Page last updated: 2024-09-02

opc 21268 and mozavaptan

opc 21268 has been researched along with mozavaptan in 46 studies

Compound Research Comparison

Studies
(opc 21268)
Trials
(opc 21268)
Recent Studies (post-2010)
(opc 21268)
Studies
(mozavaptan)
Trials
(mozavaptan)
Recent Studies (post-2010) (mozavaptan)
13336165824

Protein Interaction Comparison

ProteinTaxonomyopc 21268 (IC50)mozavaptan (IC50)
Vasopressin V2 receptorHomo sapiens (human)0.6373
Vasopressin V1a receptorRattus norvegicus (Norway rat)3.2
Vasopressin V1a receptorHomo sapiens (human)1.1373
Vasopressin V1b receptorHomo sapiens (human)2
Vasopressin V1b receptorRattus norvegicus (Norway rat)5
Vasopressin V2 receptor Rattus norvegicus (Norway rat)0.012

Research

Studies (46)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's34 (73.91)18.2507
2000's11 (23.91)29.6817
2010's1 (2.17)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Berti-Mattera, LN; Dulin, N; Mattera, R; Preston, JA; Thibonnier, M; Wilkins, PL1
Hirano, T; Itai, A; Kan, K; Kondo, K; Kurimura, M; Mori, T; Nakamura, S; Ogawa, H; Shinohara, T; Tanada, Y; Tominaga, M; Yamamura, Y; Yamashita, H1
Chiba, S; Tsukada, M2
Chiba, S; Furukawa, Y; Inoue, Y; Ren, LM; Sawaki, S; Takayama, S1
Harada, K; Hashimoto, M; Mimura, Y; Ogura, T; Oishi, T; Ota, Z; Otsuka, F; Yamauchi, T1
Kanno, Y; Okada, H; Saruta, T; Suzuki, H2
Abe, K; Funyu, T; Inoue, M; Kimura, T; Ohta, M; Ota, K; Sato, K; Shoji, M; Yamamoto, T1
Asano, N; Harada, K; Hashimoto, M; Kageyama, J; Mimura, Y; Ogura, T; Oishi, T; Ota, Z; Yamauchi, T1
Arakawa, K; Ichihara, A; Matsumoto, A; Murakami, M; Naitoh, M; Nakamoto, H; Oka, K; Saruta, T; Suzuki, H; Yamamura, Y1
Kanno, Y; Okada, H; Saruta, T; Suzuki, H; Yamamura, Y2
Burrell, LM; Buxton, BF; Johnston, CI; Liu, JJ; Phillips, PA; Rolls, KA1
Abe, Y; Aki, Y; Fujisawa, Y; Hayashida, Y; Kimura, S; Miyatake, A; Tamaki, T1
Hoshino, J; Kurashina, T; Murata, K; Nakamura, T; Ono, Z; Sakamaki, T; Sato, K1
Burrell, LM; Buxton, BB; Johnston, CI; Liu, JJ; Phillips, PA1
Fujiwara, Y; Nakahama, H; Nakanishi, T; Orita, Y; Sugita, M; Takamitsu, Y; Uyeda, N; Yamada, Y; Yamamura, Y; Yamauchi, A1
Abe, K; Abe, T; Obinata, M; Takahashi, N; Takeuchi, K; Tsutsumi, E; Yanai, N1
Ichihara, A; Matsumoto, A; Murakami, M; Naitoh, M; Nakamoto, H; Saruta, T; Suzuki, H; Yamamura, Y1
Fujisawa, G; Ishikawa, S; Okada, K; Saito, T; Tsuboi, Y1
Hirai, S; Kosaka, K; Mizuno, K; Nishioka, N; Ohno, S; Osada, S; Suzuki, A1
Bax, WA; Bos, E; Nisato, D; Saxena, PR; Stam, WB; Van der Graaf, PH1
Abe, K; Hashimoto, J; Imai, Y; Minami, N; Munakata, M1
Kawano, Y; Matsuoka, H; Nishikimi, T; Saito, Y1
Hanaoka, K; Imai, M; Kurokawa, K; Naruse, M; Yamamura, Y; Yoshitomi, K1
Calò, G; Regoli, D; Rizzi, A; Traina, L1
Goto, A; Hayakawa, H; Hirata, Y; Hirobe, M; Kakoki, M; Kikuchi, K; Kimura, K; Nagano, T; Nagata, D; Omata, M; Suzuki, E; Tojo, A1
Aldred, KL; Burrell, LM; Johnston, CI; Naitoh, M; Phillips, PA; Risvanis, J; Rockell, MD1
Hashimoto, M; Hayakawa, N; Makino, H; Mimura, Y; Ogawa, N; Ogura, T; Otsuka, F; Yamauchi, T1
Bie, P; Christensen, P; Grove, L1
Ishii, N; Kusayama, T; Tahara, A; Tanaka, A; Tomura, Y; Tsukada, J; Uchida, W; Wada, K; Yatsu, T1
Fujita, H; Iwao, H; Miura, K; Omura, T; Takeuchi, K; Yamagishi, H; Yoshikawa, J; Yoshiyama, M1
Ishii, N; Kusayama, T; Saito, M; Sugimoto, T; Tahara, A; Tanaka, A; Tomura, Y; Tsukada, J; Uchida, W; Wada, K; Yatsu, T1
Burrell, LM; Sampey, DB; Widdop, RE1
Haneda, T; Kikuchi, K; Miyata, S; Nakamura, Y; Osaki, J1
Ishiguro, S; Iwasaki, T; Miyamoto, A; Mori, T; Nishio, A1
Otsubo, K1
Japundzic-Zigon, N1
Ferguson, JW; Hayes, PC; Newby, DE; Therapondos, G1
Japundzić-Zigon, N; Jovanović, A; Milutinović, S1
Ishikawa, SE; Sasaki, M1
Cowley, AW; O'Connor, PM1
Kawago, K; Matsuda, K; Nishio, T; Sano, Y; Uchiyama, M; Yamada, T1
Hamada, T; Maejima, S; Matsuda, K; Uchiyama, M; Yamada, T1
Fujimaki-Aoba, K; Hokari, S; Takada, M1

