oxazepam and nordazepam

oxazepam has been researched along with nordazepam in 114 studies

Research

Studies (114)

TimeframeStudies, this research(%)All Research%
pre-199045 (39.47)18.7374
1990's23 (20.18)18.2507
2000's19 (16.67)29.6817
2010's23 (20.18)24.3611
2020's4 (3.51)2.80

Authors

AuthorsStudies
Collins, RJ; Gall, M; Kamdar, BV1
Babbini, M; Barbaro, AM; Bartoletti, M; Biagi, GL; Borea, PA; Gaiardi, M; Guerra, MC1
Johnston, GA; Maddalena, DJ1
Karplus, M; So, SS1
Ghuloum, AM; Jain, AN; Sage, CR1
Carrupt, PA; Crivori, P; Cruciani, G; Testa, B1
Topliss, JG; Yoshida, F1
Ertl, P; Rohde, B; Selzer, P1
Artursson, P; Luthman, K; Norinder, U; Stenberg, P1
Gao, F; Lombardo, F; Obach, RS; Shalaeva, MY1
Caron, G; Ermondi, G1
Du-Cuny, L; Huwyler, J; Kansy, M; Wiese, M1
Lombardo, F; Obach, RS; Waters, NJ1
Campillo, NE; Guerra, A; Páez, JA1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Carmona, AV; Kumari, S; Tiwari, AK; Trippier, PC1
Golovenko, NIa; Zin'kovskii, VG1
Erkkola, R; Kangas, L; Kanto, J; Piiroinen, O1
Greenblatt, DJ; Shader, RI1
Liljequist, R; Linnoila, M; Palva, E1
Baars, AM; Hekster, YA; O'Reilly, WJ; van der Kleijn, E; Vree, TB1
Kabra, PM; Marton, LJ; Stevens, GL1
Haataja, M; Hurme, P; Kanto, J; Sellman, R1
Allen, MD; Greenblatt, DJ; Orsulak, PJ; Shader, RI; Woo, E1
Clarke, CH; Nicholson, AN1
Sun, SR1
Klotz, U1
Azarnoff, DL; Cathcart-Rake, WF; Shoeman, DW; Straughan, JL1
Cohen, ME; Duffner, PK; Jusko, WJ; MacKichan, JJ1
Kanto, J; Mäenpää, M; Mäntylä, R; Sellman, R; Valovirta, E1
Aderjan, R; Schmidt, G1
Sellers, EM; Wong, GB1
Constant, H; Duthel, JM; Miachon, S; Rochet, T; Vallon, JJ1
Martin, WR; Sloan, JW; Wala, EP2
Guentert, TW; Stebler, T1
Wong, PT1
Dusci, LJ; Good, SM; Hall, RW; Ilett, KF1
Chenery, RJ; Lockwood, GF; Seddon, T1
Minder, EI1
Klockowski, PM; Levy, G2
Frey, HH; Scherkl, R1
Brase, DA; Dewey, WL; Glennon, RA; Young, R1
Alazia, M; Cano, JP; Crevat-Pisano, P; Drouet, C; Francois, G; Lacarelle, B1
Kanto, J; Scheinin, M1
Bareggi, SR; Ferrario, P; Pirola, R; Zecca, L1
Igarashi, T; Kitagawa, H; Ohmori, S; Okiyama, M; Ueno, K1
Martin, WR; McNicholas, LF; Sloan, JW; Wala, E1
Brown, C; File, SE; Greenblatt, DJ; Martin, IL1
Moroji, T; Motomura, H; Noguchi, T; Sekiguchi, R; Tada, K1
Berwish, NJ; Bond, WS; Swift, B1
Martin, WR; McNicholas, LF; Pruitt, TA1
Meeles, MT; Thys, CP; Tjaden, UR; van der Kaay, M1
Vozeh, S1
El-Hazmi, MA1
Löscher, W1
Agrawal, KK; Gupta, A; Tayal, G; Tekur, U1
Booij, LH; Crul, JF; Driessen, JJ; van Egmond, J; Vree, TB1
Aranko, K; Aranko, S; Mattila, MJ; Seppälä, T1
Coffman, WB; McFarland, SA; Meyer, EA; Mumford, R; Wynn, RL1
Klotz, U; Reimann, I1
Kölle, EU1
Dixon, R1
Frey, HH; Löscher, W1
Chiba, K; Chiba, T; Hirano, T; Horii, H; Ishizaki, T; Kato, Y1
Berrueta, LA; Gallo, B; Vicente, F1
Pang, KS; St-Pierre, MV2
Alcorn, J; Papich, MG1
Liu, JF; Zhang, Y1
Cirimele, V; Kintz, P; Mangin, P; Vayssette, F2
Sloan, JW; Wala, EP1
Miyazawa, M; Okamura, T; Sugiura, W1
Jing, X; Sloan, JW; Wala, EP1
Ali, HM; Azzam, RM; Notarianni, LJ1
Hemmersbach, P; Ragnar Norli, H; Rasmussen, KE; Reubsaet, KJ1
Carter, J; Mozayani, A; Nix, R1
Mørland, J; Olsen, KM; Skuterud, B; Smith-Kielland, A1
Contel, N; Grossman, S; Liu, Z; Ren, S; Rose, A; Short, J; Unger, S1
Djeridane, Y; Touitou, Y1
Boonen, T; De Boeck, G; Grootaert, P; Laloup, M; Pien, K; Pipeleers-Marichal, M; Samyn, N; Vits, K; Wood, M1
Atta-Politou, J; Panderi, I; Valavani, P1
Musteata, FM; Musteata, ML; Pawliszyn, J1
Baud, FJ; Bouchonnet, S; Hervé, F; Perrin, B; Pirnay, S; Ricordel, I1
Bouchonnet, S; Kinani, S; Milan, N; Ricordel, I1
Bévalot, F; Fanton, L; Gaillard, Y; Grait, H; Le Meur, C; Malicier, D1
Acikgöz, A; Bader, A; Giri, S; Karim, N; Schmidt-Heck, W1
Iannello, C; Mandrioli, R; Matrisciano, F; Mercolini, L; Nicoletti, F; Raggi, MA1
Allen, KR; Glover, SJ1
Chronister, CW; Goldberger, BA; Merves, ML1
Marin, SJ; McMillin, GA1
Gunn, J; Kriger, S; Terrell, AR1
Dawson, M; Fu, S; Keegan, J; Lewis, J; Wang, H1
Acikgöz, A; Bader, A; Giri, S; Maringka, M; Nieber, K1
Mariani, CL; Musulin, SE; Papich, MG1
KuKanich, B; Nauss, JL1
Marin, SJ; McMillin, GA; Roberts, M; Wood, M1
Liang, C; Ni, C; Rao, Y; Wang, R; Wang, X; Xiong, L; Zhang, Y1
Atayee, RS; Best, BM; Luk, S; Ma, JD1
Bertol, E; Boscolo Berto, R; Favretto, D; Mannaioni, G; Mari, F; Vaiano, F1
Bankstahl, M; Gramer, M; Hausknecht, M; Klein, S; Löscher, W1
Li, J; Liu, H; Wu, L; Zhang, J1
Darwish, WS; Hayami, A; Ikenaka, Y; Ishizuka, M; Kawai, YK; Mizukawa, H; Nakayama, SM; Watanabe, KP1
Jia, J; Jiang, F; Johansen, SS; Linnet, K; Rao, Y; Wang, X; Zhang, Y1
Castro, A; Costa, P; Franco, JM; Melo, P; Quintas, MJ; Tarelho, S; Teixeira, HM1
Boxho, P; Charlier, C; Denooz, R; Dubois, N; Lemaire, E; Schmidt, C1
Ali, SM; Baud, FJ; Garnier, R; Jouffroy, R; Raphalen, JH; Sacre, L; Villa, A1
Bugelli, V; Campobasso, CP; Chericoni, S; Fornaro, S; Giusiani, M; Papi, L; Stefanelli, F; Vanin, S1
Limoges, JF; Sarris, GG1
Concheiro, M; Cruz, A; de-Castro-Ríos, A; Lendoiro, E; López-Rabuñal, A; López-Rivadulla, M1
Falcon, M; Fernadez-Lopez, L; Luna, A; Mancini, R; Pellegrini, M; Rotolo, M1
Coulter, C; Garnier, M; Moore, C1

