ouabain and cyclosporine

ouabain has been researched along with cyclosporine in 17 studies

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (17.65)18.2507
2000's5 (29.41)29.6817
2010's8 (47.06)24.3611
2020's1 (5.88)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Batista-Gonzalez, A; Brunhofer, G; Fallarero, A; Gopi Mohan, C; Karlsson, D; Shinde, P; Vuorela, P1
Byun, SY; Choi, I; Jeon, S; Kim, S; Ko, M; Lee, J; Park, S; Shum, D1
Charuk, J; De Lannoy, IA; Klein, J; Koren, G; Silverman, M1
Ballarín, J; Barceló, P; Casado, FJ; Felipe, A; Ferrer-Martínez, A; Pastor-Anglada, M1
Ivanova, AE; Marakhova, II; Toropova, FV; Vereninov, AA; Vinogradova, TA1
Madsen, SS; Tipsmark, CK1
Ishida, H1
Coqueiro, VM; Marques-Santos, LF; Rumjanek, VM1
Abe, T; Goto, J; Hishinuma, T; Mano, N; Mikkaichi, T; Okada, M; Shimada, M; Sugie, M; Toyohara, T; Yamaguchi, H1
Jablonska, A; Janowski, M; Lukomska, B1
Aschauer, L; Jennings, P; Limonciel, A; Pfaller, W; Wilmes, A1

Reviews

2 review(s) available for ouabain and cyclosporine

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010
[The research method for investigating the role of the mitochondrial permeability transition pore in cell death].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 2004, Volume: 123, Issue:5

    Topics: Apoptosis; Arsenicals; Calcium; Cyclosporine; Cytochromes c; Diazoxide; Humans; Ion Channels; Mitochondria; Mitochondrial Membrane Transport Proteins; Mitochondrial Permeability Transition Pore; Myocardial Reperfusion Injury; Myocardium; Necrosis; Ouabain

2004

Other Studies

15 other study(ies) available for ouabain and cyclosporine

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.
    Bioorganic & medicinal chemistry, 2012, Nov-15, Volume: 20, Issue:22

    Topics: Acetylcholinesterase; Amyloid beta-Peptides; Benzophenanthridines; Binding Sites; Butyrylcholinesterase; Catalytic Domain; Cholinesterase Inhibitors; Humans; Isoquinolines; Kinetics; Molecular Docking Simulation; Structure-Activity Relationship

2012
Identification of Antiviral Drug Candidates against SARS-CoV-2 from FDA-Approved Drugs.
    Antimicrobial agents and chemotherapy, 2020, 06-23, Volume: 64, Issue:7

    Topics: Animals; Anti-Inflammatory Agents; Antiviral Agents; Betacoronavirus; Cell Line; Chlorocebus aethiops; Coronavirus Infections; COVID-19; Drug Evaluation, Preclinical; Drug Repositioning; Humans; Niclosamide; Pandemics; Pneumonia, Viral; Pregnenediones; SARS-CoV-2; Vero Cells

2020
Cyclosporin and quinidine inhibition of renal digoxin excretion: evidence for luminal secretion of digoxin.
    The American journal of physiology, 1992, Volume: 263, Issue:4 Pt 2

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Digoxin; Dogs; Female; Kidney; Male; Membrane Glycoproteins; Ouabain; Quinidine

1992
Effects of cyclosporine A on Na,K-ATPase expression in the renal epithelial cell line NBL-1.
    Kidney international, 1996, Volume: 50, Issue:5

    Topics: Animals; Biological Transport, Active; Carrier Proteins; Cattle; Cell Line; Cell Membrane; Cyclosporine; Diuretics; DNA; Enzyme Inhibitors; Epithelium; Furosemide; Immunosuppressive Agents; Kidney; Membrane Proteins; Ouabain; RNA, Messenger; Rubidium; Sodium-Potassium-Chloride Symporters; Sodium-Potassium-Exchanging ATPase; Thymidine

1996
Functional expression of the Na/K pump is controlled via a cyclosporin A-sensitive signalling pathway in activated human lymphocytes.
    FEBS letters, 1999, Aug-06, Volume: 456, Issue:2

    Topics: Cyclosporine; DNA; Humans; Immunosuppressive Agents; In Vitro Techniques; Interleukin-2; Ion Transport; Ionomycin; Lymphocyte Activation; Lymphocytes; Ouabain; Phorbol 12,13-Dibutyrate; Phytohemagglutinins; Rubidium; Signal Transduction; Sodium-Potassium-Exchanging ATPase

1999
Rapid modulation of Na+/K+-ATPase activity in osmoregulatory tissues of a salmonid fish.
    The Journal of experimental biology, 2001, Volume: 204, Issue:Pt 4

    Topics: Animals; Bucladesine; Colforsin; Cyclic AMP; Cyclosporine; Enzyme Inhibitors; Fresh Water; Gills; In Vitro Techniques; Kidney; Okadaic Acid; Ouabain; Phosphodiesterase Inhibitors; Rubidium Radioisotopes; Seawater; Sodium-Potassium-Exchanging ATPase; Theophylline; Trout

2001
Cyclosporin A does not protect the disruption of the inner mitochondrial membrane potential induced by potassium ionophores in intact K562 cells.
    Cell biology international, 2006, Volume: 30, Issue:3

    Topics: Carbonyl Cyanide m-Chlorophenyl Hydrazone; Cell Size; Cells, Cultured; Cyclosporine; Drug Resistance, Multiple; Humans; Ionophores; K562 Cells; Membrane Potentials; Mitochondrial Membranes; Nigericin; Ouabain; Potassium; Time Factors; Valinomycin

2006
Transport of estrone 3-sulfate mediated by organic anion transporter OATP4C1: estrone 3-sulfate binds to the different recognition site for digoxin in OATP4C1.
    Drug metabolism and pharmacokinetics, 2010, Volume: 25, Issue:3

    Topics: Animals; Binding, Competitive; Biological Transport; Cell Line; Chenodeoxycholic Acid; Cyclosporine; Digoxin; Dogs; Epithelial Cells; Estrone; Humans; Kidney; Organic Anion Transporters; Ouabain; Pharmacokinetics; Sulfobromophthalein; Triiodothyronine

2010
Different methods of immunosuppresion do not prolong the survival of human cord blood-derived neural stem cells transplanted into focal brain-injured immunocompetent rats.
    Acta neurobiologiae experimentalis, 2013, Volume: 73, Issue:1

    Topics: Analysis of Variance; Animals; Antigens, CD; Brain Injuries; Cells, Cultured; Cyclosporine; Enzyme Inhibitors; Fetal Blood; Graft Rejection; Graft Survival; Humans; Immunocompetence; Immunosuppressive Agents; Male; Nerve Tissue Proteins; Neural Stem Cells; Ouabain; Rats; Rats, Wistar; Stem Cell Transplantation; Time Factors; Transplantation, Heterologous

2013
Evidence for a role of claudin 2 as a proximal tubular stress responsive paracellular water channel.
    Toxicology and applied pharmacology, 2014, Sep-01, Volume: 279, Issue:2

    Topics: Cell Culture Techniques; Cells, Cultured; Claudins; Cyclosporine; Electric Impedance; Enzyme Inhibitors; Humans; Immunosuppressive Agents; Kidney Tubules, Proximal; Osmotic Pressure; Ouabain; Porosity; RNA Interference; RNA, Messenger; Sodium-Potassium-Exchanging ATPase; Stress, Physiological; Tight Junctions; Time Factors; Transfection; Water

2014