Page last updated: 2024-09-05

opc 4392 and lisuride

opc 4392 has been researched along with lisuride in 2 studies

Compound Research Comparison

Studies
(opc 4392)
Trials
(opc 4392)
Recent Studies (post-2010)
(opc 4392)
Studies
(lisuride)
Trials
(lisuride)
Recent Studies (post-2010) (lisuride)
16107568031

Protein Interaction Comparison

ProteinTaxonomyopc 4392 (IC50)lisuride (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.02
Beta-2 adrenergic receptorHomo sapiens (human)0.041
Beta-1 adrenergic receptorHomo sapiens (human)0.559
Alpha-2A adrenergic receptorHomo sapiens (human)0.0003
Cytochrome P450 2D6Homo sapiens (human)0.016
D(2) dopamine receptorHomo sapiens (human)0.0029
Alpha-2B adrenergic receptorHomo sapiens (human)0.0005
Alpha-2C adrenergic receptorHomo sapiens (human)0.0043
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0005
D(1A) dopamine receptorHomo sapiens (human)0.173
Histamine H2 receptorHomo sapiens (human)1.04
Alpha-1D adrenergic receptorHomo sapiens (human)0.041
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.003
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.02
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.0005
Histamine H1 receptorHomo sapiens (human)0.16
D(3) dopamine receptorHomo sapiens (human)0.0002
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0051
5-hydroxytryptamine receptor 6Homo sapiens (human)0.012

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (100.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Burris, KD; Kikuchi, T; Miwa, T; Mori, T; Stark, A; Tadori, Y; Tottori, K1
Chen, R; Johnson, JL; Jordan, S; Kambayashi, J; Kikuchi, T; Kitagawa, H; McQuade, R; Regardie, K; Tadori, Y1

Other Studies

2 other study(ies) available for opc 4392 and lisuride

ArticleYear
Aripiprazole's low intrinsic activities at human dopamine D2L and D2S receptors render it a unique antipsychotic.
    European journal of pharmacology, 2005, May-16, Volume: 515, Issue:1-3

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; DNA, Complementary; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Humans; Lisuride; Piperazines; Piperidines; Quinolones; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Risperidone; Transfection; Tritium

2005
In vitro functional characteristics of dopamine D2 receptor partial agonists in second and third messenger-based assays of cloned human dopamine D2Long receptor signalling.
    Journal of psychopharmacology (Oxford, England), 2007, Volume: 21, Issue:6

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Calcium Signaling; CHO Cells; Cloning, Molecular; Cricetinae; Cricetulus; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Humans; Immunoblotting; Lisuride; MAP Kinase Signaling System; Microscopy, Confocal; Mitogen-Activated Protein Kinase 1; Phosphorylation; Piperazines; Piperidines; Quinolones; Raclopride; Receptors, Dopamine D2; Schizophrenia; Time Factors; Transfection

2007
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