Page last updated: 2024-09-05

orantinib and zm 447439

orantinib has been researched along with zm 447439 in 2 studies

Compound Research Comparison

Studies
(orantinib)
Trials
(orantinib)
Recent Studies (post-2010)
(orantinib)
Studies
(zm 447439)
Trials
(zm 447439)
Recent Studies (post-2010) (zm 447439)
110193625017
80725017

Protein Interaction Comparison

ProteinTaxonomyorantinib (IC50)zm 447439 (IC50)
Aurora kinase AHomo sapiens (human)0.1315
Epidermal growth factor receptorHomo sapiens (human)0.11
Cyclin-dependent kinase 4Homo sapiens (human)0.039
G1/S-specific cyclin-D1Homo sapiens (human)0.039
Aurora kinase AMus musculus (house mouse)0.039
Aurora kinase B-AXenopus laevis (African clawed frog)0.045
Aurora kinase BHomo sapiens (human)0.1213

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bhatt, HG; Borisa, AC1
Hajduk, PJ; Johnson, EF; Kifle, L; Merta, PJ; Metz, JT; Soni, NB1

Reviews

1 review(s) available for orantinib and zm 447439

ArticleYear
A comprehensive review on Aurora kinase: Small molecule inhibitors and clinical trial studies.
    European journal of medicinal chemistry, 2017, Nov-10, Volume: 140

    Topics: Animals; Antineoplastic Agents; Aurora Kinases; Cell Proliferation; Clinical Trials as Topic; Humans; Molecular Structure; Protein Kinase Inhibitors; Small Molecule Libraries

2017

Other Studies

1 other study(ies) available for orantinib and zm 447439

ArticleYear
Navigating the kinome.
    Nature chemical biology, 2011, Volume: 7, Issue:4

    Topics: Drug Design; Pharmacogenetics; Protein Kinases; Proteome; Systems Biology

2011