ouabain and cimetidine

ouabain has been researched along with cimetidine in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-199011 (42.31)18.7374
1990's3 (11.54)18.2507
2000's6 (23.08)29.6817
2010's6 (23.08)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cha, SH; Endou, H; Kanai, Y; Kojima, R; Kusuhara, H; Sekine, T; Sugiyama, Y; Tsuda, M; Utsunomiya-Tate, N1
Cha, SH; Endou, H; Fukushima , JI; Goya, T; Kanai, Y; Kobayashi, Y; Sekine, T1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Axe, FU; Bembenek, SD; Butler, CR; Coles, F; Dunford, PJ; Edwards, JP; Fourie, AM; Grice, CA; Karlsson, L; Lundeen, K; Riley, JP; Savall, BM; Tays, KL; Wei, J; Williams, KN; Xue, X1
Austin, CP; Fidock, DA; Hayton, K; Huang, R; Inglese, J; Jiang, H; Johnson, RL; Su, XZ; Wellems, TE; Wichterman, J; Yuan, J1
Campillo, NE; Guerra, A; Páez, JA1
Benet, LZ; Brouwer, KL; Chu, X; Dahlin, A; Evers, R; Fischer, V; Giacomini, KM; Hillgren, KM; Hoffmaster, KA; Huang, SM; Ishikawa, T; Keppler, D; Kim, RB; Lee, CA; Niemi, M; Polli, JW; Sugiyama, Y; Swaan, PW; Tweedie, DJ; Ware, JA; Wright, SH; Yee, SW; Zamek-Gliszczynski, MJ; Zhang, L1
Annand, R; Gozalbes, R; Jacewicz, M; Pineda-Lucena, A; Tsaioun, K1
Artursson, P; Haglund, U; Karlgren, M; Kimoto, E; Lai, Y; Norinder, U; Vildhede, A; Wisniewski, JR1
Cantin, LD; Chen, H; Kenna, JG; Noeske, T; Stahl, S; Walker, CL; Warner, DJ1
Brodsky, JL; Chiang, A; Chung, WJ; Denny, RA; Goeckeler-Fried, JL; Havasi, V; Hong, JS; Keeton, AB; Mazur, M; Piazza, GA; Plyler, ZE; Rasmussen, L; Rowe, SM; Sorscher, EJ; Weissman, AM; White, EL1
Nishimura, H; Yamaguchi, K1
Trzeciakowski, JP1
Fu, SX; Li, CG; Li, YS1
Bounous, H; Cagin, N; Levitt, B; Somberg, JC1
McKinney, TD; Speeg, KV1
Fu, SX; Li, YS1
Faller, L; Jackson, R; Malinowska, D; Mukidjam, E; Rabon, E; Saccomani, G; Sachs, G; Smolka, A1
Kappagoda, T; Senaratne, M1
Carrasquer, G; Chu, TC; Holloman, TL; Rehm, WS; Schwartz, M1
McKinney, TD; Myers, P; Speeg, KV1
Miyazaki, M; Toda, N1
Abbott, NJ; Jones, HC; Revest, PA1
Bevan, JA; Henrion, D; Klaasen, A; Laher, I1
Hagen, SJ; Morrison, SW; Wu, H1
Braun, EJ; Dudas, PL; Pelis, RM; Renfro, JL1

Reviews

1 review(s) available for ouabain and cimetidine

ArticleYear
Membrane transporters in drug development.
    Nature reviews. Drug discovery, 2010, Volume: 9, Issue:3

    Topics: Animals; Computer Simulation; Decision Trees; Drug Approval; Drug Discovery; Drug Evaluation, Preclinical; Drug Interactions; Humans; Membrane Transport Proteins; Mice; Mice, Knockout; Prescription Drugs

2010

Other Studies

25 other study(ies) available for ouabain and cimetidine

ArticleYear
Molecular cloning and characterization of a new multispecific organic anion transporter from rat brain.
    The Journal of biological chemistry, 1999, May-07, Volume: 274, Issue:19

