; Hippocampus; Hypothalamus; Ketones; Male; Mesencephalon; Motor Cortex; Motor Neurons; Nictitating Membrane; Oxazoles; Rabbits; Reflex; Reticular Formation; Spinal Cord; Thalamic Nuclei; Tranquilizing Agents

1972
Studies on the metabolism of oxazolam. II. Isolation and identification of the metabolites of oxazolam in rats.
    Chemical & pharmaceutical bulletin, 1971, Volume: 19, Issue:9

    Topics: Animals; Benzazepines; Benzophenones; Bile; Brain; Chromatography, Thin Layer; Diazepam; Feces; Glucuronates; Kidney; Liver; Male; Oxazepam; Oxazoles; Rats; Spectrum Analysis; Ultraviolet Rays

1971
[Anticonvulsants. 2. Pharmacodynamics].
    Lakartidningen, 1971, Oct-18, Volume: 68

    Topics: Anticonvulsants; Barbiturates; Carbamazepine; Diazepam; Epilepsy; Humans; Hydantoins; Oxazoles; Primidone; Pyrrolidines

1971
Granuloma disciformis (Miescher).
    The Australasian journal of dermatology, 1969, Volume: 10, Issue:3

    Topics: Diazepam; Female; Granuloma; Humans; Middle Aged; Oxazoles; Skin Diseases; Trifluoperazine

1969
Autonomic response to pentamethylenetetrazol following trimetadione and benzodiazepines administration.
    Archives internationales de pharmacodynamie et de therapie, 1968, Volume: 173, Issue:1

    Topics: Animals; Anticonvulsants; Autonomic Nervous System; Blood Glucose; Blood Pressure; Chlordiazepoxide; Curare; Diazepam; Drug Antagonism; Female; Hyperglycemia; Male; Oxazoles; Pentylenetetrazole; Pupil; Rabbits; Trimethadione

1968
Effects of CS-386 and diazepam upon the gastric contraction and excitation of lumbar gamma-motoneurons following stimulation of the hypothalamus in the cat.
    Journal of pharmacobio-dynamics, 1980, Volume: 3, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Cats; Diazepam; Electric Stimulation; Gastrointestinal Motility; Hypothalamus; Lumbosacral Region; Male; Motor Neurons; Motor Neurons, Gamma; Oxazoles; Vagus Nerve

1980
Tofizopam affects binding of [3H]muscimol to gamma-amino-butyric acid receptors in rat and mouse brains.
    Pharmacological research communications, 1982, Volume: 14, Issue:8

    Topics: Animals; Anti-Anxiety Agents; Benzodiazepines; Binding, Competitive; Brain; Diazepam; Kinetics; Male; Mice; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter

1982
[Differences in the mechanism of the antihypoxic action of benzodiazepine receptor agonists and muscimol].
    Biulleten' eksperimental'noi biologii i meditsiny, 1984, Volume: 98, Issue:10

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Drug Evaluation, Preclinical; gamma-Aminobutyric Acid; Hypoxia; Ligands; Mice; Muscimol; Oxazoles; Receptors, GABA-A

1984
Potentiation by intraventricular muscimol of the anticonflict effect of benzodiazepines.
    Brain research, 1980, Sep-08, Volume: 196, Issue:2

    Topics: Animals; Conditioning, Operant; Conflict, Psychological; Diazepam; Dose-Response Relationship, Drug; Drinking; Eating; Fear; gamma-Aminobutyric Acid; Injections, Intraventricular; Male; Muscimol; Oxazoles; Rats; Receptors, Neurotransmitter

1980
The insensitivity of developing benzodiazepine receptors to chronic treatment with diazepam, GABA and muscimol in brain cell cultures.
    Brain research, 1981, Apr-06, Volume: 210, Issue:1-2

    Topics: Animals; Brain; Cell Membrane; Cells, Cultured; Diazepam; Female; Fetus; gamma-Aminobutyric Acid; Kinetics; Mice; Mice, Inbred C57BL; Muscimol; Oxazoles; Pregnancy; Receptors, Drug; Receptors, GABA-A; Receptors, Neurotransmitter

1981
Diazepam stimulates the binding of GABA and muscimol but not THIP to rat brain membranes.
    Neuroscience letters, 1983, Aug-08, Volume: 38, Issue:3

    Topics: Analgesics; Animals; Brain; Diazepam; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Isoxazoles; Kinetics; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A

1983
Effects of valproic acid on spinal reflexes and [3H]muscimol and [3H]diazepam binding in brain membranes in rats.
    Journal of pharmacobio-dynamics, 1983, Volume: 6, Issue:3

    Topics: Animals; Brain; Diazepam; Male; Membranes; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Reflex; Spinal Cord; Valproic Acid

1983
Diazepam antagonizes GABA- and muscimol-induced changes of acetylcholine release in slices of guinea-pig cerebral cortex.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 324, Issue:1

    Topics: Acetylcholine; Animals; Benzodiazepinones; Cerebral Cortex; Diazepam; Flumazenil; GABA Antagonists; Guinea Pigs; In Vitro Techniques; Muscimol; Oxazoles

