oxazoles has been researched along with benzofurans in 49 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 3 (6.12) | 18.7374 |
1990's | 26 (53.06) | 18.2507 |
2000's | 14 (28.57) | 29.6817 |
2010's | 6 (12.24) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Allen, DG; Westerblad, H | 2 |
Davies, JE; Garrido, MC; Ng, LL | 1 |
Baylor, SM; Harkins, AB; Hollingworth, S; Konishi, M | 1 |
Bartschat, DK; Lattanzio, FA | 1 |
Gallagher, KL; Schachter, M; Sever, PS | 1 |
Karaki, H; Obara, K; Ozaki, H; Someya, T; Usuki, T; Yabu, H; Yoshino, M | 1 |
Freudenrich, CC; Levy, LA; Lieberman, M; London, RE; Murphy, E | 1 |
Hall, RD; Levy, LA; London, RE; Murphy, E; Raju, B | 1 |
Földes, O; Gschwendtová, K; Langer, P | 1 |
Mintz, IM; Regehr, WG; Sabatini, BL | 1 |
Goldman, WF; Sugiyama, T | 1 |
Atluri, PP; Regehr, WG | 1 |
Capiod, T; Carter, T; Khodakhah, K; Ogden, D; Thomas, M | 1 |
Casteels, R; De Smedt, H; Henning, RH; Missiaen, L; Parys, JB; Sienaert, I | 1 |
Geven, WB; Kruse, J; Monnens, LA; Vis, P; Willems, HL | 1 |
Hongo, K; Konishi, M; Kurihara, S | 1 |
Garner, CW; Smith, LK; Turnbow, MA | 1 |
Berlin, JR; Konishi, M | 2 |
Simons, TJ | 1 |
Konishi, M; Kurihara, S; Suda, N | 1 |
Freund, P; Heitzmann, T; Neidlein, R; Reiff, K; Strein, K | 1 |
Chan, CK; Head, GA | 1 |
Clark, DA; Genereux, PE; Gibbs, EM; Hulin, B; Lewis, DM; Newton, LS | 1 |
Chu, TC; Gluchowski, C; Hughes, BW; Potter, DE; Wong, W | 1 |
Gundlach, AL; Hosseini, AR; Iakovidis, D; Jackman, GP; King, PR; Louis, WJ; Nero, TL; Suzuki, S | 1 |
Bock, C; Niederhoffer, N; Szabo, B | 1 |
Gundlach, AL; King, PR; Louis, WJ | 1 |
Vedejs, E; Wang, J | 1 |
Abdel-Rahman, AA; El-Mas, MM; Zhang, J | 1 |
Godwin, SJ; Head, GA; Parkin, ML | 1 |
Jungermann, K; Nath, A; Pestel, S; Schieferdecker, HL | 1 |
Ernsberger, P; Koletsky, RJ; Velliquette, RA | 1 |
Burgdorf, C; Engelhardt, A; Kurz, T; Raasch, W; Richardt, G; Schäfer, U | 1 |
Abelson, KS; Höglund, AU | 1 |
Merwid-Lad, A; Misiuk-Hojło, M; Pieśniewska, M; Szaliński, M; Trocha, M | 1 |
Abdel-Rahman, AA; Zhang, J | 1 |
Abdel-Rahman, AA; Li, G; Wang, X | 2 |
Kumar, MP; Liu, RS | 1 |
Khansefid, N; Ladgevardi, MA; Sabetkasaie, M | 1 |
Gerstenberger, BS; Konopelski, JP; Lin, J; Stessman, NY | 1 |
Brimble, MA; Liu, YC; Sperry, J | 1 |
Chen, MF; Cheng, JT; Chou, MT; Chung, HH; Yang, TT | 1 |
Agbaba, D; Gemovic, B; Nikolic, K; Srdic-Rajic, T; Veljkovic, N | 1 |
Beall, HD; Bibby, JM; Hassani, M; Moody, CJ; Newsome, JJ; Swann, E | 1 |
Das, U; Fan, YS; Hsiao, MY; Lin, W; Liu, MH | 1 |
Hussar, DA | 1 |
49 other study(ies) available for oxazoles and benzofurans
Article | Year |
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Myoplasmic free Mg2+ concentration during repetitive stimulation of single fibres from mouse skeletal muscle.