    Topics: Amino Acid Sequence; Animals; Brain; Carrier Proteins; Cloning, Molecular; DNA, Complementary; Estrone; Molecular Sequence Data; Ochratoxins; Organic Anion Transporters, Sodium-Independent; p-Aminohippuric Acid; Rats; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sequence Homology, Amino Acid; Xenopus laevis

1999
Identification and characterization of human organic anion transporter 3 expressing predominantly in the kidney.
    Molecular pharmacology, 2001, Volume: 59, Issue:5

    Topics: Amino Acid Sequence; Animals; Carrier Proteins; Chromosome Mapping; Chromosomes, Human, Pair 11; Cloning, Molecular; Gene Library; Humans; Kidney Tubules, Proximal; Molecular Sequence Data; Oocytes; Organic Anion Transporters, Sodium-Independent; Sequence Homology, Amino Acid; Tissue Distribution; Transfection; Xenopus laevis

2001
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Identification of a potent, selective, and orally active leukotriene a4 hydrolase inhibitor with anti-inflammatory activity.
    Journal of medicinal chemistry, 2008, Jul-24, Volume: 51, Issue:14

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Catalysis; Dogs; Drug Evaluation, Preclinical; Enzyme Inhibitors; Epoxide Hydrolases; Humans; Magnetic Resonance Spectroscopy; Mice; Structure-Activity Relationship

2008
Genetic mapping of targets mediating differential chemical phenotypes in Plasmodium falciparum.
    Nature chemical biology, 2009, Volume: 5, Issue:10

    Topics: Animals; Antimalarials; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chromosome Mapping; Crosses, Genetic; Dihydroergotamine; Drug Design; Drug Resistance; Humans; Inhibitory Concentration 50; Mutation; Plasmodium falciparum; Quantitative Trait Loci; Transfection

2009
Neural computational prediction of oral drug absorption based on CODES 2D descriptors.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:3

    Topics: Administration, Oral; Humans; Models, Chemical; Neural Networks, Computer; Permeability; Quantitative Structure-Activity Relationship; Technology, Pharmaceutical

2010
QSAR-based permeability model for drug-like compounds.
    Bioorganic & medicinal chemistry, 2011, Apr-15, Volume: 19, Issue:8

    Topics: Caco-2 Cells; Cell Membrane Permeability; Drug Discovery; Humans; Pharmaceutical Preparations; Pharmacokinetics; Quantitative Structure-Activity Relationship

2011
Classification of inhibitors of hepatic organic anion transporting polypeptides (OATPs): influence of protein expression on drug-drug interactions.
    Journal of medicinal chemistry, 2012, May-24, Volume: 55, Issue:10

    Topics: Atorvastatin; Biological Transport; Drug Interactions; Estradiol; Estrone; HEK293 Cells; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Least-Squares Analysis; Liver; Liver-Specific Organic Anion Transporter 1; Models, Molecular; Multivariate Analysis; Organic Anion Transporters; Organic Anion Transporters, Sodium-Independent; Protein Isoforms; Pyrroles; Solute Carrier Organic Anion Transporter Family Member 1B3; Structure-Activity Relationship; Transfection

2012
Mitigating the inhibition of human bile salt export pump by drugs: opportunities provided by physicochemical property modulation, in silico modeling, and structural modification.
    Drug metabolism and disposition: the biological fate of chemicals, 2012, Volume: 40, Issue:12

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 11; ATP-Binding Cassette Transporters; Bile Acids and Salts; Cell Line; Chemical and Drug Induced Liver Injury; Humans; Quantitative Structure-Activity Relationship

2012
Increasing the Endoplasmic Reticulum Pool of the F508del Allele of the Cystic Fibrosis Transmembrane Conductance Regulator Leads to Greater Folding Correction by Small Molecule Therapeutics.
    PloS one, 2016, Volume: 11, Issue:10