1983
Methylphenidate, apomorphine, THIP, and diazepam in monkeys: dopamine-GABA behavior related to psychoses and tardive dyskinesia.
    Psychopharmacology, 1984, Volume: 82, Issue:1-2

    Topics: Animals; Apomorphine; Chlorocebus aethiops; Diazepam; Dopamine; Drug Interactions; Dyskinesia, Drug-Induced; Female; gamma-Aminobutyric Acid; Hallucinations; Humans; Isoxazoles; Male; Methylphenidate; Motor Activity; Oxazoles; Psychoses, Substance-Induced

1984
Histological study of ibotenic acid-induced modifications of rat retina and their attenuation by diazepam.
    Cell and tissue research, 1984, Volume: 238, Issue:1

    Topics: Animals; Diazepam; Drug Interactions; Ibotenic Acid; Oxazoles; Rats; Rats, Inbred Strains; Retina; Time Factors

1984
Diazepam enhances the action but not the binding of the GABA analog, THIP.
    Brain research, 1984, Apr-09, Volume: 297, Issue:1

    Topics: Animals; Brain; Chlorides; Culture Techniques; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Ganglia, Spinal; Isoxazoles; Membrane Potentials; Mice; Oxazoles; Rats; Spinal Cord

1984
A new method for the evaluation of benzodiazepines based on their ability to block muscimol-induced myoclonic jerks in mice.
    Psychopharmacology, 1981, Volume: 75, Issue:3

    Topics: Animals; Benzodiazepines; Diazepam; Drug Evaluation; Flunitrazepam; Male; Mice; Muscimol; Myoclonus; Oxazoles; Spinal Cord

1981
Therapeutics of monomethylhydrazine intoxication.
    Toxicology and applied pharmacology, 1982, Volume: 63, Issue:2

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Drug Therapy, Combination; Male; Methylhydrazines; Mice; Mice, Inbred ICR; Monomethylhydrazine; Muscimol; Oxazoles; Pyridoxine; Seizures

1982
Effects of muscimol alone and in combination with diazepam on shuttle-box performance in rats.
    Arzneimittel-Forschung, 1981, Volume: 31, Issue:10

    Topics: Animals; Avoidance Learning; Bicuculline; Diazepam; Drug Interactions; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains

1981
Decrease in effects of muscimol on the dorsal root after repeated administration of diazepam in rats.
    Journal of pharmacobio-dynamics, 1981, Volume: 4, Issue:12

    Topics: Animals; Bicuculline; Diazepam; gamma-Aminobutyric Acid; Male; Membrane Potentials; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Spinal Nerve Roots; Time Factors

1981
Neuroleptic-induced prolactin rise: influence of pharmacological alterations of different neurotransmitter system.
    Experientia, 1980, Apr-15, Volume: 36, Issue:4

    Topics: Animals; Apomorphine; Diazepam; Diphenhydramine; Haloperidol; Kinetics; Male; Metergoline; Muscimol; Oxazoles; Piperazines; Prolactin; Rats

1980
Distinct features of seizures induced by cocaine and amphetamine analogs.
    European journal of pharmacology, 1999, Jul-21, Volume: 377, Issue:2-3

    Topics: Animals; Central Nervous System Agents; Central Nervous System Stimulants; Diazepam; Dose-Response Relationship, Drug; Flunarizine; Hallucinogens; Male; Methamphetamine; Mice; N-Methyl-3,4-methylenedioxyamphetamine; Oxazoles; Rats; Rats, Sprague-Dawley; Seizures; Time Factors; Valproic Acid

1999
Effects of lorazepam and WAY-200070 in larval zebrafish light/dark choice test.
    Neuropharmacology, 2015, Volume: 95

    Topics: Animals; Anti-Anxiety Agents; Anxiety; Boron Compounds; Choice Behavior; Diazepam; Estradiol; Estrogen Receptor beta; Habenula; Hypothalamus; Larva; Light; Lorazepam; Models, Animal; Neuropsychological Tests; Oxazoles; Phenols; Phenylalanine; Proto-Oncogene Proteins c-fos; Pyrazoles; Pyrimidines; Visual Perception; Zebrafish; Zebrafish Proteins

2015
Effects of the α2/α3-subtype-selective GABAA receptor positive allosteric modulator KRM-II-81 on pain-depressed behavior in rats: comparison with ketorolac and diazepam.
    Behavioural pharmacology, 2019, Volume: 30, Issue:5

    Topics: Analgesics; Animals; Behavior, Animal; Conditioning, Operant; Diazepam; Electric Stimulation; Ketorolac; Male; Oxazoles; Pain; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Self Stimulation

2019
Imidazodiazepine Anticonvulsant, KRM-II-81, Produces Novel, Non-diazepam-like Antiseizure Effects.
    ACS chemical neuroscience, 2020, 09-02, Volume: 11, Issue:17

    Topics: Animals; Anticonvulsants; Diazepam; Humans; Mice; Oxazoles; Receptors, GABA-A

2020
Comparative anticonvulsant activity of the GABAkine KRM-II-81 and a deuterated analog.
    Drug development research, 2023, Volume: 84, Issue:3

    Topics: Animals; Anticonvulsants; Diazepam; Mice; Oxazoles; Seizures

2023