Reviews

2 review(s) available for oxazepam and nordazepam

ArticleYear
Amide Bond Bioisosteres: Strategies, Synthesis, and Successes.
    Journal of medicinal chemistry, 2020, 11-12, Volume: 63, Issue:21

    Topics: Amides; Carbamates; Click Chemistry; Drug Design; Pyridines; Structure-Activity Relationship; Triazoles; Urea

2020
[Clinical pharmacokinetics of diazepam and its biologically active metabolites (author's transl)].
    Klinische Wochenschrift, 1978, Sep-15, Volume: 56, Issue:18

    Topics: Biotransformation; Diazepam; Half-Life; Humans; Kinetics; Models, Biological; Nordazepam; Oxazepam

1978

Trials

5 trial(s) available for oxazepam and nordazepam

ArticleYear
Effects on learning and memory of 2-week treatments with chlordiazepoxide lactam, N-desmethyldiazepam, oxazepam and methyloxazepam, alone or in combination with alcohol.
    International pharmacopsychiatry, 1979, Volume: 14, Issue:4

    Topics: Adult; Anti-Anxiety Agents; Chlordiazepoxide; Drug Interactions; Ethanol; Humans; Learning; Memory; Memory, Short-Term; Nordazepam; Oxazepam; Temazepam; Time Factors

1979
Immediate and residual effects in man of the metabolites of diazepam.
    British journal of clinical pharmacology, 1978, Volume: 6, Issue:4

    Topics: Adult; Choice Behavior; Diazepam; Humans; Male; Motor Skills; Nordazepam; Oxazepam; Placebos; Reaction Time; Temazepam; Time Factors

1978
Absorption of diazepam after its rectal administration in dogs.
    American journal of veterinary research, 1995, Volume: 56, Issue:12

    Topics: Absorption; Administration, Rectal; Animals; Anticonvulsants; Chromatography, High Pressure Liquid; Cross-Over Studies; Diazepam; Dogs; Dose-Response Relationship, Drug; Fluorescence Polarization Immunoassay; Injections, Intravenous; Male; Nordazepam; Oxazepam; Time Factors

1995
Urinary excretion of diazepam metabolites in healthy volunteers and drug users.
    Scandinavian journal of clinical and laboratory investigation, 2001, Volume: 61, Issue:3

    Topics: Adult; Anti-Anxiety Agents; Chromatography, Gas; Chromatography, High Pressure Liquid; Creatinine; Diazepam; Female; Humans; Male; Middle Aged; Nordazepam; Oxazepam; Substance Abuse Detection; Substance-Related Disorders; Temazepam

2001
Diazepam pharmacokinetics after nasal drop and atomized nasal administration in dogs.
    Journal of veterinary pharmacology and therapeutics, 2011, Volume: 34, Issue:1

    Topics: Administration, Intranasal; Animals; Anticonvulsants; Diazepam; Dogs; Dosage Forms; Drug Administration Routes; Female; Half-Life; Male; Nordazepam; Oxazepam

2011

Other Studies

107 other study(ies) available for oxazepam and nordazepam

ArticleYear
Pharmacology of some metabolites of triazolam, alprazolam, and diazepam prepared by a simple, one-step oxidation of benzodiazepines.
    Journal of medicinal chemistry, 1978, Volume: 21, Issue:12

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Benzodiazepines; Diazepam; Hydroxylation; Male; Methods; Mice; Oxidation-Reduction; Triazolam; Triazoles

1978
Rm values and structure-activity relationship of benzodiazepines.
    Journal of medicinal chemistry, 1980, Volume: 23, Issue:2

    Topics: Animals; Benzodiazepines; Chromatography, Thin Layer; Conflict, Psychological; Exploratory Behavior; Models, Biological; Rats; Solubility; Structure-Activity Relationship

1980
Prediction of receptor properties and binding affinity of ligands to benzodiazepine/GABAA receptors using artificial neural networks.
    Journal of medicinal chemistry, 1995, Feb-17, Volume: 38, Issue:4

    Topics: Binding Sites; Ligands; Neural Networks, Computer; Predictive Value of Tests; Receptors, GABA-A; Structure-Activity Relationship

1995
Genetic neural networks for quantitative structure-activity relationships: improvements and application of benzodiazepine affinity for benzodiazepine/GABAA receptors.
    Journal of medicinal chemistry, 1996, Dec-20, Volume: 39, Issue:26

    Topics: Algorithms; Benzodiazepines; Models, Genetic; Nerve Net; Protein Binding; Receptors, GABA-A; Structure-Activity Relationship

1996
Molecular hashkeys: a novel method for molecular characterization and its application for predicting important pharmaceutical properties of molecules.
    Journal of medicinal chemistry, 1999, May-20, Volume: 42, Issue:10

    Topics: Drug Design; Intestinal Absorption; Models, Molecular; Pharmaceutical Preparations; Structure-Activity Relationship

1999
Predicting blood-brain barrier permeation from three-dimensional molecular structure.
    Journal of medicinal chemistry, 2000, Jun-01, Volume: 43, Issue:11

    Topics: Blood-Brain Barrier; Databases, Factual; Models, Chemical; Molecular Conformation; Multivariate Analysis; Permeability; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
QSAR model for drug human oral bioavailability.
    Journal of medicinal chemistry, 2000, Jun-29, Volume: 43, Issue:13

    Topics: Administration, Oral; Biological Availability; Humans; Models, Biological; Models, Molecular; Pharmaceutical Preparations; Pharmacokinetics; Structure-Activity Relationship