Reviews

3 review(s) available for opc 21268 and mozavaptan

ArticleYear
[Studies on the efficient syntheses of the drug metabolites].
    Yakugaku zasshi : Journal of the Pharmaceutical Society of Japan, 2000, Volume: 120, Issue:11

    Topics: Animals; Anti-Infective Agents; Benzazepines; Chemistry, Organic; Cytochrome P-450 Enzyme System; Fluoroquinolones; Imidazoles; Indans; Lipase; Organic Chemistry Phenomena; Piperazines; Piperidines; Platelet Aggregation Inhibitors; Quinolones; Stereoisomerism; Sulfur Compounds

2000
Therapeutic role of vasopressin receptor antagonism in patients with liver cirrhosis.
    Clinical science (London, England : 1979), 2003, Volume: 105, Issue:1

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Azepines; Benzamides; Benzazepines; Controlled Clinical Trials as Topic; Diuretics; Heart Failure; Homeostasis; Humans; Inappropriate ADH Syndrome; Liver Cirrhosis; Models, Animal; Morpholines; Piperidines; Pyrroles; Quinolones; Rats; Spiro Compounds; Vasopressins

2003
[Renal action of vasopressin].
    Nihon rinsho. Japanese journal of clinical medicine, 2006, Volume: 64 Suppl 2

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Aquaporin 2; Arginine Vasopressin; Benzazepines; Diabetes Insipidus; Diabetes Insipidus, Nephrogenic; Drug Design; Humans; Hyponatremia; Inappropriate ADH Syndrome; Mutation; Piperidines; Quinolones; Receptors, Vasopressin

2006

Other Studies

43 other study(ies) available for opc 21268 and mozavaptan

ArticleYear
The human V3 pituitary vasopressin receptor: ligand binding profile and density-dependent signaling pathways.
    Endocrinology, 1997, Volume: 138, Issue:10

