Page last updated: 2024-09-05

organophosphonates and atropine

organophosphonates has been researched along with atropine in 17 studies

Compound Research Comparison

Studies
(organophosphonates)
Trials
(organophosphonates)
Recent Studies (post-2010)
(organophosphonates)
Studies
(atropine)
Trials
(atropine)
Recent Studies (post-2010) (atropine)
9,9688803,59626,7111,2591,697

Protein Interaction Comparison

ProteinTaxonomyorganophosphonates (IC50)atropine (IC50)
cystic fibrosis transmembrane conductance regulatorHomo sapiens (human)21.41
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)1.012
Muscarinic acetylcholine receptor M2Homo sapiens (human)0.0067
Muscarinic acetylcholine receptor M4Homo sapiens (human)0.0007
Muscarinic acetylcholine receptor M1Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M3Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M4Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M5Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M5Homo sapiens (human)0.0009
Muscarinic acetylcholine receptor M2Rattus norvegicus (Norway rat)0.001
Muscarinic acetylcholine receptor M1Homo sapiens (human)0.0015
Muscarinic acetylcholine receptor M3Homo sapiens (human)0.0021
Alpha-1D adrenergic receptorHomo sapiens (human)1.354
5-hydroxytryptamine receptor 2CHomo sapiens (human)1.012

Research

Studies (17)

TimeframeStudies, this research(%)All Research%
pre-199016 (94.12)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (5.88)2.80

Authors

AuthorsStudies
Kimmerle, G; Lorke, D1
Berry, WK; Davies, DR; Gordon, JJ1
Adams, N; Bay, E; Von Bredow, J1
Michelson, MJ; Muske, GA; Protas, LL1
Fleisher, JH; Harris, LW; Yamamura, HI1
Aly, HI; Haroon, E; Helmy, R1
Jović, R; Milosević, M1
McPhillips, JJ; Perrine, SE1
Cohen, EM; Polak, RL1
Berry, WK; Davies, DR1
Moroi, K; Ogura, Y; Sato, T; Yoshida, S1
Aldous, FA; Brimblecombe, RW; Green, DM; Thompson, PB1
Bosković, B; Maksimović, M; Minic, D1
Casida, JE; Chambers, HW1
Cliff, WJ; Fleisher, JH; Harris, LW; Vick, JA1
Fleisher, JH; Harris, LW1
Thiermann, H; Wille, T; Worek, F1

Reviews

1 review(s) available for organophosphonates and atropine

ArticleYear
Organophosphorus compounds and oximes: a critical review.
    Archives of toxicology, 2020, Volume: 94, Issue:7

    Topics: Animals; Antidotes; Atropine; Cholinesterase Reactivators; Humans; Nerve Agents; Organophosphate Poisoning; Organophosphonates; Oximes; Pesticides; Treatment Outcome

2020

Other Studies

16 other study(ies) available for organophosphonates and atropine

ArticleYear
[Action of reactivators in phosphoric acid ester poisoning].
    Naunyn-Schmiedebergs Archiv fur experimentelle Pathologie und Pharmakologie, 1969, Volume: 263, Issue:1

    Topics: Animals; Antidotes; Atropine; Cholinesterase Inhibitors; Diphosphates; Humans; Organophosphonates; Parathion; Phosphoric Acids; Pralidoxime Compounds; Rats; Triazines

1969
Protection of animals against soman (1,2,2-trimethylpropyl methylphosphono-fluoridate) by pretreatment with some other organophosphorus compounds, followed by oxime and atropine.
    Biochemical pharmacology, 1971, Volume: 20, Issue:1

    Topics: Amitriptyline; Animals; Atropine; Bromides; Carbamates; Cholinesterase Inhibitors; Diphosphates; Drug Antagonism; Female; Fluorine; Guinea Pigs; Hydroxamic Acids; Isoflurophate; Lethal Dose 50; Nitrates; Nitrophenols; Nitroso Compounds; Organophosphonates; Organophosphorus Compounds; Orphenadrine; Oximes; Parasympatholytics; Physostigmine; Poisoning; Pyridinium Compounds; Rabbits; Rats; Salicylates; Scopolamine; Species Specificity; Sulfonic Acids; Sulfuric Acids; Thiazoles; Time Factors

1971
Drug actions on the central nervous system as studied by the effects on the electroretinogram.
    Experimental neurology, 1971, Volume: 33, Issue:1

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Atropine; Carbachol; Cats; Central Nervous System; Cholinesterase Inhibitors; Electroretinography; Neurotransmitter Agents; Norepinephrine; Organophosphonates; Physostigmine; Retina; Synaptic Transmission

1971
On the role of blood and muscle cholinesterases in the hydrolysis of subecholine and acetylcholine in the cat.
    Pharmacological research communications, 1974, Volume: 6, Issue:3

    Topics: Acetylcholine; Animals; Atropine; Caprylates; Cats; Choline; Cholinesterase Inhibitors; Cholinesterases; Dicarboxylic Acids; Electric Stimulation; Hydrolysis; Muscle Contraction; Muscles; Nitrobenzenes; Organophosphonates; Organophosphorus Compounds

1974
De novo synthesis of acetylcholinesterase in guinea pig retina after inhibition by pinacolyl methylphosphonofluoridate.
    Biochemical pharmacology, 1971, Volume: 20, Issue:10

    Topics: Acetylcholinesterase; Animals; Atropine; Cholinesterase Inhibitors; Cycloheximide; Guinea Pigs; Organophosphonates; Phosphates; Phosphorus Isotopes; Retina

