ouabain and proscillaridin

ouabain has been researched along with proscillaridin in 15 studies

Research

Studies (15)

TimeframeStudies, this research(%)All Research%
pre-19903 (20.00)18.7374
1990's2 (13.33)18.2507
2000's5 (33.33)29.6817
2010's3 (20.00)24.3611
2020's2 (13.33)2.80

Authors

AuthorsStudies
Ball, WJ; Farr, CD; Fishwild, DM; Nair, AC; Tabet, MR; Wang, X; Welsh, WJ1
Bohlin, L; Felth, J; Fryknäs, M; Gullbo, J; Lindskog, M; Rickardson, L; Rosén, J; Wickström, M1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Byun, SY; Choi, I; Jeon, S; Kim, S; Ko, M; Lee, J; Park, S; Shum, D1
Neugebauer, G1
Graumann, G; Haustein, KO; Stephan, B1
Kawaguchi, M; Nishida, H; Saito, H1
Eim, C; Kirch, U; Li, SQ; Schneider, R; Schoner, W; Sich, B1
Eim, C; Kirch, U; Lang, RE; Li, S; Schoner, W1
Bielawska, A; Bielawski, K; Winnicka, K1
Bielawska, A; Bielawski, K; Miltyk, W; Winnicka, K2
Bielawska, A; Bielawski, K; Surazyński, A; Winnicka, K1
Arribas, J; Barradas, M; Bernadó, C; Collado, M; Da Silva-Álvarez, S; Del Pino, P; Domínguez, E; Fernández-Marcos, PJ; Ferreirós, A; García-Caballero, T; Gómez, M; González, P; González-Barcia, M; Hernández-González, F; Ikonomopoulou, MP; Lalinde, M; Llanos, S; Loza, MI; Pedrosa, P; Picallos-Rabina, P; Pietrocola, F; Prats, N; Rodilla, V; Serrano, M; Soprano, E; Triana-Martínez, F; Vidal, A1
Ferreira, RS; Qayed, WS; Silva, JRA1

Other Studies

15 other study(ies) available for ouabain and proscillaridin

ArticleYear
Three-dimensional quantitative structure-activity relationship analysis of ligand binding to human sequence antidigoxin monoclonal antibodies using comparative molecular field analysis.
    Journal of medicinal chemistry, 2002, Jul-18, Volume: 45, Issue:15

    Topics: Amino Acid Sequence; Animals; Antibodies, Monoclonal; Antibody Specificity; Binding Sites, Antibody; Binding, Competitive; Carbohydrate Sequence; Digoxin; Enzyme-Linked Immunosorbent Assay; Humans; Immunoglobulin Fab Fragments; Mice; Mice, Transgenic; Models, Molecular; Molecular Sequence Data; Ouabain; Progesterone; Quantitative Structure-Activity Relationship; Radioligand Assay

2002
Cytotoxic effects of cardiac glycosides in colon cancer cells, alone and in combination with standard chemotherapeutic drugs.
    Journal of natural products, 2009, Volume: 72, Issue:11

    Topics: Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Camptothecin; Cardenolides; Colonic Neoplasms; Digitoxin; Digoxin; Drug Screening Assays, Antitumor; HT29 Cells; Humans; Irinotecan; NF-kappa B; Proscillaridin; Strophanthins

2009
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Identification of Antiviral Drug Candidates against SARS-CoV-2 from FDA-Approved Drugs.
    Antimicrobial agents and chemotherapy, 2020, 06-23, Volume: 64, Issue:7

    Topics: Animals; Anti-Inflammatory Agents; Antiviral Agents; Betacoronavirus; Cell Line; Chlorocebus aethiops; Coronavirus Infections; COVID-19; Drug Evaluation, Preclinical; Drug Repositioning; Humans; Niclosamide; Pandemics; Pneumonia, Viral; Pregnenediones; SARS-CoV-2; Vero Cells

2020
[Influence of high intravenous doses of D-penicillamine on toxic actions of cardiac glycosides in the guinea pig. Short communication (author's transl)].
    Arzneimittel-Forschung, 1977, Volume: 27, Issue:11

    Topics: Animals; Binding, Competitive; Blood Proteins; Bufanolides; Digoxin; Electrocardiography; Guinea Pigs; Injections, Intravenous; Ouabain; Penicillamine; Proscillaridin; Protein Binding

1977
Studies on cardioactive steroids. III. Characterization of different cardiac glycosides by their effects on contractility and rhythmicity at different extracellular potassium concentrations.
    Acta biologica et medica Germanica, 1975, Volume: 34, Issue:6

    Topics: Animals; Arrhythmias, Cardiac; Cardiac Glycosides; Cymarine; Digitoxin; Digoxin; Dimethylformamide; Female; Guinea Pigs; Heart Conduction System; Male; Myocardial Contraction; Ouabain; Potassium; Proscillaridin; Stimulation, Chemical