    Topics: Animals; Arachidonic Acid; Base Sequence; Calcium-Calmodulin-Dependent Protein Kinases; Cell Division; CHO Cells; Cricetinae; Cyclic AMP; DNA; Dose-Response Relationship, Drug; Female; Humans; Ligands; Pertussis Toxin; Phenotype; Phosphorylation; Pituitary Gland; Protein Binding; Protein Kinase C; Receptors, Vasopressin; Signal Transduction; Thymidine; Tritium; Type C Phospholipases; Virulence Factors, Bordetella

1997
Novel design of nonpeptide AVP V(2) receptor agonists: structural requirements for an agonist having 1-(4-aminobenzoyl)-2,3,4, 5-tetrahydro-1H-1-benzazepine as a template.
    Journal of medicinal chemistry, 2000, Nov-16, Volume: 43, Issue:23

    Topics: Administration, Oral; Animals; Arginine Vasopressin; Benzazepines; Cyclic AMP; Diuresis; Drug Design; Female; HeLa Cells; Humans; Models, Molecular; Molecular Conformation; Radioligand Assay; Rats; Receptors, Vasopressin; Structure-Activity Relationship

2000
Blocking effects of OPC-21268 and OPC-31260 (vasopressin V1- and V2-receptor antagonists) on vasopressin-induced constrictions in isolated, perfused dog femoral arteries.
    Japanese journal of pharmacology, 1992, Volume: 59, Issue:1

    Topics: Angiotensin Receptor Antagonists; Animals; Benzazepines; Dogs; Dose-Response Relationship, Drug; Femoral Artery; Norepinephrine; Piperidines; Quinolones; Receptors, Vasopressin; Vasoconstriction; Vasopressins

1992
Potent antagonistic action of OPC-31260, a vasopressin V2 receptor antagonist, on [Arg8]vasopressin-induced vasoconstriction in isolated simian femoral arteries.
    European journal of pharmacology, 1992, Oct-20, Volume: 221, Issue:2-3

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Female; Femoral Artery; In Vitro Techniques; Macaca; Male; Norepinephrine; Piperidines; Quinolones; Vasoconstriction

1992
Blocking effects of V1 (OPC-21268) and V2 (OPC-31260) antagonists on the negative inotropic response to vasopressin in isolated dog heart preparations.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 263, Issue:2

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Deamino Arginine Vasopressin; Dogs; Heart; Heart Atria; Perfusion; Piperidines; Quinolones; Receptors, Vasopressin

1992
Effect of vasopressin V1- and V2-receptor stimulation on blood pressure in DOCA-salt hypertensive rats.
    Acta medica Okayama, 1995, Volume: 49, Issue:4

    Topics: Animals; Benzazepines; Blood Pressure; Desoxycorticosterone; Disease Models, Animal; Heart Rate; Male; Piperidines; Quinolones; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Vasopressin; Time Factors

1995
Effect of nonpeptide vasopressin receptor antagonists on developing, and established DOCA-salt hypertension in rats.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 1995, Volume: 17, Issue:3

    Topics: Administration, Oral; Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Blood Pressure; Body Weight; Desoxycorticosterone; Hypertension; Male; Piperidines; Quinolones; Random Allocation; Rats; Rats, Wistar; Sodium Chloride

1995
Effects of V1- and V2-vasopressin (AVP) antagonists on the pressor, AVP and atrial natriuretic peptide responses to a hypertonic saline infusion in conscious anephric rats.
    European journal of endocrinology, 1995, Volume: 133, Issue:1

    Topics: Animals; Atrial Natriuretic Factor; Benzazepines; Blood Pressure; Heart Rate; Hemodynamics; Kidney; Male; Nephrectomy; Neurons, Afferent; Osmolar Concentration; Piperidines; Plasma Volume; Quinolones; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Vasopressin; Saline Solution, Hypertonic; Vasopressins