2000
Fast calculation of molecular polar surface area as a sum of fragment-based contributions and its application to the prediction of drug transport properties.
    Journal of medicinal chemistry, 2000, Oct-05, Volume: 43, Issue:20

    Topics: Biological Availability; Biological Transport; Models, Molecular; Molecular Structure; Pharmaceutical Preparations; Reproducibility of Results

2000
Experimental and computational screening models for the prediction of intestinal drug absorption.
    Journal of medicinal chemistry, 2001, Jun-07, Volume: 44, Issue:12

    Topics: Biological Transport; Carbon Radioisotopes; Cell Line; Cell Membrane; Cell Membrane Permeability; Ciprofloxacin; Computational Biology; Drug Design; Foscarnet; Humans; Hydrogen Bonding; Intestinal Absorption; Intestinal Mucosa; Lactulose; Mannitol; Models, Biological; Raffinose; Surface Properties; Tritium; Verapamil

2001
Prediction of human volume of distribution values for neutral and basic drugs. 2. Extended data set and leave-class-out statistics.
    Journal of medicinal chemistry, 2004, Feb-26, Volume: 47, Issue:5

    Topics: Algorithms; Blood Proteins; Half-Life; Humans; Hydrogen-Ion Concentration; Models, Biological; Pharmaceutical Preparations; Pharmacokinetics; Protein Binding; Statistics as Topic; Tissue Distribution

2004
Calculating virtual log P in the alkane/water system (log P(N)(alk)) and its derived parameters deltalog P(N)(oct-alk) and log D(pH)(alk).
    Journal of medicinal chemistry, 2005, May-05, Volume: 48, Issue:9

    Topics: 1-Octanol; Alkanes; Hydrogen-Ion Concentration; Least-Squares Analysis; Mathematics; Models, Chemical; Models, Molecular; Solvents; Water

2005
Computational aqueous solubility prediction for drug-like compounds in congeneric series.
    European journal of medicinal chemistry, 2008, Volume: 43, Issue:3

    Topics: Benzodiazepines; Computer Simulation; Crystallography, X-Ray; Databases, Factual; Least-Squares Analysis; Models, Chemical; Organic Chemicals; Pharmaceutical Preparations; Principal Component Analysis; Solubility; Sulfonamides; Water

2008
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
[Analysis of the structure of the components of the convulsive action of corazole following administration of sulazepam and its metabolites to mice].
    Biulleten' eksperimental'noi biologii i meditsiny, 1976, Volume: 82, Issue:9

    Topics: Animals; Anti-Anxiety Agents; Diazepam; Dose-Response Relationship, Drug; Male; Mice; Mice, Inbred CBA; Nordazepam; Oxazepam; Pentylenetetrazole; Seizures; Time Factors

1976
Feto-maternal concentrations of diazepam and W-demethyldiazepam after intra-amniotic diazepam injection.
    International journal of gynaecology and obstetrics: the official organ of the International Federation of Gynaecology and Obstetrics, 1976, Volume: 14, Issue:3

    Topics: Adolescent; Adult; Amniotic Fluid; Brain Chemistry; Diazepam; Female; Fetal Blood; Humans; Injections; Injections, Intramuscular; Kinetics; Liver; Maternal-Fetal Exchange; Nordazepam; Oxazepam; Pregnancy

1976
Pharmacokinetic understanding of antianxiety drug therapy.
    Southern medical journal, 1978, Volume: 71 Suppl 2

    Topics: Adult; Anti-Anxiety Agents; Chlordiazepoxide; Clorazepate Dipotassium; Diazepam; Dose-Response Relationship, Drug; Humans; Nordazepam; Oxazepam; Prazepam

1978
Simultaneous determination of diazepam and its metabolies N-desmethyldiazepam, oxydiazepam and oxazepam in plasma and urine of man and dog by means of high-performance liquid chromatography.
    Journal of chromatography, 1979, Apr-11, Volume: 162, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Dogs; Humans; Nordazepam; Oxazepam; Species Specificity; Temazepam

1979
High-pressure liquid chromatographic analysis of diazepam, oxazepam and N-desmethyldiazepam in human blood.
    Journal of chromatography, 1978, Mar-21, Volume: 150, Issue:2

    Topics: Chromatography, High Pressure Liquid; Diazepam; Humans; Nordazepam; Oxazepam

1978
Plasma and urine concentrations of diazepam and its metabolites in children, adults and in diazepam-intoxicated patients.
    International journal of clinical pharmacology and biopharmacy, 1978, Volume: 16, Issue:6

    Topics: Adult; Aging; Biotransformation; Child; Creatinine; Diazepam; Female; Humans; Infant; Infant, Newborn; Kinetics; Male; Nordazepam; Oxazepam

1978
Rapid recovery from massive diazepam overdose.
    JAMA, 1978, Oct-20, Volume: 240, Issue:17

    Topics: Adult; Biotransformation; Diazepam; Female; Half-Life; Humans; Male; Middle Aged; Nordazepam; Oxazepam; Remission, Spontaneous; Suicide, Attempted; Temazepam; Time Factors

1978
Fluorescence--TLC densitometric determination of diazepam and other 1,4-benzodiazepines in serum.
    Journal of pharmaceutical sciences, 1978, Volume: 67, Issue:10

    Topics: Benzodiazepines; Chromatography, Thin Layer; Densitometry; Diazepam; Humans; Methods; Nordazepam; Oxazepam; Spectrometry, Fluorescence

1978
Quantitation of chlordiazepoxide and its metabolites in biological fluids by thin-layer chromatography.
    Journal of chromatography, 1978, Nov-01, Volume: 146, Issue:3

    Topics: Benzodiazepinones; Chlordiazepoxide; Chromatography, Thin Layer; Humans; Nordazepam; Oxazepam; Spectrometry, Fluorescence

1978
Liquid-chromatographic assay of diazepam and its major metabolites in plasma.
    Clinical chemistry, 1979, Volume: 25, Issue:6

    Topics: Chromatography, High Pressure Liquid; Diazepam; Humans; Nordazepam; Oxazepam

1979
Effect of age on the pharmacokinetics of diazepam given in conjunction with spinal anesthesia.
    Anesthesiology, 1979, Volume: 51, Issue:2

    Topics: Adult; Age Factors; Aged; Anesthesia, Spinal; Body Water; Diazepam; Humans; Kinetics; Middle Aged; Nordazepam; Oxazepam; Temazepam

1979
[A screening radioimmunoassay for 1,4-benzodiazepines in human blood, serum, and urine using anti-oxazepam-hemisuccinate-antibodies (author's transl)].
    Zeitschrift fur Rechtsmedizin. Journal of legal medicine, 1979, Volume: 83, Issue:3

    Topics: Benzodiazepines; Chromatography, Gas; Chromatography, Thin Layer; Diazepam; Humans; Nordazepam; Oxazepam; Radioimmunoassay; Succinates

1979
Intravascular factors affecting diazepam binding to human serum albumin.
    Biochemical pharmacology, 1979, Nov-15, Volume: 28, Issue:22