Topics: Adenosine Triphosphate; Animals; Benzofurans; Fura-2; Hydrogen-Ion Concentration; Magnesium; Male; Mice; Muscle Contraction; Muscles; Oxazoles; Sodium | 1992 |
Intracellular free magnesium in human lymphocytes and the response to lectins.
Topics: Benzofurans; Calcium; Cell Division; Fluorescent Dyes; Fluorometry; Fura-2; Humans; Intracellular Fluid; Lectins; Lymphocytes; Magnesium; Oxazoles; Stimulation, Chemical | 1991 |
Myoplasmic calcium transients in intact frog skeletal muscle fibers monitored with the fluorescent indicator furaptra.
Topics: Action Potentials; Animals; Benzofurans; Calcium; Coloring Agents; Diffusion; Fluorescent Dyes; Fura-2; In Vitro Techniques; Indicators and Reagents; Kinetics; Magnesium; Muscles; Oxazoles; Rana temporaria; Spectrometry, Fluorescence | 1991 |
The effect of pH on rate constants, ion selectivity and thermodynamic properties of fluorescent calcium and magnesium indicators.
Topics: Aniline Compounds; Benzofurans; Calcium; Fluorescent Dyes; Fura-2; Hydrogen-Ion Concentration; Indoles; Magnesium; Oxazoles; Spectrometry, Fluorescence; Thermodynamics; Xanthenes | 1991 |
Intracellular free magnesium in a vascular smooth muscle cell line.
Topics: Animals; Benzofurans; Cell Line; Fluorescent Dyes; Fura-2; Intracellular Fluid; Magnesium; Muscle, Smooth, Vascular; Oxazoles | 1990 |
Modification by calyculin A of inward Ca currents in smooth muscle cells isolated from guinea pig taenia coli.
Topics: Animals; Benzofurans; Calcium; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Guinea Pigs; In Vitro Techniques; Intestine, Large; Marine Toxins; Muscle Contraction; Muscle, Smooth; Oxazoles | 1990 |
Monitoring cytosolic free magnesium in cultured chicken heart cells by use of the fluorescent indicator Furaptra.
Topics: Animals; Benzofurans; Cells, Cultured; Chick Embryo; Cytosol; Fura-2; Magnesium; Myocardium; Oxazoles; Spectrometry, Fluorescence; Time Factors | 1989 |
A fluorescent indicator for measuring cytosolic free magnesium.
Topics: Animals; Benzofurans; Cells, Cultured; Cytosol; Fluorescent Dyes; Fura-2; Indicators and Reagents; Liver; Magnesium; Male; Oxazoles; Rats; Rats, Inbred Strains; Spectrometry, Fluorescence | 1989 |
In vivo effect of amiodarone, thiocyanate, perchlorate and goitrin on thyroxine deiodination in rat liver.
Topics: Amiodarone; Animals; Benzofurans; Diiodothyronines; Iodine; Liver; Male; Oxazoles; Oxazolidinones; Perchlorates; Rats; Rats, Inbred Strains; Thiocyanates; Thyroxine; Triiodothyronine | 1984 |
Calcium control of transmitter release at a cerebellar synapse.
Topics: Animals; Benzofurans; Cadmium; Calcium; Calcium Channel Blockers; Calcium Channels; Cerebellum; Electric Conductivity; Fluorescent Dyes; Fura-2; Neurotransmitter Agents; omega-Agatoxin IVA; omega-Conotoxin GVIA; Oxazoles; Peptides; Purkinje Cells; Rats; Spider Venoms; Synapses | 1995 |
Measurement of SR free Ca2+ and Mg2+ in permeabilized smooth muscle cells with use of furaptra.
Topics: Animals; Benzofurans; Calcium; Cell Line; Cell Membrane Permeability; Fluorescent Dyes; Fura-2; Inositol 1,4,5-Trisphosphate; Magnesium; Muscle, Smooth; Osmolar Concentration; Oxazoles; Rats; Saponins; Sarcoplasmic Reticulum | 1995 |
Calcium transients in cerebellar granule cell presynaptic terminals.