1995
Effects of novel, nonpeptide vasopressin antagonists on progressive nephrosclerosis in rats.
    Journal of cardiovascular pharmacology, 1995, Volume: 25, Issue:5

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Biomarkers; Blood Pressure; Body Weight; Disease Models, Animal; Diuresis; Glomerulosclerosis, Focal Segmental; Hypertension; Kidney; Male; Nephrectomy; Nephrosclerosis; Piperidines; Proteinuria; Quinolones; Rats; Rats, Inbred SHR

1995
Enhanced pressor response in spontaneously hypertensive rats induced by stimulation of vasopressin-V1 receptors.
    Acta medica Okayama, 1995, Volume: 49, Issue:1

    Topics: Animals; Arginine Vasopressin; Benzazepines; Blood Pressure; Heart Rate; Hypertension; Male; Piperidines; Quinolones; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Vasopressin; Stimulation, Chemical

1995
Effects of oral AVP receptor antagonists OPC-21268 and OPC-31260 on congestive heart failure in conscious dogs.
    The American journal of physiology, 1994, Volume: 267, Issue:6 Pt 2

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Body Weight; Capillary Resistance; Cardiac Output; Cardiac Pacing, Artificial; Diuresis; Dogs; Heart Failure; Hemodynamics; Kidney; Male; Natriuresis; Osmolar Concentration; Piperidines; Potassium; Quinolones; Renin; Sodium

1994
Chronic and selective vasopressin blockade in spontaneously hypertensive rats.
    The American journal of physiology, 1994, Volume: 267, Issue:6 Pt 2

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Blood Pressure; Hypertension; Male; Osmolar Concentration; Piperidines; Quinolones; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Vasopressin; Urine; Vasopressins

1994
Vascular responses to vasopressin antagonists in man and rat.
    Clinical science (London, England : 1979), 1994, Volume: 87, Issue:4

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Culture Techniques; Dose-Response Relationship, Drug; Female; Humans; Mammary Arteries; Mesenteric Artery, Superior; Piperidines; Quinolones; Rats; Rats, Sprague-Dawley; Species Specificity; Vasoconstriction

1994
Role of vasopressin on cardiovascular changes during hemorrhage in conscious rats.
    The American journal of physiology, 1994, Volume: 267, Issue:5 Pt 2

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Blood Pressure; Heart Rate; Hemorrhage; In Vitro Techniques; Kidney; Male; Piperidines; Quinolones; Rats; Rats, Sprague-Dawley; Renal Artery; Sympathetic Nervous System; Time Factors

1994
Effect of vasopressin V (OPC-21268) and V2 (OPC-31260) antagonists on renal hemodynamics and excretory function.
    Life sciences, 1994, Volume: 55, Issue:4

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Blood Pressure; Glomerular Filtration Rate; Kidney; Male; Osmolar Concentration; Piperidines; Quinolones; Rats; Rats, Wistar; Renal Circulation; Urine

1994
Human internal mammary artery responses to non-peptide vasopressin antagonists.
    Clinical and experimental pharmacology & physiology, 1994, Volume: 21, Issue:2

    Topics: Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Arteries; Benzazepines; Breast; Female; Humans; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Piperidines; Quinolones; Receptors, Vasopressin; Regional Blood Flow

1994
Organic osmolytes in rat renal inner medulla are modulated by vasopressin V1 and/or V2 antagonists.
    The American journal of physiology, 1994, Volume: 267, Issue:1 Pt 2

    Topics: Aldehyde Reductase; Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Diuresis; Kidney Medulla; Male; Osmolar Concentration; Osmosis; Piperidines; Quinolones; Rats; Rats, Wistar; RNA, Messenger; Urine; Water Deprivation

1994
Different cellular mechanisms of vasopressin receptor V1 and V2 subtype in vasopressin-induced adenosine 3', 5'-monophosphate formation in an immortalized renal tubule cell line, TKC2.
    Biochemical and biophysical research communications, 1994, Jul-29, Volume: 202, Issue:2

