Page last updated: 2024-08-21

oxazoles and bradykinin

oxazoles has been researched along with bradykinin in 21 studies

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19905 (23.81)18.7374
1990's7 (33.33)18.2507
2000's5 (23.81)29.6817
2010's3 (14.29)24.3611
2020's1 (4.76)2.80

Authors

AuthorsStudies
Kitakaze, T; Ogawa, Y; Tonda, K; Yoshizaki, T1
Begany, AJ; Datko, SL; Dervinis, A; Gluckman, MI; Malis, JL; Rosenthale, ME; Shriver, DA1
Bates, HM; Berger, FM; Diamantis, W; Kletzkin, M; Plekss, OJ; Sofia, RD; Spencer, HJ1
Hrdina, PD; Ling, GM1
Green, AY; Green, D1
Advenier, C; Biyah, K1
Hosoi, K; Kurihara, K; Ueha, T1
Cesare, P; McNaughton, P1
Chueh, SH; Ho, MY; Hu, SY; Song, SL1
Blaukat, A; Müller-Esterl, W1
Catlin, MC; Costa, LG; Gafni, J; Lam, TH; Molinski, TF; Munsch, JA; Pessah, IN1
Hoffmann, EK; Jakobsen, LD; Jensen, BS; Krarup, T1
Dolhun, B; Geiger, JD; Haughey, NJ; Holden, CP; Nath, A; Shepel, PN1
Halayko, AJ; Kahraman, S; Mitchell, RW; Solway, J; Wylam, ME1
Erdös, EG; Marcic, BM1
Huang, Y; Kong, SK; Kwan, HY; Yao, X1
Huang, Y; Kwan, HY; Leung, PC; Yao, X1
Brown, BM; Coleman, N; Köhler, R; Oliván-Viguera, A; Olmstead, MM; Singh, V; Valero, MS; Wulff, H1
Amor, S; Badorrey, R; Calvín-Tienza, V; Coleman, N; Díaz-de-Villegas, MD; Fernández-Fernández, JM; Gálvez, JA; García-Otín, ÁL; García-Villalón, ÁL; Köhler, R; Laría, C; Murillo, MD; Oliván-Viguera, A; Pinilla, E; Rivera, L; Simonsen, U; Valero, MS; Wulff, H1
Biwer, LA; Hoehn, KL; Isakson, BE; Kenwood, BM; Straub, AC; Taddeo, EP1
Adams, J; Espinosa, R; Lopez, JR; Mijares, A1

Other Studies

21 other study(ies) available for oxazoles and bradykinin

ArticleYear
Drug-induced adrenaline release and blood glucose in rats: 3-phenyl-5(2-piperidinoethyl)-isoxazole citrate.
    Japanese journal of pharmacology, 1975, Volume: 25, Issue:5

    Topics: Adrenal Glands; Adrenalectomy; Aminopyrine; Animals; Bradykinin; Epinephrine; Histamine; Hypophysectomy; Male; Oxazoles; Phenylbutazone; Piperidines; Rats; Splanchnic Nerves

1975
Anti-inflammatory properties of 4,5-diphenyl-2-oxazolepropionic acid (oxaprozin).
    Agents and actions, 1974, Volume: 4, Issue:3

    Topics: Airway Obstruction; Analgesics; Animals; Anti-Inflammatory Agents; Arthritis, Rheumatoid; Aspirin; Bradykinin; Carrageenan; Dogs; Edema; Emulsions; Encephalomyelitis, Autoimmune, Experimental; Female; Fever; Freund's Adjuvant; Indazoles; Male; Molecular Weight; Mycobacterium; Oxazoles; Peptic Ulcer; Propionates; Rats; Sulfanilamides; Synovitis; Time Factors; Uric Acid; Yeasts

1974
The pharmacological properties of seclazone (7-chloro-3,3a-dihydro-2H, 9H-isoxazolo (3,2-b) (1,3) benzoxazin-9-one) a new anti-inflammatory agent.
    Pharmacology, 1973, Volume: 9, Issue:3