Topics: Animals; Benzofurans; Calcium; Cerebellum; Coumarins; Fluorescent Dyes; Fura-2; In Vitro Techniques; Kinetics; Nerve Fibers; Neurons; Organic Chemicals; Oxazoles; Rats; Spectrometry, Fluorescence; Synapses; Tetrodotoxin; Time Factors | 1995 |
Analogue computation of transient changes of intracellular free Ca2+ concentration with the low affinity Ca2+ indicator furaptra during whole-cell patch-clamp recording.
Topics: Aniline Compounds; Animals; Benzofurans; Calcium; Fluorescence; Fura-2; Guinea Pigs; Kinetics; Oxazoles; Patch-Clamp Techniques; Pituitary Gland; Rats; Swine; Xanthenes | 1995 |
Opening up Ca2+ stores with InsP3.
Topics: Benzofurans; Calcium; Calcium Channels; Fluorescent Dyes; Fura-2; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Muscle, Smooth; Oxazoles; Receptors, Cytoplasmic and Nuclear | 1995 |
Defibrination essential in the assay of ionized magnesium in mononuclear cells.
Topics: Benzofurans; Blood Platelets; Fibrin; Fluorescent Dyes; Fura-2; Humans; Ions; Leukocytes, Mononuclear; Magnesium; Oxazoles; Spectrometry, Fluorescence; Trypan Blue | 1995 |
Relaxation, [Ca2+]i and [Mg2+]i during prolonged tetanic stimulation of intact, single fibres from mouse skeletal muscle.
Topics: Acidosis; Animals; Benzofurans; Calcium; Electric Stimulation; Fluorescent Dyes; Fura-2; In Vitro Techniques; Indoles; Magnesium; Male; Mice; Muscle Fibers, Skeletal; Muscle Relaxation; Muscle, Skeletal; Oxazoles; Parvalbumins; Sarcoplasmic Reticulum; Troponin | 1994 |
Cytoplasmic free Mg2+ in rat ventricular myocytes studied with the fluorescent indicator furaptra.
Topics: Animals; Benzofurans; Calibration; Carbonyl Cyanide p-Trifluoromethoxyphenylhydrazone; Cytoplasm; Fluorescent Dyes; Fura-2; Heart Ventricles; In Vitro Techniques; Magnesium; Male; Mitochondria, Heart; Myocardium; Oxazoles; Rats; Rats, Wistar; Spectrometry, Fluorescence | 1994 |
The oxazolidinedione CP-92,768-2 partially protects insulin receptor substrate-1 from dexamethasone down-regulation in 3T3-L1 adipocytes.
Topics: 3T3 Cells; Adipocytes; Animals; Benzofurans; Dexamethasone; Down-Regulation; Gene Expression Regulation; Insulin; Insulin Receptor Substrate Proteins; Mice; Mifepristone; Oxazoles; Oxazolidinones; Phosphoenolpyruvate Carboxykinase (GTP); Phosphoproteins; Receptors, Glucocorticoid; RNA, Messenger | 1995 |
Ca2+ transients in cardiac myocytes measured with high and low affinity Ca2+ indicators.
Topics: Animals; Benzofurans; Biophysical Phenomena; Biophysics; Buffers; Calcimycin; Calcium; Fluorescent Dyes; Fura-2; In Vitro Techniques; Kinetics; Models, Biological; Myocardium; Oxazoles; Rats; Sarcomeres; Spectrometry, Fluorescence | 1993 |
Measurement of free Zn2+ ion concentration with the fluorescent probe mag-fura-2 (furaptra).
Topics: Animals; Benzofurans; Calcium; Fluorescent Dyes; Fura-2; Histidine; Humans; Indicators and Reagents; Magnesium; Oxazoles; Protein Binding; Serum Albumin, Bovine; Spectrometry, Fluorescence; Zinc | 1993 |
Fluorescence signals from the Mg2+/Ca2+ indicator furaptra in frog skeletal muscle fibers.
Topics: Animals; Benzofurans; Biophysical Phenomena; Biophysics; Calcium; Fluorescent Dyes; Fura-2; In Vitro Techniques; Magnesium; Muscles; Oxazoles; Rana temporaria; Spectrometry, Fluorescence; Spectrophotometry, Ultraviolet | 1993 |
Ca transients in cardiac myocytes measured with a low affinity fluorescent indicator, furaptra.