    Topics: Binding, Competitive; Dialysis; Diazepam; Fatty Acids; Humans; Nordazepam; Oleic Acids; Oxazepam; Palmitic Acids; Protein Binding; Serum Albumin

1979
Quantitation by gas chromatography with selected-ion monitoring mass spectrometry of "natural" diazepam, N-desmethyldiazepam and oxazepam in normal human serum.
    Journal of chromatography, 1992, Aug-07, Volume: 579, Issue:1

    Topics: Adult; Analysis of Variance; Diazepam; Female; Gas Chromatography-Mass Spectrometry; Humans; Male; Nordazepam; Oxazepam

1992
Distribution of diazepam, nordiazepam, and oxazepam between brain extraneuronal space, brain tissue, plasma, and cerebrospinal fluid in diazepam and nordiazepam dependent dogs.
    Psychopharmacology, 1991, Volume: 105, Issue:4

    Topics: Animals; Brain; Diazepam; Dogs; Extracellular Space; Female; Nordazepam; Oxazepam; Substance-Related Disorders

1991
Determination of diazepam and nordazepam in milk and plasma in the presence of oxazepam and temazepam.
    Journal of chromatography, 1991, Mar-08, Volume: 564, Issue:1

    Topics: Chromatography, High Pressure Liquid; Diazepam; Flurazepam; Humans; Hydrogen-Ion Concentration; Milk, Human; Nordazepam; Oxazepam; Temazepam

1991
Characterization by saturation studies of the in vivo binding of [3H]flunitrazepam in mouse brain.
    Canadian journal of physiology and pharmacology, 1991, Volume: 69, Issue:2

    Topics: Animals; Brain; Chromatography, High Pressure Liquid; Clonazepam; Diazepam; Flunitrazepam; Kinetics; Mice; Nordazepam; Oxazepam

1991
Excretion of diazepam and its metabolites in human milk during withdrawal from combination high dose diazepam and oxazepam.
    British journal of clinical pharmacology, 1990, Volume: 29, Issue:1

    Topics: Adult; Diazepam; Drug Combinations; Female; Humans; Infant; Milk, Human; Nordazepam; Oxazepam; Substance Withdrawal Syndrome; Substance-Related Disorders; Temazepam

1990
In vitro drug metabolism and pharmacokinetics of diazepam in cynomolgus monkey hepatocytes during culture for six days.
    Biochemical pharmacology, 1989, Aug-15, Volume: 38, Issue:16

    Topics: Animals; Cells, Cultured; Cytochrome P-450 Enzyme System; Diazepam; Liver; Macaca fascicularis; Male; Models, Biological; Nordazepam; Oxazepam; Oxygenases; Temazepam; Time Factors

1989
Toxicity in a case of acute and massive overdose of chlordiazepoxide and its correlation to blood concentration.
    Journal of toxicology. Clinical toxicology, 1989, Volume: 27, Issue:1-2

    Topics: Anti-Anxiety Agents; Benzodiazepines; Benzodiazepinones; Biotransformation; Chlordiazepoxide; Chromatography, High Pressure Liquid; Female; Humans; Middle Aged; Nordazepam; Oxazepam

1989
Kinetics of drug action in disease states. XXIV. Pharmacodynamics of diazepam and its active metabolites in rats.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 244, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Brain; Diazepam; Female; Nordazepam; Oxazepam; Rats; Rats, Inbred Lew; Reflex; Temazepam

1988
Clorazepate, correlation between metabolism and anticonvulsant activity.
    European journal of pharmacology, 1988, Dec-13, Volume: 158, Issue:3

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Brain; Clorazepate Dipotassium; Half-Life; Male; Mice; Nordazepam; Oxazepam; Pentylenetetrazole; Seizures; Time Factors

1988
Potencies of diazepam metabolites in rats trained to discriminate diazepam.
    Life sciences, 1986, Jul-07, Volume: 39, Issue:1

    Topics: Animals; Conditioning, Operant; Diazepam; Discrimination, Psychological; Dose-Response Relationship, Drug; Male; Nordazepam; Oxazepam; Rats; Rats, Inbred Strains; Temazepam

1986
Validation of a radioreceptor assay technique for monitoring pharmacological active material during intensive diazepam tetanus therapy.
    International journal of clinical pharmacology, therapy, and toxicology, 1987, Volume: 25, Issue:7

    Topics: Biotransformation; Chromatography, Gas; Cimetidine; Diazepam; Humans; Kinetics; Middle Aged; Nordazepam; Oxazepam; Radioligand Assay; Tetanus

1987
Placental and blood-CSF transfer of orally administered diazepam in the same person.
    Pharmacology & toxicology, 1987, Volume: 61, Issue:1

    Topics: Adult; Biotransformation; Diazepam; Female; Fetal Blood; Humans; Maternal-Fetal Exchange; Nordazepam; Oxazepam; Pregnancy

1987
Analysis of chlorodesmethyldiazepam and its metabolites in plasma and urine.
    Journal of chromatography, 1987, Sep-25, Volume: 420, Issue:2

    Topics: Anti-Anxiety Agents; Benzodiazepines; Chromatography, Gas; Diazepam; Glucuronates; Humans; Lorazepam; Nordazepam; Oxazepam

1987
Simultaneous determination of diazepam and its active metabolites in rat serum, brain and cerebrospinal fluid by high-performance liquid chromatography.
    Journal of chromatography, 1987, Nov-27, Volume: 422

    Topics: Animals; Brain Chemistry; Chromatography, High Pressure Liquid; Diazepam; Female; Nordazepam; Oxazepam; Postural Balance; Rats; Rats, Inbred Strains; Temazepam

1987
Imipramine treatment alters the pharmacokinetics and pharmacodynamics of diazepam.
    Journal of pharmaceutical sciences, 1987, Volume: 76, Issue:12

    Topics: Animals; Blood Proteins; Brain Chemistry; Diazepam; Drug Interactions; Imipramine; Liver; Male; Nordazepam; Oxazepam; Pentylenetetrazole; Protein Binding; Rats; Rats, Inbred Strains; Temazepam

1987
Precipitation of abstinence in nordiazepam- and diazepam-dependent dogs.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:1

    Topics: Analysis of Variance; Animals; Diazepam; Dogs; Flumazenil; Nordazepam; Oxazepam; Pyrazoles; Seizures; Substance Withdrawal Syndrome; Substance-Related Disorders

1988
Long-lasting anticonvulsant effects of diazepam in different mouse strains: correlations with brain concentrations and receptor occupancy.
    Psychopharmacology, 1985, Volume: 86, Issue:1-2

    Topics: Animals; Anticonvulsants; Brain Chemistry; Diazepam; Mice; Mice, Inbred C3H; Nordazepam; Oxazepam; Pentylenetetrazole; Seizures; Species Specificity; Time Factors