    Topics: Adjuvants, Immunologic; Albumins; Analgesics; Animals; Anti-Inflammatory Agents; Arthritis; Benzoxazoles; Blood Proteins; Bradykinin; Carrageenan; Diuretics; Fibrinogen; Globulins; Guinea Pigs; In Vitro Techniques; Inflammation; Male; Oxazines; Oxazoles; Rats; Stomach Ulcer; Time Factors

1973
The in vivo antibradykinin activity of seclazone (7-chloro-3,3a-dihydro-2H,9H-isoxazolo(3,2-b) (1,3)benzoxazin-9-one), a new anti-inflammatory agent.
    Pharmacology, 1973, Volume: 10, Issue:3

    Topics: Airway Resistance; Animals; Anti-Inflammatory Agents; Blood Pressure; Bradykinin; Bronchi; Capillary Permeability; Guinea Pigs; In Vitro Techniques; Lung; Oxazines; Oxazoles; Skin Absorption

1973
Wy 23205, a new non-steroidal anti-inflammatory agent.
    British journal of pharmacology, 1971, Volume: 42, Issue:4

    Topics: Animals; Anti-Inflammatory Agents; Arthritis; Aspirin; Bradykinin; Gastrointestinal Diseases; Guinea Pigs; Hindlimb; In Vitro Techniques; Indomethacin; Inflammation; Oxazoles; Phenylbutazone; Propionates; Rats

1971
Effects of three alpha 2-adrenoceptor agonists, rilmenidine, UK 14304 and clonidine on bradykinin- and substance P-induced airway microvascular leakage in guinea-pigs.
    Neuropeptides, 1995, Volume: 28, Issue:4

    Topics: Acetylcholine; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Bradykinin; Brimonidine Tartrate; Capillaries; Capillary Permeability; Clonidine; Dioxanes; Extravascular Lung Water; Guinea Pigs; Idazoxan; Oxazoles; Prazosin; Quinoxalines; Rilmenidine; Substance P; Trachea

1995
Bradykinin-stimulated transient modulation of epidermal growth factor receptors in A-431 human epidermoid carcinoma cells.
    Journal of cellular physiology, 1993, Volume: 157, Issue:1

    Topics: Alkaloids; Binding, Competitive; Bradykinin; Carcinoma, Squamous Cell; ErbB Receptors; Humans; Marine Toxins; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Kinase C; Staurosporine; Tumor Cells, Cultured

1993
A novel heat-activated current in nociceptive neurons and its sensitization by bradykinin.
    Proceedings of the National Academy of Sciences of the United States of America, 1996, Dec-24, Volume: 93, Issue:26

    Topics: Animals; Animals, Newborn; Bradykinin; Cells, Cultured; Enzyme Activation; Enzyme Inhibitors; Ganglia, Spinal; Hot Temperature; Kinetics; Marine Toxins; Membrane Potentials; Neurons; Neurons, Afferent; Nociceptors; Oxazoles; Pain; Protein Kinase C; Protein Tyrosine Phosphatases; Rats; Rats, Wistar; Staurosporine; Tetradecanoylphorbol Acetate; Time Factors

1996
Inhibition of bradykinin-induced calcium increase by phosphatase inhibitors in neuroblastoma x glioma hybrid NG108-15 cells.
    Journal of neurochemistry, 1997, Volume: 68, Issue:2

    Topics: Animals; Bradykinin; Calcium; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glioma; Hybrid Cells; Marine Toxins; Mice; Neuroblastoma; Okadaic Acid; Oxazoles; Phosphoric Monoester Hydrolases; Phosphorylation; Signal Transduction; Thapsigargin; Type C Phospholipases

1997
Inhibition of B2 receptor internalization delays its dephosphorylation.
    Immunopharmacology, 1997, Volume: 36, Issue:2-3

    Topics: Autoradiography; Bradykinin; Bradykinin Receptor Antagonists; Cantharidin; Cell Line; Concanavalin A; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Fibroblasts; Humans; Irritants; Marine Toxins; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Precipitin Tests; Radioligand Assay; Receptor, Bradykinin B2; Receptors, Bradykinin; Skin; Sucrose