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Antigens, Polyomavirus Transforming; Benzazepines; Calcium; Cell Line, Transformed; Cyclic AMP; Dinoprostone; Indomethacin; Kidney Tubules; Mice; Mice, Transgenic; Piperidines; Quinolones; Receptors, Vasopressin; Vasopressins

1994
Effects of vasopressin V1 and V2 receptor antagonists on progressive renal failure in rats.
    Clinical science (London, England : 1979), 1994, Volume: 86, Issue:4

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Kidney; Kidney Failure, Chronic; Male; Piperidines; Quinolones; Rats; Rats, Wistar; Urine

1994
Arginine vasopressin produces renal vasodilation via V2 receptors in conscious dogs.
    The American journal of physiology, 1993, Volume: 265, Issue:4 Pt 2

    Topics: Animals; Arginine Vasopressin; Benzazepines; Deamino Arginine Vasopressin; Diuresis; Dogs; Drug Combinations; Hemodynamics; Male; Natriuresis; Osmolar Concentration; Piperidines; Quinolones; Receptors, Vasopressin; Renal Circulation; Vasodilation

1993
Nonpeptide vasopressin antagonist and its application in the correction of experimental hyponatremia in rats.
    Regulatory peptides, 1993, Apr-29, Volume: 45, Issue:1-2

    Topics: Animals; Benzazepines; Cells, Cultured; Hyponatremia; Inappropriate ADH Syndrome; Kidney Tubules, Collecting; Muscle, Smooth, Vascular; Piperidines; Quinolones; Rats; Rats, Brattleboro; Rats, Sprague-Dawley; Vasopressins

1993
Wortmannin inhibits the activation of MAP kinase following vasopressin V1 receptor stimulation.
    FEBS letters, 1995, Dec-27, Volume: 377, Issue:3

    Topics: Androstadienes; Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Deamino Arginine Vasopressin; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Fibroblasts; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Piperidines; Quinolones; Rats; Receptors, Vasopressin; Signal Transduction; Tetradecanoylphorbol Acetate; Wortmannin

1995
[Arg8]vasopressin-induced responses of the human isolated coronary artery: effects of non-peptide receptor antagonists.
    European journal of pharmacology, 1995, Oct-16, Volume: 285, Issue:2

    Topics: Adolescent; Adult; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Child; Coronary Vessels; Endothelium, Vascular; Female; Humans; In Vitro Techniques; Indoles; Male; Middle Aged; Muscle, Smooth, Vascular; Piperidines; Potassium; Pyrrolidines; Quinolones; Vasoconstrictor Agents

1995
Effects of vasopressin V1 and V2 receptor antagonists on the development of salt-induced hypertension in Dahl rats.
    Journal of cardiovascular pharmacology, 1995, Volume: 26, Issue:4

    Topics: Analysis of Variance; Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Blood Pressure; Blood Pressure Determination; Diuresis; Hypertension; Male; Piperidines; Quinolones; Rats; Sodium Chloride

1995
Effect of long-term treatment with selective vasopressin V1 and V2 receptor antagonist on the development of heart failure in rats.
    Journal of cardiovascular pharmacology, 1996, Volume: 27, Issue:2

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Drug Administration Schedule; Heart Failure; Hemodynamics; Male; Organ Size; Piperidines; Quinolones; Random Allocation; Rats; Rats, Wistar

1996
Functional characterization of vasopressin V1 and V2 receptors in the rabbit renal cortical collecting duct.
    Kidney international. Supplement, 1996, Volume: 55

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Calcium; Cyclic AMP; Electrophysiology; In Vitro Techniques; Kidney Cortex; Kidney Tubules, Collecting; Male; Membrane Potentials; Patch-Clamp Techniques; Piperidines; Quinolones; Rabbits; Receptors, Vasopressin; Renal Agents; Sodium

1996
Pharmacological characterization of a vasopressin V1 receptor in the isolated human gastric artery.
    Life sciences, 1997, Volume: 60, Issue:4-5