1985
Liquid-chromatographic assay of diazepam and its major metabolites in serum, and application to pharmacokinetic study of high doses of diazepam in schizophrenics.
    Clinical chemistry, 1985, Volume: 31, Issue:10

    Topics: Administration, Oral; Chromatography, High Pressure Liquid; Diazepam; Female; Humans; Kinetics; Nordazepam; Oxazepam; Schizophrenia; Temazepam

1985
Severe withdrawal syndrome after substitution of a short-acting benzodiazepine for a long-acting benzodiazepine.
    Drug intelligence & clinical pharmacy, 1985, Volume: 19, Issue:10

    Topics: Diazepam; Female; Half-Life; Humans; Middle Aged; Nordazepam; Oxazepam; Substance Withdrawal Syndrome

1985
N-desmethyldiazepam physical dependence in dogs.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 235, Issue:2

    Topics: Analysis of Variance; Animals; Body Weight; Diazepam; Dogs; Drinking; Energy Intake; Female; Lorazepam; Muscle Spasticity; Nordazepam; Oxazepam; Paresthesia; Substance Withdrawal Syndrome; Temazepam; Time Factors

1985
Determination of some benzodiazepines and metabolites in serum, urine and saliva by high-performance liquid chromatography.
    Journal of chromatography, 1980, Feb-08, Volume: 181, Issue:2

    Topics: Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Humans; Mathematics; Nordazepam; Oxazepam; Saliva; Temazepam

1980
[Pharmacokinetic of benzodiazepines in old age].
    Schweizerische medizinische Wochenschrift, 1981, Nov-21, Volume: 111, Issue:47

    Topics: Adult; Aged; Aging; Anti-Anxiety Agents; Chlordiazepoxide; Diazepam; Half-Life; Humans; Lorazepam; Metabolic Clearance Rate; Middle Aged; Nitrazepam; Nordazepam; Oxazepam

1981
Aspects of the interaction of thyroxine and its binding serum proteins with 1,4-benzodiazepine tranquillizers.
    Biochemical medicine, 1981, Volume: 26, Issue:2

    Topics: Anti-Anxiety Agents; Autoradiography; Binding, Competitive; Chlordiazepoxide; Diazepam; Electrophoresis, Polyacrylamide Gel; Humans; Male; Nordazepam; Oxazepam; Temazepam; Thyroxine; Thyroxine-Binding Proteins

1981
Rapid gas chromatographic measurement of diazepam and its metabolites desmethyldiazepam, oxazepam, and 3-hydroxydiazepam (temazepam) in small samples of plasma.
    Therapeutic drug monitoring, 1982, Volume: 4, Issue:3

    Topics: Anti-Anxiety Agents; Biotransformation; Chromatography, Gas; Diazepam; Humans; Nordazepam; Oxazepam; Temazepam

1982
Blood concentrations of diazepam and its metabolites in children and neonates with tetanus.
    The Journal of pediatrics, 1983, Volume: 102, Issue:1

    Topics: Child; Diazepam; Female; Humans; Infant, Newborn; Infant, Newborn, Diseases; Male; Nordazepam; Oxazepam; Tetanus

1983
In vitro interaction of diazepam and oxazepam with pancuronium and suxamethonium.
    British journal of anaesthesia, 1984, Volume: 56, Issue:10

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; In Vitro Techniques; Muscle Contraction; Neuromuscular Junction; Nordazepam; Oxazepam; Pancuronium; Rats; Rats, Inbred Strains; Succinylcholine; Temazepam

1984
The contribution of the active metabolites to the tolerance developing to diazepam in man: relationship to bioassayed serum benzodiazepine levels.
    Medical biology, 1984, Volume: 62, Issue:5

    Topics: Adult; Benzodiazepines; Biological Assay; Diazepam; Double-Blind Method; Drug Tolerance; Female; Humans; Male; Nordazepam; Oxazepam; Psychomotor Performance

1984
Structure activity relationships of selected benzodiazepines as anticonvulsants to local anesthetics.
    Pharmacology and therapeutics in dentistry, 1980, Volume: 5, Issue:1-2

    Topics: Anesthetics, Local; Animals; Anticonvulsants; Benzodiazepines; Diazepam; Lidocaine; Male; Mepivacaine; Mice; Nitrazepam; Nordazepam; Oxazepam; Prilocaine; Seizures; Structure-Activity Relationship; Temazepam

1980
Influence of cimetidine on the pharmacokinetics of desmethyldiazepam and oxazepam.
    European journal of clinical pharmacology, 1980, Volume: 18, Issue:6

    Topics: Adult; Cimetidine; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Female; Guanidines; Humans; Kinetics; Liver; Male; Nordazepam; Oxazepam

1980
[Pharmacokinetics of oral prazepam].
    Fortschritte der Medizin, 1981, Jun-11, Volume: 99, Issue:22

    Topics: Administration, Oral; Biotransformation; Half-Life; Humans; Kinetics; Metabolic Clearance Rate; Nordazepam; Oxazepam; Prazepam

1981
Radioimmunoassay of benzodiazepines.
    Methods in enzymology, 1982, Volume: 84

    Topics: Benzodiazepines; Chlordiazepoxide; Clonazepam; Diazepam; Flurazepam; Humans; Microchemistry; Nitrazepam; Nordazepam; Oxazepam; Radioimmunoassay

1982
Anticonvulsant potency of unmetabolized diazepam.
    Pharmacology, 1982, Volume: 25, Issue:3

    Topics: Animals; Anticonvulsants; Brain; Diazepam; Male; Mice; Nordazepam; Oxazepam; Pentylenetetrazole; Time Factors

1982
Development and preliminary application of high-performance liquid chromatographic assay of urinary metabolites of diazepam in humans.
    Journal of chromatography. B, Biomedical applications, 1995, Jun-09, Volume: 668, Issue:1

    Topics: Chromatography, High Pressure Liquid; Diazepam; Humans; Nordazepam; Oxazepam; Reference Values; Reproducibility of Results; Temazepam

1995
Analysis of oxazepam in urine using solid-phase extraction and high-performance liquid chromatography with fluorescence detection by post-column derivatization.
    Journal of chromatography, 1993, Jul-02, Volume: 616, Issue:2

    Topics: Chromatography, High Pressure Liquid; Humans; Indicators and Reagents; Nordazepam; Oxazepam; Spectrometry, Fluorescence

1993
Pharmacokinetics of nordiazepam in physical dependence and precipitated abstinence in dogs.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:4

    Topics: Administration, Oral; Animals; Blood Proteins; Diazepam; Dogs; Female; Flumazenil; Hydrolysis; Injections, Intravenous; Nordazepam; Oxazepam; Protein Binding; Substance Withdrawal Syndrome; Substance-Related Disorders

1993
Kinetics of sequential metabolism. I. Formation and metabolism of oxazepam from nordiazepam and temazepam in the perfused murine liver.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:3

    Topics: Animals; Kinetics; Male; Mice; Microsomes, Liver; Nordazepam; Oxazepam; Perfusion; Proteins; Temazepam