Topics: Animals; Benzofurans; Biophysical Phenomena; Biophysics; Calcium; Fluorescent Dyes; Fura-2; In Vitro Techniques; Intracellular Fluid; Kinetics; Magnesium; Membrane Potentials; Myocardium; Oxazoles; Rats; Spectrometry, Fluorescence | 1993 |
Dose proportionality studies of novel thiazolidinedione derivatives as potent antidiabetic agents in mice.
Topics: Animals; Benzofurans; Chromatography, High Pressure Liquid; Half-Life; Hypoglycemic Agents; Male; Mice; Mice, Inbred Strains; Naphthalenes; Oxazoles; Oxazolidinones; Spectrophotometry, Ultraviolet; Thiazoles; Thiazolidinediones | 1995 |
Relative importance of central imidazoline receptors for the antihypertensive effects of moxonidine and rilmenidine.
Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Cardiac Catheterization; Clonidine; Dose-Response Relationship, Drug; Female; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Injections, Intravenous; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine; Time Factors | 1996 |
Hypoglycemic activity of a series of alpha-alkylthio and alpha-alkoxy carboxylic acids related to ciglitazone.
Topics: 3T3 Cells; Adipocytes; Animals; Benzofurans; Carboxylic Acids; Diabetes Mellitus, Type 2; Hypoglycemic Agents; Mice; Mice, Mutant Strains; Mice, Obese; Molecular Structure; Oxazoles; Stereoisomerism; Structure-Activity Relationship; Thiazoles; Thiazolidinediones | 1996 |
Rilmenidine-induced ocular hypotension: role of imidazoline1 and alpha 2 receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzofurans; Calcium; Ciliary Body; Cyclic AMP; Female; Imidazoles; Imidazoline Receptors; Intraocular Pressure; Iris; Male; Norepinephrine; Ocular Hypotension; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathectomy; Sympathetic Nervous System; Yohimbine | 1996 |
[3H]Rilmenidine-labelled imidazoline-receptor binding sites co-localize with [3H]2-(benzofuranyl)-2-imidazoline-labelled imidazoline-receptor binding sites and monoamine oxidase-B in rabbit, but not rat, kidney.
Topics: Adrenergic alpha-Agonists; Animals; Autoradiography; Benzofurans; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isoenzymes; Kidney; Male; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Rabbits; Rats; Rats, Inbred WKY; Receptors, Drug; Rilmenidine; Species Specificity; Thiazoles | 1998 |
Analysis of the receptor involved in the central hypotensive effect of rilmenidine and moxonidine.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzazepines; Benzofurans; Blood Pressure; Dose-Response Relationship, Drug; Drug Interactions; Female; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Methyldopa; Norepinephrine; Oxazoles; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Yohimbine | 1999 |
Identification of imidazoline-receptor binding sites in cortex and medulla of the bovine adrenal gland. Colocalization with MAO-A and MAO-B.
Topics: Adrenal Cortex; Adrenal Medulla; Adrenergic beta-Agonists; Animals; Autoradiography; Benzofurans; Binding Sites; Cattle; Clonidine; Imidazoles; Imidazoline Receptors; Isoenzymes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Rats; Receptors, Drug; Rilmenidine; Thiazoles; Tritium | 1999 |
A tyrosine-derived benzofuranone related to diazonamide A.
Topics: Animals; Benzofurans; Chromatography, High Pressure Liquid; Cricetinae; Crystallography, X-Ray; Heterocyclic Compounds, 4 or More Rings; Molecular Structure; Oxazoles; Tyrosine | 2000 |
Imidazoline I(1) receptor-induced activation of phosphatidylcholine-specific phospholipase C elicits mitogen-activated protein kinase phosphorylation in PC12 cells.
Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzofurans; Choline; Diglycerides; Enzyme Activation; Imidazoles; Imidazoline Receptors; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nerve Growth Factor; Oxazoles; PC12 Cells; Phosphorylation; Phosphorylcholine; Rats; Receptors, Drug; Rilmenidine; Signal Transduction; Type C Phospholipases | 2001 |
Importance of imidazoline-preferring receptors in the cardiovascular actions of chronically administered moxonidine, rilmenidine and clonidine in conscious rabbits.