    Topics: Alleles; Benzoates; Cells, Cultured; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Furans; Gene Deletion; HEK293 Cells; HeLa Cells; High-Throughput Screening Assays; Humans; Hydroxamic Acids; Microscopy, Fluorescence; Protein Folding; Protein Structure, Tertiary; Pyrazoles; RNA, Messenger; Small Molecule Libraries; Ubiquitination; Vorinostat

2016
Angiotensin II-induced relaxation of fowl aorta.
    The American journal of physiology, 1988, Volume: 255, Issue:4 Pt 2

    Topics: 5,8,11,14-Eicosatetraynoic Acid; Angiotensin II; Animals; Aorta, Abdominal; Chickens; Cimetidine; Cyclic AMP; Cyclic GMP; In Vitro Techniques; Indomethacin; Methysergide; Microscopy, Electron; Muscle, Smooth, Vascular; Ouabain; Proadifen; Propranolol; Pyrilamine; Vasodilation

1988
Synergistic interaction between histamine and ouabain on ventricular fibrillation threshold.
    British journal of pharmacology, 1985, Volume: 85, Issue:1

    Topics: Animals; Cimetidine; Coronary Circulation; Drug Synergism; Electrocardiography; Guinea Pigs; Heart Rate; Histamine; Histamine H1 Antagonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Myocardial Contraction; Ouabain; Pyrilamine; Ventricular Fibrillation

1985
[Effects of histamine on ouabain-induced ventricular fibrillation in guinea pigs].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1986, Volume: 7, Issue:3

    Topics: Animals; Cimetidine; Drug Synergism; Female; Guinea Pigs; Heart Rate; Histamine; In Vitro Techniques; Male; Ouabain; Receptors, Histamine; Stimulation, Chemical; Ventricular Fibrillation

1986
Histamine antagonists as antiarrhythmic agents in ouabain cardiotoxicity in the cat.
    The Journal of pharmacology and experimental therapeutics, 1980, Volume: 214, Issue:2

    Topics: Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Cimetidine; Female; Histamine; Histamine Antagonists; Histamine H1 Antagonists; Male; Ouabain; Promethazine; Rats; Spinal Cord

1980
Cimetidine and procainamide secretion by proximal tubules in vitro.
    The American journal of physiology, 1982, Volume: 242, Issue:6

    Topics: Absorption; Acecainide; Animals; Carbon Dioxide; Chromatography, High Pressure Liquid; Cimetidine; Guanidines; Hypothermia; Kidney Tubules, Proximal; Kinetics; Ouabain; Probenecid; Procainamide; Quinidine; Rabbits

1982
[Anti-arrhythmic action of cimetidine].
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1983, Volume: 4, Issue:2

    Topics: Aconitine; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Cimetidine; Female; Guanidines; Guinea Pigs; Heart; In Vitro Techniques; Male; Ouabain; Rabbits; Rats; Refractory Period, Electrophysiological

1983
Mechanistic aspects of gastric (H+ + K+)-ATPase.
    Annals of the New York Academy of Sciences, 1982, Volume: 402

    Topics: Adenosine Triphosphatases; Adenosine Triphosphate; Animals; Azides; Biological Transport, Active; Bucladesine; Cimetidine; Gastric Juice; H(+)-K(+)-Exchanging ATPase; Kinetics; Microsomes; Ouabain; Potassium; Stomach; Vanadates; Vanadium

1982
Tetrodotoxin-resistant relaxation to transmural nerve stimulation in isolated saphenous vein.
    The American journal of physiology, 1984, Volume: 247, Issue:6 Pt 2

    Topics: Aminophylline; Animals; Biomechanical Phenomena; Cimetidine; Cyproheptadine; Dogs; Drug Resistance; In Vitro Techniques; Indomethacin; Microscopy, Electron, Scanning; Muscle Contraction; Muscle Relaxation; Ouabain; Reaction Time; Saphenous Vein; Stimulation, Chemical; Tetrodotoxin