1971
Effect of dipterex on the acetylcholine content and cholinesterase activity of the brain of male albino rats.
    The Journal of the Egyptian Medical Association, 1969, Volume: 52, Issue:2

    Topics: Acetylcholine; Animals; Atropine; Brain Chemistry; Cholinesterases; Male; Organophosphonates; Rats

1969
Inhibitory action of soman and some cholinolytics on the uptake of oxygen in the brain of rats and mice.
    European journal of pharmacology, 1970, Volume: 9, Issue:3

    Topics: Animals; Atropine; Benactyzine; Brain; Cerebral Cortex; Cholinesterase Inhibitors; Cyclopentanes; Esters; Fluorine; Male; Medulla Oblongata; Mice; Organophosphonates; Oxygen Consumption; Parasympatholytics; Rats

1970
Specific subsensitivity of the rat atrium to cholinergic drugs.
    The Journal of pharmacology and experimental therapeutics, 1970, Volume: 175, Issue:2

    Topics: Acetylcholine; Animals; Atropine; Bethanechol Compounds; Carbachol; Cholinesterase Inhibitors; Drug Synergism; Epinephrine; Female; Heart Atria; Heart Rate; In Vitro Techniques; Methacholine Compounds; Organophosphonates; Parasympathomimetics; Rats; Time Factors; Veratrine

1970
The influence of oximes on the distribution of 32P in the body of the rat after injection of 32P-sarin.
    Biochemical pharmacology, 1970, Volume: 19, Issue:3

    Topics: Acetylcholinesterase; Animals; Atropine; Brain; Brain Chemistry; Cholinesterase Inhibitors; Cholinesterases; Female; Injections, Intravenous; Kidney; Liver; Lung; Male; Muscles; Organophosphonates; Oximes; Phosphorus Isotopes; Pralidoxime Compounds; Rats; Time Factors

1970
The use of carbamates and atropine in the protection of animals against poisoning by 1,2,2-trimethylpropyl methylphosphonofluoridate.
    Biochemical pharmacology, 1970, Volume: 19, Issue:3

    Topics: Animals; Atropine; Carbamates; Chickens; Cholinesterase Inhibitors; Dogs; Esters; Female; Fluorine; Guinea Pigs; Male; Mice; Neostigmine; Organophosphate Poisoning; Organophosphonates; Physostigmine; Poisoning; Pyridinium Compounds; Rabbits; Rats; Species Specificity; Time Factors

1970
[Effect of ethyl-p-nitrophenyl phenylphosphonothiate (EPN) on tryptophan pyrrolase activity in relation to miosis and change in serum cholinesterase activities].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1970, Jul-20, Volume: 66, Issue:4

    Topics: Adrenal Glands; Alloxan; Animals; Atropine; Cholinesterases; Depression, Chemical; Dilatation; Ergotamine; Insecticides; Male; Monoamine Oxidase Inhibitors; Nitrobenzenes; Organophosphonates; Phosphorus; Pralidoxime Compounds; Propranolol; Pupil; Rats; Sympatholytics; Tryptophan Oxygenase

1970
Central and peripheral actions of anticholinergic drugs when administered with triflupromazine.
    Neuropharmacology, 1971, Volume: 10, Issue:1

    Topics: Animals; Arousal; Atropine; Benzilates; Cyclopentanes; Drug Synergism; Electroencephalography; Mandelic Acids; Mice; Mydriatics; Organophosphonates; Parasympatholytics; Pyrrolidinones; Salivation; Scopolamine; Tremorine; Triflupromazine

1971
Ageing and reactivation of acetylcholinesterase inhibited with Soman and its thiocholine-like analogue.
    Biochemical pharmacology, 1968, Volume: 17, Issue:8

    Topics: Aging; Animals; Antidotes; Antineoplastic Agents; Atropine; Binding Sites; Cholinesterase Inhibitors; Erythrocytes; Humans; Mice; Organophosphonates; Pralidoxime Compounds; Rabbits

1968
Protective activity of 1,3-disubstituted 2- and 6-pyridones against selected neurotoxic agents.
    Toxicology and applied pharmacology, 1969, Volume: 14, Issue:2

    Topics: Animals; Atropine; Carbamates; Chemical Phenomena; Chemistry; Cholinesterase Inhibitors; Decamethonium Compounds; Hexamethonium Compounds; Male; Mice; Neuromuscular Junction; Organophosphonates; Phosphates; Pyridones; Tubocurarine

1969
Effects of 2-pyridinium aldoxine methochloride and atropine in relation to elevation of blood pH in soman-poisoned dogs.
    Biochemical pharmacology, 1969, Volume: 18, Issue:2

    Topics: Acetylcholinesterase; Acid-Base Equilibrium; Animals; Atropine; Blood Pressure; Cholinesterase Inhibitors; Dogs; Electrocardiography; Erythrocytes; Female; Heart Rate; Hydrogen-Ion Concentration; Hypertension; Injections, Intravenous; Male; Organophosphonates; Phenoxybenzamine; Pralidoxime Compounds; Respiration; Stimulation, Chemical; Time Factors

1969
Dealkylation as a mechanism for aging of cholinesterase after poisoning with pinacolyl methylphosphonofluoridate.
    Biochemical pharmacology, 1965, Volume: 14, Issue:5

    Topics: Acetylcholinesterase; Aging; Animals; Atropine; Brain; Brain Chemistry; Cholinesterase Inhibitors; Diaphragm; Liver; Lung; Organophosphonates; Phosphorus Isotopes; Physostigmine; Rats

1965