1997
Xestospongins: potent membrane permeable blockers of the inositol 1,4,5-trisphosphate receptor.
    Neuron, 1997, Volume: 19, Issue:3

    Topics: Alkaloids; Animals; Antineoplastic Agents; Astrocytes; Biological Transport; Bradykinin; Caffeine; Calcium; Calcium Channels; Central Nervous System Stimulants; Cytosol; Dose-Response Relationship, Drug; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Ionomycin; Ionophores; Macrocyclic Compounds; Membrane Proteins; Neurons; Oxazoles; PC12 Cells; Porifera; Quinolizines; Rabbits; Rats; Receptors, Cytoplasmic and Nuclear; Ryanodine

1997
Na+-K+-2Cl- cotransport in Ehrlich cells: regulation by protein phosphatases and kinases.
    The American journal of physiology, 1998, Volume: 275, Issue:1

    Topics: Animals; Azepines; Bradykinin; Carbazoles; Carcinoma, Ehrlich Tumor; Carrier Proteins; Chlorides; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Homeostasis; Hypertonic Solutions; Indoles; Isoquinolines; Kinetics; Marine Toxins; Mice; Myosin-Light-Chain Kinase; Naphthalenes; Osmolar Concentration; Oxazoles; Phosphoprotein Phosphatases; Potassium; Protein Kinases; Pyrroles; Sodium-Potassium-Chloride Symporters; Sulfonamides; Tumor Cells, Cultured

1998
Diadenosine pentaphosphate increases levels of intracellular calcium in astrocytes by a mechanism involving release from caffeine/ryanodine- and IP3-sensitive stores.
    Journal of neuroscience research, 2000, Jan-15, Volume: 59, Issue:2

    Topics: Adenosine Triphosphate; Astrocytes; Bradykinin; Caffeine; Calcium; Central Nervous System Stimulants; Dinucleoside Phosphates; Extracellular Space; Fetus; Humans; Inositol 1,4,5-Trisphosphate; Macrocyclic Compounds; Oxazoles; Receptors, Purinergic P2; Receptors, Purinergic P2X; Receptors, Purinergic P2Y1; Ryanodine; Ryanodine Receptor Calcium Release Channel; Vasoconstrictor Agents

2000
Selective restoration of calcium coupling to muscarinic M(3) receptors in contractile cultured airway myocytes.
    American journal of physiology. Lung cellular and molecular physiology, 2000, Volume: 278, Issue:5

    Topics: Acetylcholine; Animals; Atropine; Blood Proteins; Blotting, Western; Bradykinin; Calcium; Calcium Channels; Cells, Cultured; Diamines; Dogs; Dose-Response Relationship, Drug; Fluorescent Dyes; Fura-2; Inositol 1,4,5-Trisphosphate Receptors; Macrocyclic Compounds; Muscarinic Antagonists; Muscle, Smooth; Oxazoles; Parasympatholytics; Phenotype; Piperidines; Pirenzepine; Receptor, Muscarinic M3; Receptors, Bradykinin; Receptors, Cytoplasmic and Nuclear; Receptors, Muscarinic; Trachea; Vasodilator Agents

2000
Protein kinase C and phosphatase inhibitors block the ability of angiotensin I-converting enzyme inhibitors to resensitize the receptor to bradykinin without altering the primary effects of bradykinin.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:2

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Arachidonic Acid; Bradykinin; Bradykinin Receptor Antagonists; Calcium; Cells, Cultured; CHO Cells; Cricetinae; Drug Interactions; Enalaprilat; Endothelium, Vascular; Enzyme Inhibitors; Humans; Marine Toxins; Naphthalenes; Okadaic Acid; Oxazoles; Phosphoric Monoester Hydrolases; Phosphorylation; Protein Kinase C; Pulmonary Artery; Receptor, Bradykinin B2; Receptors, Bradykinin; Transfection

2000
cGMP abolishes agonist-induced [Ca(2+)](i) oscillations in human bladder epithelial cells.
    American journal of physiology. Renal physiology, 2001, Volume: 281, Issue:6