1975
[Effect of proscillaridin on active cation transport across human red cell membrane (author's transl)].
    [Hokkaido igaku zasshi] The Hokkaido journal of medical science, 1974, Volume: 49, Issue:3

    Topics: Adenosine Triphosphate; Adult; Biological Transport, Active; Bufanolides; Cell Membrane; Erythrocytes; Humans; In Vitro Techniques; Ouabain; Potassium; Proscillaridin; Sodium

1974
Proscillaridin A immunoreactivity: a new endogenous cardiac glycoside?
    Annals of the New York Academy of Sciences, 1997, Nov-03, Volume: 834

    Topics: Animals; Cardiac Glycosides; Cattle; Cross Reactions; Enzyme-Linked Immunosorbent Assay; Humans; Hypothalamus; Immunoglobulin G; Muscle, Skeletal; Organ Specificity; Ouabain; Proscillaridin; Rats

1997
Bovine adrenals and hypothalamus are a major source of proscillaridin A- and ouabain-immunoreactivities.
    Life sciences, 1998, Volume: 62, Issue:11

    Topics: Adrenal Glands; Animals; Cardiotonic Agents; Cattle; Chromatography, High Pressure Liquid; Cross Reactions; Enzyme-Linked Immunosorbent Assay; Humans; Hypothalamus; Ouabain; Proscillaridin; Sodium-Potassium-Exchanging ATPase

1998
Inhibition of DNA topoisomerases I and II, and growth inhibition of breast cancer MCF-7 cells by ouabain, digoxin and proscillaridin A.
    Biological & pharmaceutical bulletin, 2006, Volume: 29, Issue:7

    Topics: Breast Neoplasms; Cell Line, Tumor; Cell Survival; Digoxin; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Humans; Kinetics; Models, Molecular; Ouabain; Proscillaridin; Topoisomerase I Inhibitors; Topoisomerase II Inhibitors

2006
Apoptosis-mediated cytotoxicity of ouabain, digoxin and proscillaridin A in the estrogen independent MDA-MB-231 breast cancer cells.
    Archives of pharmacal research, 2007, Volume: 30, Issue:10

    Topics: Antineoplastic Agents, Phytogenic; Apoptosis; Breast Neoplasms; Calcium; Caspase 3; Cell Line, Tumor; Cell Proliferation; Cell Survival; Digoxin; Dose-Response Relationship, Drug; Enzyme Activation; Female; Humans; Inhibitory Concentration 50; Ouabain; Proscillaridin; Time Factors

2007
Antiproliferative activity of derivatives of ouabain, digoxin and proscillaridin A in human MCF-7 and MDA-MB-231 breast cancer cells.
    Biological & pharmaceutical bulletin, 2008, Volume: 31, Issue:6

    Topics: Blotting, Western; Calcium; Carbohydrate Sequence; Caspase 3; Cell Line, Tumor; Cell Proliferation; Cell Survival; Digoxin; DNA, Neoplasm; Electrophoresis, Polyacrylamide Gel; Enzyme Inhibitors; Female; Flow Cytometry; Humans; Immunoprecipitation; Indicators and Reagents; Microscopy, Fluorescence; Molecular Sequence Data; Ouabain; Proscillaridin; Topoisomerase I Inhibitors; Topoisomerase II Inhibitors

2008
Dual effects of ouabain, digoxin and proscillaridin A on the regulation of apoptosis in human fibroblasts.
    Natural product research, 2010, Volume: 24, Issue:3

    Topics: Apoptosis; Digoxin; Dose-Response Relationship, Drug; Enzyme Activation; Fibroblasts; Humans; Mitogen-Activated Protein Kinase Kinases; Ouabain; Proscillaridin; Signal Transduction

2010
Identification and characterization of Cardiac Glycosides as senolytic compounds.
    Nature communications, 2019, 10-21, Volume: 10, Issue:1

    Topics: A549 Cells; Animals; Antibiotics, Antineoplastic; Apoptosis; Bleomycin; Breast Neoplasms; Cardiac Glycosides; Cell Line, Tumor; Cell Membrane; Cellular Senescence; Chondrocytes; Digoxin; Female; Fibroblasts; Humans; Hydrogen-Ion Concentration; Mice; Osteoarthritis; Ouabain; Proscillaridin; Pulmonary Fibrosis; Xenograft Model Antitumor Assays

2019
In Silico Study towards Repositioning of FDA-Approved Drug Candidates for Anticoronaviral Therapy: Molecular Docking, Molecular Dynamics and Binding Free Energy Calculations.
    Molecules (Basel, Switzerland), 2022, Sep-14, Volume: 27, Issue:18

    Topics: Antiviral Agents; COVID-19; Cysteine Endopeptidases; Digitoxin; Digoxin; Drug Repositioning; Humans; Molecular Docking Simulation; Molecular Dynamics Simulation; Niclosamide; Ouabain; Papain; Proscillaridin; RNA-Dependent RNA Polymerase; SARS-CoV-2

2022