1993
Kinetics of sequential metabolism. II. Formation and metabolism of nordiazepam and oxazepam from diazepam in the perfused murine liver.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:3

    Topics: Animals; Diazepam; Kinetics; Male; Mice; Microsomes, Liver; Nordazepam; Oxazepam; Perfusion

1993
[Determination of N-demethyldiazepam and its metabolite oxazepam in plasma by HPLC and their pharmacokinetics in rats].
    Yao xue xue bao = Acta pharmaceutica Sinica, 1995, Volume: 30, Issue:9

    Topics: Animals; Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Humans; Male; Nordazepam; Oxazepam; Rats; Rats, Sprague-Dawley

1995
Hair analysis for nordiazepam and oxazepam by gas chromatography--negative-ion chemical ionization mass spectrometry.
    Journal of chromatography. B, Biomedical applications, 1996, Mar-03, Volume: 677, Issue:2

    Topics: Adult; Anti-Anxiety Agents; Gas Chromatography-Mass Spectrometry; Hair; Humans; Nordazepam; Oxazepam; Reproducibility of Results; Substance Abuse Detection

1996
Flumazenil, diazepam, nordiazepam and oxazepam interactions on plasma protein binding.
    Pharmacological research, 1995, Volume: 32, Issue:5

    Topics: Animals; Anti-Anxiety Agents; Biotransformation; Blood Proteins; Diazepam; Dogs; Drug Interactions; Flumazenil; In Vitro Techniques; Nordazepam; Oxazepam; Protein Binding

1995
[Detection of nordiazepam in the hair of drug addicts].
    Annales pharmaceutiques francaises, 1996, Volume: 54, Issue:5

    Topics: Gas Chromatography-Mass Spectrometry; Hair; Heroin Dependence; Humans; Nordazepam; Oxazepam

1996
Reduction of oxazepam to desmethyldiazepam by human intestinal bacteria.
    Biological & pharmaceutical bulletin, 1996, Volume: 19, Issue:4

    Topics: Bifidobacterium; Biotransformation; Humans; Intestines; Magnetic Resonance Spectroscopy; Mass Spectrometry; Molecular Structure; Nordazepam; Oxazepam; Oxidation-Reduction; Spectrophotometry

1996
The effect of chronic benzodiazepines exposure on body weight in rats.
    Pharmacological research, 1998, Volume: 37, Issue:3

    Topics: Analysis of Variance; Animals; Anti-Anxiety Agents; Body Weight; Diazepam; Dose-Response Relationship, Drug; Female; Flumazenil; Flunitrazepam; GABA Modulators; Male; Nordazepam; Oxazepam; Rats; Rats, Sprague-Dawley; Sex Factors; Time Factors; Weight Gain

1998
Rapid and simple chromatographic method for the determination of diazepam and its major metabolites in human plasma and urine.
    Journal of chromatography. B, Biomedical sciences and applications, 1998, Apr-24, Volume: 708, Issue:1-2

    Topics: Calibration; Chromatography, High Pressure Liquid; Clonazepam; Diazepam; Humans; Nordazepam; Oxazepam; Reference Values; Temazepam

1998
Determination of benzodiazepines in human urine and plasma with solvent modified solid phase micro extraction and gas chromatography; rationalisation of method development using experimental design strategies.
    Journal of pharmaceutical and biomedical analysis, 1998, Volume: 18, Issue:4-5

    Topics: Alprazolam; Anti-Anxiety Agents; Benzodiazepines; Chromatography, Gas; Diazepam; Flunitrazepam; Humans; Hydrogen-Ion Concentration; Models, Chemical; Nordazepam; Oxazepam; Research Design

1998
Distribution of topiramate in a medical examiner's case.
    Journal of analytical toxicology, 1999, Volume: 23, Issue:6

    Topics: Adolescent; Anticonvulsants; Autopsy; Bile; Ethanol; Fatal Outcome; Female; Fructose; Gas Chromatography-Mass Spectrometry; Humans; Liver; Nordazepam; Oxazepam; Stomach; Tissue Distribution; Topiramate; Vitreous Body

1999
The simultaneous determination of diazepam and its three metabolites in dog plasma by high-performance liquid chromatography with mass spectroscopy detection.
    Journal of pharmaceutical and biomedical analysis, 2001, Volume: 26, Issue:2

    Topics: Animals; Anti-Anxiety Agents; Chromatography, High Pressure Liquid; Diazepam; Dogs; Mass Spectrometry; Nordazepam; Oxazepam; Reproducibility of Results; Temazepam

2001
Effects of diazepam and its metabolites on nocturnal melatonin secretion in the rat pineal and Harderian glands. A comparative in vivo and in vitro study.
    Chronobiology international, 2003, Volume: 20, Issue:2

    Topics: Animals; Circadian Rhythm; Diazepam; Harderian Gland; In Vitro Techniques; Male; Melatonin; Nordazepam; Oxazepam; Perfusion; Pineal Gland; Rats; Rats, Wistar; Temazepam

2003
Toxicological data and growth characteristics of single post-feeding larvae and puparia of Calliphora vicina (Diptera: Calliphoridae) obtained from a controlled nordiazepam study.
    International journal of legal medicine, 2004, Volume: 118, Issue:4

    Topics: Animals; Anti-Anxiety Agents; Chromatography, Liquid; Diptera; Forensic Medicine; Larva; Mass Spectrometry; Nordazepam; Oxazepam

2004
Development and validation of a liquid chromatographic/electrospray ionization mass spectrometric method for the quantitation of prazepam and its main metabolites in human plasma.
    Journal of mass spectrometry : JMS, 2005, Volume: 40, Issue:4

    Topics: Calibration; Chromatography, Liquid; Diazepam; Humans; Molecular Structure; Nordazepam; Oxazepam; Prazepam; Reference Standards; Reproducibility of Results; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization

2005
Fast in vivo microextraction: a new tool for clinical analysis.
    Clinical chemistry, 2006, Volume: 52, Issue:4

    Topics: Animals; Biocompatible Materials; Blood Chemical Analysis; Blood Specimen Collection; Calibration; Chemistry Techniques, Analytical; Chromatography, Liquid; Diazepam; Dogs; Mass Spectrometry; Nordazepam; Oxazepam; Polyethylene Glycols; Polymers; Pyrroles; Silicon Dioxide

2006
Liquid chromatographic-electrospray ionization mass spectrometric quantitative analysis of buprenorphine, norbuprenorphine, nordiazepam and oxazepam in rat plasma.
    Journal of pharmaceutical and biomedical analysis, 2006, Jun-16, Volume: 41, Issue:4

    Topics: Animals; Buprenorphine; Chromatography, Liquid; Male; Nordazepam; Oxazepam; Rats; Rats, Sprague-Dawley; Spectrometry, Mass, Electrospray Ionization

2006
A sensitive and selective method for the detection of diazepam and its main metabolites in urine by gas chromatography-tandem mass spectrometry.
    Journal of chromatography. A, 2007, Feb-02, Volume: 1141, Issue:1