    Topics: Aged; Aged, 80 and over; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Arteries; Benzazepines; Humans; In Vitro Techniques; Indoles; Middle Aged; Muscle, Smooth, Vascular; Oxytocin; Piperidines; Pyrrolidines; Quinolones; Receptors, Vasopressin; Stomach; Vasoconstrictor Agents

1997
Receptor subtype for vasopressin-induced release of nitric oxide from rat kidney.
    Hypertension (Dallas, Tex. : 1979), 1997, Volume: 29, Issue:1 Pt 1

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Desoxycorticosterone; Dinoprost; Dose-Response Relationship, Drug; Enzyme Inhibitors; In Vitro Techniques; Kidney; Male; Nitric Oxide; omega-N-Methylarginine; Perfusion; Piperidines; Quinolones; Rats; Rats, Wistar; Receptors, Vasopressin; Renal Agents

1997
Modulation of genetic hypertension by short-term AVP V1A or V2 receptor antagonism in young SHR.
    The American journal of physiology, 1997, Volume: 272, Issue:2 Pt 2

    Topics: Angiotensin-Converting Enzyme Inhibitors; Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Blood Pressure; Hypertension; Male; Myocardium; Organ Size; Piperidines; Quinolones; Ramipril; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Systole; Time Factors

1997
In vitro macro- and microautoradiographic localization of V1 and V2 receptors in the rat kidney using OPC-21268 and OPC-31260.
    Nephron, 1997, Volume: 76, Issue:3

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Autoradiography; Benzazepines; In Vitro Techniques; Kidney; Ligands; Male; Piperidines; Quinolones; Rats; Rats, Wistar; Receptors, Vasopressin; Tissue Distribution; Tritium; Vasopressins

1997
Effects of receptor blockade on metabolism and renal actions of vasopressin in conscious dogs.
    Acta physiologica Scandinavica, 1998, Volume: 163, Issue:1

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Dimethyl Sulfoxide; Dogs; Female; Glomerular Filtration Rate; Hemodynamics; Hormones; Kidney; Natriuresis; Piperidines; Quinolones; Solvents; Vasopressins

1998
Effect of YM087, a potent nonpeptide vasopressin antagonist, on vasopressin-induced protein synthesis in neonatal rat cardiomyocyte.
    Cardiovascular research, 1998, Volume: 38, Issue:1

    Topics: Analysis of Variance; Animals; Animals, Newborn; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Leucine; Myocardium; Piperidines; Protein Biosynthesis; Quinolones; Rats; Rats, Wistar; Receptors, Vasopressin; Stimulation, Chemical; Thymidine

1998
The effect of vasopressin V1- and V2-receptor antagonists on hemodynamics in early and late phase after myocardial infarction in rats.
    Japanese journal of pharmacology, 1998, Volume: 78, Issue:2

    Topics: Administration, Oral; Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Heart Ventricles; Hemodynamics; Male; Myocardial Infarction; Organ Size; Piperidines; Quinolones; Rats; Rats, Wistar; Time Factors; Vasopressins; Ventricular Function, Left

1998
Pharmacological characterization of the human vasopressin receptor subtypes stably expressed in Chinese hamster ovary cells.
    British journal of pharmacology, 1998, Volume: 125, Issue:7

    Topics: Animals; Benzazepines; Binding, Competitive; Calcium; CHO Cells; Cricetinae; Cyclic AMP; Humans; Indoles; Morpholines; Piperidines; Pyrrolidines; Quinolones; Receptors, Vasopressin; Spiro Compounds; Transfection; Tritium

1998
Vasopressin V2 receptor enhances gain of baroreflex in conscious spontaneously hypertensive rats.
    The American journal of physiology, 1999, Volume: 276, Issue:3

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Baroreflex; Benzazepines; Blood Pressure; Heart Rate; Injections, Intravenous; Male; Piperidines; Quinolones; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Receptors, Vasopressin

1999
Hypertrophic growth of cultured neonatal rat heart cells mediated by vasopressin V(1A) receptor.
    European journal of pharmacology, 2000, Mar-10, Volume: 391, Issue:1-2

