organophosphonates has been researched along with cyclophostin in 5 studies
| Studies (organophosphonates) | Trials (organophosphonates) | Recent Studies (post-2010) (organophosphonates) | Studies (cyclophostin) | Trials (cyclophostin) | Recent Studies (post-2010) (cyclophostin) |
|---|---|---|---|---|---|
| 9,968 | 880 | 3,596 | 13 | 0 | 9 |
| Protein | Taxonomy | organophosphonates (IC50) | cyclophostin (IC50) |
|---|---|---|---|
| Acetylcholinesterase | Homo sapiens (human) | 0.0286 | |
| Carboxylic ester hydrolase | Musca domestica (house fly) | 0.0008 |
| Timeframe | Studies, this research(%) | All Research% |
|---|---|---|
| pre-1990 | 0 (0.00) | 18.7374 |
| 1990's | 0 (0.00) | 18.2507 |
| 2000's | 1 (20.00) | 29.6817 |
| 2010's | 4 (80.00) | 24.3611 |
| 2020's | 0 (0.00) | 2.80 |
| Authors | Studies |
|---|---|
| Bandyopadhyay, S; Dupureur, CM; Dutta, S; Rath, NP; Spilling, CD | 1 |
| Bandyopadhyay, S; Dupureur, CM; Dutta, S; Malla, RK; Spilling, CD | 1 |
| Canaan, S; Carriere, F; Cavalier, JF; Delorme, V; Diomande, S; Malla, RK; Martin, BP; Point, V; Rath, NP; Spilling, CD | 1 |
| Canaan, S; Carrière, F; Cavalier, JF; Malla, RK; Point, V; Spilling, CD | 1 |
| Dupureur, CM; Martin, BP; Spilling, CD; Vasilieva, E | 1 |
5 other study(ies) available for organophosphonates and cyclophostin
| Article | Year |
|---|---|
Synthesis and biological evaluation of a phosphonate analog of the natural acetyl cholinesterase inhibitor cyclophostin.
Topics: Cholinesterase Inhibitors; Cyclization; Hydrogenation; Lactones; Organophosphonates; Organophosphorus Compounds; Structure-Activity Relationship | 2008 |
Synthesis and kinetic analysis of some phosphonate analogs of cyclophostin as inhibitors of human acetylcholinesterase.
Topics: Acetylcholinesterase; Binding Sites; Cholinesterase Inhibitors; Humans; Kinetics; Mass Spectrometry; Molecular Structure; Organophosphonates; Organophosphorus Compounds; Stereoisomerism; Structure-Activity Relationship | 2010 |
Synthesis and kinetic evaluation of cyclophostin and cyclipostins phosphonate analogs as selective and potent inhibitors of microbial lipases.
Topics: Carboxylic Ester Hydrolases; Enzyme Inhibitors; Fusarium; Kinetics; Lipase; Molecular Structure; Mycobacterium tuberculosis; Organophosphonates; Organophosphorus Compounds; Structure-Activity Relationship | 2012 |
Enantioselective inhibition of microbial lipolytic enzymes by nonracemic monocyclic enolphosphonate analogues of cyclophostin.
Topics: Bacterial Proteins; Carboxylic Ester Hydrolases; Fungal Proteins; Fusarium; Lipase; Lipolysis; Monoacylglycerol Lipases; Mycobacterium tuberculosis; Organophosphonates; Organophosphorus Compounds; Stereoisomerism | 2013 |
Synthesis and comparison of the biological activity of monocyclic phosphonate, difluorophosphonate and phosphate analogs of the natural AChE inhibitor cyclophostin.
Topics: Acetylcholinesterase; Cholinesterase Inhibitors; Halogenation; Humans; Organophosphates; Organophosphonates; Organophosphorus Compounds | 2015 |