    Topics: Benzodiazepinones; Diazepam; Gas Chromatography-Mass Spectrometry; Nordazepam; Oxazepam; Reproducibility of Results; Tandem Mass Spectrometry; Time Factors

2007
Fatal intoxication with milnacipran.
    Journal of forensic and legal medicine, 2008, Volume: 15, Issue:6

    Topics: Adult; Anti-Anxiety Agents; Antidepressive Agents; Chromatography, High Pressure Liquid; Cyclopropanes; Female; Fluoxetine; Forensic Toxicology; Gas Chromatography-Mass Spectrometry; Humans; Milnacipran; Nordazepam; Oxazepam; Phenothiazines; Selective Serotonin Reuptake Inhibitors; Sertraline; Suicide

2008
Two compartment model of diazepam biotransformation in an organotypical culture of primary human hepatocytes.
    Toxicology and applied pharmacology, 2009, Jan-15, Volume: 234, Issue:2

    Topics: Anti-Inflammatory Agents; Antithyroid Agents; Biotransformation; Cell Separation; Chlorodiphenyl (54% Chlorine); Chromatography, High Pressure Liquid; Cytochrome P-450 Enzyme System; Dexamethasone; Diazepam; Enzyme Induction; Hepatocytes; Humans; Hypnotics and Sedatives; Models, Biological; Models, Statistical; Nordazepam; Organ Culture Techniques; Oxazepam; Phenobarbital; Temazepam

2009
Simultaneous analysis of diazepam and its metabolites in rat plasma and brain tissue by HPLC-UV and SPE.
    Talanta, 2009, Nov-15, Volume: 80, Issue:1

    Topics: Animals; Brain; Brain Chemistry; Chromatography, High Pressure Liquid; Diazepam; Nordazepam; Oxazepam; Rats; Reproducibility of Results; Solid Phase Extraction; Spectrophotometry, Ultraviolet; Temazepam

2009
Measurement of benzodiazepines in urine by liquid chromatography-tandem mass spectrometry: confirmation of samples screened by immunoassay.
    Annals of clinical biochemistry, 2010, Volume: 47, Issue:Pt 2

    Topics: Benzodiazepines; Biological Assay; Calibration; Chromatography, Liquid; European Union; Immunoassay; Limit of Detection; Nitrazepam; Nordazepam; Oxazepam; Sensitivity and Specificity; Tandem Mass Spectrometry; Temazepam

2010
Quantitation of benzodiazepines in blood and urine using gas chromatography-mass spectrometry (GC-MS).
    Methods in molecular biology (Clifton, N.J.), 2010, Volume: 603

    Topics: Alprazolam; Benzodiazepines; Diazepam; Gas Chromatography-Mass Spectrometry; Humans; Lorazepam; Nordazepam; Oxazepam; Solid Phase Extraction; Triazolam

2010
LC-MS/MS analysis of 13 benzodiazepines and metabolites in urine, serum, plasma, and meconium.
    Methods in molecular biology (Clifton, N.J.), 2010, Volume: 603

    Topics: Alprazolam; Benzodiazepines; Chromatography, Liquid; Clonazepam; Flurazepam; Humans; Infant, Newborn; Meconium; Nordazepam; Oxazepam; Reproducibility of Results; Solid Phase Extraction; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Triazolam

2010
Simultaneous determination and quantification of 12 benzodiazepines in serum or whole blood using UPLC/MS/MS.
    Methods in molecular biology (Clifton, N.J.), 2010, Volume: 603

    Topics: Alprazolam; Benzodiazepines; Chlordiazepoxide; Chromatography, Liquid; Clonazepam; Flunitrazepam; Humans; Lorazepam; Midazolam; Nordazepam; Oxazepam; Reproducibility of Results; Tandem Mass Spectrometry

2010
A novel reductive transformation of oxazepam to nordiazepam observed during enzymatic hydrolysis.
    Journal of analytical toxicology, 2010, Volume: 34, Issue:5

    Topics: Benzodiazepines; Glucuronidase; Humans; Hydrolysis; Nordazepam; Oxazepam; Substance Abuse Detection

2010
Biotransformation of diazepam in a clinically relevant flat membrane bioreactor model using primary porcine hepatocytes.
    Fundamental & clinical pharmacology, 2011, Volume: 25, Issue:3

    Topics: Adult; Animals; Bioreactors; Biotransformation; Cells, Cultured; Culture Media; Culture Media, Serum-Free; Diazepam; Female; Hepatocytes; Humans; Inactivation, Metabolic; Liver, Artificial; Male; Nordazepam; Oxazepam; Swine; Temazepam; Young Adult

2011
Pharmacokinetics of the cytochrome P-450 substrates phenytoin, theophylline, and diazepam in healthy Greyhound dogs.
    Journal of veterinary pharmacology and therapeutics, 2012, Volume: 35, Issue:3

    Topics: Animals; Chromatography, High Pressure Liquid; Cytochrome P-450 Enzyme System; Diazepam; Dogs; Female; Fluorescence Polarization Immunoassay; Gas Chromatography-Mass Spectrometry; Injections, Intravenous; Male; Nordazepam; Oxazepam; Phenytoin; Theophylline

2012
Sensitive UPLC-MS-MS assay for 21 benzodiazepine drugs and metabolites, zolpidem and zopiclone in serum or plasma.
    Journal of analytical toxicology, 2012, Volume: 36, Issue:7

    Topics: Azabicyclo Compounds; Benzodiazepines; Chromatography, Liquid; Humans; Liquid-Liquid Extraction; Lorazepam; Mass Spectrometry; Nordazepam; Oxazepam; Piperazines; Plasma; Pyridines; Serum; Specimen Handling; Tandem Mass Spectrometry; Temazepam; Triazolam; Zolpidem

2012
Direct determination of diazepam and its glucuronide metabolites in human whole blood by μElution solid-phase extraction and liquid chromatography-tandem mass spectrometry.
    Forensic science international, 2013, Dec-10, Volume: 233, Issue:1-3

    Topics: Chromatography, Liquid; Diazepam; Forensic Toxicology; Humans; Hypnotics and Sedatives; Limit of Detection; Nordazepam; Oxazepam; Reproducibility of Results; Solid Phase Extraction; Tandem Mass Spectrometry; Temazepam

2013
Urinary diazepam metabolite distribution in a chronic pain population.
    Journal of analytical toxicology, 2014, Volume: 38, Issue:3

    Topics: Aryl Hydrocarbon Hydroxylases; Chromatography, High Pressure Liquid; Chronic Pain; Cytochrome P-450 CYP2C19; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Diazepam; Drug Interactions; Esomeprazole; Female; Fluoxetine; Humans; Male; Methadone; Nordazepam; Oxazepam; Retrospective Studies; Specimen Handling; Temazepam

2014
A mixed MDPV and benzodiazepine intoxication in a chronic drug abuser: determination of MDPV metabolites by LC-HRMS and discussion of the case.
    Forensic science international, 2014, Volume: 243