    Topics: Animals; Animals, Newborn; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Blotting, Northern; Calcium; Cardiomegaly; Cells, Cultured; Culture Media; DNA; Kinetics; Myocardium; Piperidines; Protein Biosynthesis; Protein Kinase C; Proteins; Proto-Oncogene Proteins c-fos; Quinolones; Rats; Rats, Sprague-Dawley; Receptors, Vasopressin; RNA, Messenger; Second Messenger Systems; Vasopressins

2000
Vasopressin receptor subtypes on mesenteric and cremasteric arterioles in rat.
    European journal of pharmacology, 2000, Jul-14, Volume: 400, Issue:1

    Topics: Animals; Arginine Vasopressin; Arterioles; Benzazepines; Male; Mesenteric Arteries; Muscle, Skeletal; Piperidines; Quinolones; Rats; Rats, Wistar; Receptors, Vasopressin; Vasoconstriction

2000
Effects of nonpeptide V1a and V2 antagonists on blood pressure fast oscillations in conscious rats.
    Clinical and experimental hypertension (New York, N.Y. : 1993), 2001, Volume: 23, Issue:4

    Topics: Analysis of Variance; Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Blood Pressure; Heart Rate; Hemorrhage; Hypovolemia; Male; Piperidines; Quinolones; Rats; Receptors, Vasopressin

2001
Effects of nonpeptide and selective V1 and V2 antagonists on blood pressure short-term variability in spontaneously hypertensive rats.
    Journal of pharmacological sciences, 2004, Volume: 95, Issue:1

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Blood Pressure; Hypertension; Male; Piperidines; Quinolones; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Vasopressin

2004
Vasopressin-induced nitric oxide production in rat inner medullary collecting duct is dependent on V2 receptor activation of the phosphoinositide pathway.
    American journal of physiology. Renal physiology, 2007, Volume: 293, Issue:2

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Calcium; Calcium-Transporting ATPases; Cyclic AMP-Dependent Protein Kinases; Kidney Medulla; Kidney Tubules, Collecting; Male; Nitric Oxide; Phosphatidylinositols; Piperidines; Quinolones; Rats; Rats, Sprague-Dawley; Receptors, Vasopressin; Signal Transduction; Spectrometry, Fluorescence; Type C Phospholipases; Vasopressins

2007
Effects of arginine vasotocin and vasopressin receptor antagonists on Na+ and Cl- transport in the isolated skin of two frog species, Hyla japonica and Rana nigromaculata.
    General and comparative endocrinology, 2008, May-15, Volume: 157, Issue:1

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Anura; Benzazepines; Biological Transport; Chlorides; Colforsin; Dose-Response Relationship, Drug; Electrophysiology; Female; In Vitro Techniques; Male; Piperidines; Quinolones; Receptors, Vasopressin; Skin; Sodium; Species Specificity; Time Factors; Vasotocin

2008
Effects of hypertonic stimuli and arginine vasotocin (AVT) on water absorption response in Japanese treefrog, Hyla japonica.
    General and comparative endocrinology, 2008, Volume: 157, Issue:2

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Biological Transport; Central Nervous System; Dose-Response Relationship, Drug; Glucose Solution, Hypertonic; Hypertonic Solutions; Osmotic Pressure; Piperidines; Quinolones; Ranidae; Receptors, Vasopressin; Saline Solution, Hypertonic; Vasotocin; Water; Water-Electrolyte Balance

2008
Effects of arginine vasotocin and mesotocin on the activation and development of amiloride-blockable short-circuit current across larval, adult, and cultured larval bullfrog skins.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 2010, Volume: 180, Issue:3

    Topics: Adrenal Cortex Hormones; Amiloride; Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Colforsin; Electrophysiological Phenomena; Epithelial Sodium Channel Blockers; Epithelial Sodium Channels; Epithelium; Gene Expression; Larva; Oxytocin; Piperidines; Quinolones; Rana catesbeiana; Receptors, Oxytocin; Receptors, Pituitary Hormone; Receptors, Vasopressin; Skin; Vasotocin

2010