Topics: Adrenergic alpha-2 Receptor Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Cardiovascular System; Clonidine; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Fourth Ventricle; Heart Rate; Idazoxan; Imidazoles; Imidazoline Receptors; Injections, Intraventricular; Male; Oxazoles; Rabbits; Receptors, Drug; Rilmenidine | 2003 |
Inhibition of prostaglandin D2 clearance in rat hepatocytes by the thromboxane receptor antagonists daltroban and ifetroban and the thromboxane synthase inhibitor furegrelate.
Topics: Animals; Benzofurans; Bridged Bicyclo Compounds, Heterocyclic; Cells, Cultured; Complement C5a; Enzyme Inhibitors; Hepatocytes; Liver; Male; Metabolic Clearance Rate; Oxazoles; Perfusion; Phenylacetates; Prostaglandin D2; Rats; Rats, Wistar; Receptors, Thromboxane; Sulfonamides; Thromboxane B2; Thromboxane-A Synthase | 2003 |
The role of I(1)-imidazoline receptors and alpha(2)-adrenergic receptors in the modulation of glucose and lipid metabolism in the SHROB model of metabolic syndrome X.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzofurans; Blood Pressure; Disease Models, Animal; Female; Glucagon; Glucose; Glucose Tolerance Test; Humans; Imidazoles; Imidazoline Receptors; Lipid Metabolism; Male; Metabolic Syndrome; Obesity; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Yohimbine | 2003 |
Moxonidine displays a presynaptic alpha-2-adrenoceptor-dependent synergistic sympathoinhibitory action at imidazoline-1 receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Agmatine; Animals; Benzofurans; Bridged Bicyclo Compounds; Brimonidine Tartrate; Drug Synergism; Heart; Heptanes; Imidazoles; Imidazoline Receptors; Norepinephrine; Oxazoles; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Sympatholytics; Yohimbine | 2003 |
The effects of the alpha2-adrenergic receptor agonists clonidine and rilmenidine, and antagonists yohimbine and efaroxan, on the spinal cholinergic receptor system in the rat.
Topics: Acetylcholine; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Animals; Benzofurans; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Injections, Spinal; Ligands; Male; Microdialysis; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Cholinergic; Rilmenidine; Spinal Cord; Time Factors; Yohimbine | 2004 |
[Effect of rilmenidine on intraocular pressure in rabbits, interaction with efaroxan and rauwolscine].
Topics: Administration, Topical; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzofurans; Drug Interactions; Glaucoma; Imidazoles; Intraocular Pressure; Male; Oxazoles; Rabbits; Rilmenidine; Time Factors; Yohimbine | 2004 |
Mitogen-activated protein kinase phosphorylation in the rostral ventrolateral medulla plays a key role in imidazoline (i1)-receptor-mediated hypotension.
Topics: Animals; Benzofurans; Blood Pressure; Heart Rate; Imidazoles; Imidazoline Receptors; Male; Medulla Oblongata; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Oxazoles; Phosphorylation; Rats; Rats, Sprague-Dawley; Receptors, Drug; Rilmenidine; Signal Transduction | 2005 |
Site-dependent inhibition of neuronal c-jun in the brainstem elicited by imidazoline I1 receptor activation: role in rilmenidine-evoked hypotension.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Benzazepines; Benzofurans; Blood Pressure; Brain Stem; Cerebrospinal Fluid; Clonidine; Consciousness; Gene Expression; Heart Rate; Hydralazine; Hypotension; Imidazoles; Imidazoline Receptors; Immunohistochemistry; Male; Medulla Oblongata; Neurons; Nordefrin; Oxazoles; Proto-Oncogene Proteins c-jun; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; RNA, Messenger; Time Factors; Vasoconstrictor Agents; Vasodilator Agents | 2005 |
Neuronal norepinephrine responses of the rostral ventrolateral medulla and nucleus tractus solitarius neurons distinguish the I1- from the alpha2-receptor-mediated hypotension in conscious SHRs.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Area Postrema; Benzazepines; Benzofurans; Blood Pressure; Clonidine; Consciousness; Heart Rate; Hypotension; Imidazoles; Interleukin-1; Male; Motor Activity; Neurons; Nordefrin; Norepinephrine; Oxazoles; Rats; Rats, Inbred SHR; Receptors, Adrenergic, alpha-2; Rilmenidine; Solitary Nucleus | 2005 |
Zn(OTf)2-catalyzed cyclization of proparyl alcohols with anilines, phenols, and amides for synthesis of indoles, benzofurans, and oxazoles through different annulation mechanisms.