1984
Effects of ouabain on frog gastric mucosa in vitro.
    Biochimica et biophysica acta, 1981, Jan-22, Volume: 640, Issue:2

    Topics: Animals; Cimetidine; Electric Conductivity; Gastric Juice; Gastric Mucosa; Hydrogen-Ion Concentration; In Vitro Techniques; Membrane Potentials; Ouabain; Rana pipiens; Sodium; Sodium Chloride; Sulfates

1981
Cimetidine secretion by rabbit renal tubules in vitro.
    The American journal of physiology, 1981, Volume: 241, Issue:1

    Topics: Animals; Biological Transport; Chromatography, High Pressure Liquid; Cimetidine; Creatinine; Guanidines; In Vitro Techniques; Kidney Tubules; Kinetics; Ouabain; p-Aminohippuric Acid; Perfusion; Phlorhizin; Quinine; Rabbits; Tolazoline

1981
Angiotensin-induced relaxation in isolated dog renal and cerebral arteries.
    The American journal of physiology, 1981, Volume: 240, Issue:2

    Topics: Aminophylline; Angiotensin II; Animals; Arteries; Aspirin; Atropine; Brain; Cimetidine; Cocaine; Depression, Chemical; Dogs; Female; Hexamethonium Compounds; In Vitro Techniques; Kidney; Male; Muscle Contraction; Muscle, Smooth, Vascular; Ouabain; Propranolol; Prostaglandins F; Saralasin

1981
Transendothelial electrical potential across pial vessels in anaesthetised rats: a study of ion permeability and transport at the blood-brain barrier.
    Brain research, 1994, Jul-25, Volume: 652, Issue:1

    Topics: Anesthesia; Animals; Blood-Brain Barrier; Cell Membrane Permeability; Cimetidine; Electrophysiology; Endothelium, Vascular; Histamine; Ion Channels; Kinetics; Microelectrodes; Ouabain; Pia Mater; Potassium Channels; Rats; Rats, Inbred Strains; Sodium Channels

1994
Myogenic tone of rabbit facial vein and posterior cerebral artery is influenced by changes in extracellular sodium.
    The American journal of physiology, 1994, Volume: 266, Issue:2 Pt 2

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Analysis of Variance; Animals; Bicarbonates; Cerebral Arteries; Cimetidine; Histamine; In Vitro Techniques; Isometric Contraction; Meglumine; Monensin; Mouth; Muscle Tonus; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Ouabain; Propranolol; Rabbits; Sodium; Veins

1994
NH(4)Cl inhibition of acid secretion: possible involvement of an apical K(+) channel in bullfrog oxyntic cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2000, Volume: 279, Issue:2

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adenosine Triphosphate; Ammonia; Ammonium Chloride; Animals; Barium; Biological Transport; Bumetanide; Carbachol; Carbon Radioisotopes; Cholinergic Agents; Cimetidine; Clotrimazole; Diuretics; Enzyme Inhibitors; Gastric Mucosa; Growth Inhibitors; Histamine; Hydrochloric Acid; Hypoglycemic Agents; Imidazoles; Methylamines; Microscopy, Electron; Omeprazole; Ouabain; Parietal Cells, Gastric; Potassium Channel Blockers; Potassium Channels; Protons; Rana catesbeiana; Tetraethylammonium; Tolbutamide

2000
Transepithelial urate transport by avian renal proximal tubule epithelium in primary culture.
    The Journal of experimental biology, 2005, Volume: 208, Issue:Pt 22

    Topics: Animals; Biological Transport, Active; Bromcresol Green; Carbon Radioisotopes; Chickens; Cimetidine; Cytochalasins; DNA Primers; Electric Impedance; Epithelium; Estrone; Glutarates; Hydrogen-Ion Concentration; Kidney Tubules, Proximal; Lithium; Membrane Potentials; Nocodazole; Organic Anion Transporters; Ouabain; p-Aminohippuric Acid; Probenecid; Reverse Transcriptase Polymerase Chain Reaction; Time Factors; Uric Acid

2005