    Topics: Acetylcholine; Alkaloids; Bradykinin; Calcium Signaling; Calcium-Transporting ATPases; Carbazoles; Cell Line; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Dipyridamole; Drug Antagonism; Enzyme Inhibitors; Epithelial Cells; Humans; Indoles; Kinetics; Macrocyclic Compounds; Oxazoles; Phosphodiesterase Inhibitors; Urinary Bladder

2001
Depletion of intracellular Ca2+ stores sensitizes the flow-induced Ca2+ influx in rat endothelial cells.
    Circulation research, 2003, Feb-21, Volume: 92, Issue:3

    Topics: Adenosine Triphosphate; Aniline Compounds; Animals; Bradykinin; Calcium; Calcium Channels; Calcium Signaling; Cells, Cultured; Cyclic GMP-Dependent Protein Kinases; Endothelium, Vascular; Enzyme Inhibitors; Fluorescent Dyes; Inositol 1,4,5-Trisphosphate Receptors; Intracellular Fluid; Macrocyclic Compounds; Male; Manganese; Ochratoxins; Oxazoles; Poloxamer; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, Cytoplasmic and Nuclear; Spectrometry, Fluorescence; Type C Phospholipases; Xanthenes

2003
New positive Ca2+-activated K+ channel gating modulators with selectivity for KCa3.1.
    Molecular pharmacology, 2014, Volume: 86, Issue:3

    Topics: Animals; Benzothiazoles; Blood Pressure; Bradykinin; Chlorocebus aethiops; Coronary Vessels; COS Cells; Crystallography, X-Ray; HEK293 Cells; Humans; Intermediate-Conductance Calcium-Activated Potassium Channels; Ion Channel Gating; Isometric Contraction; Male; Mice, Inbred C57BL; Muscle, Smooth, Vascular; Oxazoles; Structure-Activity Relationship; Swine; Vasodilator Agents

2014
Vascular Reactivity Profile of Novel KCa 3.1-Selective Positive-Gating Modulators in the Coronary Vascular Bed.
    Basic & clinical pharmacology & toxicology, 2016, Volume: 119, Issue:2

    Topics: Animals; Bradykinin; Cells, Cultured; Coronary Circulation; Coronary Vessels; Endothelial Cells; Endothelium, Vascular; Gene Expression Regulation; Heart; Intermediate-Conductance Calcium-Activated Potassium Channels; Male; Nitric Oxide Synthase Type III; Oxazoles; Patch-Clamp Techniques; Pyrazoles; Rats; Rats, Sprague-Dawley; RNA, Messenger; Swine; Vasodilation; Vasodilator Agents

2016
Two functionally distinct pools of eNOS in endothelium are facilitated by myoendothelial junction lipid composition.
    Biochimica et biophysica acta, 2016, Volume: 1861, Issue:7

    Topics: Biological Transport; Bradykinin; Calcium; Calcium Signaling; Cell Communication; Coculture Techniques; Cyclic GMP; Diglycerides; Egtazic Acid; Endoplasmic Reticulum; Endothelial Cells; Gap Junctions; Gene Expression Regulation; Humans; Inositol 1,4,5-Trisphosphate; Macrocyclic Compounds; Myocytes, Smooth Muscle; Nitric Oxide Synthase Type III; Oxazoles; Phenylephrine; Phosphatidylserines; Phosphorylation; Primary Cell Culture; Protein Kinase C; Protein Kinase Inhibitors; Thapsigargin

2016
Increases in [IP3]i aggravates diastolic [Ca2+] and contractile dysfunction in Chagas' human cardiomyocytes.
    PLoS neglected tropical diseases, 2020, Volume: 14, Issue:4

    Topics: Adult; Bradykinin; Calcium; Cell Membrane Permeability; Chagas Cardiomyopathy; Endothelins; Female; Humans; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Macrocyclic Compounds; Male; Middle Aged; Myocytes, Cardiac; Oxazoles; Quality of Life; Sarcoplasmic Reticulum; Sodium

2020