ornithine and icatibant

ornithine has been researched along with icatibant in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's7 (77.78)29.6817
2010's2 (22.22)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cialdai, C; Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Quartara, L; Tramontana, M; Valenti, C1
Bellucci, F; Bressan, A; Catalani, C; Cucchi, P; Faiella, A; Giolitti, A; Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Quartara, L; Rotondaro, L; Santicioli, P1
Bellucci, F; Cucchi, P; Lazzeri, M; Meini, S; Santicioli, P; Turini, D1
Cialdai, C; Giuliani, S; Maggi, CA; Quartara, L; Tramontana, M; Valenti, C1
Bellucci, F; Catalani, C; Cucchi, P; Giuliani, S; Maggi, CA; Meini, S; Santicioli, P1
Cialdai, C; Giuliani, S; Maggi, CA; Tramontana, M; Valenti, C1
Bellucci, F; Catalani, C; Cucchi, P; Giuliani, S; Maggi, CA; Meini, S2
Bellucci, F; Catalani, C; Cucchi, P; Giolitti, A; Giuliani, S; Maggi, CA; Meini, S; Quartara, L; Rotondaro, L; Zappitelli, S1

Other Studies

9 other study(ies) available for ornithine and icatibant

ArticleYear
MEN16132, a novel potent and selective nonpeptide kinin B2 receptor antagonist: in vivo activity on bradykinin-induced bronchoconstriction and nasal mucosa microvascular leakage in anesthetized guinea pigs.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 315, Issue:2

    Topics: Anesthesia; Animals; Blood Pressure; Blood Proteins; Bradykinin; Bradykinin B2 Receptor Antagonists; Bronchoconstriction; Capillary Permeability; Dose-Response Relationship, Drug; Guinea Pigs; Hypotension; In Vitro Techniques; Injections, Intravenous; Male; Microcirculation; Nasal Mucosa; Ornithine; Regional Blood Flow; Sulfonamides

2005
MEN16132, a novel potent and selective nonpeptide antagonist for the human bradykinin B2 receptor. In vitro pharmacology and molecular characterization.
    European journal of pharmacology, 2005, Dec-28, Volume: 528, Issue:1-3

    Topics: Animals; Binding, Competitive; Bradykinin; Bradykinin B2 Receptor Antagonists; Cells, Cultured; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Guinea Pigs; Humans; In Vitro Techniques; Inositol Phosphates; Middle Aged; Muscle Contraction; Muscle, Smooth; Myocytes, Smooth Muscle; Ornithine; Point Mutation; Quinolines; Receptor, Bradykinin B2; Sulfonamides; Transfection

2005
Characterization of kinin receptors in human cultured detrusor smooth muscle cells.
    British journal of pharmacology, 2007, Volume: 150, Issue:2

    Topics: Bradykinin; Bradykinin B1 Receptor Antagonists; Cells, Cultured; Dinoprostone; Humans; Inositol Phosphates; Interleukin-1beta; Kallidin; Male; Middle Aged; Muscle, Smooth; Ornithine; Radioligand Assay; Receptor, Bradykinin B1; Sulfonamides; Transforming Growth Factor alpha; Urinary Bladder

2007
MEN16132, a kinin B2 receptor antagonist, prevents the endogenous bradykinin effects in guinea-pig airways.
    European journal of pharmacology, 2008, Jan-28, Volume: 579, Issue:1-3

    Topics: Administration, Intranasal; Aerosols; Animals; Blood Proteins; Bradykinin; Bradykinin B2 Receptor Antagonists; Bronchoconstriction; Dextran Sulfate; Dose-Response Relationship, Drug; Guinea Pigs; Kallikrein-Kinin System; Male; Nasal Mucosa; Ornithine; Sulfonamides

2008
Pharmacological characterization of the bradykinin B2 receptor antagonist MEN16132 in rat in vitro bioassays.
    European journal of pharmacology, 2009, Aug-01, Volume: 615, Issue:1-3

    Topics: Animals; Binding, Competitive; Bradykinin; Bradykinin B2 Receptor Antagonists; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nasal Mucosa; Ornithine; Radioligand Assay; Rats; Rats, Wistar; Species Specificity; Sulfonamides; Urinary Bladder; Uterus

2009
Effect of Intra-articular 4-(S)-amino-5-(4-{4-[2,4-dichloro-3-(2,4-dimethyl-8-quinolyloxymethyl)phenylsulfonamido]-tetrahydro-2H-4-pyranylcarbonyl} piperazino)-5-oxopentyl](trimethyl)ammonium chloride hydrochloride (MEN16132), a kinin B2 receptor antagoni
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 331, Issue:3

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Bradykinin; Bradykinin B2 Receptor Antagonists; Dinoprostone; Disease Models, Animal; Dose-Response Relationship, Drug; Hindlimb; Injections, Intra-Articular; Iodoacetates; Male; Ornithine; Osteoarthritis; Pain; Rats; Rats, Wistar; Sulfonamides; Synovial Fluid

2009
Novel effects mediated by bradykinin and pharmacological characterization of bradykinin B2 receptor antagonism in human synovial fibroblasts.
    British journal of pharmacology, 2009, Volume: 158, Issue:8

    Topics: Bradykinin; Bradykinin B2 Receptor Antagonists; Cells, Cultured; Fibroblasts; Humans; Inhibitory Concentration 50; Inositol Phosphates; Interleukin-6; Interleukin-8; Ornithine; Radioligand Assay; Receptor, Bradykinin B2; Sulfonamides; Synovial Membrane; Synovitis

2009
Bradykinin and B₂ receptor antagonism in rat and human articular chondrocytes.
    British journal of pharmacology, 2011, Volume: 162, Issue:3

    Topics: Animals; Bradykinin; Bradykinin B2 Receptor Antagonists; Cartilage, Articular; Cells, Cultured; Chondrocytes; Humans; Inositol Phosphates; Interleukin-6; Interleukin-8; Knee; Ornithine; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Bradykinin B2; Sulfonamides

2011
Comparison of the molecular interactions of two antagonists, MEN16132 or icatibant, at the human kinin B₂ receptor.
    British journal of pharmacology, 2011, Volume: 162, Issue:5

    Topics: Amino Acid Substitution; Animals; Binding Sites; Bradykinin; Bradykinin B2 Receptor Antagonists; CHO Cells; Cricetinae; Cricetulus; Humans; In Vitro Techniques; Kinetics; Models, Molecular; Mutagenesis, Site-Directed; Mutant Proteins; Oligopeptides; Ornithine; Peptides, Cyclic; Receptor, Bradykinin B2; Recombinant Proteins; Sulfonamides

2011