Topics: Alcohols; Amides; Aniline Compounds; Benzofurans; Catalysis; Cyclization; Indoles; Mesylates; Molecular Structure; Oxazoles; Phenols; Stereoisomerism | 2006 |
Possible role of NMDA receptors in antinociception induced by rilmenidine in mice in the formalin test.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analgesics; Animals; Benzofurans; Binding Sites; Binding, Competitive; Dizocilpine Maleate; Dose-Response Relationship, Drug; Drug Synergism; Excitatory Amino Acid Antagonists; Imidazoles; Imidazoline Receptors; Male; Mice; Nervous System; Neurons, Afferent; Nociceptors; Oxazoles; Pain; Pain Measurement; Receptors, Drug; Receptors, N-Methyl-D-Aspartate; Rilmenidine; Yohimbine | 2007 |
Diazonamide support studies: stereoselective formation of the C10 chiral center in both the CDEFG and AEFG fragments.
Topics: Benzofurans; Heterocyclic Compounds, 4 or More Rings; Indoles; Oxazoles; Oxindoles; Stereoisomerism; Substrate Specificity; Tyrosine | 2008 |
Synthesis of natural products containing spiroketals via intramolecular hydrogen abstraction.
Topics: Anthelmintics; Anti-Bacterial Agents; Antineoplastic Agents; Benzofurans; Biological Products; Bridged-Ring Compounds; Ciguatoxins; Cyclization; Ethers; Ethers, Cyclic; Furans; Hydrogen; Ivermectin; Marine Toxins; Molecular Structure; Oxazoles; Oxidation-Reduction; Phenazines; Phosphoprotein Phosphatases; Pyrans; Spiro Compounds | 2010 |
Improvement of hyperphagia by activation of cerebral I(1)-imidazoline receptors in streptozotocin-induced diabetic mice.
Topics: Animals; Benzofurans; Cerebrum; Diabetes Mellitus, Type 1; Disease Models, Animal; Eating; Female; Humans; Hyperphagia; Hypothalamus; Imidazoles; Imidazoline Receptors; Male; Mice; Mice, Inbred BALB C; Neuropeptide Y; Oxazoles; Rilmenidine; Streptozocin | 2012 |
Imidazoline-1 receptor ligands as apoptotic agents: pharmacophore modeling and virtual docking study.
Topics: Antineoplastic Agents; Apoptosis; Benzofurans; Cell Proliferation; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Imidazoles; Imidazoline Receptors; K562 Cells; Ligands; Models, Molecular; Molecular Docking Simulation; Oxazoles; Quantitative Structure-Activity Relationship; Rilmenidine; Tumor Cells, Cultured | 2013 |
Benzofuran-, benzothiophene-, indazole- and benzisoxazole-quinones: excellent substrates for NAD(P)H:quinone oxidoreductase 1.
Topics: Antineoplastic Agents; Benzofurans; Cell Line, Tumor; Enzyme Assays; Humans; Indazoles; NAD(P)H Dehydrogenase (Quinone); Oxazoles; Oxidation-Reduction; Quinones; Thiophenes | 2013 |
Chemoselective intramolecular Wittig reactions for the synthesis of oxazoles and benzofurans.
Topics: Benzofurans; Indicators and Reagents; Molecular Structure; Oxazoles | 2014 |
New drugs 2015, part 2.
Topics: Antibodies, Monoclonal, Humanized; Benzhydryl Compounds; Benzofurans; Cyclopropanes; Diphosphates; Drug Approval; Drug Therapy; Glucagon-Like Peptide 1; Glucosides; Glycopeptides; Humans; Lactones; Lipoglycopeptides; Organophosphates; Oxazoles; Pyridines; Sulfates; Teicoplanin; United States; United States Food and Drug Administration | 2015 |