Page last updated: 2024-09-05

opc 28326 and piperidines

opc 28326 has been researched along with piperidines in 9 studies

Compound Research Comparison

Studies
(opc 28326)
Trials
(opc 28326)
Recent Studies (post-2010)
(opc 28326)
Studies
(piperidines)
Trials
(piperidines)
Recent Studies (post-2010) (piperidines)
91140,2355,22114,545

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (11.11)18.2507
2000's7 (77.78)29.6817
2010's1 (11.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fujiki, H; Imaizumi, T; Kambayashi, J; Kimura, Y; Kishi, M; Mori, T; Orito, K; Shimizu, H; Tanaka, M; Teramoto, S; Tominaga, M; Yoshida, K1
Chen, R; Kambayashi, JI; Li, J; Lockyer, S; Sun, B; Yoshitake, M1
Hashimoto, A; Imaizumi, T; Kambe, T; Kishi, M; Mori, T; Nakazawa, T; Orito, K1
Fujiki, H; Imaizumi, T; Kishi, M; Mori, T; Orito, K; Yoshida, K1
Robins, P1
Czerwiec, FS; Kambayashi, J; Krasa, H; Leatherman, G; Orlandi, C; White, B; Wigley, FM; Wise, RA; Zhong, J1
Chiba, S; Fukui, D; Yang, XP1
Hashimoto, A; Imaizumi, T; Mori, T; Nagai, R; Ohki, T; Sata, M; Sumi, M; Yanaga, K1
Fujiwara, H; Fujiwara, T; Goto, K; Hashimoto, A; Kanamori, H; Kawasaki, M; Minatoguchi, S; Miyakoda, G; Nagashima, K; Nakagawa, M; Ogino, A; Okada, H; Takemura, G; Tsujimoto, A; Yabuuchi, Y1

Trials

1 trial(s) available for opc 28326 and piperidines

ArticleYear
Efficacy and tolerability of a selective alpha(2C)-adrenergic receptor blocker in recovery from cold-induced vasospasm in scleroderma patients: a single-center, double-blind, placebo-controlled, randomized crossover study.
    Arthritis and rheumatism, 2004, Volume: 50, Issue:12

    Topics: Administration, Oral; Adolescent; Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Aniline Compounds; Cold Temperature; Cross-Over Studies; Dose-Response Relationship, Drug; Double-Blind Method; Female; Fingers; Humans; Male; Middle Aged; Piperidines; Raynaud Disease; Regional Blood Flow; Scleroderma, Systemic; Skin Temperature; Vasodilation

2004

Other Studies

8 other study(ies) available for opc 28326 and piperidines

ArticleYear
Mechanisms of action of OPC-28326, a selective hindlimb vasodilator.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:2

    Topics: Adrenergic Antagonists; Anesthesia; Aniline Compounds; Animals; Blood Pressure; Brimonidine Tartrate; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Female; Femoral Artery; Hemodynamics; Hindlimb; In Vitro Techniques; Male; Perfusion; Phenylephrine; Piperidines; Prazosin; Quinoxalines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Vasodilator Agents; Yohimbine

1999
OPC-28326, a selective femoral vasodilator, is an alpha2C-adrenoceptor-selective antagonist.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 299, Issue:2

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Antagonists; Alprostadil; Aniline Compounds; Animals; CHO Cells; Cloning, Molecular; Cricetinae; Femoral Vein; Hindlimb; In Situ Hybridization; In Vitro Techniques; Luciferases; Male; Piperidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Vasodilator Agents; Yohimbine

2001
alpha(2)-adrenoceptor antagonist properties of OPC-28326, a novel selective peripheral vasodilator.
    British journal of pharmacology, 2001, Volume: 134, Issue:4

    Topics: Adrenergic alpha-Antagonists; Aniline Compounds; Animals; Azepines; Binding, Competitive; Blood Pressure; Brimonidine Tartrate; Decerebrate State; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Contraction; Mydriasis; Piperidines; Quinoxalines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Synaptic Transmission; Vas Deferens; Vasodilator Agents; Yohimbine

2001
Effect of oral OPC-28326, a selective femoral arterial vasodilator, on hindlimb subcutaneous tissue temperature in conscious dogs under buprenorphine sedation.
    Japanese journal of pharmacology, 2002, Volume: 88, Issue:1

    Topics: Analgesics, Opioid; Aniline Compounds; Animals; Blood Circulation; Body Temperature; Buprenorphine; Consciousness; Dogs; Femoral Artery; Hindlimb; Male; Piperidines; Rectum; Regional Blood Flow; Thigh; Time Factors; Vasodilation; Vasodilator Agents

2002
Japanese Pharmacological Society--77th Annual Meeting. Part I. 8-10 March 2004, Osaka, Japan.
    IDrugs : the investigational drugs journal, 2004, Volume: 7, Issue:4

    Topics: Aniline Compounds; Animals; Arthritis, Rheumatoid; Bridged Bicyclo Compounds; Dicarboxylic Acids; Drugs, Investigational; Humans; Japan; Myopia; Pharmacology, Clinical; Piperidines; Receptors, Metabotropic Glutamate; Societies, Medical

2004
Neurogenic double-peaked vasoconstriction of human gastroepiploic artery is mediated by both alpha1- and alpha2-adrenoceptors.
    British journal of pharmacology, 2005, Volume: 144, Issue:6

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Aged; Aniline Compounds; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Female; Gastroepiploic Artery; Humans; Male; Middle Aged; Norepinephrine; Perfusion; Piperidines; Prazosin; Receptors, Adrenergic, alpha; Time Factors; Vasoconstriction; Vasoconstrictor Agents; Vasodilator Agents; Yohimbine

2005
OPC-28326, a selective femoral arterial vasodilator, augments ischemia induced angiogenesis.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2007, Volume: 61, Issue:4

    Topics: Aniline Compounds; Animals; Aorta; Blotting, Western; Cells, Cultured; Dose-Response Relationship, Drug; Endothelial Cells; Endothelium, Vascular; Hindlimb; Humans; In Vitro Techniques; Ischemia; Laser-Doppler Flowmetry; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Neovascularization, Physiologic; Nitric Oxide Synthase Type III; Phosphorylation; Piperidines; Rats; Regional Blood Flow; Vasodilator Agents

2007
OPC-28326, a selective peripheral vasodilator with angiogenic activity, mitigates postinfarction cardiac remodeling.
    American journal of physiology. Heart and circulatory physiology, 2015, Jul-01, Volume: 309, Issue:1

    Topics: Angiogenesis Inducing Agents; Aniline Compounds; Animals; Cell Proliferation; Heart; Ki-67 Antigen; Mice; Myocardial Infarction; Myocardium; Myofibroblasts; Nitric Oxide Synthase Type III; Piperidines; Proto-Oncogene Proteins c-akt; Survival Rate; Vasodilator Agents; Ventricular Dysfunction, Left; Ventricular Remodeling

2015