    Topics: Adult; Alprazolam; Benzodiazepines; Benzodioxoles; Chlordiazepoxide; Chromatography, Liquid; Diazepam; Humans; Hypnotics and Sedatives; Male; Mass Spectrometry; Nordazepam; Oxazepam; Psychotropic Drugs; Pyrrolidines; Substance-Related Disorders; Synthetic Cathinone; Temazepam

2014
Low doses of ethanol markedly potentiate the anti-seizure effect of diazepam in a mouse model of difficult-to-treat focal seizures.
    Epilepsy research, 2014, Volume: 108, Issue:10

    Topics: Animals; Anticonvulsants; Brain; Diazepam; Disease Models, Animal; Drug Compounding; Drug Synergism; Electroencephalography; Epilepsy, Temporal Lobe; Ethanol; Female; Kainic Acid; Mice; Nordazepam; Oxazepam; Seizures; Solvents; Temazepam; Water

2014
A comparative study of primary secondary amino (PSA) and multi-walled carbon nanotubes (MWCNTs) as QuEChERS absorbents for the rapid determination of diazepam and its major metabolites in fish samples by high-performance liquid chromatography-electrospray
    Journal of the science of food and agriculture, 2016, Jan-30, Volume: 96, Issue:2

    Topics: Adsorption; Animals; Chromatography, High Pressure Liquid; Diazepam; Fishes; Food Contamination; Nanotubes, Carbon; Nordazepam; Oxazepam; Seafood; Sensitivity and Specificity; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Temazepam

2016
Characterization of equine cytochrome P450: role of CYP3A in the metabolism of diazepam.
    Journal of veterinary pharmacology and therapeutics, 2016, Volume: 39, Issue:5

    Topics: Animals; Chlorocebus aethiops; COS Cells; Cytochrome P-450 CYP3A; Diazepam; Horses; Hypnotics and Sedatives; Male; Microsomes, Liver; Nordazepam; Oxazepam; Phylogeny; Protein Isoforms; Rats; Rats, Sprague-Dawley; Species Specificity; Temazepam

2016
Deposition of diazepam and its metabolites in hair following a single dose of diazepam.
    International journal of legal medicine, 2017, Volume: 131, Issue:1

    Topics: Adult; Asian People; Chromatography, Liquid; Diazepam; Female; Hair; Healthy Volunteers; Humans; Hypnotics and Sedatives; Male; Nordazepam; Oxazepam; Tandem Mass Spectrometry; Temazepam; Young Adult

2017
Pentobarbital in the context of possible suicides: Analysis of a Case.
    Forensic science international, 2017, Volume: 274

    Topics: Adult; Central Nervous System Depressants; Diazepam; Ethanol; Gastrointestinal Contents; Humans; Male; Nordazepam; Oxazepam; Pentobarbital; Suicide; Temazepam

2017
Site-, Technique-, and Time-Related Aspects of the Postmortem Redistribution of Diazepam, Methadone, Morphine, and their Metabolites: Interest of Popliteal Vein Blood Sampling.
    Journal of forensic sciences, 2017, Volume: 62, Issue:6

    Topics: Adult; Blood Specimen Collection; Chromatography, Liquid; Diazepam; Female; Femoral Vein; Forensic Toxicology; Humans; Male; Methadone; Middle Aged; Morphine; Morphine Derivatives; Nordazepam; Oxazepam; Popliteal Vein; Postmortem Changes; Subclavian Vein; Young Adult

2017
Toxicodynetics in nordiazepam and oxazepam overdoses.
    Annales pharmaceutiques francaises, 2017, Volume: 75, Issue:3

    Topics: Adolescent; Adult; Aging; Central Nervous System Depressants; Child; Child, Preschool; Drug Overdose; Ethanol; Female; GABA Modulators; Humans; Male; Middle Aged; Nordazepam; Oxazepam; Retrospective Studies; Toxicokinetics; Young Adult

2017
Entomotoxicology in burnt bodies: a case of maternal filicide-suicide by fire.
    International journal of legal medicine, 2017, Volume: 131, Issue:5

    Topics: Adult; Animals; Automobiles; Burns; Carbon Monoxide Poisoning; Carboxyhemoglobin; Child; Child, Preschool; Diazepam; Diptera; Feeding Behavior; Female; Fires; Gasoline; Homicide; Humans; Hypnotics and Sedatives; Kidney; Larva; Liver; Male; Nordazepam; Oxazepam; Postmortem Changes; Suicide

2017
Demoxepam Derivatization and GC-MS Analysis Produces Erroneous Nordiazepam and Oxazepam Results.
    Journal of analytical toxicology, 2019, Jun-01, Volume: 43, Issue:5

    Topics: Benzodiazepines; Chlordiazepoxide; False Positive Reactions; Gas Chromatography-Mass Spectrometry; Humans; Limit of Detection; Nordazepam; Oxazepam; Reference Standards

2019
LC-MS-MS Method for the Determination of Antidepressants and Benzodiazepines in Meconium.
    Journal of analytical toxicology, 2020, Jul-31, Volume: 44, Issue:6

    Topics: Alprazolam; Antidepressive Agents; Benzodiazepines; Chromatography, Liquid; Clonazepam; Forensic Toxicology; Humans; Limit of Detection; Meconium; Nordazepam; Oxazepam; Reproducibility of Results; Solid Phase Extraction; Substance Abuse Detection; Tandem Mass Spectrometry; Venlafaxine Hydrochloride; Zolpidem

2020
Postmortem Analysis of Benzodiazepines in Human Bone by Gas Chromatography-Mass Spectrometry.
    Journal of analytical toxicology, 2021, Jan-21, Volume: 44, Issue:9

    Topics: Alprazolam; Autopsy; Benzodiazepines; Chromatography, Liquid; Clonazepam; Diazepam; Forensic Toxicology; Gas Chromatography-Mass Spectrometry; Humans; Liquid-Liquid Extraction; Lorazepam; Nordazepam; Oxazepam; Tandem Mass Spectrometry

2021
Rapid Extraction and Qualitative Screening of 30 Drugs in Oral Fluid at Concentrations Recommended for the Investigation of DUID Cases.
    Journal of analytical toxicology, 2022, Oct-14, Volume: 46, Issue:8

    Topics: 2-Propanol; 3,4-Methylenedioxyamphetamine; Alprazolam; Amphetamines; Buprenorphine; Carisoprodol; Clonazepam; Cocaine; Codeine; Dronabinol; Fentanyl; Hexanes; Hydrocodone; Hydromorphone; Lorazepam; Meprobamate; Methadone; Methamphetamine; Morphine Derivatives; N-Methyl-3,4-methylenedioxyamphetamine; Nordazepam; Oxazepam; Oxycodone; Oxymorphone; Pharmaceutical Preparations; Phencyclidine; Tandem Mass Spectrometry; Temazepam; Tramadol; Zolpidem

2022